Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
12/2000
12/14/2000WO2000074676A1 Use of riluzole for the treatment of multiple sclerosis
12/14/2000WO2000029378A3 Acyclic and cyclic guanidine- and acetamidine derivatives, their preparation and their use as pesticides, esp. as parasiticides
12/14/2000CA2375874A1 Use of riluzole for the treatment of multiple sclerosis
12/14/2000CA2371158A1 Diaminothiazoles and their use for inhibiting protein kinases
12/13/2000EP1059302A1 Factor VIIa inhibitors
12/13/2000EP1059293A1 Novel amino chlorothiazole compounds
12/13/2000EP1059288A1 Process for the ring cleavage of thiazolidine derivatives
12/13/2000EP1058682A1 Heterocyclic diarylmethylene derivatives, methods of preparing them and their uses in therapeutics
12/13/2000EP1058679A1 Synthesis of epothilones, intermediates thereto and analogues therof
12/13/2000CN1276790A Carboxamidothiazole derivs., preparation, pharmaceutical composition contg. them
12/13/2000CN1276789A 4-aminothiazole derivs, their preparation and their use as inhibitors of cyclin-dependent kinases
12/13/2000CN1276785A N-aroylphenylalanine derivs.
12/13/2000CN1059437C Method for preparation of cyanoimino-1,3-thiazolidine compounds
12/12/2000US6160129 Cyclopentane heptan(ene)oic acid, 2-heteroarylalkenyl derivatives as therapeutic agents
12/12/2000US6160126 Useful in preparing guanidine derivatives useful as insecticides and miticides
12/12/2000US6160122 Chemical intermediates for hiv protease inhibiting
12/12/2000US6160112 Inhibitors of beta-lactamase
12/12/2000US6160024 Photoactivated antiviral and antitumor compositions
12/12/2000US6160012 Leukotriene B4 derivatives, in particular oximo-LTB4 - antagonists
12/12/2000US6159998 Administered as vasodilators, analgesics, anesthetics, sedatives, and anitspasmodic agents
12/12/2000US6159996 Polycyclic thiazolidin-2-ylidene amines, process for their preparation, and their use as pharmaceuticals
12/12/2000US6159995 Substituted diaminocarboxylic acids
12/12/2000US6159979 Bicyclic aryl or a bicyclic heterocyclic ring containing compounds having a combined 5HT1A, 5HT1B and 5HT1D receptor antagonistic activity
12/12/2000US6159973 Aromatic amides, their preparation process, the compositions containing them and their use as pesticides
12/12/2000CA2038060C Iminothiazolines, their production and use as herbicides, and intermediates for their production
12/07/2000WO2000073283A1 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
12/07/2000WO2000073266A1 Novel antioxidants, preparation methods and uses
12/07/2000WO2000073252A1 6-hydroxy-2-naphthylcarbinol and process for the preparation thereof
12/07/2000WO2000031247A3 Recombinant methods and materials for producing epothilone and epothilone derivatives
12/07/2000CA2376024A1 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
12/07/2000CA2375348A1 Novel antioxidants, preparation methods and uses
12/07/2000CA2375019A1 6-hydroxy-2-naphthylcarbinol and method for preparing the same
12/06/2000EP1056743A1 Benzamine derivatives
12/06/2000EP1056732A2 4-aminothiazole derivatives, their preparation and their use as inhibitors of cyclin-dependent kinases
12/06/2000CN1275982A Novel heterocyclic compounds process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
12/06/2000CN1275909A In-modulators
12/06/2000CN1059207C Herbicidal saccharin carboxylic and itsester defivatives and method for their prepn.
12/05/2000US6156937 Nonionic surfactants; water and oil repellency
12/05/2000US6156905 Deoxy epothilones and intermediates utilized in the process for preparing epothilones
12/05/2000US6156904 2-(4-chloro-4,4-difluorobutylthio)thiazole used as agricultural nematocide
12/05/2000US6156794 Nervous system disorders or alzheimers disease
12/05/2000US6156776 Diaryl substituted thiazoles useful in the treatment of fungal infections
12/05/2000US6156773 Pharmaceutical composition
12/05/2000US6156763 Enzyme inhibitors with heterocyclic diimides
12/05/2000US6156761 Substituted tetralone derivatives for enhancing cognition
12/05/2000US6156759 Nonnucleoside inhibitors of reverse transcriptase, composite binding pocket and method for use thereof
12/05/2000US6156748 Compounds useful as neuro-protective agents
12/05/2000US6156494 Solid phase synthesis using substrate having regions, each region is an optical fiber having covalently bound reactive groups; fibers are used to direct light, heat or both to compounds tethered to its surface
11/2000
11/30/2000WO2000071540A1 Hydrochloride of fused-heterocycle compound
11/30/2000WO2000071500A1 Halogen compounds
11/30/2000WO2000043535A3 Composition and device for detecting leukocytes in urine
11/30/2000WO2000032598A9 Methods and compositions for treating inflammatory diseases utilizing inhibitors of tumor necrosis factor activity
11/29/2000EP1055665A1 3-(3-Hydroxyphenyl)-3-amino-propionamide derivatives
11/29/2000EP1054858A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
11/29/2000EP1054857A1 Biaryl-acetic acid derivatives and their use as cox-2 inhibitors
11/29/2000CN1275126A Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof
11/29/2000CN1275123A Prostaglandin agonists and their use to treat bone disorders
11/29/2000CN1058964C Branched-amino-sbustituted thiazoles, process for their preparation and the pharmaceutical compositions which contain them
11/28/2000US6153763 A microbicides comprising an imidazole ring
11/28/2000US6153759 Herbicide comprising a 5-membered or 6-membered heterocyclic, saturated or unsaturated radical containing one to three hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen
11/28/2000US6153630 Phenylpyridyl compounds for inhibiting phosphodiesterase IV and methods of using same
11/28/2000US6153622 Estrogen agonists/antagonists
11/28/2000US6153611 As non-dopaminergic antiischemic compounds for treating brain disorders
11/23/2000WO2000069838A1 Ion channel modulating agents
11/23/2000WO2000069827A1 Hydroxamic and carboxylic acid derivatives
11/23/2000WO2000069810A1 Glucagon antagonists/inverse agonists
11/23/2000WO2000043371A3 Fused ring heteroaryl and heterocyclic compounds which inhibit leukocyte adhesion mediated by vla-4
11/23/2000WO2000043354A3 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4
11/23/2000WO1999065871A3 Thiolesters and uses thereof
11/23/2000DE19922934A1 New 5,5-dihalo- or 4,5,5-trihalo-4-pentenoic acid derivatives, useful as bactericides, fungicides, insecticides, acaricides and nematocides, especially plant fungicides
11/23/2000CA2373892A1 Glucagon antagonists/inverse agonists
11/22/2000EP1053237A2 Inhibition of human telomerase by a g-quadruplex-interaction compound
11/22/2000EP1052989A1 Use of 2-amino-6- trifluoromehthoxy- benzothiazole for preventing or treating cerebellum dysfunction
11/22/2000CN1274288A Peptide-containing & alpha; -ketoamide cysteine and serine protease inhibitors
11/21/2000US6150537 Methods for the esterification of alcohols and compounds useful therefor as potential anticancer agents
11/21/2000US6150530 Amidation of amine with acid
11/21/2000US6150394 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
11/21/2000US6150389 Antidepressants; treating elevated intraocular pressure, e.g., glaucoma; antidiabetic agents for non-insulin dependent diabetes, sexual disorders, e.g., male impotence and obesity; e.g. trans-2-(3-phenyl-bicyclo(2.2.1)heptyl)-2-aminooxazoline
11/21/2000US6150384 Pharmaceutical composition
11/21/2000US6150383 Comprising an insulin sensitivity enhancer in combination with one or more other antidiabetics differing from the enhancer in mechanism of action; lipid/glycometabolism disorders; antidiabetic agents; side effect reduction
11/21/2000US6150378 Peptidyl-containing α-ketoamide cysteine and serine protease inhibitors
11/21/2000US6150370 1,3-dinitrocyclic compound treats numerous diseases caused by undesired metalloprotease activity, such as tumor metastasis, osteoarthritis, rheumatoid arthritis, skin inflammation, ulcerations, and periodontitis
11/21/2000US6150307 Heterocyclic thioethers as additives for lubricants
11/21/2000US6150129 Antimicrobial determination of N-(aminoalkyl) and/or N-(Amidoalkyl) dinitrogen heterocyclic compositions
11/21/2000US6150083 Naptho(1,2-d)thiazolium derivative cyanine dyes; high contrast black and white and multicolor printing; photosensitivity; stain resistance
11/16/2000WO2000068210A1 Benzohetero cyclylcyclo hexenones and their use as herbicides
11/16/2000WO2000068178A1 Novel compounds
11/16/2000WO2000067801A2 Prodrugs of chemotherapeutic agents with oxaalkanoic acids
11/16/2000WO2000067753A1 Parenteral formulation of 5-(2-chloroethyl)-4-methylthiazole edisylate(clomethiazole edisylate)
11/16/2000WO2000015634A3 Hiv protease inhibitors
11/16/2000DE19923001A1 New epothilone derivatives, used as mitosis regulators e.g. for treating malignant tumors, psoriasis or arthritis
11/16/2000DE19919336A1 Hydrolysis of thiazolidine derivative using acidic cation exchanger, giving 2-aminomercaptan derivative, e.g. cysteine or penicillamine, and carbonyl compound in high yield and purity
11/16/2000CA2373137A1 Benzohetero cyclylcyclo hexenones and their use as herbicides
11/16/2000CA2368831A1 Permeable, water soluble, non-irritating prodrugs of chemotherapeutic agents with oxaalkanoic acids
11/16/2000CA2336673A1 Novel compounds
11/15/2000EP1052256A1 Process for producing aminomethylated heterocyclic derivative
11/15/2000EP1052255A1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics.
11/15/2000EP1052250A1 Sulfonylalkanoylamino hydroxyethylamino sulfonamide retroviral protease inhibitors
11/15/2000EP1052238A1 Novel tricyclic compound
11/15/2000EP1051399A1 Phenylalanine derivatives useful as pharmaceutical agents