| Patents for C07D 205 - Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom (6,868) |
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| 07/08/2004 | US20040132809 Cell adhesion inhibitors |
| 07/08/2004 | US20040132713 Fluorinated cyclic amides as dipeptidyl peptidase IV inhibitors |
| 07/06/2004 | US6759554 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds |
| 07/01/2004 | DE10257785A1 Isophthalsäurederivate Isophthalic acid derivatives |
| 06/29/2004 | US6756372 For therapy of autoimmune diseases, alzheimer's disease, atherosclerosis, osteoporosis, rheumatoid arthritis, systemic lupus erythematosus, crohn's disease, ulcerative colitis, multiple sclerosis, guillain-barre syndrome, psoriasis |
| 06/24/2004 | WO2004052839A1 Isophtalic acid derivatives |
| 06/24/2004 | US20040122050 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors |
| 06/24/2004 | US20040122017 Melanin concentrating hormone (MCH) modulators; metabolic and eating disorders |
| 06/23/2004 | EP1429756A2 Treatment of xanthoma with azetidinone derivatives as sterol absorption inhibitors |
| 06/23/2004 | CN1507443A Method for producing 2-azetidinone derivative |
| 06/17/2004 | WO2004050613A2 2-substituted-3-propenamide derivatives and methods of using the same |
| 06/17/2004 | WO2004018414A3 Antibacterial agents |
| 06/17/2004 | US20040116518 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
| 06/17/2004 | US20040116353 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same |
| 06/16/2004 | EP1427409A1 Methods for treating or preventing vascular inflammation using sterol absorption inhibitor(s) |
| 06/15/2004 | US6750243 COMPETITIVE INHIBITORS OF TRYPSIN-LIKE SERINE PROTEASES, ESPECIALLY THROMBIN; chemical synthesis; anticoagulants; treatment of thrombosis |
| 06/15/2004 | US6750213 Bone disorders; urogenital system disorders; anticancer agents |
| 06/10/2004 | WO2004048326A1 Therapeutic agent for respiratory disease containing 4-hydroxypiperidine derivative as active ingredient |
| 06/10/2004 | US20040110965 Chiral ligand |
| 06/10/2004 | US20040110736 Cyclic derivatives as modulators of chemokine receptor activity |
| 06/10/2004 | CA2507509A1 Therapeutic agent for respiratory disease containing 4-hydroxypiperidine derivative as active ingredient |
| 06/09/2004 | EP1425407A2 Enzymatic resolution of t-butyl taxane derivatives |
| 06/09/2004 | CN1152859C Novel N-vinyllactam derivatives and polymer thereof |
| 06/08/2004 | US6747161 Process for cyclizing optically active 4-amino-2-halogenobutyric acids |
| 06/08/2004 | CA2079692C Novel 7-substituted-9-substituted amino-6-demethyl-6-deoxytetracyclines |
| 06/03/2004 | US20040106790 Novel compounds and method for preparing 3-methylcephams |
| 06/03/2004 | US20040106788 asymmetric hydrogenation of a lactam-enamide; multi-step synthesis |
| 06/03/2004 | US20040106593 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same |
| 06/02/2004 | EP1423362A1 New mandelic acid derivatives and their use as thrombin inhibitors |
| 05/27/2004 | WO2004043973A1 Novel intermediate for carbapenem compound for oral administration and process for producing the same |
| 05/27/2004 | WO2004043940A1 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes |
| 05/27/2004 | WO2004043939A1 Amide compounds and methods of using the same |
| 05/26/2004 | EP1421063A1 Disulfide and thiosulfonate ligands and libraries comprising these ligands |
| 05/26/2004 | EP1027332B1 Novel lactam metalloprotease inhibitors |
| 05/25/2004 | CA2048172C Substituted sulfonamids, preparation processes and drugs containing same |
| 05/21/2004 | WO2004042351A2 Piperidinyl-alpha-aminoamide modulators of chemokine receptor activity |
| 05/21/2004 | WO2004041795A1 Novel inhibitors of dipeptidyl peptidase iv |
| 05/21/2004 | CA2503844A1 Piperidinyl-alpha-aminoamide modulators of chemokine receptor activity |
| 05/20/2004 | US20040097482 Combinations of nicotinic acid and derivatives thereof and sterol absorption inhibitor(s) and treatments for vascular indications |
| 05/12/2004 | EP1417190A1 Substituted piperazines as modulators of the melanocortin receptor |
| 05/12/2004 | CN1149210C Thrombin inhibitors |
| 05/12/2004 | CN1149191C Azetidine derivatives, Preparation and medicines containing them |
| 05/12/2004 | CN1149081C Arylsubstituted piperazines useful in the threatement of bening prostatic hyperlasia |
| 05/11/2004 | US6734311 Substituted amidine derivatives as inhibitors of cell adhesion |
| 05/11/2004 | US6734176 Pharmaceutical compositions containing 3-aminoazetidine derivatives, novel derivatives and their preparation |
| 05/06/2004 | US20040087647 Enzyme inhibitors; prevent thrombosis; anticoagulants |
| 05/06/2004 | US20040087569 N-heterocyclic bicyclic lactone compounds |
| 05/06/2004 | EP1415985A1 Process for producing optically active azetidine-2-carboxylic acid |
| 05/05/2004 | CN1148346C Hydrazine derivs. |
| 05/04/2004 | US6730782 Carbamoyl substituted β-lactams |
| 04/29/2004 | WO2004035540A1 Malonic acid monoesters and process for producing the same |
| 04/29/2004 | WO2004035539A1 Process for producing carbapenem derivative and intermediate for use in the production |
| 04/29/2004 | WO2004035538A1 Process for making azetidine-3-carboxylic acid |
| 04/29/2004 | US20040082786 Piperazine based inhibitors of factor xa |
| 04/29/2004 | US20040082561 Antilipemic agents; anticholesterol agents |
| 04/28/2004 | CN1147504C New thrombin inhibitors, their preparation and use |
| 04/22/2004 | WO2004033442A2 Novel taxanes and methods related to use and preparation thereof |
| 04/22/2004 | WO2003101958A3 Flourinated cyclic amides as dipeptidyl peptidase iv inhibitors |
| 04/22/2004 | US20040077706 Piperidine and azepine derivatives; anxiolytic, analgesic, antidepressant, antiemetic, antiinflammatory, and hypotensive agents; sexual and psychological disorders; Alzheimer*s, Parkinson*s, Lesche-Nyhane, Wilson*s, and Tourette*s syndrome |
| 04/22/2004 | US20040077623 Antilepemic agents; low intestinal absorption; side effect reduction; modulating serum cholesterol concentration; preventing and treating arteriosclerotic conditions |
| 04/21/2004 | EP1049671B1 Azetidinecarboxamide derivatives for the treatment of cns disorders |
| 04/15/2004 | WO2004031137A1 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors |
| 04/15/2004 | WO2002050090A8 Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents |
| 04/15/2004 | US20040073048 Antitumor agents; anticancer agents; leukemia therapy; using metal alkoxide |
| 04/15/2004 | US20040073047 Preparation of substituted isoserine esters using beta-lactams and metal or ammonium alkoxides |
| 04/15/2004 | US20040072854 Antiemetics; psychlogical disorders; antidepressants; anxiolytic agents; antitussive agents |
| 04/15/2004 | US20040072309 Method for producing 2-azetidinone derivative |
| 04/13/2004 | US6720319 Compounds useful as reversible inhibitors of cysteine proteases |
| 04/08/2004 | US20040067913 Acid-group-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use |
| 04/07/2004 | CN1487919A New mandelic acid derivatives and their use as throbin inhibitors |
| 04/06/2004 | US6716861 Heterocyclic 1,2,4-oxadiazole or oxazole ring containing propanohydroxamic acids useful as antiscarring agent |
| 04/01/2004 | WO2004026824A1 Process for preparing intermediates |
| 04/01/2004 | WO2003075853A3 Cyclic derivatives as modulators of chemokine receptor activity |
| 04/01/2004 | CA2499426A1 Process for preparing n-hydroxylamine compounds |
| 03/25/2004 | WO2004024702A1 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof |
| 03/25/2004 | CA2496563A1 New carboxamide compounds having mch-antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture |
| 03/24/2004 | EP1214296B1 Substituted n-phenyl 2-hydroxy-2-methyl-3,3,3-trifluoropropanamide derivatives which elevate pyruvate dehydrogenase activity |
| 03/24/2004 | EP1161232B1 Hydroxy diphenyl urea sulfonamides as il-8 receptor antagonists |
| 03/24/2004 | CN1142908C Process for chloridizing dithio-aza cyclo-butanone derivatives |
| 03/23/2004 | US6710040 Fluorinated cyclic amides as dipeptidyl peptidase IV inhibitors |
| 03/18/2004 | US20040053953 Treatment of chemokine mediated diseases |
| 03/17/2004 | EP1398028A2 Taxanes having alkoxy, alkenoxy or aryloxy substituted side-chain and pharmaceutical compositions containing same |
| 03/17/2004 | EP1397340A2 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors |
| 03/17/2004 | EP1140820B1 New amidino derivatives and their use as thrombin inhibitors |
| 03/17/2004 | EP1140802B1 Substituted aryl and heteroaryl derivatives, their production and their use as medicines |
| 03/17/2004 | CN1483039A Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents |
| 03/17/2004 | CN1483021A Novel 1, 2-diphenzylazetidinones, method for producing the same, medicaments containing said compounds, and the use thereof for treating disorders of the lipid metabolism |
| 03/16/2004 | US6706712 Cyclic derivatives as modulators of chemokine receptor activity |
| 03/11/2004 | DE10238865A1 New carboxamides are melanin-concentrating hormone receptor antagonists, useful for treating e.g. metabolic diseases, diabetes, eating disorders, cardiovascular disease, emotional disorders, reproductive and memory disorders |
| 03/10/2004 | CN1481381A Diphenyl azetidinone derivatives, method for prodn. thereof medicaments contg. these compounds, and their use |
| 03/10/2004 | CN1481378A Diphenyl azetidinone derivatives, method for prodn. thereof, medicaments contg. these compounds, and their use |
| 03/09/2004 | US6703386 Treating hyperlipidemia, arteriosclerosis and hypercholesterolemia; derivatives of ezetimibe that are absorbed to a very low extent and so have a side effect reduction |
| 03/09/2004 | US6702705 Prodrugs activated by targeted catalytic proteins |
| 03/04/2004 | WO2004018414A2 Antibacterial agents |
| 03/04/2004 | US20040044233 Nucleophilic kinetic resolution of cyclic substrates using silyl azides |
| 03/03/2004 | EP1392287A2 Use of azetidinone substituted derivatives in the treatment of alzheimer's disease |
| 02/26/2004 | WO2003057144A3 Change inhibitors of dipeptidyl peptidase iv |
| 02/26/2004 | US20040039053 Administering to a patient a (3-halomethylphenoxy) (4-halophenyl) acetic acid derivatives or salt, free of its (+) stereoisomer to treat the type II diabetes, gout, insulin resistance and atherosclerosis |
| 02/25/2004 | EP1390340A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds |
| 02/25/2004 | CN1478094A Process and ester derivatives for preparing cephalosporins |