Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
06/1999
06/02/1999CN1218460A Substituted 4-hydroxy-phenylalcanoic acid derivatives with activity to ppar-'gamma'
06/02/1999CN1218046A Imide derivatives
06/02/1999CN1218045A Imide derivatives or salts thereof
06/01/1999US5908938 Base-catalyzed reaction of a hydrazone with olefin; cyclization
06/01/1999US5908931 Preorganized hexadentate ligands useful in radiographic imaging agents
06/01/1999US5908852 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation
06/01/1999CA1340567C Heterocyclic amide derivatives
05/1999
05/27/1999WO1999025702A1 Herbicidal n-alkenyl heteroarylyloxyacetamides
05/27/1999WO1999025701A1 NOVEL HETEROCYCLICALLY SUBSTITUTED α-HYDROXYCARBOXLIC ACID DERIVATIVES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS
05/27/1999WO1999025695A1 5-arylpyrazole compounds
05/27/1999WO1999025686A1 Cyclic amine derivatives and their use as drugs
05/27/1999DE19751943A1 New pyrazolyl-pyrazole derivatives are pre- and post-emergent herbicides
05/27/1999CA2308746A1 Novel heterocyclically substituted .alpha.-hydroxycarboxylic acid derivatives, method for producing the same and their use as endothelin receptor_antagonists
05/26/1999EP0917526A2 New nitrification inhibitors and the use of polyacids to treat mineral fertilizers containing a nitrification inhibitor
05/26/1999CN1217714A Substituted indazole derivatives and their use as inhibitors phosphodiesterase (PDE) type IV and production of tumor necrosis factor (TNF)
05/25/1999US5907041 Process for preparing pyrazole derivatives
05/20/1999WO1999024873A1 Compound, composition and use
05/20/1999WO1999024871A1 Compound, composition and use
05/20/1999WO1999024460A2 Dipeptide nitriles
05/20/1999WO1999016753A3 Tricyclic 3-oxo-propanenitrile compounds
05/20/1999DE19750529A1 New heterocyclic alpha-hydroxycarboxylic acid derivatives useful for treating hypertension, chronic coronary insufficiency, asthma, prostate cancer etc.
05/20/1999CA2309946A1 Compound, composition and use
05/19/1999EP0916675A2 Process for preparing sildenafil
05/19/1999EP0915873A1 Substituted pyrazolyl-pyrazole derivatives, process for their preparation and their use as agents with a herbicidal effect
05/19/1999EP0915868A1 Carbanilides used as pesticides
05/19/1999EP0915853A1 Substituted 3-phenyl pyrazoles
05/19/1999EP0915852A1 1,3-dimethyl-5-fluoro-pyrazole-4-carboxamide derivatives, their preparation and their use as microbicides
05/19/1999EP0915846A2 2- and 2,5-substituted phenylketoenols
05/19/1999EP0915829A1 Diagnostic imaging contrast agent with improved in-serum-relaxivity
05/14/1999WO1999023091A1 Aromatic heterocyclic compounds as anti-inflammatory agents
05/14/1999WO1999023077A1 Indazole bioisostere replacement of catechol in therapeutically active compounds
05/14/1999WO1999023076A1 Therapeutically active compounds based on indazole bioisostere replacement of catechol in pde4 inhibitors
05/14/1999WO1999023069A1 Heterocyclic compounds having nos inhibitory activities
05/14/1999WO1999022720A2 Selective cyclooxygenase-2 inhibitors against premature labor
05/14/1999WO1999001423A8 Glucagon antagonists/inverse agonists
05/14/1999CA2309175A1 Therapeutically active compounds based on indazole bioisostere replacement of catechol in pde4 inhibitors
05/14/1999CA2309150A1 Indazole bioisostere replacement of catechol in therapeutically active compounds
05/14/1999CA2308639A1 Method of using cyclooxygenase-2 inhibitors in maintaining the fetal ductus ateriosus during treatment and prevention of preterm labor
05/14/1999CA2308428A1 Aromatic heterocyclic compounds as anti-inflammatory agents
05/12/1999EP0915089A2 Methods of preparing 4-cyano-4-(substituted indazole)cyclohexane-carboxylic acids useful as PDE4 inhibitors
05/12/1999EP0914317A2 1-alkyl-4-benzoyl-5-hydroxypyrazole compounds and their use as herbicides
05/12/1999EP0808297B1 Use of not easily volatilised pyrazol derivatives with hydrophilic groups as nitrification inhibitors
05/12/1999EP0583433B1 Diphosphine ligands
05/12/1999CN1216535A Pyrazole compounds, processes for their production and herbicides containing them
05/12/1999CN1216533A 3-cyanoaryl pyrazoles and their use as herbicides
05/12/1999CN1216530A Ethylene derivatives and pest controlling agents
05/12/1999CN1216444A Substituted aminomethyl phenyl sulphonyl ureas, their production and their use as herbicides and plant growth regulators
05/06/1999WO1999021837A1 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
05/06/1999EP0913392A1 Ethylene derivatives and pest controlling agents
05/06/1999EP0912570A1 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
05/06/1999EP0912521A1 Substituted indazole derivatives and their use as inhibitors phosphodiesterase (pde) type iv and the production of tumor necrosis factor (tnf)
05/06/1999EP0912494A1 Coumpounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
05/06/1999CA2307815A1 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
05/05/1999CN1216043A Substd. benzenesulfonamide derivs as prodrugs of COX-2 inhibitors
05/05/1999CN1216040A N-arylsulfilimine compounds and their use as catalysts in preparation of N-arylarylsulfonamide compounds
05/04/1999US5900489 Bromination
05/04/1999CA2184604C Bicyclic carbamates
04/1999
04/29/1999WO1999020607A1 Amide derivatives or salts thereof
04/29/1999WO1999020272A1 Azapeptide acids as cell adhesion inhibitors
04/28/1999EP0911329A1 3-Substituted arylpyrazole derivatives
04/28/1999EP0910564A1 D-amino acid derived inhibitors of cysteine and serine proteases
04/22/1999WO1999019303A1 Pyrazole derivatives
04/22/1999WO1999019300A1 Prostaglandin agonists and their use to treat bone disorders
04/22/1999WO1999018941A2 Ih-MODULATORS
04/22/1999CA2305180A1 Ih-modulators
04/22/1999CA2304979A1 Pyrazole derivatives having a calcium release-activated calcium channel inhibitory effect
04/21/1999EP0712397B1 Amide derivatives as 5ht1d receptor antagonists
04/21/1999EP0579797B1 Diphosphine ligands
04/21/1999CN1214678A Butadiene derivatives and process for preparing thereof
04/21/1999CN1214339A Pyrazole derivatives, their preparation and their use in pharmaceuticals
04/15/1999WO1999018080A1 Process for preparing 3-substituted indazoles
04/15/1999WO1999018079A1 Heteroaryl butyric acids and their derivatives as inhibitors of matrix metalloproteinases
04/15/1999WO1999018076A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/15/1999WO1999017770A1 Indeno[1,2-c]pyrazole derivatives for inhibiting tyrosine kinase activity
04/15/1999WO1999017769A1 INDENO[1,2-c]-, NAPHTHO[1,2-c]- AND BENZO[6,7]CYCLOHEPTA[1,2-c]PYRAZOLE DERIVATIVES
04/15/1999WO1999007674A3 Microbicidal n-sulfonylglycin alkynyloxyphenemethyl amide derivatives
04/15/1999WO1999004770A3 A pharmaceutical composition active in reducing production of mcp-1 protein
04/15/1999WO1998055118A3 Use of nitrogen heterocyclic aromatic derivatives in the topical treatment of the epithelial tissues diseases
04/15/1999CA2306348A1 Process for preparing 3-substituted indazoles
04/15/1999CA2304565A1 Indeno[1,2-c]-, naphtho[1,2-c]- and benzo[6,7]cyclohepta[1,2-c]pyrazole derivatives
04/15/1999CA2304466A1 Indeno[1,2-c]pyrazole derivatives for inhibiting tyrosine kinase activity
04/15/1999CA2303449A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/14/1999EP0908456A1 Pyrazole derivatives, their preparation and their use in drugs
04/14/1999EP0908452A2 Process for preparing 3-substituted indazoles
04/14/1999EP0907637A1 Phenylalamine derivatives as integrin inhibitors
04/14/1999EP0810991B1 1-aryl-2-acylamino-ethane compounds and their use as neurokinin especially neurokinin 1 antagonists
04/14/1999EP0618904B1 Novel n-phenyl amino pyrazole derivatives and means and process for colouring hair
04/14/1999CN1214039A Carbamoyloxy derivatives of mutiline and their use as antibacterials
04/08/1999WO1999016753A2 Tricyclic 3-oxo-propanenitrile compounds
04/08/1999WO1999016751A1 Benzamidine derivatives as factor xa inhibitors
04/08/1999WO1999016453A1 Method for the treatment of cystic fibrosis
04/08/1999WO1999003823A3 Novel polyamine analogues as therapeutic and diagnostic agents
04/08/1999DE19743435A1 Benzamidinderivate Benzamidine derivatives
04/08/1999CA2305568A1 Benzamidinderivates
04/08/1999CA2304482A1 Method for the treatment of cystic fibrosis
04/08/1999CA2302025A1 Tricyclic 3-oxo-propanenitrile compounds
04/07/1999EP0906287A1 Substituted pyrazolyl-pyrazole derivatives and their use as herbicides
04/07/1999EP0906286A1 5-aminopyrazoles useful as selective inhibitors of the protein tyrosine kinase p56ick
04/07/1999EP0906285A1 3-cyanoaryl pyrazoles and use thereof as herbicides
04/07/1999EP0906270A1 Process for producing hydroxyarenes