Patents
Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868)
10/2001
10/04/2001WO2001072704A1 AZETIDINONE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND A METHOD FOR PRODUCING 1-β-ALKYL AZETIDINONE USING THE SAME
10/04/2001WO2001072687A1 Diphenyl ether compounds useful in therapy
10/04/2001WO2001029245A8 ENZYMATIC PROCESS FOR THE RESOLUTION OF ENANTIOMERIC MIXTURES OF β-LACTAMS
10/04/2001US20010027193 1-Diarylmethyl-4-alkyl or alkylsulfonylalkyl-azetidines; cannabinoid receptor antagonists; nervous system disorders (CNS); cardiovascular and glandular disorders; drug abuse; psychological disorders;
10/04/2001EP1137634A1 Process for the synthesis of azetidinones
10/04/2001CA2404439A1 Diphenyl ether compounds useful in therapy
10/03/2001CN1072222C Phenyloxazolidinones having C-C bond to 4-8 membered heterocyclic rings
10/02/2001CA2037541C Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
09/2001
09/27/2001US20010025103 Bactericides
09/26/2001CN1314886A Process for production of N-protected azetidinie-2-carboxylic acids (AzeOHs)
09/26/2001CN1071745C Process for synthesis of acetidinones
09/25/2001CA2214051C Beta-lactams useful in preparation of taxols
09/19/2001CN1313855A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta
09/19/2001CN1071292C Improved process for prodn. of enantiomericallypure azetidine-2-carboxylic acid
09/13/2001WO2001066534A2 Cyclic and bicyclic diamino histamine-3 receptor antagonists
09/12/2001EP0707567B1 Process for the synthesis of azetidinones
09/07/2001WO2001064634A1 Pharmaceutical compositions containing azetidine derivatives, novel azetidine derivatives and preparation thereof
09/07/2001WO2001064633A1 Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
09/07/2001WO2001064632A1 Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
09/07/2001CA2400138A1 Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
09/07/2001CA2400116A1 Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
09/05/2001CN1311679A Benzimidazole derivatives as modulators of IgE
09/05/2001CN1311675A Compounds having IgE affecting properties
09/04/2001CA2224062C Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors
08/2001
08/30/2001WO2000071510A3 INHIBITORS OF FACTOR Xa
08/30/2001US20010018423 Anticoagulant agents
08/29/2001CN1310629A Coadministration of ACAT and MMP inhibitors for the treatment of atherosclerotic lesions
08/28/2001US6281243 Derivatives of azetidine and pyrrolidine
08/23/2001WO2001060828A1 Intermediates for and synthesis of 3-methylene cephams
08/23/2001WO2000071508A3 Inhibitors of factor Xa
08/22/2001CN1309634A Hydrazine derivs.
08/21/2001CA2196845C Hydroxamic acid compounds
08/16/2001WO2001058891A2 Piperazine and piperidine derivatives for treatment or prevention of neuronal damage
08/16/2001WO2001010842A3 Melanocortin-4 receptor binding compounds and methods of use thereof
08/16/2001US20010014746 Preparation of substituted isoserine esters using metal alkoxides and beta-lactams
08/16/2001EP0788498B1 Phenyloxazolidinone antimicrobials
08/16/2001CA2398822A1 Piperazine and piperidine derivatives
08/15/2001CN1308251A Photographic element, compound and method containing azacyclo-substrated color former
08/09/2001WO2001056986A1 New coupling process
08/09/2001WO2001056985A1 Process for cyclizing optically active 4-amino-2-halogenobutyric acids
08/09/2001WO2000071511A3 INHIBITORS OF FACTOR Xa
08/09/2001US20010012857 Pharmaceutical for treatment of neurological and neuropsychiatric disorders
08/09/2001CA2396743A1 New coupling process
08/08/2001CN1307560A Amidino and guanidino beta-azetidinone tryptase inhibitors
08/07/2001US6271390 Suppression of the IgE-dependent allergic response by benzimidazole analogs
08/02/2001WO2001055104A1 Process for preparation of optically active n-substituted azetidine-2-carboxylic acids
07/2001
07/25/2001EP1118907A2 Photographic element containing nitrogen heterocycle substituted cyan coupler, compound and process
07/25/2001EP1117823A1 Resolution of trans-2 -(alkoxycarbonylethyl) -lactams useful in the synthesis of 1- (4-fluorophenyl) -3(r) - 3(s) -hydroxy-3 -(4-fluorophenyl) -propyl)] -4(s) -(4-hydroxyphenyl) -2-azetidinone
07/24/2001US6265397 Amidino derivatives and their use as thrombin inhibitors
07/19/2001WO2001051456A2 Antibacterial agents
07/19/2001CA2397575A1 Antibacterial agents
07/18/2001EP1071685A4 Titanium catalyzed preparation of carbapenem intermediates
07/17/2001US6262278 Reacting water and mixture of stereoisomers of chiral cyclic substrate in the presence of non-racemic chiral catalyst to produce by kinetic resolution stereoisomerically enriched cyclic substrate or stereoisomerically enriched hydrolyzate
07/17/2001US6262046 Azetidinylpropylpiperidine derivatives, intermediates and use as tachykinin antagonists
07/11/2001EP1007511A4 Preparation of beta-methyl carbapenem intermediates
07/11/2001EP0823896B1 Substituted oximes, hydrazones and olefins as neurokinin antagonists
07/11/2001CN1068325C Phenyloxazolidinone antimicrobials
07/05/2001WO2001047868A1 Novel phenylalanine derivatives
07/04/2001EP1112251A1 Azetidine derivatives, preparation and medicines containing them
07/04/2001EP1112250A1 Therapeutic compounds and methods
07/03/2001US6255301 Amino acid derivatives and their use as thrombin inhibitors
06/2001
06/28/2001WO2001046135A1 Synthesis of chiral 2-azetidinemethanol compounds
06/28/2001CA2395169A1 Synthesis of chiral 2-azetidinemethanol compounds
06/27/2001EP1109782A1 PROCESS FOR THE PRODUCTION OF N-PROTECTED AZETIDINE-2-CARBOXYLIC ACIDS (AzeOHs)
06/27/2001CN1067682C Anti-tumor compounds, pharmaceutica compositions, methods for preparation thereof and for treatment.
06/21/2001WO2001029245A3 ENZYMATIC PROCESS FOR THE RESOLUTION OF ENANTIOMERIC MIXTURES OF β-LACTAMS
06/20/2001EP1108717A2 C7 taxane derivatives and pharmaceutical compositions containing them
06/14/2001WO2001042249A1 Olefin polymerization cocatalysts derived from group-15 compounds and processes using them
06/14/2001WO2001041724A2 Compositions for dyeing keratinic fibres, containing paraphenylenediamine derivatives with an azetidinyl group
06/14/2001WO2001007022A3 Azetidine compounds in cns and eye diseases
06/14/2001CA2391855A1 Olefin polymerization cocatalysts derived from group-15 compounds and processes using them
06/14/2001CA2362623A1 Compositions for dyeing keratinic fibres, containing paraphenylenediamine derivatives with an azetidinyl group
06/13/2001EP0573667B1 Process for producing 4-substituted azetidinone derivative
06/06/2001EP1104395A1 Stereoselective ring opening reactions
06/06/2001CN1298389A Cyclic amino compounds
06/05/2001US6242596 Preparation of betamethyl carbapenem intermediates
06/05/2001US6242439 Azetidinone derivatives for the treatment of HCMV infections
06/05/2001US6242438 3-Azetidinylalkylpiperidines or -pyrrolidines as tachykinin antagonists
05/2001
05/30/2001CN1066438C Preparation of beta-methyl carbapenem intermediates
05/29/2001US6239175 Carbamoyloxy derivatives of mutiline and their use as antibacterials
05/29/2001US6239151 Compounds as inhibitor of tumor necrosis factor alpha release
05/29/2001US6239125 Antiviral agents against herpes viruses.
05/25/2001WO2001007023A3 Azetidine compounds in cns and eye diseases
05/16/2001EP1099690A1 MONOCYCLIC $g(b)-LACTAM COMPOUNDS AND CHYMASE INHIBITORS CONTAINING THE SAME
05/16/2001EP1098876A1 Cyclisation process
05/16/2001EP1098662A2 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
05/09/2001EP0693057B1 Process for the preparation of 4-(formylthio)-azetidin-2-one derivatives and penem derivatives
05/08/2001US6228853 Pyrrolopyrrolone derivatives as inhibitors of neutrophil elastase
05/02/2001EP0906255B1 Process for the production of enantiomerically-pure azetidine-2-carboxylic acid
05/02/2001CN1065240C Taxanes having butenyl substituted side-chain and pharmaceutical compositions containing them
05/01/2001US6225463 Reacting s-amine compound with an aldehyde; reacting with acyl chloride in presence of triethylamine to form diastereoisomeric beta-lactams; separation; treating with cerium ammonium nitrate and acetonitrile and water
05/01/2001US6225351 For therapy of asthma, arthritis, and sepsis bronchitis, chronic obstructive airways disease, psoriasis, allergic rhinitis, dermatitis, sepsis, septic shock, cachexia, acquire immuno deficiency syndrome (aids)
04/2001
04/26/2001WO2001029245A2 ENZYMATIC PROCESS FOR THE RESOLUTION OF ENANTIOMERIC MIXTURES OF β-LACTAMS
04/26/2001CA2386487A1 Enzymatic process for the resolution of enantiomeric mixtures of .beta.-lactams
04/25/2001EP0701568B1 New peptide derivatives
04/25/2001CN1064958C Method for preparation of taxol midbody
04/24/2001US6221865 Inhibitors of protein farnesyltransferase and protein geranylgeranyltransferase.
04/17/2001US6218553 Process for the preparation of taxane derivatives and β-lactam intermediates therefor
04/11/2001EP1089989A1 Inhibitors of alpha4beta1 mediated cell adhesion
04/11/2001EP1089973A1 Amidino and guanidino azetidinone tryptase inhibitors
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