Patents
Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868)
02/2000
02/23/2000CN1245496A 3-pyridyl enantiomers and their use as analgesics
02/22/2000US6028205 Antileukemia and antitumor agents as cancer chemotherapeutic agents
02/15/2000US6025487 Reacting 2-(4-azetidin-2-one)-cyclohexanone derivatives with sterically hindered organic base in presence of lewis acid
02/09/2000EP0977733A1 Arylsulfonylamino hydroxamic acid derivatives
02/08/2000CA2127677C 2-bromo- and 2-nitroxy derivatives of 3-bromo- and 3.3-dibromo-4-oxo-azetidines, processes for the preparation thereof and use thereof
02/03/2000WO2000005204A1 MONOCYCLIC β-LACTAM COMPOUNDS AND CHYMASE INHIBITORS CONTAINING THE SAME
02/03/2000WO2000004892A2 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
02/03/2000CA2335062A1 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
02/02/2000CN1048982C Method for semi-synthesis of taxalkane derivative with metal alkane oxide and beta-lactum
02/01/2000US6020368 Microbiocides
01/2000
01/27/2000WO2000003982A1 Cyclisation process
01/26/2000EP0974670A2 Process for producing optically active N-substituted azetidine-2-carboxylic acid compound
01/26/2000EP0974582A1 Process for the preparation of 4-substituted azetidinone derivatives
01/26/2000EP0973737A1 Efficient synthesis of a chiral mediator
01/26/2000CN1048719C Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxytetracyclines, prepn. method, their compositions and use thereof
01/19/2000EP0971889A1 Process for synthesizing carbapenem intermediates
01/13/2000CA2276543A1 Method for manufacturing (3s,4r)-4-¬(r)-1'-formylethyl| azetidin-2-one derivatives
01/12/2000EP0970049A1 PROCESS FOR THE PRODUCTION OF ENANTIOMERICALLY ENRICHED $i(N)-ACYLAZETIDINE-2-CARBOXYLIC ACIDS
01/12/2000CN1048240C Process for preparing 7-substed-9-substed. amino-6-demethyl-6-deoxytetracyclines
01/11/2000US6013837 Aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
01/11/2000US6013791 Process for the preparation of 4-(formylthio)-azetidin-2-one derivatives and penem derivatives
01/06/2000WO2000000465A1 Hydrazine derivatives
01/06/2000CA2335245A1 Hydrazine derivatives
01/04/2000US6011151 Process for preparing β-lactam halide compound
01/04/2000US6011150 Synthetic intermediate of a 1 beta-methylcarbapenem derivative
01/04/2000US6011056 C9 taxane derivatives and pharmaceutical compositions containing them
12/1999
12/29/1999WO1999067230A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION
12/29/1999WO1999067215A1 Amidino and guanidino azetidinone tryptase inhibitors
12/29/1999CA2342778A1 Inhibitors of .alpha.4.beta.1 mediated cell adhesion
12/29/1999CA2336003A1 Amidino and guanidino azetidinone tryptase inhibitors
12/28/1999US6008367 Intermediate for synthesis of anticoagulant agents
12/28/1999US6008347 N-substituted 2-azetidinones
12/21/1999US6005138 Antileukemia and antitumor agents
12/21/1999US6004964 Administering amide or sulfonamide derivative; analgesics
12/21/1999US6004948 Derivatives of benzosulphonamides as inhibitors of the enzyme cyclooxygenase II
12/16/1999WO1999064395A1 Heterocyclic amide compounds as cell adhesion inhibitors
12/16/1999WO1999042435A3 Myxochelines
12/08/1999EP0659177B1 4-oxo-azetidine-2-sulphonic acid amides and their salts, process for their production and their use
12/07/1999US5998656 Anticancer, antitumor agents; leukemia
12/07/1999US5998612 Antibiotic synthesis
12/07/1999US5998436 Pyridonecarboxylic acid derivatives or their salts and antibacterial agent comprising the same as the active ingredient
12/07/1999US5998399 Hypotensive agents
12/02/1999WO1999061424A1 Conformationally constrained amino acid compounds having affinity for the alpha2delta subunit of a calcium channel
12/02/1999WO1999061020A1 BENZIMIDAZOLE ANALOGS AS DOWN-REGULATORS OF IgE
12/02/1999WO1999061019A1 BENZIMIDAZOLE DERIVATIVES AS MODULATORS OF IgE
12/02/1999WO1999061013A2 COMPOUNDS HAVING IgE AFFECTING PROPERTIES
12/02/1999CA2332999A1 Compounds having ige affecting properties
12/02/1999CA2332989A1 Benzimidazole derivatives as modulators of ige
12/02/1999CA2332985A1 Benzimidazole analogs as down-regulators of ige
12/01/1999EP0655056B1 Azacyclyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
11/1999
11/30/1999US5994576 Have utility as antileukemia and antitumor agents.
11/24/1999CN1236358A Substituted N-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides
11/23/1999US5990102 Substituted azetidin-2-ones for treatment of atherosclerosis
11/17/1999EP0957090A1 Method for producing 3,3,4,4-tetramethyl-2-azetidinone
11/17/1999EP0957089A1 Method for racemization of optically active azetidine-2-carboxylate
11/17/1999CN1235596A Cyclic amine derivatives
11/16/1999US5986091 Process for preparation of β-lactam compounds
11/09/1999CA2106452C Amidinophenol derivatives
10/1999
10/28/1999WO1999054321A1 Substituted diamines and their use as cell adhesion inhibitors
10/27/1999EP0952151A2 Intermediates for use in preparing novel pyridonecarboxylic acid derivatives or their salts
10/21/1999WO1999052908A1 Titanium catalyzed preparation of carbapenem intermediates
10/21/1999CA2328219A1 Titanium catalyzed preparation of carbapenem intermediates
10/20/1999EP0950057A1 3-pyridyl enantiomers and their use as analgesics
10/20/1999EP0950046A1 3,4-disubstituted azetidin-2-one derivatives useful as cysteine proteinase regulators
10/20/1999CN1232035A Preparation of beta-methyl carbapenem intermediates
10/19/1999US5968962 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/19/1999US5968923 (Azetidin-1-ylalkyl) lactams as tachykinin antagonists
10/13/1999EP0540609B1 Cephalosporins and homologues, preparations and pharmaceutical compositions
10/06/1999EP0623622B1 Process for producing cephem compound
10/06/1999CN1045444C Preparation of beta-lactam compounds and intermediates therefor
10/05/1999CA2158147C Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment
09/1999
09/29/1999EP0944594A1 Inhibitors of the enzymatic activity of psa
09/29/1999CN1045296C Process for preparing crystalline beta-lactam monohydrate
09/28/1999US5959123 Reacating substituted amino acid with 3-amino-4-substituted-azetidine-2-one compound to form 3, 4-disubstituted-azetidine-2-one compound; useful for treating muscular dystrophy, arthritis, viral and parasitic infections
09/28/1999US5958918 Substituted (sulfinic acid, sulfonic acid, sulfonylamino or sulfinylamino) N- (aminominomethyl)phenylalkyl!-azaheterocyclylamide compounds
09/22/1999EP0943609A1 Azetidine derivative, bifidobacterium division-promoting composition containing the same, and a process for production thereof
09/22/1999CN1229076A Trimethlene imidic derivant and composition for promoting two-tailed bacterium division using the derivant as active principle and making method thereof
09/21/1999US5955606 Photoresists of polyvinyllactams
09/15/1999CN1228430A 1-isothiazolidinone derivatives of azetidine-2-one, processes for preparation thereof and use thereof
09/14/1999US5952321 Substituted azetidinones as anti-inflammatory and antidegenerative agents
09/14/1999CA2098478C Preparation of substituted isoserine esters using metal alkoxides and .beta.-lactams
09/09/1999DE19807475A1 New myxocheline derivatives useful e.g. for treating disorders associated with deficient metal ion metabolism, especially iron or aluminium metabolism, e.g. hemosiderosis, thalassemia or Alzheimer's disease
09/07/1999CA1340721C 1,4-dihydro-quinoline-and naphthyridine-3-carboxylic acid antibacterial agents
09/02/1999WO1999043648A1 Cyclic amino compounds
09/02/1999WO1999043647A1 Derivatives of azetidine and pyrrolidine
09/01/1999CN1227466A Substituted cyclopentane compounds useful as neuraminidase inhibitors
08/1999
08/26/1999WO1999042435A2 Myxochelines
08/25/1999EP0937725A2 Method for removing the protecting group for hydroxy group
08/25/1999EP0751934B1 Substituted azetidinone compounds useful as hypocholesterolemic agents
08/25/1999CN1226895A Amino acid derivatives and their use as thrombin inhibitors
08/24/1999US5942630 Process for the production of enantiomerically-pure azetidine-2-carboxylic acid
08/18/1999CN1044702C Ozonide reducing method
08/17/1999US5939561 Process for the preparation of β-phenylisoserine and β-lactam and their analogues
08/17/1999US5939392 Thrombin inhibitors, anticoagulants and antiinflammatory agents
08/11/1999EP0934928A1 Cyclic amine derivatives
08/11/1999EP0933993A1 Substituted cyclopentane compounds useful as neuraminidase inhibitors
08/10/1999US5936088 Nervous system disorders
08/04/1999EP0933360A1 Synthesis of new beta-lactams
07/1999
07/29/1999WO1999037614A1 Azetidinecarboxamide derivatives for the treatment of cns disorders
07/29/1999WO1999037613A1 Azetidinecarboxamide derivatives for treating cns disorders
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