| Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868) |
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| 09/27/2000 | EP0848703B1 Derivatives of benzosulphonamides as inhibitors of the enzyme cyclo-oxygenase ii |
| 09/26/2000 | US6124481 Ammonium alkoxides |
| 09/26/2000 | US6124474 Synthesis of chiral 2-azetidinemethanol compounds |
| 09/20/2000 | EP1036062A1 Hydroxamic acid derivatives as matrix metalloprotease (mmp) inhibitors |
| 09/19/2000 | US6121462 Complexing |
| 09/13/2000 | CN1266427A New amidino derivatives and their use as thrombin inhibitors |
| 09/06/2000 | EP1033366A2 Amide derivatives useful as Neuropeptide Y (NPY) antagonists |
| 09/05/2000 | US6114543 Process for producing optically active azetidine-2-carboxylic acid |
| 08/23/2000 | EP0805795B1 Novel aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides |
| 08/23/2000 | CN1264385A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same |
| 08/23/2000 | CN1264300A Arylsubstituted piperazines useful in the threatement of bening prostatic hyperlasia |
| 08/22/2000 | US6107329 Hypotensive agents; cardiovascular disorders |
| 08/16/2000 | EP1027332A1 Novel lactam metalloprotease inhibitors |
| 08/16/2000 | EP0690711B1 Taxanes having an amino substituted side-chain |
| 08/15/2000 | US6103911 By-product inhibition |
| 08/02/2000 | EP1023285A1 Azetidinylpropylpiperidine derivatives, intermediates and use as tachykinin antagonists |
| 08/02/2000 | EP1023265A1 Azetidinone derivatives for the treatment of hcmv infections |
| 08/02/2000 | EP0691953B1 1-amidinophenyl-pyrrolidones/ piperidinones as platelet aggregation inhibitors |
| 08/02/2000 | CN1261887A Azetidinyl propylpiperidine derivatives, intermediates and use as tachykinin antagonists |
| 08/01/2000 | US6096883 3-hydroxy gamma-lactone based enantioselective synthesis of azetidinones |
| 08/01/2000 | US6096712 Tripeptide derivative; antiallergens, male contraceptives, antiinflammatory agents, antispasmodics, hypertensive agents |
| 08/01/2000 | CA2015034C Piperazine derivatives |
| 07/26/2000 | EP1021405A1 Azetidinone derivatives for the treatment of hcmv infections |
| 07/26/2000 | EP1021404A1 Azetidinone derivatives for the treatment of hcmv infections |
| 07/26/2000 | EP0694032B1 Method for preparing beta-lactams |
| 07/26/2000 | CN1054842C 1-amidinophenyl-pyrrolidones piperidinones azetinones platelet aggregation inhibitors |
| 07/25/2000 | US6093812 Process for the stereospecific synthesis of azetidinones |
| 07/25/2000 | CA2197086C (azetidin-1-ylalkyl)lactams as tachykinin antagonists |
| 07/20/2000 | WO2000042059A1 New amidinobenzylamine derivatives and their use as thrombin inhibitors |
| 07/20/2000 | CA2355792A1 New amidinobenzylamine derivatives and their use as thrombin inhibitors |
| 07/19/2000 | EP1019406A1 Pyrrolopyrrolone derivatives as inhibitors of neutrophil elastase |
| 07/18/2000 | US6090786 Serine proteases, their activity and their synthetic inhibitors |
| 07/13/2000 | DE19900576A1 New substituted allyl-, glycidyl- or hydroxypropyl-benzene derivatives, used as intermediates for drugs, especially central nervous system drugs, particularly the antidepressants paroxetine and femoxetine |
| 07/12/2000 | EP0413762B1 Peptide analogs and their use as haptens to elicit catalytic antibodies |
| 07/11/2000 | US6087379 Cyclic amine derivatives |
| 07/11/2000 | US6087186 Synthetic library of random oligomers, each member comprising an oligomer linked to a microchip encoded with information identifying structure of oligomer; for drug screening |
| 07/06/2000 | WO2000039124A1 Thrombin inhibitors |
| 07/06/2000 | WO2000039073A1 Stereospecific ring opening of chiral azetidinium salts |
| 07/06/2000 | CA2355281A1 Thrombin inhibitors |
| 07/05/2000 | EP1014966A1 Pharmaceutical for treatment of neurological and neuropsychiatric disorders |
| 07/05/2000 | CN1258674A Pyrone carboxylic acid derivate or its salt and antibiotic with the same as effective component |
| 07/05/2000 | CN1258672A Amino-compound |
| 06/28/2000 | EP1012140A1 New amidino derivatives and their use as thrombin inhibitors |
| 06/28/2000 | EP1011663A1 BETA-LACTAM INHIBITORS OF CoA-IT |
| 06/27/2000 | US6080854 Process for synthesizing carbapenem intermediates |
| 06/27/2000 | US6080767 Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides |
| 06/27/2000 | US6080760 Treating benign prostatic hyperplasia; complement slower-acting therapeutics by providing acute relief; induce relaxation of the lower urinary tract to decrease difficulty in urination and sexual dysfunction |
| 06/22/2000 | WO2000035869A1 New amidino derivatives and their use as thrombin inhibitors |
| 06/22/2000 | WO2000035859A1 Substituted aryl and heteroaryl derivatives, their production and their use as medicines |
| 06/22/2000 | WO2000035442A1 Hydroxy diphenyl urea sulfonamides as il-8 receptor antagonists |
| 06/22/2000 | CA2355890A1 Hydroxy diphenyl urea sulfonamides as il-8 receptor antagonists |
| 06/22/2000 | CA2353151A1 Substituted aryl and heteroaryl derivatives, the preparation thereof and their use as medicaments |
| 06/15/2000 | WO2000034240A1 Process for the synthesis of azetidinones |
| 06/14/2000 | EP1007511A1 Preparation of beta-methyl carbapenem intermediates |
| 06/06/2000 | US6071915 Arylsubstituted piperazines useful in the treatment of benign prostatic hyperplasia |
| 06/06/2000 | US6071899 Azetidinone derivatives for the treatment of atherosclerosis |
| 05/31/2000 | EP1003511A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS |
| 05/30/2000 | US6069260 Stereospecific taxane derivative having metal salt of the hydroxy attached to the carbon at the 13 ring position; chemical intermediates for antitumor agents |
| 05/30/2000 | CA2024880C 10-(1-hydroxyethyl)-11-oxo-1-azatricyclo(7.2.0.0.3,8)undec-2-ene-2-2-ca rboxylic acid derivatives |
| 05/18/2000 | WO2000004892A3 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions |
| 05/17/2000 | EP1001036A2 Enzymatic processes for resolution of enantiomeric mixtures of compounds useful as intermediates in the preparation of taxanes |
| 05/17/2000 | EP1000016A1 Isocyanoalkyl carbonic acid derivatives, their conversion into secondary amidoalkyl carbonic acid derivatives by isocyanide-multicomponent reactions, as well as these secondary amidoalkyl carbonic acid derivatives. |
| 05/16/2000 | US6063935 Cultivating a bacteria of a bacillus genus capable of producing 3,3-dihydroxyazetidine or salt thereof to produce the 3,3-dihydroxyazetidine or salt in culture medium and collecting the product |
| 05/16/2000 | US6063918 Reacting a base with a 2-azetidinyl-3,4-dihalogeno-2-butenoic acid compound in an aqueous organic solvent to yield a cyclized isooxacephalosporin derivative; simplification |
| 05/10/2000 | EP0999204A1 Novel compound having effect of promoting neuron differentiation |
| 05/03/2000 | EP0996434A1 Kappa agonist anti-pruritic pharmaceutical formulations and method of treating pruritus therewith |
| 05/03/2000 | EP0736031B1 Improvements in or relating to chiral syntheses |
| 05/02/2000 | US6057336 Lactam metalloprotease inhibitors |
| 04/26/2000 | EP0973737A4 Efficient synthesis of a chiral mediator |
| 04/25/2000 | US6054594 Process for the production of enantiomerically enriched N-acylazetidine-2-carboxylic acids |
| 04/18/2000 | US6051724 An antileukemia and antitumor agents |
| 04/18/2000 | US6051716 Antimicrobial agents |
| 04/18/2000 | US6051568 Thrombin inhibitors, their preparation and use |
| 04/13/2000 | WO2000020623A1 Resolution of trans-2 -(alkoxycarbonylethyl) -lactams useful in the synthesis of 1- (4-fluorophenyl) -3(r) -[3(s) -hydroxy-3 -(4-fluorophenyl) -propyl)] -4(s) -(4-hydroxyphenyl) -2-azetidinone |
| 04/12/2000 | EP0992501A2 Pyridonecarboxylic acid derivatives as antibacterial agents |
| 04/12/2000 | EP0992491A1 Processes for producing azetidine-2-carboxylic acid and intermediates thereof |
| 04/12/2000 | EP0991654A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same |
| 04/11/2000 | US6048860 Kappa agonist anti-pruritic pharmaceutical formulations and method of treating pruritus therewith |
| 04/06/2000 | WO1999061013A3 COMPOUNDS HAVING IgE AFFECTING PROPERTIES |
| 04/05/2000 | CN1249743A Arylsulfonylamino hydroxamic acid derivs |
| 03/29/2000 | CN1050830C Hydroxy-substituted azetidinone compounds and its use in medicine |
| 03/28/2000 | US6043356 Process for preparing β-lactam compound |
| 03/28/2000 | US6043266 Microbiocides treating gram-positive bacteria infections and persons with aids |
| 03/23/2000 | WO2000015609A1 Azetidine derivatives, preparation and medicines containing them |
| 03/22/2000 | EP0986384A1 Inhibitors of protein isoprenyl transferases |
| 03/16/2000 | WO2000014063A1 Therapeutic compounds and methods |
| 03/16/2000 | CA2342858A1 Method of screening compounds useful in the treatment of a desease caused by or exacerbated by mpv |
| 03/15/2000 | EP0984778A1 Neuropeptide-y ligands |
| 03/15/2000 | EP0984777A1 Arylsubstituted piperazines useful in the treatement of benign prostatic hyperlasia |
| 03/14/2000 | US6037498 Chiral syntheses |
| 03/14/2000 | US6037472 For treating disease-states characterized by excessive activity of matrix metalloproteases such as rheumatoid arthritis, osteoarthritis, periodontal disease, aberrant angiogenesis, tumor invasion and metastasis |
| 03/09/2000 | WO2000012474A1 An efficient process for the preparation of a human leukocyte elastase inhibitor |
| 03/09/2000 | WO2000012473A1 PROCESS FOR THE PRODUCTION OF N-PROTECTED AZETIDINE-2-CARBOXYLIC ACIDS (AzeOHs) |
| 03/08/2000 | EP0982991A1 Beta lactams as antiproliferative agents |
| 03/07/2000 | US6034104 Anticoagulant agents |
| 03/07/2000 | US6034093 Anticoagulants |
| 02/29/2000 | US6031094 Beta-lactam substrates and uses thereof |
| 02/29/2000 | US6030972 2- or 5-aminomethyl,2- or 5-cyanopyrimidines as intermediates of anticoagulants in extracorporeal circulation (heart-lung machine, hemodialysis) |
| 02/24/2000 | WO2000009463A1 Stereoselective ring opening reactions |
| 02/24/2000 | CA2339618A1 Stereoselective ring opening reactions |