Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
01/2002
01/03/2002US20020002169 Protein kinase inhibitors
01/03/2002US20020002152 Methionine aminopeptidase type 2 inhibitors; n'-((2S,3R)-3-amino-2-hydroxy-5-(isopropylsulfanyl)pentanoyl)-3-chloro benzoyl hydrazide
01/03/2002US20020002138 For use in treatment of diseases associated with reduced levels of growth hormone
01/02/2002EP1167355A1 A crystalline form of celecoxib
01/02/2002EP1166785A1 Use of pyrazole derivatives for inhibiting thrombin-induced platelet aggregation
01/02/2002EP1165547A1 Substituted benzoylpyrazoles as herbicides
01/02/2002EP1165544A1 Substituted 1,4-dihydroindeno[1,2-c]pyrazoles as inhibitors of tyrosine kinase
01/02/2002EP1165516A2 Heterocyclic urea and related compounds useful as anti-inflammatory agents
01/02/2002EP1165511A2 Method of producing heterocyclic carbamates from aza-heterocyclic compounds and carbon dioxide
01/02/2002EP1165485A2 Processes for preparing pesticidal intermediates
01/02/2002EP1165472A1 Methods for the preparation of biphenyl isoxazole sulfonamides
01/02/2002EP1165072A2 Valdecoxib compositions
01/02/2002CN1329600A Method for control of arthropods in animals
01/01/2002USRE37495 As pesticide, insecticide
01/01/2002US6335440 Method for detecting oligonucleotides using energy transfer dyes with long stoke shift
01/01/2002US6335357 1-aryl-3-cyano-5-(het)arylalkylaminopyrazole derivatives; insecticides for agriculture and horticulture
01/01/2002US6335356 Method of treating a patient by parenteral administration of a lipophilic compound
01/01/2002US6335334 Hypertensive agents, anticoagulants; cardiovascular and sexual disorders, angina pectoris, and atherosclerosis
12/2001
12/27/2001WO2001098304A1 A process for preparing pyrazolopyrimidinone derivatives for the treatment of impotence
12/27/2001WO2001097810A2 Use of therapeutic benzamide derivatives
12/27/2001WO2001097806A1 Cox-2 inhibitors and the prevention of the side effects of radiation therapy
12/27/2001WO2001053268A3 Indazole compounds, pharmaceutical compositions, and their use for mediating or inhibiting cell proliferation
12/27/2001WO2000064864A9 N-protected amines and their use as prodrugs
12/27/2001US20010056189 Pyrazole substituted hydroxamic acid derivatives as cyclooxxgenase-2 and 5- lipoxygenase inhibitors
12/27/2001US20010055565 Method of detecting cyclooxygenase-2
12/27/2001CA2412362A1 Cox-2 inhibitors and the prevention of the side effects of radiation therapy
12/26/2001CN1327793A Pyrrolo-triazine and pyrimidine compounds
12/26/2001CN1076584C Use of etychlozate as plant growth regulator in production of water melon
12/25/2001US6333425 Ionic compounds derived from malononitrile in which anionic charge is delocalized; excellent properties of solubility and dissociation
12/25/2001US6333343 Diphenyl-triazole derivatives and their use as anti-gestative, immuno-suppressant and anti-tumoral agents
12/25/2001US6333330 Pyrazolopyrimidinone CGMP PDE5 inhibitors for the treatment of sexual dysfunction
12/25/2001US6333325 Method of treating cytokine mediated diseases or conditions
12/25/2001US6333296 Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them
12/20/2001WO2001096334A2 Heteroarylalkanoic acids as integrin receptor antagonists
12/20/2001WO2001096323A1 Serine protease inhibitors
12/20/2001WO2001096307A2 Cycloalkyl alkanoic acids as integrin receptor antagonists
12/20/2001WO2001096297A2 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
12/20/2001US20010053856 Sunscreen agents; ultraviolet radiation absorber
12/20/2001US20010053854 Pesticidal compounds and compositions
12/20/2001US20010053788 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity
12/20/2001CA2412618A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
12/20/2001CA2411805A1 Serine protease inhibitors
12/18/2001USRE37478 1-(arylthioalkyl, arylaminoalkyl, or arylmethylenealkyl)-4-(heteroaryl)piperazines and related compounds useful as antipsychotics and analgesics
12/18/2001US6331563 N-Hydroxy-2-(Alkyl, Aryl, or Heteroaryl, Sulfanyl, Sulfinyl or Sulfonyl)-3-Substituted Alkyl, Aryl or Heteroarylamides as Matrix Metalloproteinase inhibitors
12/18/2001US6331553 Inhibitors of nitric oxide synthase; treating cerebrovascular diseases
12/18/2001US6331542 Protease inhibitors
12/18/2001US6331507 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
12/18/2001CA2208585C Benzamidoxime derivative, process for production thereof, and agrohorticultural bactericide
12/13/2001WO2001094316A1 Processes for the preparation of pesticidal compounds and novel intermediates thereof
12/13/2001WO2001094315A2 Process for the preparation of pesticidal compounds
12/13/2001WO2001049275A3 Methods and compositions for mitigating pain using nitrate esters
12/13/2001WO2001025241A3 Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides
12/13/2001US20010051651 Administering effective amount of 1,3,6-trihydro-6-aza-3-oxapentalen-2-one derivative to the patient for inducing or promoting apoptosis and for arresting uncontrolled neoplastic cell proliferation
12/12/2001EP1161420A2 Fungicidal pyrazole carboxanilides
12/12/2001EP0917526B1 use of polyacids to treat mineral fertilizers containing a nitrification inhibitor
12/12/2001EP0772597B1 3,4-substituted pyrazoles for the treatment of inflammation
12/12/2001CN1326446A Method for producing 5-Amino-3-(thio) carbamoylpyrazoles
12/11/2001US6329531 For therapy of alzheimer's disease
12/11/2001US6329530 Method for the production of 1-substituted 5-hydroxypyrazoles
12/11/2001US6329527 Acylating substitutedaryl hydrazine, forming dipolar compound, contacting dipolarophile and subjecting to oxidation, removing protecting group
12/11/2001US6329415 Aromatic heterocyclic compounds as antiinflammatory agents
12/11/2001US6329412 Bisamidine compounds as antiproliferative agents
12/11/2001US6329402 Heterocycle-containing carboxylic acid derivative and drug containing the same
12/11/2001US6329372 Phenylalanine derivatives
12/06/2001WO2001092273A2 Benzenedicarboxylic acid derivatives
12/06/2001WO2001092241A1 Benzamide derivatives and their use as apob-100 and mtp inhibitors
12/06/2001WO2001092218A2 Polyamine analogues as therapeutic and diagnostic agents
12/06/2001US20010049374 Amidino derivatives of quinoline and naphthalene
12/06/2001CA2410935A1 Novel polyamine analogues as therapeutic and diagnostic agents
12/05/2001EP1160331A1 Enzymatic oxidations
12/05/2001EP1160248A1 N-(Isoxazol-5-yl)-sulfonamide derivatives and their use as endothelin antagonists
12/05/2001EP1159264A2 INHIBITORS OF FACTOR Xa
12/05/2001EP1159262A1 Tyrosine alkoxyguanidines as integrin inhibitors
11/2001
11/30/2001CA2349057A1 Enzymatic oxidations
11/30/2001CA2348847A1 New isoxazole-sulfonamide endothelin antagonists
11/29/2001WO2001090078A1 Pyrazole derivatives and their use as gastrin and cholecystokin in receptor ligands
11/29/2001WO2001089457A2 Thrombopoietin mimetics
11/29/2001US20010047031 Heterocyclic compounds useful as NMDA receptor selective subtype blockers
11/29/2001US20010047023 1-(p-(methylsulfonamido)phenyl)-3-trifluoromethyl-5-phenylpyra zolone and derivatives; antiinflammatory agents
11/28/2001EP1157990A2 Squarylium dye and filter for display device
11/28/2001EP1157010A1 Pyrazole-3-on-derivative as factor xa inhibitors
11/28/2001EP1157003A1 Acylated aminoacetonitriles as cysteine protease inhibitors
11/28/2001EP1157002A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy
11/28/2001EP1156804A1 Thrombopoietin mimetics
11/28/2001EP0777654B1 N-phenyltetrahydroindazoles, their preparation, and their use as crop protection agents
11/28/2001CN1075490C O-benzyl oxime ether derivatives and their use in crop production compositions
11/27/2001US6323230 Epicuaneous route in the case of dermatological illnesses like psoriasis, atopic dermatitis and other similar affections, or when administered by oral or rectal route in the case of diseases of the epithelia of the lower intestines
11/27/2001US6323227 Prodrugs
11/27/2001US6322775 For coloring the skin and/or the hair; side effects reduction; stability
11/22/2001WO2001087888A1 Pyrazolopyrimidinone derivatives, process for their preparation and their use
11/22/2001WO2001087846A2 Tricyclic pyrazole derivatives as protein kinase inhibitors
11/22/2001WO2001087830A2 Substituted thioacetamides
11/22/2001WO2001087343A2 Combination therapy using cox-2 selective inhibitor and thromboxane inhibitor and compositions therefor
11/22/2001WO2001087287A2 Use of pyrazole derivatives for treating infertility
11/22/2001WO2001047475A3 Agent for dyeing keratin containing fibers
11/22/2001WO2001005769A3 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
11/22/2001US20010044445 Azole inhibitors of cytokine production
11/22/2001CA2409225A1 Tricyclic pyrazole derivatives
11/22/2001CA2409116A1 Substituted thioacetamides
11/22/2001CA2407469A1 Combination therapy using cox-2 selective inhibitor and thromboxane inhibitor and compositions therefor