Patents
Patents for C07D 499 - Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula: , e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (3,448)
01/2002
01/03/2002US20020001616 Novel method of treatment
01/02/2002EP1165049A2 Agglomerates by crystallisation
12/2001
12/27/2001WO2001098518A2 Biotransformation of biologically active compounds made of various classes of chemical substances by means of laccase and manganese peroxidase enzymes
12/27/2001CA2413554A1 Biotransformation of biologically active compounds made of various classes of chemical substances by means of laccase and manganese peroxidase enzymes
12/19/2001EP1086109A4 Process for preparing crystalline salts of amoxycillin
12/19/2001CN1326935A Synthesis of cynnematin
12/18/2001CA2078684C Process for preparing penem esters
12/06/2001WO2001092268A1 Process for drying amoxicillin
12/05/2001EP1158995A1 Biologically active compounds of ganoderma pfeifferi dms 13239
12/05/2001CN1324795A Triphase one-step extraction process to purify penicillin
12/05/2001CN1324683A Serial self-suction type multi-channel phase dispersing extractor
11/2001
11/22/2001WO2001087299A1 Aralkyl ester soft drugs
11/22/2001CA2407099A1 Aralkyl ester soft drugs
11/21/2001CN1075064C New benzoxazinedione derivatives, and producing process thereof and use
11/15/2001WO2001085664A2 Compounds and methods for regulating bacterial growth and pathogenesis
11/01/2001US20010036930 Therapeutic azide compounds
10/2001
10/31/2001EP1149107A1 Process of preparing esters of penicillanic acid sulfoxide
10/25/2001WO2001079210A2 A process for the preparation of highly crystalline sodium cefoperazone
10/25/2001WO2000061541A8 Pharmaceutical compounds
10/17/2001EP1144418A1 3,6-disubstituted penam sulfone derivatives as antibacterials
10/17/2001EP1143991A2 Inhibitors of h+k+ -atpase
10/16/2001CA2089366C Penem compounds
10/04/2001EP1138333A1 Medicinal compositions for oral use
09/2001
09/27/2001WO2000061541A3 Pharmaceutical compounds
09/27/2001WO2000061537A3 Pharmaceutical compounds
09/25/2001US6294199 The dosage is provided by a bilayer tablet.
09/18/2001US6290948 Using certain chemokines or biologically active fragments thereof alone or in conjunction with an anti-infective agent or hematopoietic maturing agent.
09/13/2001US20010021706 Administering a beta-lactam antibiotic with a beta-lactamase inhibiting compound such as benzhydryl 2-beta-(chloroacetoxy-methyl)-6-((z)-(tert-butoxycarbonyl)methylene) penicillinate to treat beta-lactam resistant bacterial infections
09/11/2001US6288234 Fluorinated heterocyclic amido amine compounds as drugs
08/2001
08/22/2001EP1124528A1 Multivalent macrolide antibiotics
08/22/2001EP0907633B1 New synthetic catechol derivatives, method for production and use thereof
08/14/2001US6274730 Reacting with nitrous acid in a water slurry under acid conditions
08/08/2001CN1306962A Method for preparing sodium amoxicillin
08/07/2001US6271222 Antibiotic
08/07/2001US6271212 Mixture with carrier
08/02/2001WO2001054691A1 Nitrate salts of antimicrobial agents
08/02/2001CA2397754A1 Nitrate salts of antimicrobial agents
07/2001
07/25/2001CN1305375A Antibacterial agents
07/18/2001CN1304412A Process for preparing crystalline salts of amoxycillin
07/11/2001EP0660837B1 Penem derivatives, their preparation and pharmaceutical compositions containing them
07/05/2001US20010006962 Behavior of biologically active compounds favorably modified by replacing a functional group with an unsaturated fatty derivative, e.g. elaidic acid; bioavailability; membrane passage; organ targeting; drugs; agriculture
07/03/2001US6255479 Process for the preparation of α-oxolactams
06/2001
06/28/2001WO1999063937A9 Multivalent macrolide antibiotics
06/13/2001CN1067078C 2-beta-alkenyl penam sulfones, prepn. method and use thereof
06/12/2001US6245811 Fatty acid esters as bioactive compounds
06/07/2001WO1999063940A3 INHIBITORS OF H+K+-ATPase
06/06/2001CN1298408A A method for crystallizing a beta-lactam antibiotic
06/06/2001CN1298407A Preparation of beta-Lactam antibiotics in the presence of urea or amide
05/2001
05/29/2001CA2086250C Process for preparation of beta-lactams
05/15/2001US6232305 Substituted amino bicyclic-β-lactam penam and cepham derivatives as cysteine protease inhibitors
05/15/2001CA2196539C Process for making quinolonyl lactam antimicrobials and novel intermediate compounds
05/09/2001EP0693057B1 Process for the preparation of 4-(formylthio)-azetidin-2-one derivatives and penem derivatives
05/08/2001CA2045253C Dicarboximides
05/03/2001WO2001030783A1 PROCESS FOR THE PREPARATION OF A β-LACTAM ANTIBIOTIC
04/2001
04/19/2001WO2001026691A1 Medicinal compositions for oral use
04/19/2001CA2354558A1 Oral pharmaceutical composition
04/17/2001US6218138 Reacting amino-beta-lactam component and corresponding amino-group containing acylating side chain component in presence of biocatalystto form antibiotic, solubilizing by adding acid which deactivates enzyme; enzyme is reusedenzyme
04/04/2001CN1289766A Penicillene compounds and derivatives therefrom
03/2001
03/28/2001EP1086109A1 Process for preparing crystalline salts of amoxycillin
03/28/2001EP1085893A1 Phosphodiesterase-v modulator drugs and their uses
03/28/2001EP1085891A1 Multibinding inhibitors of topoisomerase
03/28/2001EP1085861A1 Inhibitors of nitric oxide synthase
03/28/2001EP1085846A2 Multibinding inhibitors of microsomal triglyceride transferase protein
03/21/2001EP1083920A1 Novel antibacterial compounds
03/21/2001EP1083919A1 Novel antiviral compounds
03/14/2001EP1082325A1 Naphthosulfamylmethyl penem antibacterials
03/08/2001WO1999064047A8 Novel antiviral compounds
03/06/2001US6197185 Process for preparing beta lactam compound
03/01/2001WO2000061115A3 Pharmaceutical formulation comprising amoxycillin
02/2001
02/22/2001WO2001012584A2 Pharmaceutical compounds
02/22/2001CA2698353A1 Pharmaceutical compounds
02/22/2001CA2381409A1 Nitric ester derivatives
02/21/2001CN1284959A Process for purifying solution of ampicillin pro-drug ester
02/21/2001CN1062272C Silylation process
02/14/2001EP1075479A1 A method for crystallizing a beta-lactam antibiotic
02/13/2001CA2001203C Novel antimicrobial dithiocarbamoyl quinolones
02/08/2001WO2001009135A1 Process for the preparation of basic antibiotic-inorganic acid addition salts and intermediate oxalates
02/07/2001EP1073663A1 Preparation of beta-lactam antibiotics in the presence of urea or amide
01/2001
01/31/2001EP1072267A1 Antibacterial agents
01/24/2001CN1280982A Preparation method of penicillin and cephalosporin
01/18/2001WO1999064049A9 Novel antibacterial agents
01/10/2001CN1279685A Process for recovery of beta-lactam antibiotic
01/10/2001CN1279684A Process for recovery of beta-lactam antibiotic
01/09/2001US6172221 Clavulanic acid extraction process
12/2000
12/28/2000DE19911680A1 New extracts and compounds from Ganoderma pfeifferi , useful e.g. as antibacterial and antiviral agents, preservatives, cosmetic, pharmaceutical and food additives and in fish farming, are protease inhibitors
12/26/2000US6165708 Electrochemiluminescent monitoring of compounds
12/19/2000CA2001225C Antimicrobial lactam-quinolones
12/12/2000US6160112 Inhibitors of beta-lactamase
12/05/2000US6156745 2β-substituted-6-alkylidene penicillanic acid derivatives as β-lactamase inhibitors
12/05/2000US6156534 Producing antibiotic cefprozil, cefadroxil or amoxicillin by reacting penicillin or cephalosporin derivitive with 4-hydroxy-d-phenylglycyl ester in presence of penicillin g amidase
11/2000
11/28/2000US6153747 Process for the preparation of 2-halomethyl-penems and their use for the preparation of antibacterial penems
11/28/2000CA2016500C Process for producing beta-lactamase inhibitor
11/08/2000EP1049702A1 Process for purifying a solution of an ampicillin pro-drug ester
11/02/2000WO2000041478A3 Agglomerates by crystallisation
10/2000
10/19/2000WO2000061549A2 Pharmaceutical compounds
10/19/2000WO2000061541A2 Pharmaceutical compounds
10/19/2000WO2000061537A2 Pharmaceutical compounds
10/19/2000WO2000061115A2 Pharmaceutical formulation comprising amoxycillin
10/19/2000CA2370425A1 Pharmaceutical compounds
10/19/2000CA2370406A1 Pharmaceutical compounds
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