Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
04/2001
04/19/2001WO2001027103A1 Fab i inhibitors
04/19/2001WO2001027081A1 6-position substituted indoline, production and use thereof as a medicament
04/19/2001WO2001027080A2 5-substituted indolinones and use thereof as kinase and cyclin/cdk complex inhibitors
04/19/2001WO2001026654A1 Fab i inhibitors
04/19/2001WO2001026653A1 V TYPE AND/OR X TYPE sPLA2 INHIBITORS
04/19/2001WO2001026652A1 Fab i inhibitors
04/19/2001WO2000046198A8 Anti-inflammatory indole derivatives
04/19/2001WO2000018767A9 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
04/19/2001DE19949209A1 In 5-Stellung substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel In the 5-position substituted indolinones, their preparation and their use as medicaments
04/19/2001DE19949208A1 New 3-(amino-methylene)-2-indolinone derivatives are kinase inhibitors and cell proliferation inhibitors useful e.g. for treating tumors, metastasis, rheumatoid arthritis or psoriasis
04/18/2001EP1092753A1 Cyanine dye
04/18/2001EP1091937A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
04/18/2001EP1091930A1 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES
04/18/2001EP1091726A2 Analogs of 2-phthalimidinoglutaric acid and their use as inhibitors of angiogenesis
04/18/2001EP0968250B1 Soluble chromophores having improved solubilising groups
04/18/2001EP0934268A4 Process for preparing 2-azadihydroxybicyclo 2.2.1]heptane compounds and the l-tartaric acid salt of the compound
04/18/2001EP0797437B1 IMMUNOTHERAPEUTIC IMIDES/AMIDES AND THEIR USE FOR REDUCING LEVELS OF TNFalpha
04/18/2001CN1291976A Indole ferivatives and medicinal compositions containing same
04/18/2001CN1291973A N-sulphonyl and N-sulphinyl phenylglycinamide
04/18/2001CN1064674C Alkoxyaryl compounds, their process of preparation and pharmaceutical compositions which contain them
04/17/2001US6218576 Process for producing a diarylamine
04/17/2001US6218548 (triarylmethyl)aminospiropyrroles
04/17/2001US6218536 1,2-bis-adducts of stable nitroxides with substituted ethylenes and stabilized compositions
04/17/2001US6218429 Tricyclic compounds, their production and use
04/17/2001US6218426 For therapy of mammalian reproductive disorders and steroid hormone-dependent tumors as well as for regulating fertility, where suppression of gonadotropin release is indicated
04/17/2001US6218419 Aminoiminoquinone and aminoquinone alkaloid compounds and methods of use
04/17/2001US6218406 As antitumor and antileukemic agents
04/17/2001US6218389 For therapy and prophylaxis of arthritis, cancer, cardiovascular disorders; skin disorders; ocular disorders; inflammation and gum diseases, multiple sclerosis, cachexia, preventing loosening of prosthetic devices
04/17/2001US6218359 Treating autoimmune, arthritic, tumor diseases
04/17/2001US6218072 Optical information recording medium
04/17/2001CA2080475C Neuroprotective indolone and related derivatives
04/17/2001CA2010963C Process for the preparation of lactam derivatives
04/12/2001WO2001025198A1 Method for improving the solubility of tricyclic amino alcohol derivatives
04/12/2001WO2001025197A1 Antifungal enediynes
04/12/2001WO2001025196A2 Slurry preparation of bis(halophthalimides) and of polyether polymers
04/12/2001WO2001025181A1 Carboxylic acid derivatives and drugs containing the same
04/12/2001WO1999057117A3 Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
04/12/2001CA2386373A1 Method for improving the solubility of tricyclic amino alcohol derivatives
04/11/2001EP1089997A1 4,5,6 and 7-indole and indoline derivatives, their preparation and use
04/11/2001EP1089964A1 Hydrazine derivatives
04/11/2001EP0775113B1 N-substituted azabicycloheptane derivatives useful as neuroleptics
04/11/2001CN1291185A Phtalimido arylpiperazines as alpha IA receptor antagonists useful in the treatment of benign prostatic hyperplasia
04/11/2001CN1291183A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl-3-substituted-alkyl, aryl or heteroarylamides) as matrix metallo protein inhibitors
04/11/2001CN1291174A Compound for use as a mineral fiber binder and process for providing such
04/11/2001CN1291095A Chemical compounds
04/11/2001CN1290697A Acylation method
04/11/2001CN1064350C Aryl and heteroaryl alkoxynaphtalene derivatives
04/11/2001CN1064349C Novel tricyclic amide, its preparing method and medicinal composition
04/10/2001US6214994 Treatment of neoplastic diseases, bacterial or fungal infections, and preventing or decreasing production of phosphorylated paired helical filament (phf) epitopes associated with alzheimer's disease
04/10/2001US6214991 3-(4,5,7-trifluorobenzothiazol-2-yl)methyl-indole-n-acetic acid, ethyl ester for example; treating complications of diabetes mellitus, such as cataracts, retinopathy, nephropathy, and neuropathy
04/10/2001US6214877 Antidiabetic agents; modulator of glucose concentration
04/10/2001US6214859 Psychological disorders; alzheimer's disorders; parkinson'sdisorders
04/10/2001US6214858 Caspases and apoptosis
04/10/2001US6214857 Substituted alkanohydroxamic acids and method of reducing TNFα levels
04/10/2001US6214856 Treating neurodegenerative disorders, e.g., alzheimer's disease, strokes, traumatic brain injury; antiischemic agents; muscular dystrophy; also cataracts; platelet aggregation
04/10/2001US6214854 Administering adrenoceptor, or antagonist thereof; cardiovascular disorders
04/10/2001US6214835 Dihalopropene compounds insecticides containing them as active ingredients, and intermediates for their production
04/10/2001US6214829 Piperazine compounds, their preparation, and methods of using them
04/10/2001US6214790 Neo-tryptophan
04/10/2001US6214481 Organic blue-emitting layer sandwiched between two electrodes
04/10/2001CA2133413C Indole derivatives as 5-ht1 antagonists
04/05/2001WO2001023496A1 Organic electroluminescent element
04/05/2001WO2001023374A1 Piperazine derivatives as 5-ht1b antagonists
04/05/2001WO2001023354A2 Trifluoromethyl-substituted spirocyclic ketoenols and use thereof as pesticides and herbicides
04/05/2001WO2001023353A2 Method for producing indole derivatives on a solid phase
04/05/2001WO2001023347A1 Novel aromatic compounds
04/05/2001WO2001023346A2 Process for phenylacetic acid derivatives
04/05/2001WO2001022966A1 Caspases and apoptosis
04/05/2001WO2001022951A2 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives for the treatment of multiple sclerosis
04/05/2001WO2001012602A8 Condensed indoline derivatives and their use as 5ht, in particular 5ht2c, receptor ligands
04/05/2001DE19955087A1 Solid phase synthesis of indole derivatives comprises bonding of the indole nitrogen to a solid phase having vicinal diol groups by trans-acetalization of dialkoxymethyl protected indoles.
04/05/2001DE19947863A1 New 3-salicyloyl-indole derivatives, useful for treating diseases dependent on protein kinase or estrogenic activity, especially tumor diseases, proliferative epidermal diseases or osteoporosis
04/05/2001DE19946625A1 Trifluormethylsubstituierte spirocyclische Ketoenole Trifluoromethyl-substituted spirocyclic ketoenols
04/05/2001DE19942700C1 Verfahren zur Herstellung cyclischer N-Hydroxydicarboximide A process for producing cyclic N-hydroxydicarboximides
04/05/2001CA2386074A1 Method for producing indole derivatives on a solid phase
04/05/2001CA2385737A1 Piperazine derivatives as 5-ht1b antagonists
04/05/2001CA2385490A1 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives for the treatment of multiple sclerosis
04/05/2001CA2384501A1 Trifluoromethyl-substituted spirocyclic ketoenols
04/04/2001EP1088824A2 Bicyclic pyrrolyl amides as glycogen phosphorylase inhibitors
04/04/2001EP1088817A2 Process for the preparation of 3-acyl-indoles
04/04/2001EP1088481A2 Fungicides for the control of take-all disease of plants
04/04/2001EP1087954A1 Cycloalkyl-substituted aryl-piperazines, piperidines and tetrahydropyridines as serotonergic agents
04/04/2001EP1087935A1 Anthracene derivatives as anti-cancer agents
04/04/2001CN1290250A Sulfonylamino derivatives which inhibit matrix-degrading metallopr teinases
04/04/2001CN1290249A Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof
04/04/2001CN1064063C Process for producing dioxazine compounds
04/03/2001US6211395 Enantioselective synthesis of 3-aminopyrrolidines
04/03/2001US6211377 Extracting aqueous reaction solution with organic solvent, separating resulting organic phase containing the (+-)-2-azabicyclo(2.2.1)hept-5-en-3-one from resulting aqueous phase, mixing resulting organic phase with water, separating
04/03/2001US6211365 Fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
04/03/2001US6211245 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
04/03/2001US6211242 Benzamide derivatives as vasopressin antagonists
04/03/2001US6211234 Substituted phenyl compounds
04/03/2001US6211224 Antagonists of gonadotropin releasing hormone
04/03/2001US6211219 Drugs, analgesics and agonists
04/03/2001US6210657 Use of isoindolinone derivatives as stabilizers for organic materials
04/03/2001CA2022486C 1,3-dihydro-1-(pyridinylamino)-2h-indol-2-ones, a process for their preparation and their use as medicaments
03/2001
03/30/2001CA2321379A1 Bicyclic pyrrolyl amides as glycogen phosphorylase inhibitors
03/29/2001WO2001021589A2 Mono- and bis-indolylquinones and prophylactic and therapeutic uses thereof
03/29/2001WO2001021588A2 Cycloalkyl bicycloheptene dicarboximides
03/29/2001WO2001021587A2 Hydroxyfunctional amide 1h-indole derivatives active as spla2 inhibitors