Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
02/2000
02/09/2000EP0977756A1 PYRAZOLOPYRIMIDINONES WHICH INHIBIT TYPE 5 CYCLIC GUANOSINE 3',5'-MONOPHOSPHATE PHOSPHODIESTERASE (cGMP PDE5) FOR THE TREATMENT OF SEXUAL DYSFUNCTION
02/09/2000EP0977725A1 New fatty acid derivatives
02/09/2000CN1244122A Method of using cyclooxygenase-2 inhibitors in the treatment and prevention of neoplasia
02/08/2000US6022979 Process for preparing pyrazoles
02/08/2000US6022870 4-(heterocycle-substituted-phenyl)-1,2,4-triazol-3-ones
02/03/2000WO2000005221A1 Substituted benzoylcyclohexandiones
02/03/2000WO2000005217A1 Imidazole compounds and their use as adenosine deaminase inhibitors
02/03/2000WO2000005216A1 Il-8 receptor antagonists
02/03/2000WO1999058504A9 Novel 1,2,5-trisubstituted 1,2-dihydro-indazol-3-ones with anti-asthmatic, anti-allergic, anti-inflammatory, immuno-modulating and neuro-protective effect, method for the production and use thereof as a medicament
02/03/2000DE19834110A1 New heterocyclyl(alkyl)-substituted pyrazolyl-pyrazole derivatives, used as herbicides and plant growth regulators, especially as pre- or post-emergence selective herbicides in crops such as rice
02/03/2000DE19834044A1 Neue substituierte Pyrazolderivate New substituted pyrazole derivatives
02/03/2000DE19833913A1 Verfahren zur Herstellung von N,N'-Carbonyldiazolen A process for the preparation of N, N'-carbonyldiazoles
02/03/2000CA2338741A1 Il-8 receptor antagonists
02/03/2000CA2338305A1 Imidazole compounds
02/03/2000CA2338304A1 Substituted benzoylcyclohexandiones
02/02/2000EP0976737A1 Pyrazole derivatives, process for preparing the same, intermediates, and pest control agent containing the same as active ingredient
02/02/2000EP0976707A1 Cycloalkyl benzyl ether compounds
02/01/2000US6020498 Process for preparing carboxamide oximes
02/01/2000US6020368 Microbiocides
02/01/2000US6020357 Nitrogen containing heteroaromatics as factor Xa inhibitors
02/01/2000US6019986 Parasiticidal pyrazoles
01/2000
01/27/2000WO2000003993A1 Pyrazole-type compounds, process for producing the same and herbicides containing the same
01/27/2000WO2000003988A1 Novel benzoic acid derivatives and processes for the preparation thereof
01/27/2000DE19921732A1 New 2-benzoyl-1,3-cyclohexanedione derivatives useful as herbicides, especially for selective weed control in monocot crops, e.g. maize
01/26/2000EP0974585A1 Method for the preparation of pyrazoles
01/26/2000EP0973774A1 1,5-dihydro-pyrazolo 3,4-d]-pyrimidinone derivatives
01/26/2000EP0973752A1 Heterocyclically substituted aromatic amino compounds with a herbicidal effect
01/26/2000EP0973747A1 Pesticidal 1-arylpyrazoles
01/26/2000EP0973512A1 N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
01/26/2000EP0973395A1 Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them
01/26/2000CN1048719C Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxytetracyclines, prepn. method, their compositions and use thereof
01/25/2000US6017965 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
01/20/2000WO2000002851A1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them
01/20/2000WO2000002850A2 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
01/20/2000WO1999059529A3 Agents and method for producing semi-permanent colorations of keratin fibers
01/20/2000DE19832146A1 Preparation of 3-methyl-pyrazole, uses mineral acid salt of hydrazine
01/20/2000DE19831656A1 Verfahren zur Herstellung von Pyrazolen A process for the preparation of pyrazoles
01/19/2000EP0971714A1 Method of using cyclooxygenase-2 inhibitors in the treatment and prevention of dementia
01/19/2000EP0971588A1 Novel cannabinoid receptor modulators
01/19/2000EP0672038B1 Herbicides
01/19/2000CN1242006A Guanidinyl heterocycle compounds useful as alpha-2 adrenoceptor agonists
01/19/2000CN1242003A Pesticidal 1-aryl and pyridylpyrazole derivatives
01/19/2000CN1242002A Pesticidal 1-arylpyrazoles
01/19/2000CN1242001A Guanidinylamino heterocycle compounds useful as alpha-2 adrenoceptor agonists
01/18/2000US6015911 Process for preparing 1-alkyl-4-(2-chloro-3-alkoxy-4-alkylsulfonylbenzoyl)-5-hydroxypyrazole and related compounds
01/18/2000US6015910 Intermediates to pesticidal 5-amino-4-ethylsulfinyl-1-arylpryazoles
01/18/2000US6015908 IL-8 receptor antagonists
01/18/2000US6015829 1-phenylpyrazole compounds and medicinal application thereof
01/18/2000US6015657 Pyrazolone magenta dye-forming couplers having particular thio coupling-off group that enables improved photographic properties
01/13/2000WO2000001673A2 Method for preparing 1-alkyl-pyrazol-5-carboxylic acid esters
01/13/2000WO1999018941A3 Ih-MODULATORS
01/13/2000DE19830431A1 Sulfonylamino-carbonsäure-N-arylamide als Guanylatcyclase-Aktivatoren Sulfonylamino-carboxylic acid N-arylamides as guanylate cyclase activators
01/13/2000CA2336310A1 Method for preparing 1-alkyl-pyrazol-5-carboxylic acid esters
01/12/2000EP0970046A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
01/12/2000EP0969835A1 Use of central cannabinoid receptor antagonists for regulating appetence
01/12/2000EP0969832A1 Pharmaceutical composition for oral administration of a n-piperidino- 3-pyrazolecarboxamide derivative, its salts and their solvates
01/12/2000CN1048246C Indazolesulfonylurea deriv., use thereof, and intermediate for production thereof
01/11/2000US6013651 Meta-azacyclic amino benzoic acid compounds and derivatives thereof
01/06/2000WO2000000477A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000WO2000000473A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000WO2000000465A1 Hydrazine derivatives
01/06/2000CA2336625A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000CA2335921A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000CA2335245A1 Hydrazine derivatives
01/05/2000EP0968179A1 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
01/05/2000DE19829616A1 Verfahren zur Herstellung von 1-Alkyl-pyrazol-5-carbonsäureestern A process for the preparation of 1-alkyl-pyrazole-5-carboxylic acid esters
01/05/2000CN1240439A Aminophenol derivates with fungicidal property
01/05/2000CN1240437A Preparation and use of ortho-sulfonamido heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
01/05/2000CN1240433A Process for preparing N-substituted 3-hydroxypyrazoles
01/05/2000CN1240432A 1-phenylpyrazole compounds and medicinal application thereof
01/05/2000CN1240419A Aromatic amine derivatives having NOS inhibitory effect
01/05/2000CN1048015C Bicyclic tetrahydro pyrazolopyridines
01/04/2000US6011159 Processes and intermediates for preparing substituted indazole derivatives
01/04/2000US6011059 Acyl guanidine sodium/proton exchange inhibitors and method
01/04/2000US6011052 Pyrazolone derivatives as MCP-1 antagonists
01/04/2000US6010981 1-alkyl-4-benzoyl-5-hydroxypyrazole compounds and their use as herbicides
01/04/2000US6010837 Silver halide photographic element comprising image dye-forming couplers
12/1999
12/29/1999WO1999067243A1 Pyrazolo(3,4-d)pyrimidines with anticonvulsive and antiallergic/antiasthmatic action
12/29/1999WO1999067235A1 Five-membered ring compounds
12/29/1999WO1999066925A1 Protease inhibitors
12/29/1999EP0967206A1 Derivatives of N-phenylpyrazoles
12/29/1999EP0966490A2 Catalyst compositions for the polymerization of olefins
12/29/1999EP0966452A1 Process for preparing sulphurous 2-chloro-3-(4,5-dihydroisoxazol-3-yl)-benzoic acids
12/29/1999EP0966445A1 Processes for preparing pesticidal intermediates
12/29/1999EP0966444A1 Process for preparing pyrazole derivatives
12/29/1999EP0612314B1 2-pyrazinylethylamine derivatives and their use as pharmaceuticals
12/29/1999CN1239953A 3-thiocarbamoylpyrazole derivatives as pesticides
12/29/1999CN1047775C N-piperidino 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl pyrazole-3-formyl amide, its preparation and drug composition
12/29/1999CA2335876A1 Protease inhibitors
12/29/1999CA2301107A1 Pyrazolo(3,4-d)pyrimidines with anticonvulsive and antiallergic/antiasthmatic action
12/28/1999US6008243 An enzyme inhibitor for preventing the degradation and remodeling of connective tissues
12/23/1999WO1999065871A2 Thiolesters and uses thereof
12/23/1999WO1999065310A1 Il-8 receptor antagonists
12/23/1999DE19827679A1 New pyrazolo(3,4-d)pyrimidine derivative adenosine A3 receptor antagonists, used for treating epilepsy, asthma or allergy
12/23/1999DE19826669A1 Production of pyrazole compounds useful as nitrification inhibitors and as intermediates for plant protection agents, dyes or polymers
12/23/1999CA2335464A1 Novel thiolesters and uses thereof
12/23/1999CA2335292A1 Il-8 receptor antagonists
12/22/1999EP0853639B1 Water dispersible blocked isocyanates
12/22/1999EP0731795B1 Substituted pyrazolyl benzenesulfonamides for the treatment of inflammation
12/21/1999US6005118 Methods of preparing 4-cyano-4 (substituted indazole) cyclohexane-carboxylic acids useful as PDE4 inhibitors