Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
07/2001
07/26/2001US20010009962 One pot process for preparing sildenafil (drug for erectile dysfunction) and derivatives by reacting for example 4-(2-methoxy-5-(4-methyl-1-piperazinylsulfonyl)benzamido)-1-methyl-3-propyl -1H-pyrazole-5-carboxamide with ethanol
07/26/2001US20010009044 Mixing with an oxidant, applying to hair, and washing out after a certain time with water and shampoo
07/26/2001CA2397686A1 Gyrase inhibitors and uses thereof
07/26/2001CA2394703A1 Amide compounds for inhibiting protein kinases
07/26/2001CA2388885A1 Indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation
07/25/2001EP1117650A2 Use of substituted 5-hydroxypyrazoles, novel 5-hydroxypyrazoles, methods for the production thereof and agents containing the same
07/25/2001EP1117397A1 Geometrically restricted 2-indolinone derivatives as modulators of protein kinase activity
07/25/2001EP0966445B1 Processes for preparing pesticidal intermediates
07/25/2001EP0888306B1 Cosmetic compositions containing pyrazolin-4,5-diones, novel pyrazolin-4,5-diones, preparation methods therefor and uses thereof
07/25/2001EP0854861B1 Oxyamino oxime ethers, methods and intermediate products for their production, and agents containing them and used for controlling harmful fungi and pests
07/25/2001CN1305462A Novel 1,5 and 3-O-substituted 1H-indazoles with anti-asthmatic, anti-allergic, anti-inflammatory, immuno-modulating and neuro-protective effect, and method for the production and use thereof as medica
07/24/2001US6265606 To control a broad spectrum of undesirable vegetation, are selective to major crops, have desirable environmental profiles,
07/24/2001US6265430 Insecticides, miticides, nematocides
07/24/2001US6265429 Administering phosphodiesrterase inhibitor
07/24/2001US6265351 Phenylpyrazoles with a herbicidal activity
07/19/2001WO2001005758A3 Indoles and indazoles for the treatment of migraine
07/19/2001WO2000076970A3 Serine protease inhibitors
07/19/2001US20010008749 3-anilino-5-pyrazolone coupler; storage stability
07/18/2001EP1116717A1 Substituted 3-phenylpyrazoles as herbicides
07/18/2001EP1116486A1 Medical composition containing nitroetheneamine derivative or salt thereof as active constituent
07/18/2001EP1115707A1 Benzamide derivatives and ther use as cytokine inhibitors
07/18/2001EP1115701A1 Arylsulfonanilide ureas
07/18/2001EP0850221B1 Meta-guanidine, urea, thiourea or azacyclic amino benzoic acid derivatives as integrin antagonists
07/18/2001CN1068589C Process for producing 3,5-diaryl pyrazolene
07/17/2001US6262044 Modulators of protein tyrosine phosphatases (PTPASES)
07/17/2001US6262040 Indazole derivatives and their use as inhibitors of phosphodiesterase (PDE) type IV and the production of tumor necrosis factor (TNF)
07/12/2001WO2001049721A2 Bacterial genes and proteins that are essential for cell viability and their uses
07/12/2001WO2001049288A1 Novel compounds and compositions as protease inhibitors
07/12/2001WO2001049275A2 Methods and compositions for mitigating pain using nitrate esters
07/12/2001US20010007876 Well tolerated by plants, nontoxic to mammals, active against normally sensitive and resistant species and all or individual development stages
07/12/2001CA2396257A1 Novel compounds and compositions as protease inhibitors
07/12/2001CA2396040A1 Novel bacterial genes and proteins that are essential for cell viability and their uses
07/12/2001CA2394184A1 Methods and compositions for mitigating pain using nitrate esters
07/11/2001EP0876350B1 Pyrazole derivatives, method for preparing same, and pharmaceutical compositions containing said derivatives
07/11/2001CN1303283A Thienylazolylal coxyethanamines, their preparation and their application as medicaments
07/11/2001CN1303281A Use of compounds for elevation of pyruvate dehydrogenase activity
07/11/2001CN1068313C 2[(dihydro)pyrazolyl-3'-oxymethyene]-anilides, prepn. method and use thereof
07/11/2001CN1068308C Substituted benzoylguanide, its preparing process and medicine and application of same
07/10/2001US6258973 Processes for preparing pesticidal intermediates
07/10/2001US6258822 Urokinase inhibitors
07/10/2001US6258806 Peptides with cyclic diazaalkanes for prevention of premature metabolism method for inhibiting an hiv protease in a mammal in need of such protease inhibition, comprising administering to said mammal an effective dosage
07/10/2001US6258751 Controlling weeds in crops
07/10/2001US6258521 Silver halide color photographic light-sensitive material, phenidone compound for use therein, and method of producing the same
07/10/2001CA2048456C The preparation of 3-methylpyrazole
07/05/2001WO2001047475A2 Agent for dyeing keratin containing fibers
07/05/2001US20010006962 Behavior of biologically active compounds favorably modified by replacing a functional group with an unsaturated fatty derivative, e.g. elaidic acid; bioavailability; membrane passage; organ targeting; drugs; agriculture
07/04/2001EP1113332A1 Photographic element, compound, and process
07/04/2001EP1113329A1 Photographic element, compound, and process
07/04/2001EP1113011A1 Aminotetrazole derivatives useful as nitric oxide synthase inhibitors
07/04/2001EP1112269A2 Hiv protease inhibitors
07/04/2001EP1112071A1 Growth hormone secretagogues
07/04/2001EP0969832B1 Pharmaceutical composition for oral administration of a n-piperidino- 3-pyrazolecarboxamide derivative, its salts and their solvates
07/04/2001CN1302298A Substituted (4-brompyrazole-3-yl) indole
07/04/2001CN1067991C Aminoalkyl substituted benzo-heterocyclic compounds
07/03/2001US6255496 Trifluoromethyl ketone analogs as selective cPLA2 inhibitors
07/03/2001US6255489 Method for producing (hetero)aromatic hydroxylamines
07/03/2001US6255342 Pesticides
07/03/2001US6255333 Humans or animals
07/03/2001US6255327 Diphenyl-substituted heterocycles, processes for preparing them and their use as pharmaceutical compositions
06/2001
06/28/2001WO2001046200A1 Novel piperidine and piperazine derivatives
06/28/2001WO2001046172A1 Pyrazole cyclic amp-specific pde inhibitors
06/28/2001WO2001046154A1 Pyrazolyl benzyl ether derivatives containing a fluoromethoxyimino group and use thereof as pesticides
06/28/2001WO2001046153A1 Pyrazolyl benzyl ether derivatives having a fluoromethoxy group and the use thereof as pesticides
06/28/2001WO2001046152A1 Herbicidal diacyl derivatives of propylene diamine
06/28/2001WO2001045703A1 Nitrosated and nitrosylated cyclooxygenase-2 inhibitors, compositions and methods of use
06/28/2001WO2001010834A3 Antibacterial agents
06/28/2001WO2000066104A3 Ace-2 inhibiting compounds and methods of use thereof
06/28/2001US20010005752 Mixing an arylsubstituted indazole compound labelled molecule with binding molecule, selectively detecting a binding event with arylsubstituted indazole labelled compound and binding molecule by fluorescence spectroscopy
06/28/2001DE19962872A1 Oxidation color for coloring keratinous fibers, e.g. fur, wool, feathers and especially human hair, with 4,5-diaminopyrazole derivative as developer contains halogenated m-aminophenol as coupler
06/28/2001DE10034129A1 New 3-substituted benzyloxy-pyrazole derivatives, useful as pesticides, particularly fungicides and insecticides for plant protection
06/28/2001CA2395113A1 Pyrazole cyclic amp-specific pde inhibitors
06/28/2001CA2394095A1 Novel piperidine and piperazine derivatives
06/28/2001CA2393724A1 Nitrosated and nitrosylated cyclooxygenase-2 inhibitors, compositions and methods of use
06/27/2001EP1110954A1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics
06/27/2001EP1110453A1 Triazolyloxybenzyl alkoxyacrylic acid esters, process for producing them and their use
06/26/2001US6252083 Fungicides, insecticides, nematocides
06/26/2001US6251907 1-(aryloxyalkyl)-4-(heteroaryl) piperazines and related compounds useful as antipsychotics and analgesics
06/26/2001US6251830 Pesticides and herbicides
06/21/2001DE19961330A1 New 3-benzyloxy-pyrazole derivatives, are useful as microbicides, pesticides or herbicides, for protection of plants and stored materials, or also as antimycotics
06/20/2001EP1109061A1 Silver halide color photographic light sensitive material
06/20/2001EP1107956A2 Use of 5-amino-pyrazol-derivatives for combating micro-organisms
06/20/2001EP1107955A2 Substituierte 3-aryl-pyrazole als herbizide
06/20/2001EP0890176B1 Proton conductor in liquid form
06/20/2001EP0740690B1 Monoazo dyes containing a fluorosulphonyl group and use thereof
06/20/2001CN1300282A Pyrazole derivatives as P-38 MAP kinase inhibitors
06/20/2001CN1067419C Reactive dyestuffs their preparation and their use
06/19/2001US6248769 Phenyl-triazole compounds for PDE-IV inhibition
06/19/2001US6248753 Bicyclic compounds
06/19/2001US6248743 Antithrombotic agents effective to inhibit the production of type 1 plasminogen activator inhibitor (pai-1)
06/14/2001WO2001042243A2 Protein kinase inhibitors
06/14/2001WO2001042223A1 Pyrazolecarboxamide and pyrazolethioamide as fungicide
06/14/2001WO2001042222A1 Polymorphic crystalline forms of celecoxib
06/14/2001WO2001042221A1 Solid-state form of celecoxib having enhanced bioavailability
06/14/2001WO2001042220A2 Podate ligands and methods of use thereof
06/14/2001WO2001042201A1 N-phenylcarbamates having a microbicide, insecticide and acaricide effect
06/14/2001WO2001041762A2 Valdecoxib compositions
06/14/2001WO2001041761A2 Valdecoxib compositions
06/14/2001WO2001041760A2 Cyclooxygenase-2 inhibitor compositions having rapid onset of therapeutic effect
06/14/2001WO2001041536A2 Solid-state form of celecoxib having enhanced bioavailability
06/14/2001CA2382921A1 Pyrazolecarboxamide and pyrazolethioamide as fungicide