Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
03/2001
03/14/2001CN1287119A Synthesis of sylekirsey
03/13/2001US6201003 Insecticides, miticides, aphidicides, anthelmintics for crops, veterinary medicine, horticulture and agriculture
03/13/2001US6200979 Administering substituted pyrazoles and pyzazolopyrimidines for treating phobias obsessive-compulsive disorder, post-traumatic stress disorder, single episode depression, recurrent depression, dysthymia, bipolar disorders
03/13/2001US6200978 For preventing or treating inflammatory diseases such as arthritis, psoriasis, asthma, or inflammatory bowel disease, disorders of respiratory function, gastrointestinal disorders such as functional bowel disease, as analgesics
03/08/2001WO2001016147A1 Glucopyranosyloxypyrazole derivatives, medicinal compositions containing the same and intermediates in the production thereof
03/08/2001WO2001016138A1 Sulfonylphenylpyrazole compounds useful as cox-2 inhibitors
03/08/2001WO2001016112A1 Benzoate compounds, herbicides and method of using the same
03/08/2001WO2001016111A2 Hypoglycemic sulfonyl pyrazolones and pyrazolines
03/08/2001WO2001016097A1 Phosphate mimics and methods of treatment using phosphatase inhibitors
03/08/2001WO2001015686A1 Selective cox-2 inhibitory novel esters from indolealkanols and novel amides from indolealkylamines
03/08/2001WO2000059506A8 HETEROCYCLIC CONTAINING BIPHENYL aP2 INHIBITORS AND METHOD
03/08/2001CA2382789A1 Phosphate mimics and methods of treatment using phosphatase inhibitors
03/08/2001CA2379421A1 Sulfonylphenylpyrazole compounds useful as cox-2 inhibitors
03/07/2001EP1080068A1 Modulators of protein tyrosine phosphatases
03/07/2001EP0808308B1 Method for separating carbinols
03/06/2001US6197973 Herbicides
03/06/2001US6197791 N-hdroxy-2-(alkyl, aryl, or heteroaryl, sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
03/01/2001WO2001014375A1 Imidazo[1,2-a]pyridine and pyrazolo[2,3-a]pyridine derivatives
03/01/2001WO2001014339A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/01/2001CA2376293A1 Imidazo[1,2-a]pyridine and pyrazolo[2,3-a]pyridine derivatives
03/01/2001CA2376275A1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
02/2001
02/28/2001EP1077971A1 1,5-DIARYL SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS
02/28/2001EP1077951A1 N,n'-azobis-nitroazoles and analogs thereof as igniter compounds for use in energetic compositions
02/28/2001EP1077948A1 Novel 1,2,5-trisubstituted 1,2-dihydro-indazol-3-ones with anti-asthmatic, anti-allergic, anti-inflammatory, immuno-modulating and neuro-protective effect, method for the production and use thereof as a medicament
02/28/2001EP1077947A1 Novel 1,5 and 3-o-substituted 1h-indazoles with anti-asthmatic, anti-allergic, anti-inflammatory, immuno-modulating and neuro-protective effect, method for the production and use thereof as medicaments
02/28/2001EP0712853B1 Pyrazole derivative
02/27/2001US6194443 Aminophenol derivatives with fungicidal property
02/27/2001US6194410 Antiserotonine agents; nervous system and psychological disorders
02/27/2001US6194132 Photographic element, compound, and process
02/22/2001WO2001012609A1 Pyrazoloanthrone and derivatives thereof as jnk inhibitors and their compositions
02/22/2001WO2001012600A1 INHIBITORS OF FACTOR Xa
02/22/2001WO2001012189A1 3(5)-amino-pyrazole derivatives, process for their preparation and their use as antitumor agents
02/22/2001WO2001012188A1 3(5)-ureido-pyrazole derivatives, process for their preparation and their use as antitumor agents
02/22/2001WO2000059862A3 Processes for preparing pesticidal intermediates
02/22/2001CA2383268A1 Pyrazoloanthrone and derivatives thereof as jnk inhibitors and their compositions
02/22/2001CA2380786A1 3(5)-ureido-pyrazole derivatives, process for their preparation and their use as antitumor agents
02/21/2001EP1077214A1 An improved process for preparing a pyrazolopyrimidinone derivative
02/21/2001EP1076660A1 Substituted (4-brompyrazole-3-yl)benzazoles
02/21/2001EP1076557A1 Ccr-3 receptor antagonists
02/21/2001CN1284948A Indezole bioisostere replacement of catechol in therafeutically active compounds
02/20/2001US6191283 Pyrazole intermediates in a method of preparation of β-amino acids
02/20/2001US6191159 Anticoagulants
02/20/2001US6191158 Respiratory system disorders; cardiovascular disorders; anticholesterol agents
02/20/2001US6190853 Photographic elements containing novel yellow couplers
02/20/2001US6190850 Photographic element, compound, and process
02/20/2001CA2223624C Tricyclic 5,6-dihydro-9h-pyrazolo[3,4-c]-1,2,4-triazolo[4,3-.alpha.]pyridines
02/15/2001WO2001010864A1 1-cycloalkylpyrazoyl-benzoyl derivatives
02/15/2001WO2001010834A2 Antibacterial agents
02/14/2001EP1076053A1 3-arylphenyl sulfide derivatives and insecticides and miticides
02/14/2001EP1075467A1 Pyrazole derivatives as p-38 map kinase inhibitors
02/14/2001EP0836593B1 5-pyrazolylbenzoic acid derivatives as herbicides
02/14/2001EP0833820B1 Benzisoxazole and indazole derivatives as antipsychotic agents
02/14/2001CN1061816C Process for agrochemical treatment of grasslands
02/13/2001US6187930 Reacting selected amine with optically active acid selected from (+)-ditoluyl-l-tartaric acid and/or (-)-ditoluyl-l-tartaric acid in solvent to form diasteroisomeric salt, separating, isolating enantiomer
02/13/2001US6187774 Fused heterocyclic compounds and pharmaceutical applications thereof
02/08/2001WO2001009128A1 Thiourea and isothiourea derivatives for inhibiting ras-transformed cell growth
02/08/2001WO2001009121A2 2-pyrazolin-5-ones_as tyrosine kinase inhibitors
02/08/2001WO2001009102A2 Process for preparing 1,5-diaryl-3-substituted pyrazoles
02/08/2001CA2380644A1 2-pyrazolin-5-ones
02/08/2001CA2380371A1 Thiourea and isothiourea derivatives for inhibiting ras-transformed cell growth
02/07/2001EP1074551A2 Phenylpyrazoles with a herbicidal activity
02/07/2001EP1073633A2 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
02/07/2001EP1073626A1 Azine used as fungicides
02/07/2001EP1073431A1 Use of nmda antagonists for treatment of irritable bowel syndrome
02/07/2001CN1283192A Inhibition of raf kinase using aryl and hetroaryl substituted heterocyclic ureas
02/07/2001CN1283191A Benzylidene pyrazolones and its preparation and use
02/07/2001CN1283190A Substituted benzene compounds, process for their preparation and herbicidal and defoliant composition containing them
02/07/2001CN1282740A Intermediate compound for preparing xibo ketone
02/06/2001USH1942 Made by reacting 1-methyl-5-difluoromethoxy-4-chloro-3-(2-fluoro-4-chloro-5 -aminophenyl)pyrazole with t-butyl nitrite, copper chloride, and ethyl acrylate in acetonitrile, for example
02/06/2001US6184241 Aspartic protease inhibitors
02/01/2001WO2001007413A1 1-aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
02/01/2001WO2001007411A1 Biarylurea derivatives
02/01/2001WO2001007405A2 New vitamin d derivatives with cyclic substructures in the side chains, method and intermediates for their production and their use in the preparation of medicaments
02/01/2001WO2001007020A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof
02/01/2001DE19935771A1 Neue Vitamin D-Derivate mit cyclischen Substrukturen in den Seitenketten, Verfahren und Zwischenprodukte zu ihrer Herstellung und die Verwendung zur Herstellung von Arzneimitteln New vitamin D derivatives with cyclic substructures in the side chains, to processes and intermediates for their preparation and to the use for the preparation of medicaments
02/01/2001DE19935219A1 Carbonsäureamide, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Herstellung Carboxamides, medicaments containing these compounds, their use and production
02/01/2001CA2380389A1 Biarylurea derivatives
02/01/2001CA2376465A1 New vitamin d derivatives with cyclic substructures in the side chains, method and intermediates for their production and their use in the preparation of medicaments
01/2001
01/31/2001EP1072598A1 Pyrazolinone derivatives
01/31/2001EP1072597A1 Pyrazoles and their use as endothelin antagonists
01/31/2001EP1072576A1 Fluorinating agent, process for producing the same, and use thereof
01/31/2001EP1072266A1 Thienylazolylalcoxyethanamines, their preparation and their application as medicaments
01/31/2001EP1071701A1 Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereof
01/31/2001EP1071682A2 Fungicidal benzoheterocyclyloxime
01/31/2001EP1071670A1 Novel diphenyl-substituted 5-ring-heterocycles, method for producing them and their use as medicaments
01/31/2001EP1071668A1 5-aminoindeno(1,2-c)pyrazol-4-ones as anti-cancer and anti-proliferative agents
01/31/2001EP1071661A1 Process for preparing 4-hydroxy indole, indazole and carbazole compounds
01/31/2001CN1281851A Useful sypolyphenol intermediate and its preparation method
01/31/2001CN1061339C Novel sulfonamide inhibitors of aspartyl protease
01/30/2001US6180798 Chemical intermediates for insecticides and pesticides
01/30/2001US6180796 Sulfonamide derivatives
01/30/2001US6180653 Aminopyrazole derivatives
01/30/2001US6180637 Therapy for parkinson, alzheimer disease
01/25/2001WO2001005774A1 Heteroaromatic ring compounds
01/25/2001WO2001005769A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/25/2001WO2001005758A2 Indoles and indazoles for the treatment of migraine
01/25/2001WO2000044740A3 Heteroaryl acetylenic sulfonamide and phosphinic acid amide hydroxamic acid tace inhibitors
01/25/2001CA2378047A1 Heterocyclic compounds for the treatment of migraine
01/25/2001CA2377527A1 Heteroaromatic ring compounds
01/24/2001EP1070052A1 Fungicide compositions comprising a hydroximic or hydrazonic group