Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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11/11/2009 | EP1915379B1 Olanzapine analogs and methods of use thereof |
11/11/2009 | CN101578287A Conjugates of disorazoles and their derivatives with cell-binding molecules, novel disorazole derivatives, processes of manufacturing and uses thereof |
11/11/2009 | CN101575344A Method for preparing high-purity pseudo-polymorphic lavo-ofloxacin hemihydrate |
11/11/2009 | CN100558730C Garcinia acid derivatives, preparation method and application thereof in pharmacy |
11/11/2009 | CN100558728C Calcitonin gene related peptide receptor antagonists |
11/11/2009 | CN100558428C Calcitonin gene related peptide receptor antagonists |
11/10/2009 | US7615573 Via amino ceramide-like compounds; lowering glycosphingolipid concentrations; Fabry's disease, Gaucher's disease |
11/10/2009 | CA2476257C O-alkylated rapamycin derivatives and their use, particularly as immunosuppressants |
11/10/2009 | CA2382117C 4-substituted piperidine compound |
11/05/2009 | WO2009134952A2 Potent conjugates and hydrophilic linkers |
11/05/2009 | WO2009133135A1 Spiro (piperidine-4, 2 ' -pyrrolidine) -1- (3, 5- trifluoromethyl phenyl) methylcarboxamides as nk1 tachikynin receptor antagonists |
11/05/2009 | WO2009132986A1 Imidazolidinone derivatives as 11b-hsd1 inhibitors |
11/05/2009 | WO2009132921A1 Spiro-indole derivatives for the treatment of parasitic diseases |
11/05/2009 | WO2009104147A3 Azatricyclic antibiotic compounds |
11/05/2009 | WO2009006243A8 Processes for preparing bicyclic oxazine carboxaldehyde and beta-lactamase inhibitors |
11/05/2009 | US20090275573 Imidazolidinone Derivatives as 11B-HSD1 Inhibitors |
11/05/2009 | US20090275572 Fab i inhibitors |
11/05/2009 | US20090275558 Substituted sulfonamide compounds |
11/05/2009 | US20090275523 Spirocyclic nitriles as protease inhibitors |
11/05/2009 | US20090275062 Extracting tacrolimus in a non-precipitating, non-denaturing aqueous environment, eliminates use of organic solvents and centrifugation, also fulfills the requirements for full automation of tacrolimus quantification assays |
11/05/2009 | US20090274947 Imidazolidinone nitroxides as electrode materials for energy storage devices |
11/05/2009 | US20090274656 Hepatitis c virus inhibitors |
11/05/2009 | CA2723062A1 Spiro (piperidine-4, 2 ' -pyrrolidine) -1- (3, 5- trifluoromethylphenyl) methylcarboxamides as nk1 tachikynin receptor antagonists |
11/05/2009 | CA2722487A1 Imidazolidinone derivatives as 11b-hsd1 inhibitors |
11/05/2009 | CA2720516A1 Indoline anti-cancer agents |
11/05/2009 | CA2719365A1 Spiro-indole derivatives for the treatment of parasitic diseases |
11/04/2009 | EP2113230A2 Drug-Delivery Endovascular Stent and Method for Treating Restenosis |
11/04/2009 | EP1617806B1 Selective spirocyclic glucocorticoid receptor modulators |
11/04/2009 | EP1481077B1 Mitotic kinesin inhibitors |
11/04/2009 | EP0879236B1 Derivatives of camptothecin for use in treating cancer |
11/04/2009 | CN101573360A Heteroaryl compounds, compositions thereof, and methods of treatment therewith |
11/03/2009 | US7612199 Polymorphic forms α, β, and γ of rifaximin |
11/03/2009 | US7612089 N-[4-(1-methyl-4,5-dihydro-1H-imidazol-2-yl)phenyl]-2N-(4-chlorophenylaminocarbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide; thrombosis; inhibits coagulation of a blood sample |
11/03/2009 | US7612087 Heterocyclic compounds as inhibitors of beta-lactamases |
11/03/2009 | US7612086 Jun N-terminal kinase inhibitors; 1H-pyrrolo[2,3-b]pyridines 3-substituted with a C 5-7 carbocycle and 5-substituted by a 5-member heterocycle; 3-(p-(dimethylamino)phenyl)-5-(2-thiazolyl-1H-pyrrolo[2,3-b]pyridine; neurodegenerative disorders related to apoptosis and/or inflammation |
11/03/2009 | US7612078 Piperidinylamino-thieno[2,3-D] pyrimidine compounds |
11/03/2009 | US7612063 antibiotics, fungicides, viricides; treating microbial infections; fused rings based on 4-oxo-4H-pyrido[3,2,1-kl]benzo[g]-phenoxazine for example; Tumor suppression agents with reduced side effects; anticancer |
11/03/2009 | US7612055 Macrocyclic lactams and pharmaceutical use thereof |
11/03/2009 | CA2383327C Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists |
11/03/2009 | CA2360767C Tricyclic benzodiazepines as vasopressin receptor antagonists |
11/03/2009 | CA2316356C Benzoxazine compounds for enhancing synaptic response |
10/29/2009 | WO2009131926A1 Quinuclidine compounds as alpha-7 nicotinic acetylcholine receptor ligands |
10/29/2009 | WO2009131237A1 Harmful arthropod control composition, and fused heterocyclic compound |
10/29/2009 | WO2009131065A1 Long-chain fatty acid elongation enzyme inhibitor comprising arylsulfonyl derivative as active ingredient |
10/29/2009 | WO2009130560A1 Fused pyrimidineone compounds as trpv3 modulators |
10/29/2009 | US20090270621 N-4-[3-Chloro-4-(3-fluoro-benzyloxy)-phenyl]-N6-(3-ethyl-oxazolidin-2-ylidene)-quinazoline-4,6-diamine; use as type I receptor tyrosine kinase inhibitor; hyperproliferation diseases such as cancer; antiinflammatory agents |
10/29/2009 | US20090270467 5-[(1S,3S,4R)-3-Amino-4-(2,4,5-trifluorophenyl)cyclohexyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-amine, used for treating insulin resistance, hyperglycemia and non-insulin dependent diabetes in mammals |
10/29/2009 | US20090270446 Diamine derivatives |
10/29/2009 | US20090270441 Macrolides |
10/29/2009 | US20090270405 nicotinic receptor ligands such as N-(benzo[d]thiazol-2-yl)-4H-1'-azaspiro[oxazole-5,3'-bicyclo[2.2.2]octan]-2-amine, used for the treatment of nervous system, psychological and neurodegenerative disorders; treatment of schizophrenia or Alzheimer's Disease |
10/29/2009 | US20090270383 Novel Oxabispidine Compounds And Their Use In The Treatment Of Cardiac Arrhythmias |
10/29/2009 | US20090270382 Soluble epoxide hydrolase inhibitors |
10/29/2009 | US20090270379 Quinolone derivatives useful as antibacterial agents |
10/29/2009 | CA2722325A1 Quinuclidine compounds as alpha-7 nicotinic acetylcholine receptor ligands |
10/29/2009 | CA2722159A1 Substituted phenylimidazole compounds and their use as ido inhibitors |
10/29/2009 | CA2722075A1 Long-chain fatty acyl elongase inhibitor comprising arylsulfonyl derivative as active ingredient |
10/29/2009 | CA2721270A1 Harmful arthropod control composition, and fused heterocyclic compound |
10/29/2009 | CA2720357A1 Fused pyrimidineone compounds as trpv3 modulators |
10/28/2009 | EP2111396A1 Hcv inhibiting macrocyclic phenylcarbamates |
10/28/2009 | EP1745052B9 Hiv integrase inhibitors: cyclic pyrimidinone compounds |
10/28/2009 | EP1696914B1 3-cyano-quinoline derivatives with antiproliferative activity |
10/28/2009 | CN101568543A Macrocyclic peptides as hepatitis c virus inhibitors |
10/28/2009 | CN101568336A Macrocyclic peptides as hepatitis C virus inhibitors |
10/28/2009 | CN101564571A Medical apparatus containing rapamycin analogue |
10/27/2009 | US7608613 Soluble 17-amino-analogs of geldanamycin in acid addition salt form; water solubility; anticancer agents; storage stability |
10/27/2009 | US7608564 Herbicide; in crops such as wheat, rice, maize, soybeans and cotton they act against broad-leaved weeds and grass weeds without damaging the crop plants; compounds are based on 3-(5,5-disubstituted 2-isoxazolin-3-yl)benzoic acid, esters, thioesters and pyrazolyl ketones thereof |
10/27/2009 | US7608420 Adding tetrahydrofuran to the fermentation broth, ultrafiltering the dilute broth, concentrating the permeate, adjusting the pH of the concentrate to at least pH 8.5 and collecting the precipitated staurosporine |
10/27/2009 | CA2465534C Agents useful for reducing amyloid precursor protein and treating dementia and methods of use thereof |
10/27/2009 | CA2415050C Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepines |
10/27/2009 | CA2381885C Isomeric fused pyrrolocarbazoles and isoindolones |
10/27/2009 | CA2318976C Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives |
10/22/2009 | WO2009077956A3 HETEROCYCLIC INHIBITORS OF AN Hh-SIGNAL CASCADE, MEDICINAL COMPOSITIONS BASED THEREON AND METHODS FOR TREATING DISEASES CAUSED BY THE ABERRANT ACTIVITY OF AN Hh-SIGNAL SYSTEM |
10/22/2009 | WO2008071961A8 2-quinolinone and 2-quinoxalinone- derivatives and their use as antibacterial agents |
10/22/2009 | US20090264405 Cetp Inhibitors |
10/21/2009 | EP1781673B1 Selected fused heterocyclics and uses thereof |
10/21/2009 | EP1346993B1 Lactam compounds and medical use thereof |
10/21/2009 | CN101563347A Vasopressin V1a antagonists |
10/21/2009 | CN101563345A Pharmaceutical compounds |
10/20/2009 | US7605258 Preparing an individual isomer of mono-pegylated rapamycin 42 ester with 3-hydroxy-2-(hydroxymethyl)-2-methylpropionic acid (CCI-779) by reacting an isomer of rapamycin with 3-hydroxy-2-(hydroxymethyl)-2-methylpropionic acid; use in treating nerve system cancer, leukemia, breast cancer, prostate cancer |
10/20/2009 | US7605257 Acylation in presence of lipase |
10/20/2009 | US7605169 Antibacterial agents |
10/20/2009 | US7605157 Tricyclic tetrahydroquinoline antibacterial agents |
10/20/2009 | CA2450122C Novel heterocyclic antibacterial compounds |
10/20/2009 | CA2380852C Tricyclic compounds having spiro union |
10/20/2009 | CA2378183C Antibacterial heterobicyclic substituted phenyl oxazolidinones |
10/15/2009 | WO2009125809A1 Piperidine derivatives |
10/15/2009 | WO2009125808A1 Aminocyclohexyl derivative |
10/15/2009 | WO2009124746A1 Substituted sulfonamide derivatives |
10/15/2009 | WO2009065920A3 Compounds |
10/15/2009 | US20090258891 Macrocyclic Compounds As Antiviral Agents |
10/15/2009 | US20090258864 Pyrimidine-2-amine compounds and their use as inhibitors of jak kinases |
10/15/2009 | CA2720879A1 Substituted sulfonamide derivatives |
10/14/2009 | CN101558074A Epothilone analogues modified at positions C12-C13 as anticancer drugs |
10/14/2009 | CN101555212A Synthesized micromolecule compound capable of conveying bioactivator and application thereof |
10/14/2009 | CN100549008C Substituted oxazolidinones and their use in the field of blood coagulation |
10/14/2009 | CN100549007C Broadspectrum 2-amino-benzoxazole sulfonamide HIV protease inhibitors |
10/14/2009 | CN100548296C Mitotic kinesin inhibitors |
10/14/2009 | CN100548236C Medical devices containing rapamycin analogs |
10/13/2009 | US7601836 Pyrido[2,3-D]pyrimidine inhibitors of phosphodiesterase (PDE) 7 |
10/13/2009 | US7601745 Nuclear factor kappa beta (NF-kB) inhibitors such as [4-(1H-Indol-3-yl)-piperidin-1-yl]-{2-[1-(pyrazine-2-carbonyl)-piperidin-4-yl]-thiazol-4-yl}-methanone |