Patents
Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868)
03/1998
03/26/1998CA2266639A1 3,4-disubstituted azetidin-2-one derivatives useful as cysteine proteinase regulators
03/24/1998USRE35754 Cephem derivatives
03/24/1998US5731431 Process for preparing 4-substituted azetidinone derivatives
03/24/1998US5731315 Inhibitors of factor xa
03/17/1998US5728850 Antitumor agents
03/17/1998US5728827 Intermediates in synthesis of penems and hypocholesterolemic agents
03/17/1998US5728725 C2 taxane derivaties and pharmaceutical compositions containing them
03/11/1998EP0827961A1 Process for the preparation of beta-lactam compounds
03/11/1998EP0827954A1 Process for producing optically active azetidine-2-carboxylic acid
03/11/1998EP0827496A1 Catalic enantioselective synthesis of a spiro-fused azetidinone
03/11/1998CN1175953A Novel dipeptide amidines as thrombin inhibitors
03/11/1998CN1037680C Novel method of producing 7 -(substd.) -9 -£(substd. glycyl) -amino| -6 -demethyl 6 -deoxytetra -cylines
03/10/1998US5726159 Peptide thrombin inhibitors
03/05/1998WO1998008811A1 Cyclic amine derivatives
03/04/1998CN1175246A Substituted azetidin-2-ones for treatment of atherosclerosis
03/03/1998US5723634 Metal alkoxide compounds
03/03/1998US5723627 Bactericides
03/03/1998US5723444 Enzyme inhibitors and anticoagulants
02/1998
02/26/1998WO1998007691A1 Process for stereoselective preparation of trans-azetidinones
02/26/1998WO1998007690A1 Process for stereoselective preparation of 4-acetoxyazetidinones
02/26/1998WO1998007420A1 Neuropeptide-y ligands
02/26/1998CA2268051A1 Neuropeptide-y ligands
02/25/1998CN1174548A Sulfur-substituted azetidinone compounds useful as hypocholesterolemic agents
02/24/1998US5721366 Phenylamidine derivatives
02/24/1998US5721360 Blocking the nitrogen of 3-phenylacetamido-4-acetoxyazetidin-2-one; cyclization; deblocking
02/24/1998US5721268 Anticarcinogenic agents
02/18/1998EP0823896A1 Substituted oximes, hydrazones and olefins as neurokinin antagonists
02/18/1998EP0823893A1 Novel tetracycline derivatives
02/17/1998US5719275 Reacting silyl enol ether with azetidinone derivative to form intermediate for penicillin-type antibiotic
02/17/1998US5719186 Central muscle relaxants, anxiolytic agents, antiinflammatory agents, analgesics, anticonvulsants
02/11/1998CN1173170A Matrix metalloprotease inhibitors
02/10/1998US5717115 Intermediates for taxane derivatives
02/03/1998US5714513 Antitumor and -carcinogenic agents; leukemia
01/1998
01/28/1998EP0619826B1 Azetidinol reaction products
01/28/1998CN1037177C Process for preparation of substituted propargyl azacyclic butanone
01/27/1998US5712388 Method of preparing a derivative of optically active azetidin-2-one
01/22/1998WO1998002568A1 The bioresolution of n-acylazetidine-2-carboxylic acids
01/22/1998WO1998002417A1 Process for the production of enantiomerically enriched n-acylazetidine-2-carboxylic acids
01/22/1998CA2259714A1 Process for the production of enantiomerically enriched n-acylazetidine-2-carboxylic acids
01/22/1998CA2259402A1 The bioresolution of n-acylazetidine-2-carboxylic acids
01/20/1998US5710287 Taxanes having an amino substituted side-chain and pharmaceutical compositions containing them
01/20/1998US5710146 Antibiotics for bactericides
01/20/1998US5710100 Safening imidazolinone herbicides
01/14/1998CN1036996C Preparation of £1R-oxo-3S-thiolanylthio (thiocarbonyl)-thio|-2-azetidinones
01/13/1998US5707966 Peptide derivatives
01/07/1998EP0816376A1 Trombin inhibitors as anticoagulant agents
01/06/1998US5705636 Chemical intermediate for preparation of antibacterial compounds
01/06/1998US5705508 Forming taxol derivatives
01/06/1998US5705487 Antithrombotic agents
12/1997
12/31/1997WO1997049404A1 Anticoagulant agents
12/31/1997CA2258915A1 Anticoagulant agents
12/30/1997US5703234 Chemical intermediate for 1-methylcarbapenem antibiotics
12/30/1997CA2134964C Bridged aza-bicyclic derivatives as substance p antagonists
12/23/1997US5700930 4-substituted azetidinones as precursors to 2-substituted-3-carboxy carbapenem antibiotics and a method of producing them
12/18/1997WO1997047621A1 Process for the preparation of carbapenem derivatives and intermediates thereof
12/18/1997WO1997047194A1 Substituted cyclopentane compounds useful as neuraminidase inhibitors
12/16/1997US5698548 Spirocycloalkyl-substituted azetidinones useful as hypocholesterolemic agents
12/11/1997WO1997046577A1 New amino acid derivatives and their use as thrombin inhibitors
12/11/1997CA2255625A1 New amino acid derivatives and their use as thrombin inhibitors
12/09/1997US5696267 Substituted oximes, hydrazones and olefins as neurokinin antagonists
12/09/1997US5696256 Process for preparing and using guanidine derivatives
12/04/1997WO1997045406A1 3-hydroxy gamma-lactone based enantioselective synthesis of azetidinones
12/04/1997WO1997045115A1 Pharmaceutical for treatment of neurological and neuropsychiatric disorders
12/04/1997CA2619901A1 Pharmaceutical for treatment of neurological and neuropsychiatric disorders
12/03/1997CN1166489A Prep. of novel alkyl-substituted alpha-ketone ester
12/02/1997US5693792 β-lactam and cephem compounds and processes for their production
11/1997
11/20/1997WO1997043255A1 Inhibitors of microsomal triglyceride transfer protein and method
11/18/1997US5688990 Forming chemical intermediates for azetidinone compounds that inhibit cholesterol biosynthesis for prevention of atherosclerosis
11/18/1997US5688942 Process for preparing 2-isocephem derivatives
11/18/1997US5688787 Substituted β-lactam compounds useful as hypochlesterolemic agents and processes for the preparation thereof
11/18/1997US5688785 Substituted azetidinone compounds useful as hypocholesterolemic agents
11/13/1997WO1997042170A1 A process for the preparation of azetidinones
11/12/1997EP0805795A1 Novel aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
11/12/1997CN1164531A Novel derivatives of 3-bromo-and 3,3-dibromo-4-oxo-1-azetidines, processes for preparation thereof and their use
11/11/1997US5686588 Amine acid salt compounds and process for the production thereof
11/06/1997WO1997041099A1 Azetidinone derivatives for the treatment of atherosclerosis
11/06/1997WO1997041098A1 Azetidinone derivatives for the treatment of atherosclerosis
11/06/1997WO1997041084A1 Improved process for the production of enantiomerically-pure azetidine-2-carboxylic acid
11/06/1997CA2252696A1 Azetidinone derivatives for the treatment of atherosclerosis
11/04/1997CA2126557C Azetidinol reaction products
10/1997
10/28/1997US5681951 Metal catalyzed displacement process
10/22/1997EP0630365B1 Method for preparing beta-phenylisoserine and analogues thereof
10/15/1997EP0594608B1 Chiral catalysts for enantioselective synthesis
10/15/1997CN1162312A Phenyloxazolidinone antimicrobials
10/14/1997US5677283 Antiinflammatory agents, nervous system disorders
10/09/1997WO1997036867A1 Benzyl(idene)-lactam derivatives, their preparation and their use as selective (ant)agonists of 5-ht1a- and/or 5-ht1d receptors
10/09/1997CA2249603A1 Benzyl(idene)-lactam derivatives, their preparation and their use as selective (ant)agonists of 5-ht1a- and/or 5-ht1d receptors
10/08/1997EP0799200A1 Substituted azetidin-2-ones for treatment of atherosclerosis
10/07/1997US5674976 Coupling first modular component to third modular component to yield precyclized gamma turn mimetic, cyclizing
10/01/1997EP0596015B1 Substituted beta-lactam compounds useful as hypocholesterolemic agents and processes for the preparation thereof
10/01/1997CN1036006C Antibiotic compound carbapenem
09/1997
09/30/1997US5672701 4-substituted alkyl carbapenem antibiotics
09/30/1997US5672681 Conformationally restricted mimetics of gamma turns and peptides containing the same
09/30/1997CA2020097C Azetidines, their preparation and their application as intermediates for the preparation of compounds with antimicrobial activity
09/23/1997US5670638 2-bromo- and 2-nitroxy derivatives of 3-bromo- and 3,3-dibromo-4-oxo-azetidines, and preparation
09/23/1997US5670155 Confomationally restricted mimetics of beta turns and beta bulges and peptides containing the same
09/18/1997WO1997033891A1 PROCESS FOR THE PREPARATION OF ss-LACTAM COMPOUNDS
09/10/1997EP0793643A1 Matrix metalloprotease inhibitors
09/09/1997CA1339450C Stable oxapenem-3-carboxylic acids
09/04/1997WO1997031922A1 Process for the preparation of 2-halomethyl-penems and their use for the preparation of antibacterial penems
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