Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
05/2000
05/30/2000US6069247 Reacting an acetylenecarboxy amide and an aryl or heterocyclyl halide or a group enhancing the electrophilicity of the atom to which it is attached for displacement; using a palladium compound catalyst, a base and an acid
05/30/2000US6069163 Azapeptide acids as cell adhesion inhibitors
05/30/2000US6069157 Parasiticidal compounds
05/25/2000WO2000012482A3 Indazole derivatives with 5-ht2 receptor activity
05/25/2000WO2000011951A3 Use of 5-amino-pyrazol-derivatives for combating micro-organisms
05/25/2000DE19853560A1 Single-stage preparation of 4-substituted pyrazole compounds useful e.g. as insecticides, from new or known 4-unsubstituted compound and halide
05/24/2000EP1002798A1 An improved process for preparing a therapeutically active pyrazolopyrimidinone derivative
05/24/2000EP1001941A1 Fused heterocyclic compounds and their use as kynurenine-3-hydroxylase inhibitors
05/24/2000EP1001940A1 Condensed pyrazole compounds
05/24/2000EP1001939A1 Heterocyclic substituted 4-benzoyl-pyrazole as herbicides
05/24/2000EP1001938A1 2-benzoyl-cyclohexane-1,3-dione as herbicides
05/24/2000EP1001937A1 Method for producing 2-(3-pyrazolyl-oxymethylene) nitrobenzenes
05/24/2000EP1001927A2 Novel polyamine analogues as therapeutic and diagnostic agents
05/24/2000EP0626969B1 CoA-IT AND PAF INHIBITORS
05/24/2000CN1254330A Cycloalkyl benzyl ether compounds
05/23/2000US6066756 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
05/23/2000US6066735 Treatment of erectile dysfunction
05/18/2000WO2000027822A2 Tricyclic pyrazole derivatives
05/18/2000WO2000027821A1 Method for producing 1-substituted 5-hydroxypyrazoles
05/18/2000WO2000027627A1 Aryloxime linkers in the solid-phase synthesis of 3-aminobenzisoxazoles
05/18/2000WO2000027394A1 Activators of soluble guanylate cyclase
05/18/2000CA2350235A1 Tricyclic pyrazole derivatives
05/18/2000CA2349244A1 Method for producing 1-substituted 5-hydroxypyrazoles
05/17/2000EP1000930A2 Tachykinin antagonists
05/17/2000EP1000617A2 Treatment of platelet derived growth factor related disorders such as cancers using inhibitors of platelet derived growth receptor
05/17/2000EP1000062A1 Tricyclic vasopressin agonists
05/17/2000EP1000025A1 Substituted naphthopyrans
05/17/2000EP1000018A2 Urokinase inhibitors
05/17/2000EP1000012A1 Process for converting propargylic amine-n-oxides to enaminones
05/17/2000EP0999836A1 A pharmaceutical composition active in reducing production of mcp-1 protein
05/17/2000EP0848701B1 O-benzyl oxime ether derivatives and their use in crop protection compositions
05/17/2000EP0804191B1 Use of inhibitors of platelet derived growth receptor for the manufacture of a medicament for the treatment of cancers
05/17/2000CN1253561A Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3', 5'-monophosphate phosphodiesterase (cGMP PDE5) for treatment of sexual dysfunction
05/17/2000CN1253502A Method of using cyclooxygenase-2 inhibitors in prevention of cardiovascular disorders
05/17/2000CN1253501A IL-8 receptor antagonists
05/16/2000US6063860 A polyisocyanate is blocked with a substituted pyrazole forms polyetherurethane copolymer or polylactone-urethane copolymer or polyurethane polymer; used as a coating
05/16/2000US6063800 Modulators of molecules with phosphotyrosine recognition units
05/16/2000US6063798 Substituted N-methylenethioureas as pesticides
05/16/2000US6063734 Agricultural chemicals, agents for preventing attachment of aquatic organisms
05/11/2000WO2000007542A3 Utilization of aryl(or heteroaryl)azolylcarbinol derivatives in the preparation of a medicament for the treatment of troubles mediated by an excess of substance p
05/10/2000CN1252803A Herbicidal sulfonamides
05/10/2000CN1252790A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
05/10/2000CN1252713A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
05/09/2000US6060605 Process for producing substituted arylpyrazoles
05/09/2000US6060502 Agriculture; pesticides for control of arthropods, helminths, nematodes, protozoa
05/09/2000US6060495 Pesticidal sulfur compounds
05/09/2000US6060432 Synergistic mixture; crops, agriculture
05/04/2000WO2000024745A1 PYRAZOLOPYRIMIDINONE cGMP PDE5 INHIBITORS FOR THE TREATMENT OF SEXUAL DYSFUNCTION
05/03/2000EP0997153A1 Formulations for lipophilic compounds
05/03/2000CN1252059A Pesticidal 1-aryl-3-iminopyrazoles
05/02/2000US6057362 Protease inhibitors
05/02/2000US6057354 Pesticidal 1-arylpyrazoles
05/02/2000US6057335 Treatment of bulimia, obesity or diabetes
05/02/2000US6057270 Herbicides
04/2000
04/27/2000WO2000023421A1 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES
04/27/2000CA2347792A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
04/26/2000EP0995750A1 Pyrazolopyrimidinone cGMP PDE5 inhibitors for the treatment of sexual dysfunction
04/26/2000EP0995747A1 Substituted sulfonylphenylheterocycles as cyclooxygenase-2 and 5-lipoxygenase inhibitors
04/26/2000EP0995742A1 Sulfonamide compounds and medicinal use thereof
04/26/2000EP0995439A1 Use of indazole derivatives in the manufacture of a medicament for treating congestive heart failure
04/26/2000EP0994848A1 Glucagon antagonists/inverse agonists
04/26/2000EP0810998B1 Phenyl diketone derivatives as herbicides
04/26/2000CN1251578A Pyrazole derivative
04/26/2000CN1251524A Pharmaceutical composition for oral administration of N-piperidino-3-phrazolecarboxamide derivative, its salts and their solvates
04/25/2000US6054592 Chemical intermediate for pesticide, fungicide
04/25/2000US6054473 1,3-dimethyl-5-fluoro-pyrazole-4-carboxamide derivatives, their preparation and their use as microbicides
04/25/2000US6054460 Anticonvulsive and antiallergic/antiasthmatic pyrazolo-[3,4-d]pyrimidines, and process for preparing
04/25/2000US6054413 1-sulfonyl-3-phenylpyrazoles and their use as herbicides and for desiccating or defoliating plants
04/25/2000US6054412 Substituted 4,5-di(trifluoromethyl)pyrazoles and their use as herbicides and for desiccating/defoliating plants
04/25/2000CA2004776C Process for the preparation of perfluoroalkylthioethers
04/21/2000CA2287139A1 Method for treating congestive heart failure
04/20/2000WO2000022129A1 Non-endogenous, constitutively activated human g protein-coupled receptors
04/20/2000WO2000021987A2 A method of identifying modulators of cell surface membrane receptors useful in the treatment of disease
04/20/2000WO1999048868A9 Heterocyclic classes of compounds for the modulating tyrosine protein kinase
04/20/2000CA2342314A1 Non-endogenous, constitutively activated human g protein-coupled receptors
04/19/2000EP0994115A2 Process for preparation of pyrazolo-(4,3-d)pyrimidin-7-ones and intermediates thereof
04/19/2000EP0993441A1 INHIBITORS OF p38
04/18/2000US6051573 Treatment of GLC1A glaucoma with non-steroidal glucocorticoid antagonists
04/18/2000CA2010180C Pesticidal 3-cyano-5-alkoxy-1-arylpyrazoles
04/13/2000WO2000020399A2 Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for the production thereof and agents containing the same
04/13/2000WO2000019994A1 Estrogen receptor ligands
04/13/2000WO2000002850A3 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
04/12/2000EP0991638A1 NOVEL GUANIDINE MIMICS AS FACTOR Xa INHIBITORS
04/12/2000EP0991625A2 Inhibitors of factor xa with a neutral p1 specificity group
04/12/2000CN1250447A 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
04/12/2000CN1250441A Pesticidal 1-arylpyrazoles
04/12/2000CN1250440A Process for preparing pyrazole derivatives
04/11/2000US6048885 Fungicides
04/11/2000US6048852 Bactericides
04/11/2000CA2009503C Ethers of 1-benzyl-3-hydroxymethyl-indazole with aliphatic 2-hydroxyacids
04/06/2000WO2000018741A2 Pyrazole compounds as cox-2 inhibitors
04/06/2000WO2000018738A1 Benzamide derivatives and their use as cytokine inhibitors
04/06/2000CA2340454A1 Benzamide derivatives and their use as cytokine derivatives
04/05/2000EP0990650A1 Tricyclic pyrrole or pyrazole derivatives
04/05/2000EP0990649A1 Benzoylpyrazole derivatives having specified substituents and herbicides
04/05/2000EP0990645A1 Novel sulfonamide derivatives
04/05/2000EP0989971A1 Glyoxylic acid amides
04/05/2000EP0785923B1 Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production
04/05/2000CN1249747A Processes for preparing pesticidal intermediates
04/05/2000CN1051078C Pyrazolinyl compounds contg. composition for preventing crop from detriment of herbicides, method for preparing same