| Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868) |
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| 11/18/2004 | US20040229860 For enhancing bone formation; for therapy of diseases or disorders associated with abnormal bone or mineral homeostasis |
| 11/18/2004 | US20040229848 For therapy of non-insulin dependent diabetes |
| 11/18/2004 | CA2523235A1 3-(1-naphthyl)-2-cyanopropanoic acid derivatives as estrogen receptor ligands |
| 11/11/2004 | WO2004096794A1 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disordrs |
| 11/11/2004 | WO2004096763A1 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders |
| 11/11/2004 | WO2004096287A2 Inosine monophosphate dehydrogenase inhibitory phosphonate compounds |
| 11/11/2004 | WO2004096286A2 Antiviral phosphonate analogs |
| 11/11/2004 | WO2004096236A2 Immunomodulator phosphonate conjugates |
| 11/11/2004 | WO2004096235A2 Anti-cancer phosphonate analogs |
| 11/11/2004 | CA2524251A1 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders |
| 11/11/2004 | CA2523083A1 Antiviral phosphonate analogs |
| 11/11/2004 | CA2519840A1 Anti-cancer phosphonate analogs |
| 11/10/2004 | CN1545555A Enzymatic resolution of t-butyl taxane derivatives |
| 11/04/2004 | WO2004071454A3 Substituted azetidine compounds as inhibitors of dipeptidyl peptidase iv |
| 11/04/2004 | WO2004042351A3 Piperidinyl-alpha-aminoamide modulators of chemokine receptor activity |
| 11/04/2004 | US20040220191 Substituted N-aryl heterocycles, process for their preparation and their use as medicaments |
| 11/04/2004 | DE10314610A1 Neues Diphenylazetidinon mit verbesserten physiologischen Eigenschaften, Verfahren zu dessen Herstellung, diese Verbindungen enthaltende Arzneimittel und dessen Verwendung New diphenylazetidinone with improved physiological properties, process for its preparation, pharmaceutical compositions containing them and their use |
| 10/28/2004 | WO2004092116A1 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof |
| 10/28/2004 | CA2521937A1 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof |
| 10/27/2004 | EP1470137A1 Edg receptor agonists |
| 10/27/2004 | CN1541211A Derivatives of N-(arylsulfonyl) beta-aminoacids comprising substituted aminomethyl group, prepn. method thereof and pharmaceutical compsns. contg same |
| 10/21/2004 | WO2004089885A1 Novel compounds |
| 10/21/2004 | WO2004089876A1 Biphenylcarboxylic amide derivatives as p38 kinease inhibitors |
| 10/21/2004 | US20040209846 Heterocyclic analgesic compounds and methods of use thereof |
| 10/14/2004 | WO2004087655A1 Novel diphenyl azetidinone with improved physiological characteristics, corresponding production method, medicaments containing said compound and use of the latter |
| 10/14/2004 | WO2004087650A2 Process and intermediates for the preparation of beta-amino acid amide dipeptidyl peptidase-iv inhibitors |
| 10/14/2004 | US20040202734 Method for preparing nicotianamine or nicotianamine-containing product |
| 10/14/2004 | CA2520689A1 Novel diphenyl azetidinone with improved physiological characteristics, corresponding production method, medicaments containing said compound and use of the latter |
| 10/13/2004 | EP1465891A2 Inhibitors of dipeptidyl peptidase iv |
| 10/13/2004 | EP1347987B1 Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents |
| 10/13/2004 | EP0999204B1 Novel compound having effect of promoting neuron differentiation |
| 10/13/2004 | EP0934928B1 Cyclic amine derivatives |
| 10/13/2004 | EP0736036B1 Kininogen inhibitors |
| 10/13/2004 | CN1170842C New amidinobenzylamine derivatives and their use as thrombin inhibitors |
| 10/07/2004 | WO2004033442A3 Novel taxanes and methods related to use and preparation thereof |
| 10/07/2004 | US20040199005 Method for producing (R) -3- [4- (trifluoromethyl) phenylamino] -pentanoic acid amide derivative |
| 10/07/2004 | US20040198700 Administering to a patient an azetidinone compound containing at least 3 phenyl rings fo rprevention of a vascular condition, diabetes, obesity, stroke, lowering a concentration of a sterol or stanol in plasma of a mammal, preventing demyelination or treating Alzheimer's disease |
| 10/05/2004 | US6800766 Catalyzing the decyclization of racemic and diastereomeric epoxides mixtures in the presence of a non-racemic, chiral catalyst; pharmaceutical synthesis |
| 10/05/2004 | CA2103837C Novel method of producing 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines |
| 09/30/2004 | WO2004083166A1 Processes for production of (r)-3-[4-(trifluoromethyl)- phenylamino]pentanamide derivatives |
| 09/30/2004 | WO2003051314A3 Antibiotic compounds |
| 09/30/2004 | US20040192742 Antiarthritic agents; muscular dystrophy; antiinflammatory agents; glomerulonephritis; malaria; oral diseases |
| 09/30/2004 | US20040192676 Ligands of melanocortin receptors and compositions and methods related thereto |
| 09/30/2004 | CA2515789A1 Method for producing(r)-3-[4-(trifluoromethyl)phenylamino]-pentanoic acid amide derivative |
| 09/29/2004 | EP1461315A2 Catalytic carbonylation of three and four membered heterocycles |
| 09/29/2004 | EP1012140B1 New amidino derivatives and their use as thrombin inhibitors |
| 09/28/2004 | US6797833 Taxane derivatives having a tricyclic or tetracyclic core; remarkable properties in vitro; valuable antileukemia, antitumor and anticarcinogenic agents; human cancer cell line comparable to that of taxol and taxotere |
| 09/28/2004 | CA2299013C Neuropeptide y antagonists |
| 09/23/2004 | WO2004081643A1 Lenslet array with polarization conversion |
| 09/23/2004 | WO2004081002A1 Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholesterolemia |
| 09/23/2004 | WO2004050613A3 2-substituted-3-propenamide derivatives and methods of using the same |
| 09/23/2004 | US20040186090 New amidino derivatives and their use as thrombin inhibitors |
| 09/23/2004 | US20040186088 Mercapto-cycloalkyl or heterocyclyl ring-sulfonyl-aryl or heteroaryl derivatives; preventing the cleavage Of tumor necrosis factor- alpha from cell membranes in mammal; treating autoimmune diseases, inflammation, inflammatory bowel disease, Crohn's disease, asthma, sepsis and septic shock |
| 09/22/2004 | EP1458413A2 Pharmaceutical compositions based on azetidine derivatives |
| 09/21/2004 | US6794523 Anticancer agents, antitumor agents; leukemia |
| 09/21/2004 | US6794359 Vertebrate intestinal protein which absorbs cholesterol, its inhibitors and mehtod of identifying the same |
| 09/16/2004 | WO2004058149A3 1-(amino)indanes and (1,2-dihydro-3-amino)-benzofurans, benzothiophenes and indoles |
| 09/15/2004 | EP1456393A1 Cyclisation process for the preparation of c-2 beta-lactam compounds |
| 09/15/2004 | EP1456171A1 Substituted cyclohexane derivatives |
| 09/15/2004 | EP0986384A4 Inhibitors of protein isoprenyl transferases |
| 09/10/2004 | WO2004007444A3 N-hydroxyamide derivatives possessing antibacterial activity |
| 09/09/2004 | DE10306250A1 Substituierte N-Arylheterozyklen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Substituted N-Arylheterozyklen, processes for their preparation and their use as medicaments |
| 09/08/2004 | EP1453501A1 N- aryl-n'-arylcycloalkyl-urea derivatives as mch antagonists for the treatment of obesity |
| 09/08/2004 | CN1527876A Compounds, compositions, and methods for controlling biofilms |
| 09/08/2004 | CN1527707A The use of substituted azetidinone compounds for the treatment of sitosterolemia |
| 09/07/2004 | US6787540 Compounds useful as reversible inhibitors of cysteine proteases |
| 09/02/2004 | US20040171849 Halogenation a 4-amino-2-hydroxybutyric acid ; cyclization; in aqueous solution |
| 08/26/2004 | WO2004072025A2 Substituted n-arylheterocycles, method for production and use thereof as medicaments |
| 08/26/2004 | WO2004071454A2 Substituted azetidine compounds as inhibitors of dipeptidyl peptidase iv |
| 08/26/2004 | US20040167115 induction apoptosis; Dna replication inhibition; p38 MAP kinase activation or caspase cascading activation, or cytochromic C release from mitochondria into cytoplasm |
| 08/26/2004 | CA2516118A1 Substituted n-arylheterocycles, method for production and use thereof as medicaments |
| 08/25/2004 | EP1448523A1 Heterocyclic compounds and methods of use |
| 08/25/2004 | EP1278728B1 Pyrrolidine and piperidine derivatives and their use for the treatment of neurodegenerative disorders |
| 08/24/2004 | US6780858 Hydroxyamidines and related compounds |
| 08/19/2004 | WO2004069793A2 Novel 2-substituted cyclic amines as calcium sensing receptor modulators |
| 08/12/2004 | US20040157823 Pharmaceutical compositions containing 3-aminoazetidine derivatives, novel derivatives and their preparation |
| 08/12/2004 | US20040157822 Azetidinyl diamines useful as ligands of the nociceptin receptor ORL-1 |
| 08/11/2004 | EP1444200A1 Azetidinyl diamines useful as ligands of the nociceptin receptor orl-1 |
| 08/11/2004 | EP1443922A1 Mch antagonists for the treatment of obesity |
| 08/11/2004 | EP1140918B1 Thrombin inhibitors |
| 08/04/2004 | EP1441728A2 Modulators of the cholesterol biosynthetic pathway |
| 08/04/2004 | EP0667772B9 Taxanes having an alkyl substituted side-chain and pharmaceutical compositions containing them |
| 08/04/2004 | CN1518534A Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds |
| 08/03/2004 | CA2136836C Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension |
| 07/29/2004 | US20040147502 Beta lactam compounds and their use as inhibitors of tryptase |
| 07/28/2004 | CN1516687A 3,4-di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands |
| 07/28/2004 | CN1515563A Aryl substituted piperazine for curing benign prostatauxe |
| 07/28/2004 | CN1515556A Intermediate compound for preparing aryl substituted piperazine |
| 07/27/2004 | CA2103861C Novel 7-(substituted)-8-(substituted-9-(substituted amino)-6-demethyl-6-deoxytetracyclines |
| 07/22/2004 | US20040142999 Novel compounds and compositions as cathepsin inhibitors |
| 07/22/2004 | US20040142986 Controlling transforming growth facor; artificial skin; wound healing agents |
| 07/15/2004 | WO2004058735A2 Ligands of melanocortin receptors and compositions and methods related thereto |
| 07/15/2004 | WO2004058149A2 1-(amino)indanes and (1,2-dihydro-3-amino)-benzofurans, benzothiophenes and indoles |
| 07/14/2004 | EP1436255A1 Novel compounds and compositions as cathepsin inhibitors |
| 07/14/2004 | EP1436009A1 Pharmaceutical formulation |
| 07/14/2004 | CN1512983A Compounds and compositions as cathepsins inhibitors |
| 07/13/2004 | US6762309 Antileukemia and antitumor agents |
| 07/13/2004 | US6762306 Chiral ligand |
| 07/08/2004 | WO2004056766A1 Inhibitors of tace |
| 07/08/2004 | US20040132991 Novel taxanes and methods related to use and preparation thereof |