Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
03/2001
03/13/2001US6200988 Tetrahydroquinoline derivates; inhibitors of acyl coa:cholesterol acyltransferase and lipoperoxidation; arteriosclerosis: cardiovascular and brain disorders
03/13/2001US6200987 Cyclic amides
03/13/2001US6200978 For preventing or treating inflammatory diseases such as arthritis, psoriasis, asthma, or inflammatory bowel disease, disorders of respiratory function, gastrointestinal disorders such as functional bowel disease, as analgesics
03/13/2001US6200971 For treating atherosclerosis
03/13/2001US6200967 Used as thrombin inhibitors, coagulation inhibitors and agents for the treatment of thromboembolic disorders
03/08/2001WO2001016130A1 Substituted indolinones as tyrosine kinase inhibitors
03/08/2001WO2001016108A2 Bicyclic androgen and progesterone receptor modulator compounds and methods
03/08/2001WO2001016104A1 Cyclopropylindole derivatives
03/08/2001WO2001016103A1 Fused pyrrolecarboxamides: gaba brain receptor ligands
03/08/2001WO2001016102A1 ISOLATION OF NATURAL L-β-3-INDOLYLALANINE AND ENRICHMENT OF NATURAL ALIPHATIC AMINO ACID MIXTURES WITH NATURAL L-β-3-INDOLYLALANINE
03/08/2001WO2001016101A1 Process for the preparation of indole derivatives or salts thereof
03/08/2001WO2001016097A1 Phosphate mimics and methods of treatment using phosphatase inhibitors
03/08/2001WO2001016058A1 Catalyst for pauson-khand reaction
03/08/2001WO2001015686A1 Selective cox-2 inhibitory novel esters from indolealkanols and novel amides from indolealkylamines
03/08/2001WO2001015673A2 Pharmaceutical formulations and use thereof in the prevention of stroke, diabetes and/or congestive heart failure
03/08/2001WO2000059885A8 Method for the preparation of tricyclic amino alcohol derivatives through azides
03/08/2001WO1999063930A8 Novel angiotensin receptor modulators and their uses
03/08/2001WO1999019296A8 Aminobutanoic acid derivatives
03/08/2001DE19937537A1 Substituierte 2-Dialkylaminoalkylbiphenyl-Derivate 2-substituted derivatives Dialkylaminoalkylbiphenyl
03/08/2001CA2417639A1 Isolation of natural l-.beta.-3-indolylalanine and enrichment of natural aliphatic amino acid mixtures with natural l-.beta.-3-indolylalanine
03/08/2001CA2384435A1 Bicyclic androgen and progesterone receptor modulator compounds and methods
03/08/2001CA2382789A1 Phosphate mimics and methods of treatment using phosphatase inhibitors
03/08/2001CA2382116A1 Process for the preparation of indole derivatives or salts thereof
03/08/2001CA2381821A1 Substituted indolinones, their manufacture and their use as medicaments
03/08/2001CA2381553A1 Fused pyrrolecarboxamides: gaba brain receptor ligands
03/07/2001EP1081136A1 Optically active tetrahydrobenzindole derivatives
03/07/2001EP1081135A2 1H-indole-3-glyoxylamide spla2 inhibitors
03/07/2001EP1081132A1 Hydroxamic acid derivatives and medicinal utilization thereof
03/07/2001EP1080095A1 Modulators of protein tyrosine phosphatases (ptpases)
03/07/2001EP1080080A1 Novel therapeutic agents that modulate neurokinin receptors
03/07/2001EP1080078A1 Heterocyclic compounds and methods to treat cardiac failure and other disorders
03/07/2001EP1080074A1 New heterocyclically substituted amides, their production and their use
03/07/2001EP1080073A1 Compositions comprising 2-phenyl-indole compounds and estrogen formulations
03/07/2001EP1080068A1 Modulators of protein tyrosine phosphatases
03/07/2001EP1080066A1 Bioreductive cytotoxic agents
03/07/2001EP1079830A1 BENZIMIDAZOLE ANALOGS AS DOWN-REGULATORS OF IgE
03/07/2001EP1079828A1 New use
03/07/2001EP1079826A2 Use of indigoid bisindole derivatives for the manufacture of a medicament to inhibit cyclin dependent kinases
03/07/2001EP1079763A2 Serotonergic 5ht 7? receptor compounds for treating ocular and cns disorders
03/07/2001EP0777650B1 Biphenylamide derivatives as 5ht 1d antagonists
03/07/2001EP0730579B1 Substituted indoles as phosphodiesterase type iv inhibitors
03/07/2001CN2422282Y Light-weight and small metal phthalocyanine device
03/07/2001CN1286683A Tetrahydrobenzindole derivs
03/07/2001CN1062865C Process for production of amidinobenzofuran and amidinobenzothiophen derivs. and salt thereof
03/06/2001US6198000 Intermediates useful in the synthesis of quinoline antibiotics
03/06/2001US6197975 7-azabicyclo(2.2.1)heptane-7-carbonyl-substituted 2-phenylindole derivatives; sexual disorders; anticarcinogenic agents
03/06/2001US6197974 Enantioselective synthesis of 3-aminopyrrolidines
03/06/2001US6197968 Storage stability; colorless after solution treatment
03/06/2001US6197956 Cyanine dyes and synthesis methods thereof
03/06/2001US6197791 N-hdroxy-2-(alkyl, aryl, or heteroaryl, sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
03/06/2001US6197773 N-acyl and N-aroyl aralkyl amides as serotonergic agents
03/06/2001US6197770 Alkenyl- and alkynl-containing metalloprotease inhibitors
03/06/2001US6197750 C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases
03/06/2001CA2223081C Heterocyclic ring-fused pyrimidine derivatives
03/06/2001CA1341196C Process for the preparation of substituted imino diacids
03/01/2001WO2001014380A1 Isomeric fused pyrrolocarbazoles and isoindolones
03/01/2001WO2001014330A2 Phenylpiperazines as serotonin reuptake inhibitors
03/01/2001WO2001014328A2 Substituted ureas as cell adhesion inhibitors
03/01/2001WO2001014320A1 Compounds that inhibit tryptase activity
03/01/2001WO2001014316A1 Substituted chiral allosteric hemoglobin modifiers
03/01/2001WO2000068223A8 Ureas and their use as cell adhesion modulators
03/01/2001DE19940829A1 New 3-(anilino-methylidene)-2-indolinone derivatives, are kinase inhibitors and cell proliferation inhibitors, useful e.g. for treating tumors, metastasis, rheumatoid arthritis or psoriasis
03/01/2001DE19939910A1 Neue Verbindungen, die Tryptase-Aktivität hemmen Novel compounds that inhibit tryptase activity
03/01/2001CA2384511A1 Substituted chiral allosteric hemoglobin modifiers
03/01/2001CA2381096A1 Compounds that inhibit tryptase activity
03/01/2001CA2316767A1 Somatostatin antagonists and agonists that act at the sst subtype 2 receptor
02/2001
02/28/2001EP1077978A1 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors
02/28/2001EP1077969A1 Benzothiophenes, benzofurans, and indoles useful in the treatment of insulin resistance and hyperglycemia
02/28/2001EP1077968A1 Naphtho[2,3-b]heteroar-4-yl derivatives
02/28/2001EP1077944A1 Carboxamide compounds, compositions, and methods for inhibiting parp activity
02/28/2001EP1077941A1 Compounds with growth hormone releasing properties
02/28/2001EP1077939A1 Method for making substituted indoles
02/28/2001EP1077929A1 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
02/28/2001EP1077928A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
02/28/2001EP1077927A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
02/28/2001EP1077700A1 BENZIMIDAZOLE DERIVATIVES AS MODULATORS OF IgE
02/28/2001EP1077695A2 COMPOUNDS HAVING IgE AFFECTING PROPERTIES
02/28/2001EP1077694A1 Aryl nitrone therapeutics for the treatment of inflammatory bowel disease
02/28/2001EP0888339A4 Synthesis of indolylmaleimides
02/28/2001CN1285817A Novel tricyclic compounds, preparation method and pharmaceutical compositions containing same
02/27/2001US6194586 Selective sulphonation of the primary alcohol of a diol containing both primary and secondary alcohols
02/27/2001US6194439 Tricyclic polyhydroxylic tyrosine kinase inhibitors
02/27/2001US6194437 Non-peptide bombesin receptor antagonists
02/27/2001US6194424 Arylacetamides and their use as medicaments
02/27/2001US6194416 Central nervous system disorders; alzheimer's disease
02/27/2001US6194396 Benzimidazole compounds as bradykinin antagonists
02/27/2001US6194132 Photographic element, compound, and process
02/27/2001CA2124206C Indole derivatives
02/27/2001CA2111204C Piperidine derivatives having anxiolytic effect
02/27/2001CA2101316C Gnrh analogs
02/27/2001CA1341195C Tinctorial compositions for keratinic fibers and dyeing process using these compositions
02/22/2001WO2001012699A1 Electrically conductive polymers capable of being covalently grafted on by light, method for obtaining same and uses as supports in probes for specific identification in electronic biosensors
02/22/2001WO2001012603A1 Indole derivatives, process for their preparation, pharmaceutical compositions containing them and their medicinal application
02/22/2001WO2001012602A1 Condensed indoline derivatives and their use as 5ht, in particular 5ht2c, receptor ligands
02/22/2001WO2001012601A1 Novel anilide derivatives or salts thereof and drugs containing the same
02/22/2001WO2001012600A1 INHIBITORS OF FACTOR Xa
02/22/2001WO2001012587A1 Aminosalicylclic acid amides and their use for combating organisms that are harmful to plants
02/22/2001WO2001012576A1 Synthesis of cyclooctatetraene derivatives and their use as electron transporters in organic light emitting diodes
02/22/2001WO2001012575A1 Methods for preparing perfluorinated [18f]-radiolabelled nitroimidazole derivatives for cellular hypoxia detection
02/22/2001WO2001012187A2 Benzoic acid derivatives and their use as ppar receptor agonists