Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
04/2001
04/26/2001WO2001029007A1 Pyrazole derivatives as cannabinoid receptor antagonists
04/26/2001WO2001029006A1 Synthesis of 1,3,5-trisubstituted pyrazoles and intermediates therefore
04/26/2001WO2001028987A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/26/2001WO2001028493A2 Small molecule inhibitors of necrosis
04/26/2001WO2001004095A3 Α-α'-SUBSTITUTED N-ALKYL-3-ALKENYLBENZOYL-PYRAZOL-DERIVATIVES
04/26/2001WO2000055139A3 Heterocyclic urea and related compounds useful as anti-inflammatory agents
04/26/2001CA2387892A1 Pyrazole derivatives as cannabinoid receptor antagonists
04/26/2001CA2387031A1 Small molecule modulators of non-endogenous, constitutively activated human serotonin receptors
04/26/2001CA2384240A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/26/2001CA2382212A1 Synthesis of 1,3,5-trisubstituted pyrazoles and intermediates therefore
04/25/2001EP1093367A1 Protease inhibitors
04/25/2001CN1292791A Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
04/25/2001CN1292787A Fungicidal benzoheterocyclyloxime
04/24/2001US6221810 3-hydroxy-4-aryl-5-oxo-pyrazoline derivatives
04/19/2001WO2001027113A2 PYRAZOLO `4,3-d! PYRIMIDINE DERIVATIVES
04/19/2001WO2001027107A2 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001WO2001027068A1 Biaryl ether derivatives useful as monoamine reuptake inhibitors
04/19/2001WO2001026652A1 Fab i inhibitors
04/19/2001WO2000045894A3 Use of pyrazole carboxamides
04/19/2001US20010000345 Compounds such as (4,7-dimethylbenzimidazol-5-yl)guanidine; treating nasal congestion, otitis media, asthma, pain, migraine, gastrointestinal disorder, ulcer
04/19/2001CA2388813A1 Heterocyclic sodium/proton exchange inhibitors and method
04/18/2001EP1091943A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
04/18/2001EP1091940A1 Method for preparing 1-alkyl-pyrazol-5-carboxylic acid esters
04/18/2001EP1091937A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
04/17/2001US6218426 For therapy of mammalian reproductive disorders and steroid hormone-dependent tumors as well as for regulating fertility, where suppression of gonadotropin release is indicated
04/17/2001US6218418 Therapy of cell proliferative disorders associated with an altered cell dependent kinase activity by administering amino pyrazole derivative to mammal
04/17/2001US6218397 For therapy of stress-related illnesses, such as stress-induced depression, anxiety, and headache; abdominal bowel syndrome; inflammatory diseases; immune suppression; alzheimer's disease; gastronintestinal diseases
04/12/2001WO2001025241A2 Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides
04/12/2001WO2001025181A1 Carboxylic acid derivatives and drugs containing the same
04/12/2001WO1999063939A9 Multibinding inhibitors of cyclooxygenase-2
04/12/2001DE19948101A1 New substituted aryl- and heteroaryl-alkanes are serine protease and thrombin inhibitors, used for treatment of e.g. deep vein thrombosis or stroke
04/11/2001EP1089964A1 Hydrazine derivatives
04/11/2001CN1290699A New pyrazolone compound and eye plastic lens made therefrom
04/10/2001US6214994 Treatment of neoplastic diseases, bacterial or fungal infections, and preventing or decreasing production of phosphorylated paired helical filament (phf) epitopes associated with alzheimer's disease
04/10/2001US6214880 Lowering plasma cholesterol levels and inhibiting abnormal cell proliferation with said compound; treatment of cancer, psoriasis, vascular restenosis, infections, atherosclerosis and hypercholesterolemia
04/10/2001US6214835 Dihalopropene compounds insecticides containing them as active ingredients, and intermediates for their production
04/10/2001US6214813 Azopyrazoles
04/05/2001WO2001023358A1 Pyrazole derivatives, intermediates for the preparation thereof, processes for the preparation of both and herbicides containing the derivatives as the active ingredient
04/05/2001WO2001023349A1 Acylsulfonamide derivatives
04/05/2001WO2000057877A8 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof
04/05/2001US20010000179 Inhibitors of typsin-like serine protease; anticoagulants
04/04/2001EP1087941A2 Thiolesters and uses thereof
04/04/2001EP1087661A1 Il-8 receptor antagonists
04/04/2001CN1290262A Heteroaromatic derivatives
04/04/2001CN1290249A Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof
04/04/2001CN1290164A Inhibition of RAF kinase using substituted heterocyclic ureas
04/03/2001US6211403 Process for preparing 2-chloro-3-alkoxy-4-alkylsulfonyl-benzoic acids and esters
04/03/2001US6211245 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
04/03/2001US6211234 Substituted phenyl compounds
04/03/2001US6211222 Substituted indazole derivatives and related compounds
03/2001
03/29/2001WO2001021618A1 Acrylonitrile compounds and pest control agent
03/29/2001WO2001021591A1 Pyrazole derivatives
03/29/2001WO2001021584A1 Tyrosine derivatives
03/29/2001WO2001021180A1 Thrombopoietin mimetics
03/29/2001WO2001021160A2 Carboxymide and aniline derivatives as selective inhibitors of pathogens
03/29/2001WO2001020993A1 Insecticidal and acaricidal agents
03/29/2001WO2001002350A3 Novel amino sulfonamides and amido sulfonamides as antiviral agents
03/29/2001CA2385447A1 Pyrazole derivatives
03/29/2001CA2383157A1 Insecticidal and acaricidal agents
03/28/2001EP1086682A2 Utilization of aryl(or heteroaryl)azolylcarbinol derivatives in the preparation of a medicament for the treatment of neurogenic inflammation
03/28/2001EP1085845A2 Multibinding inhibitors of cyclooxygenase-2
03/28/2001CN1289326A N-[(substituted five-membered di-or thiaza diunsaturated ring) carbonyl] guanidine derivatives for the treatment of ischemia
03/27/2001US6207831 A benzopyrazole compound
03/27/2001US6207829 Cyclization of a corresponding pyrazole compound
03/27/2001US6207693 Benzamide derivatives having a vasopressin antagonistic activity
03/27/2001US6207680 Heteroarylpiperidines and their use as antipsychotics and analgesics
03/27/2001US6207618 Heterocyclic substituted 4-benzoyl-pyrazole as herbicides
03/27/2001US6207363 Cyan ?nb coupler?
03/22/2001WO2001019798A2 INHIBITORS OF FACTOR Xa
03/22/2001WO2001019778A1 Novel dicarboxylic acid derivatives with pharmaceutical properties
03/22/2001CA2385589A1 Inhibitors of factor xa
03/21/2001EP1085016A1 Heterocycle-bearing thio phenol compounds, intermediates for the preparation of the same and processes for the preparation of both
03/21/2001EP1085011A1 Novel polyamine analogues as therapeutic and diagnostic agents
03/21/2001EP1084111A1 Substituted 3-thiocarbamoylpyrazoles
03/21/2001EP1083897A1 Hiv integrase inhibitors
03/21/2001CN1288457A Inhibitors of & alpha; 4 mediated cell adhesion
03/21/2001CN1063440C Aromatic pyrozol fungicide
03/20/2001US6204391 Water soluble fullerenes with antiviral activity
03/20/2001US6204383 Processes for preparing sildenafil
03/20/2001CA2213111C Substituted carboxanilide derivative and plant disease control agent comprising same as active ingredient
03/15/2001WO2001018171A2 Novel class of cytodifferentiating agents and histone deacetylase inhibitors, and methods of use thereof
03/15/2001WO2001018004A2 PYRAZOLO[4,3-d]PYRIMIDINES
03/15/2001WO2001017982A1 Benzophenones as inhibitors of reverse transcriptase
03/15/2001WO2001017973A2 Novel herbicides
03/15/2001WO2001017972A2 Novel herbicides
03/15/2001WO2001017353A1 Herbicidal composition
03/15/2001WO2001017349A1 Thrombopoietin mimetics
03/15/2001WO2000058286A3 Method of producing heterocyclic carbamates from aza-heterocyclic compounds and carbon dioxide
03/15/2001WO2000051972A8 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy
03/15/2001WO2000049007A8 Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsin s
03/15/2001DE19943636A1 Neuartige Dicarbonsäurederivate mit pharmazeutischen Eigenschaften Novel dicarboxylic acid derivatives with pharmaceutical properties
03/15/2001DE19942474A1 Pyrazolo[4,3-d]pyrimidine Pyrazolo [4,3-d] pyrimidines
03/15/2001CA2723014A1 A herbicidal composition comprising a 3-hydroxy-4-aryl-5-oxopyrazoline derivative and an isoxadifen derivative
03/15/2001CA2383999A1 Novel class of cytodifferentiating agents and histone deacetylase inhibitors, and methods of use thereof
03/15/2001CA2383782A1 Compounds for the treatment of viral infections
03/15/2001CA2382432A1 Novel herbicides
03/15/2001CA2318004A1 Novel polyamine analogues as therapeutic and diagnostic agents
03/14/2001EP1083171A1 Pyrazoline derivatives, their preparation and application as medicaments
03/14/2001EP1082127A1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME
03/14/2001EP1082110A1 Use of compounds for the elevation of pyruvate dehydrogenase activity