Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
01/2001
01/24/2001EP0837852B1 Pesticidal sulfur compounds
01/24/2001CN1281441A Therapeutically active compounds based on indazole bioisostere replacement of catechol in PDE4 inhibitors
01/24/2001CN1061044C Tricyclic 5,6-dihydro-9H-pyrazolo [3,4-C]-1,2,4-triaolo [4,3-alpha] pyridines
01/24/2001CN1061037C 取代的1-芳基吡唑 Substituted 1-aryl-pyrazole
01/24/2001CN1061036C Substituted pyrazolyl benzenesulfonamides for treating inflammation
01/23/2001USRE37029 Antipsychotic and analgesic agents
01/23/2001US6177459 Substituted heterocyclic compounds and their use as fungicides
01/23/2001US6177427 Treatment of glaucoma and ocular hypertension
01/23/2001US6177401 Use of organic compounds for the inhibition of Flk-1 mediated vasculogenesis and angiogenesis
01/23/2001US6177379 Containing diels-alder adduct obtained by reacting specified azo compound and conjugated diene
01/23/2001CA2033479C Process for preparing (1r,5s,6s)-2-[(6,7-dihydro-5h-pyrazolo[1,2-a][1,2,4] triazolium-6-yl)] thio-6- [(r)-1-hydroxyethyl] -1-methyl-carbapenem-3-carboxylate and starting materialsthereof
01/18/2001WO2001004115A2 Novel process for synthesis of heteroaryl-substituted urea compounds
01/18/2001WO2001004097A2 Cyclic delocalized cations connected by spacer groups
01/18/2001WO2001004096A2 N-cycloalkyl-3-alkenylbenzoyl-pyrazole derivatives as herbicides
01/18/2001WO2001004095A2 Α-α'-SUBSTITUTED N-ALKYL-3-ALKENYLBENZOYL-PYRAZOL-DERIVATIVES
01/18/2001CA2378780A1 .alpha.-.alpha.'-substituted n-alkyl-3-alkenylbenzoyl-pyrazol-derivatives
01/18/2001CA2378592A1 N-cycloalkyl-3-alkenylbenzoyl-pyrazole derivatives as herbicides
01/17/2001EP1068187A1 Pyrazole inhibitors of cytokine production
01/17/2001EP1068178A1 NON-PEPTIDE GnRH AGENTS
01/17/2001CN1280568A Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
01/17/2001CN1280565A Heterocyclic compounds having NOS inhibitory activities
01/17/2001CN1280560A Adamantane derivatives
01/17/2001CN1280127A 5-aminopyrazole-4-carboxylic ester derivatives and its preparing method
01/17/2001CN1280126A Substituted pyrazolyl benzene sulfone amides compounds for curing inflammation
01/17/2001CN1280125A Substituted pyrazolyl benzene sulfone amides compounds for curing inflammation
01/17/2001CN1060768C Pyrazoles and pyrazolopyrimidines
01/16/2001US6174915 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses
01/16/2001US6174889 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
01/16/2001US6174884 1,5-dihydro-pyrazolo[34-D]-pyrimidinone derivatives
01/16/2001US6174839 As herbicide
01/16/2001CA2025932C Pyrazole-3-carboxamides
01/11/2001WO2001002369A2 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
01/11/2001WO2001002356A1 Indoline or tetrahydroquinoline derivatives
01/11/2001WO2001002354A1 Phthalamide derivatives, intermediates in the production thereof, and agricultural/horticultural insecticides and method of using the same
01/11/2001WO2001002350A2 Novel amino sulfonamides and amido sulfonamides as antiviral agents
01/10/2001EP1067121A2 5-Aminopyrazole-4-carboxylate derivative and process for preparing the same
01/10/2001EP1066257A2 Heterocylic classes of compounds for the modulating tyrosine protein kinase
01/10/2001CN1279671A Pyrazolylpyrazoles substituted by 1-methyl-5-alkylsulphonyl, 1-methyl-5-alkylsuphinyl and 1-methyl-5-alkylthio, methods for preparing them and use as herbicides
01/10/2001CN1060478C Substituted pyrazole derivatives
01/09/2001US6172261 Biosynthesis using chain extension
01/09/2001US6172239 Psychological, nervous system disorders
01/09/2001US6172225 Herbicides
01/09/2001US6172222 Diaminopyrazoles
01/09/2001US6172170 Initiators for radical polymerization
01/09/2001US6172096 Administering 4-pyrazolylbenzenesulfonamide derivatives to treat autoimmune diseases
01/09/2001US6172057 Antiinflammatory agents; antiarthritic agents; antitumor agents
01/09/2001US6171522 Heterocyclic aromatic anion salts, and their uses as ionic conducting materials
01/04/2001WO2001000585A1 Pyrazolidinol compounds
01/04/2001WO2001000576A1 Indole and indazole urea-peptoids as thrombin receptor antagonists
01/04/2001WO2001000575A1 Heterocyclic dicarboxylic acid diamide derivatives, agricultural/horticultural insecticides and method of using the same
01/04/2001WO2001000229A1 Combination of tumors necrocis factor (tnf) antagonists and cox-2 inhibitors for the treatment of inflammation
01/04/2001DE19930075A1 Neue Amino- und Amidosulfonamide als antivirale Mittel New amino and Amidosulfonamide as antiviral agents
01/04/2001CA2377200A1 Pyrazolidinol compounds
01/04/2001CA2369145A1 Combination of tumors necrocis factor (tnf) antagonists and cox-2 inhibitors for the treatment of inflammation
01/03/2001EP1065205A1 Heteroaromatic derivatives
01/03/2001EP1065203A2 Heterocyclic compounds as retinoic acid receptor antagonists
01/03/2001EP1064964A2 Compositions containing aldose reductase inhibitors and selective cyclooxygenase inhibitors for the treatment of diabetic complications
01/03/2001EP1064270A2 Disubstituted pyrazolines and triazolines as factor xa inhibitors
01/03/2001EP1063992A1 Sulfurpenta fluorophenyl pyrazoles for controlling ectoparasitic infestations
01/03/2001EP1063982A2 Antagonists for treatment of cd11/cd18 adhesion receptor mediated disorders
01/03/2001CN1278807A Herbicidal N-alkenyl Heteroaryloxyacetamides
01/03/2001CN1278805A Novel heterocyclioally substituted and a-hydroxycarboxlic acid derivatives, method for producing the same and their use as endothelin receptor antagonists
01/03/2001CN1278725A Indeno [1,2-c]-naphtho [1,2-C]- and benzo [6,7] cyclohepta [1,2-C] pyrazole derivatives
01/03/2001CN1278724A Indeno [1,2-c] pyrazole derivatives for inhibiting tyrosine kinase activty
01/02/2001US6169089 Nitric oxide synthase inhibitors; treatment of arthritis
01/02/2001US6169086 Pyrazole derivatives
01/02/2001CA2009604C Diaryl-substituted heterocyclic compounds, their preparation and drugs and cosmetics obtained therefrom
12/2000
12/30/2000CA2313131A1 Compositions and treatment for diabetic complications
12/28/2000WO2000078723A1 Process for the preparation of butoxycarbonylimino compounds and intermediates therefor
12/28/2000WO2000078712A1 Substituted arylmalonic acid dinitriles as intermediates for the prepartion of herbicides
12/28/2000CA2368827A1 New intermediates
12/27/2000EP1063227A1 Hydrazide fixed to resin and derivative thereof, and method for synthesizing pyrazolones in solid phase
12/27/2000EP1062218A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
12/27/2000EP1062217A1 Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
12/27/2000EP1062208A1 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
12/27/2000EP1062204A1 Modulators of protein tyrosine phosphatases (ptpases)
12/27/2000CN1278244A Dipeptide nitriles
12/26/2000US6166055 Antiinflammatory agents
12/26/2000US6166038 Aminopyrazole derivatives
12/26/2000US6166023 1,5- and 3-O-substituted 1H-indazoles having anti-asthmatic, anti-allergic, anti-inflammatory, immunomodulating and neuroprotective action, process for their preparation and their use as medicaments
12/26/2000US6165944 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
12/21/2000WO2000077027A2 Serine protease inhibitors
12/21/2000WO2000076983A1 1-(4-arylsulfonyl)-3-substituted-5-aryl-2-pyrazolines as inhibitors of cyclooxygenase-2
12/21/2000WO2000076971A2 Serine protease inhibitors
12/21/2000WO2000076970A2 Serine protease inhibitors
12/21/2000WO2000076503A1 1-(4-sulfamylaryl)-3-substituted-5-aryl-2-pyrazolines as inhibitors of cyclooxygenase-2
12/21/2000WO2000076489A2 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
12/21/2000CA2383008A1 Compounds
12/21/2000CA2377153A1 1-(4-sulfamylaryl)-3-substituted-5-aryl-2-pyrazolines as inhibitors of cyclooxygenase-2
12/21/2000CA2375920A1 Compounds
12/21/2000CA2375551A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
12/20/2000EP1061075A2 Substituted triazoles, imidazoles and pyrazoles as herbicides
12/19/2000US6162819 Pyrazole derivatives, their preparation and their use in pharmaceuticals
12/14/2000WO2000075138A1 Oxime derivatives, process for the preparation thereof and pesticides
12/14/2000WO2000046210A3 New process for preparing pesticidal intermediates
12/13/2000CN1276785A N-aroylphenylalanine derivs.
12/12/2000US6160002 1-arylpyrazole derivatives; pesticides, parasiticides; veterinary medicine
12/07/2000WO2000073264A1 Cell proliferation inhibitors
12/07/2000CA2371092A1 Cell proliferation inhibitors
12/06/2000EP1057812A1 Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof