| Patents for C07D 499 - Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula: , e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (3,448) |
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| 06/03/2004 | CA2503316A1 Method and compositions for temporarily incapacitating subjects |
| 06/03/2004 | CA2503312A1 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs |
| 06/02/2004 | CN1500788A Method for extracting penicillin using membrane separation |
| 05/20/2004 | US20040097402 Therapy for infections; bactericides; synergistic mixtures |
| 05/13/2004 | WO2004039776A2 A process for the preparation of benzyl 2-oxo-4- (heteroaryl) dithio-alpha-isoprenyl-1- azetidineazetate derivatives |
| 05/06/2004 | WO2004037163A2 STERICALLY-AWKWARD β-LACTAMASE INHIBITORS |
| 04/27/2004 | US6726911 Biologically active compounds of Ganoderma pfeifferi DSM 13239 |
| 04/22/2004 | US20040077622 penicillins and oxapenicillins with a fused bicyclic N-heteroarymethylene group; 6-[(5-benzyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)methylene]-7-oxo-4-thia-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid; antibiotic resistance is reduced when administered alone or with other B-lactam antibiotics |
| 04/22/2004 | US20040077035 Mutated penicillin expandase and process for preparing 7-ADCA using the same |
| 04/22/2004 | US20040077034 Mutated penicillin expandase and process for preparing 7-ADCA using the same |
| 04/20/2004 | CA2282461C 2-.beta.-substituted-6-alkylidene penicillanic acid derivatives as .beta.-lactamase inhibitors |
| 04/15/2004 | WO2004031196A1 Processes for preparation of organic compounds |
| 04/14/2004 | EP1406619A1 Antiviral and antimicrobial guanidine or biguanidine derivatives |
| 04/14/2004 | CN1145629C Synthesis of cynnematin |
| 04/14/2004 | CN1145628C Synthesis of cynnematin |
| 04/08/2004 | US20040067925 Multilayer tablet containing amyoxycillin, or sodium salt thereof |
| 04/07/2004 | EP0946525B1 Method for producing metal complex carboxylic acid amides |
| 04/01/2004 | US20040063677 Omega monounsaturated fatty acid derivativatized biologically active materials; drug delivery; drug resistance; bioavail-ability |
| 03/31/2004 | CN1143851C Penicillene compounds and derivatives therefrom |
| 03/18/2004 | US20040053913 Process for preparing 6-alkylidene penem derivatives |
| 03/17/2004 | EP0804441B1 Clavulanic acid extraction process |
| 03/16/2004 | US6706878 Spiroazabicyclic heterocyclic compounds |
| 03/09/2004 | US6703502 Spiroazo bicyclic heterocyclic |
| 03/04/2004 | WO2004018484A1 Beta-lactamase inhibitor prodrug |
| 03/04/2004 | CA2494953A1 Beta-lactamase inhibitor prodrug |
| 03/02/2004 | US6699989 Antiviral and antimicrobial guanidine or biguanidine derivatives |
| 03/02/2004 | US6699699 Having a better substrate specificity to penicillin g, wherein the mutated penicillin expandase comprises an amino acid substitution at one or more residual positions corresponding to those of a wild-type |
| 02/25/2004 | EP1165049B1 Agglomerates by crystallisation |
| 02/25/2004 | EP1138333B1 Medicinal compositions for oral use |
| 02/19/2004 | US20040033969 Such as penicillin G coupled to 2'deoxyazithromycin; drug delivery |
| 02/12/2004 | US20040030127 Process for the preparation of highly crystalline sodium cefoperazone |
| 02/05/2004 | US20040023290 Novel therapeutic agents that modulate enzymatic processes |
| 01/07/2004 | CN1133428C Antibacterial composition for topical administration containing antibiotics |
| 01/02/2004 | EP1375492A1 Process for producing (dioxolenon-4-yl)methyl ester derivative |
| 01/01/2004 | US20040002600 Antibiotics |
| 12/31/2003 | WO2004000848A1 Process for the conversion of penam ring system to cepham ring system |
| 12/31/2003 | CN1132652C Serial self-suction type multi-channel phase dispersing extractor |
| 12/25/2003 | US20030236243 Sterically-awkward beta-lactamase inhibitors |
| 12/18/2003 | WO2003104241A1 Process for preparation of penam derivatives from cepham derivatives |
| 12/18/2003 | US20030232983 Process for preparation of penam derivatives from cepham derivatives |
| 12/17/2003 | EP1370296A2 Catecholate beta-lactam conjugates, method for producing the same and the use thereof |
| 12/17/2003 | EP0999213B1 Process for producing exo-methylenepenam compounds |
| 12/09/2003 | US6660855 Crystal of diphenylmethyl 2-methyl-2-triazolylmethylpenam-3-carboxylate; given X-ray powder diffraction pattern; storage stability |
| 12/09/2003 | US6660299 Treating a bacterial infection in a human by administering a specified high dosage of amoxycillin over given time |
| 11/20/2003 | WO2001085664A8 Compounds and methods for regulating bacterial growth and pathogenesis |
| 11/20/2003 | US20030216372 Inhibitors of serine and metallo-beta-lactamases |
| 11/13/2003 | WO2003093279A1 BICYCLIC 6-ALKYLIDENE-PENEMS AS ß-LACTAMASES INHIBITORS |
| 11/13/2003 | WO2003093277A1 Process for preparing 6-alkylidene penem derivatives |
| 11/13/2003 | WO2003092851A1 Preparation of small crystals |
| 11/13/2003 | WO2002055486A3 Triazene compounds and use thereof |
| 11/13/2003 | CA2483538A1 Bicyclic 6-alkylidene-penems as .szlig.-lactamases inhibitors |
| 11/13/2003 | CA2483533A1 Process for preparing 6-alkylidene penem derivatives |
| 11/04/2003 | US6642377 Process for the preparation of basic antibiotic-inorganic acid addition salts and intermediate oxalates |
| 10/29/2003 | CN1125825C Process for producing halogenated beta lactam compound |
| 10/23/2003 | WO2003087105A1 INHIBITORS OF SERINE AND METALLO-ß-LACTAMASES |
| 10/15/2003 | CN1124277C Preparation method of penicillin and cephalosporin |
| 10/09/2003 | US20030190695 Mutated penicillin expandase and process for preparing 7-ADCA using the same |
| 10/08/2003 | CN1446908A Method of using saltative ring enlargement enzyme to prepare 7-amino-desacetoxy cephalosporin acid |
| 10/02/2003 | WO2003080543A1 Process for producing cyclic compound |
| 10/02/2003 | US20030186956 Using inert gas; controlling humidity |
| 10/02/2003 | US20030186354 Mutated penicillin expandase and process for preparing 7- ADCA using the same |
| 10/01/2003 | EP1348759A1 Mutated penicillin expandase and process for preparing 7-ADCA using the same |
| 09/25/2003 | US20030180893 Biotransformation of biologically active compounds made of various classes of chemical substance by means of laccase and manganese peroxidase enzymes |
| 09/18/2003 | US20030176670 Multivalent macrolide antibiotics |
| 09/17/2003 | CN1121405C Triphase one step extraction process to purify penicillin |
| 09/04/2003 | US20030166935 Spiroazabicyclic heterocyclic compounds |
| 09/03/2003 | EP1340762A1 Cephalosporin synthesis |
| 09/03/2003 | EP0837066B1 Improved process for producing penicillin g phenyl ester |
| 08/28/2003 | WO2003070254A1 Antibiotic conjugates |
| 08/28/2003 | CA2476448A1 Antibiotic conjugates |
| 08/19/2003 | CA2045972C Optically active n-.alpha.-fluoroacryloylamino acid derivatives and optically active polymers thereof for the resolution of racemates |
| 08/14/2003 | US20030153544 Fatty acid derivatives |
| 08/13/2003 | CN1117755C Spiroazabicyclic heterocyclic compounds, method for preparing same and use thereof |
| 07/31/2003 | US20030143653 Method and kit for detecting, or determining the quantity of, beta-lactam penicillins |
| 07/30/2003 | CN1433396A Pharmaceutical compounds |
| 07/30/2003 | CN1432572A Penicillin purifying process |
| 07/30/2003 | CN1116298C Process for preparation of 2-halomethyl-penems and their use for preparation of antibacterial penems |
| 07/30/2003 | CN1116297C Method for preparing sodium amoxicillin |
| 07/29/2003 | US6600035 6-(substituted methylene) penems and intermediates |
| 07/23/2003 | EP0757051B1 Penem derivatives and antimicrobial agent containing the same |
| 07/23/2003 | CN1115147C Improved method for preparing potassium clavulanate |
| 07/10/2003 | US20030130236 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs |
| 07/09/2003 | CN1113885C Process for producing beta-lactam derivs. |
| 07/02/2003 | EP0757691B1 Cephalosporin synthesis |
| 06/18/2003 | EP1158995B1 Biologically active compounds of ganoderma pfeifferi dms 13239 |
| 06/11/2003 | CN1422858A Penicillin static continuous extraction process and its special apparatus |
| 06/11/2003 | CN1111163C Method of eliminating water and other impurities from coarse penicillin G sulfoxide |
| 06/05/2003 | US20030105066 For use in producing antiviral, antifungal and antibacterial medicaments |
| 06/04/2003 | EP1044204B1 Process for the preparation of alpha-oxolactams |
| 05/28/2003 | CN1109688C Preparation and use of tazobactam semihydrate |
| 05/22/2003 | US20030096858 The parent drug compound is modified by forming one or more of predetermined chemical arrangement within parent drug structure for programming specific course and rate of metabolism for drug that leads to inactive nontoxic metabolite |
| 05/22/2003 | US20030095992 Altering a drug's distribution, metabolism and elimination properties, especially by modifying with aralkyl ester moieties to increase rate of metabolism to inactive and nontoxic metabolites when exposure is halted; surgery, riots |
| 05/21/2003 | CN1419450A Nitrite salts of antimicrobial agents |
| 05/20/2003 | US6566509 Compound for use as bactericide |
| 05/13/2003 | CA2299959C Procedure for the preparation of dioxopenicillanic acid derivatives |
| 05/06/2003 | US6559176 A method for regulating the activity of an autoinducer-2 receptor comprising contacting an autoinducer-2 receptor with an AI-2 agonist or antagonist compound. |
| 04/29/2003 | US6555700 1,3-propane diol esters and ethers and methods for their use in drug delivery |
| 04/23/2003 | EP1303631A2 Biotransformation of biologically active compounds made of various classes of chemical substances by means of laccase and manganese peroxidase enzymes |
| 04/23/2003 | CN1106380C New synthetic catechol derivatives, method for production and use thereof |
| 04/16/2003 | EP0871632B1 Production of a crystalline salt of amoxicillin |