| Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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| 10/13/2009 | US7601736 Pyridine derivatives, a process for their preparation and a pharmaceutical composition containing the same |
| 10/13/2009 | US7601713 Kinase inhibitors and their uses |
| 10/08/2009 | WO2009123536A1 NEW CLASSES OF GABAa/BZR LIGANDS |
| 10/08/2009 | WO2009122176A2 Rapamycin carbonate esters |
| 10/08/2009 | WO2009121872A2 Tetrahydroisoquinolines, pharmaceutical compositions containing them, and their use in therapy |
| 10/08/2009 | WO2009099736A3 Benzoxazole carboxamide inhibitors of poly(adp-ribose)polymerase (parp) |
| 10/08/2009 | US20090253733 Rapamycin carbonate esters |
| 10/08/2009 | US20090253732 Production Of Polyketides And Other Natural Products |
| 10/08/2009 | US20090253692 Crystalline form of n-[[4-fluoro-2-(5-methyl-1h-1,2,4-triazol-1-yl)phenyl]methyl]-4,6,7,9-tetrahydro-3-hydroxy-9,9-dimethyl-4-oxo-pyrimido[2,1-c][1,4]oxazine-2-carboxamide, sodium salt monohydrate |
| 10/08/2009 | US20090253681 HIV Integrase Inhibitors |
| 10/08/2009 | US20090253677 HIV Integrase Inhibitors |
| 10/08/2009 | US20090253653 Soluble 17-amino-analogs of geldanamycin in acid addition salt form; water solubility; anticancer agents; storage stability |
| 10/08/2009 | CA2720461A1 New classes of gabaa/bzr ligands |
| 10/08/2009 | CA2720004A1 Tetrahydroisoquinolines, pharmaceutical compositions containing them, and their use in therapy |
| 10/07/2009 | EP0741700B1 1-h-3-arylpyrrolidine-2,4-dione derivatives as pest-control agents |
| 10/07/2009 | CN101550143A Industrial compounding method of mule (benzo (e) (1,3) oxazine-2, 4'-piperidine)-4(3H)-ketonic |
| 10/06/2009 | US7598389 Silylated carboxamides |
| 10/06/2009 | US7598383 mitogen activated protein kinase inhibitors; 4-(2-fluoro-4-methylphenylamino)-1,3-dimethyl-6,7-dihydro-1H-pyrrolo[3,4-b]pyridine-2,5-dione; used in the treatment of hyperproliferative diseases, such as cancer and inflammation in mammals |
| 10/06/2009 | US7598376 Reaction of N,N'-diacyl-hydrazines with 2,2'-disubstituted diethyl ethers to form 4,5-diacyl-[1,4,5]-oxadiazepines; tetrahydropyrazolodione type herbicides |
| 10/06/2009 | US7598282 (3R,5S,7as)-(3,5-bis(4-fluorophenyl)tetrahydro-1H-oxazolo[3,4-c]oxazol-7a-yl)methanol; does not involve microtubule stabilization; Alzheimer's |
| 10/06/2009 | US7598266 Fused heterocyclic derivatives as PPAR modulators |
| 10/06/2009 | US7598264 HIV integrase inhibitors |
| 10/06/2009 | US7598254 Substituted 1,3-thiazolo[5,4-d]pyrimidines as xanthine oxidase inhibitors |
| 10/06/2009 | US7598253 Reverse-turn mimetics and methods relating thereto |
| 10/06/2009 | US7598237 7-aryl 1,5-dihydro-4,1-benzoxazepin-2(3H)-one derivatives and their use as progesterone receptor modulators |
| 10/01/2009 | WO2009120841A1 Crystalline form of n-[[4-fluoro-2-(5-methyl-1h-1,2,4-triazol-1-yl)phenyl]methyl]-4,6,7,9-tetrahydro-3-hydroxy-9,9-dimethyl-4-oxo-pyrimido[2,1-c][1,4]oxazine-2-carboxamide, sodium salt monohydrate |
| 10/01/2009 | WO2009120789A1 Bicyclic nitroimidazoles covalently linked to substituted phenyl oxazolidinones |
| 10/01/2009 | US20090247747 preparation of N-demethyl-tiotropium by reacting methyl-di-(2-thienyl)-glycolate with a scopine salt in presence of a weak base, a polar organic solvent; industrial scale production |
| 10/01/2009 | US20090247746 Fused heterocyclic compound |
| 10/01/2009 | US20090247509 for treating central nervous system disorders such as psychological disorders, drug dependence and abuse, dyskinesia, dementia, anxiety disorders, sleep disorders and mood disorders |
| 10/01/2009 | US20090247502 Substituted pyridoxazines |
| 10/01/2009 | US20090246134 Compositions and methods for modulating gated ion channels |
| 10/01/2009 | CA2712613A1 Bicyclic nitroimidazoles covalently linked to substituted phenyl oxazolidinones |
| 09/30/2009 | EP2105435A1 Hydrazone derivative |
| 09/30/2009 | CN101547927A 8-sulfonyl-l, 3, 4, 8-tetrahydr0-2h- [1, 4] oxazepino [6, 7-e] indole derivatives and their use as 5-ht6 receptor ligands |
| 09/30/2009 | CN101544658A (3R)-3-benzyl-7a-(difluoromethyl)tetrahydropyrrolo[2,1-b]oxazole-5(6H)-ketone and synthesis method thereof |
| 09/30/2009 | CN101544657A 3a-(trifluoromethyl)-3,3a-dihydrobenzene[d]pyrrole[2,1-b]oxazole-1(2H)-ketone and synthesis method thereof |
| 09/30/2009 | CN101544656A (3R)-3-benzyl-7a-(trifluoromethyl)tetrahydropyrrolo[2,1-b]oxazole-5(6H)-ketone and synthesis method thereof |
| 09/30/2009 | CN101544643A New method of synthesizing 1, 2, 3-triazol 1, 3-diazacyclo compound |
| 09/30/2009 | CN101544637A Pyridone heterocyclic compound and synthesizing method thereof |
| 09/30/2009 | CN101544636A Polyhalogenated isoquinoline class derivate and synthetic method thereof |
| 09/30/2009 | CN100545160C Diamine derivatives |
| 09/29/2009 | US7595400 Synthesis of antitumor agents including camptothecin derivative 9-ethyl-9-hydroxy-1-pentyl-1H,12H-pyrano[3'',4'':6',7']-indolizino[1',2':6,5]pyrido[4,3,2-de]quinazoline-10,13(9H,15H)-dione |
| 09/29/2009 | US7595343 Inhibitors of histone deacetylase |
| 09/24/2009 | WO2009117728A2 Compounds and compositions for the detection and treatment of alzheimer's disease and related disorders |
| 09/24/2009 | WO2009117540A1 Bridged heterocycles as hiv integrase inhibitors |
| 09/24/2009 | WO2009117036A2 Bioactive molecules from co-cultivation of microbes |
| 09/24/2009 | WO2009116801A2 Caspase inhibitor prodrug |
| 09/24/2009 | WO2009076440A3 Fungicidal bicyclic pyrazoles |
| 09/24/2009 | WO2009062990A3 Equilibrative nucleoside transporter ent1 inhibitors |
| 09/24/2009 | US20090240051 New process for the production of oxabispidines |
| 09/24/2009 | CA2719008A1 Fluorinated macrocyclic compounds as hepatitis c virus inhibitors |
| 09/24/2009 | CA2718950A1 Bridged heterocycles as hiv integrase inhibitors |
| 09/24/2009 | CA2718936A1 Novel heterocyclic compounds and uses therof |
| 09/24/2009 | CA2718035A1 Compounds and compositions for the detection and treatment of alzheimer's disease and related disorders |
| 09/23/2009 | EP2103618A1 Novel ansamitocin derivatives |
| 09/23/2009 | EP2102217A2 4- (2-oxo-oxazolidin-3yl)-phenoxymethyle derivativeas as antibacterials |
| 09/23/2009 | EP2102208A1 Novel substituted diaza spiro pyridinone derivatives for use in mch-1 mediated diseases |
| 09/23/2009 | EP2102170A2 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
| 09/23/2009 | EP1819713B1 Isoxazoline-indole derivatives with an improved antipsychotic and anxiolytic a ivity |
| 09/23/2009 | EP1648893B1 Nicotine addiction reducing heteroaryl fused azapolycyclic compounds |
| 09/22/2009 | US7592361 Indole acetic acid derivatives and their use as pharmaceutical agents |
| 09/22/2009 | US7592354 Administering a stimulantfor the endogenous production/ release of somatotropins; 3-((1-(2-aminoprop-2-yl)carbonylamino-),2-(phenylmethoxymethyl-)ethyl-),5-(morpholino-carbonyloxymethyl-)-5,6,7,8-tetrahydro-1,2,4-triazolo(4,3-)pyridine; osteoporosis; obesity;improving bone densisty, muscle mass/strength |
| 09/22/2009 | US7592353 Substituted 3-amino-thieno[2,3-b]pyridine-2-carboxylic acid amide compounds and processes for preparing and their uses |
| 09/22/2009 | US7592351 5,7-Dimethyl-2-thiophen-3-yl-imidazo[1,2-a]pyridin-3-yl)-(1,1,3,3-tetramethylbutyl)-amine;vanilloid/cannabinoid receptor antagonists; analgesics, neuropathic pain; headaches; antiepileptic agents; emetic agents; eating disorders; hypotensive agents; antidepressants; glaucoma; incontinence; prion disease |
| 09/22/2009 | US7592339 Substituted oxazolidinones and their use in the field of blood coagulation |
| 09/22/2009 | US7592335 3-{3-fluoro-4-[(7aE)-hexahydropyrrolo[3,4-b][1,4]oxazin-4(4aH)-yl]phenyl}-5-(iodomethyl)-1,3-oxazolidin-2-one; antibiotics; preventing catheter infections; good activity against multiply resistant gram positive pathogens |
| 09/22/2009 | US7592334 6-[({3-hydroxy-8-[6-(methyloxy)-1,5-naphthyridin-4-yl]-8-azaspiro[4.5]dec-2-yl}amino)methyl]-2H-pyrido[3,2-b][1,4]thiazin-3-on; bacterial infections; antibiotic resistance; Staphylococcus aureus, Streptococcus pneumoniae and pyogenes, Enterococcus; Haemophilus influenzae, Moraxella catarrhalis, E-coli |
| 09/22/2009 | CA2145407C New reagents for peptide couplings |
| 09/17/2009 | WO2009114677A1 Pyridazine derivatives as factor xia inhibitors |
| 09/17/2009 | WO2009112439A1 4-aryl-2-anilino-pyrimidines as plk kinase inhibitors |
| 09/17/2009 | US20090233274 Drug development target protein and target gene, and method of screening |
| 09/17/2009 | CA2716079A1 4-aryl-2-anilino-pyrimidines as plk kinase inhibitors |
| 09/16/2009 | EP2099806A1 Spiropiperidine derivatives as nk3 antagonists |
| 09/16/2009 | EP2099799A1 Spiro-piperidine derivatives |
| 09/16/2009 | EP1486500B1 10-(3-cyclopropylaminomethyl-1-pyrrolidinyl)pyridobenzoxazinecarboxylic acid derivative effective against resistant bacteria |
| 09/16/2009 | CN101531670A 7-methyl-3a-(trifluoromethyl)-3, 3a-dihydrobenzo (d) pyrrole (2, 1-b)-oxazole-1(2H)-ketone and synthetic method thereof |
| 09/16/2009 | CN101531669A 7-chlorine-3a-(trifluoromethyl)-3, 3a-dihydrobenzo (d) pyrrole (2, 1-b)-oxazole-1(2H)-ketone and synthetic method thereof |
| 09/16/2009 | CN101531668A (3s)-3-benzyl-7a-(trifluoromethyl) tetrahydropyrrolo [2, 1-b] oxazole-5(6H)-ketone and synthetic method thereof |
| 09/16/2009 | CN100540547C Inhibitors of histone deacetylase |
| 09/15/2009 | US7589194 Crystalline k-252b, sodium salt, methanolate pentahydrate |
| 09/15/2009 | US7589128 Process for preparation of amorphous form of a drug |
| 09/15/2009 | US7589102 Heterocyclic aromatic compounds useful as growth hormone secretagogues |
| 09/15/2009 | US7589100 Non-hygroscopic and powdery amorphous pimecrolimus |
| 09/15/2009 | US7589077 such as 5-iodo-O6-5'-cyclo-5,6-dihydro-3'-azido-3'-deoxythymidine for prophylaxis or diagnosis of viral diseases caused by hepatitis virus, herpes viruses such as Epstein-Barr virus |
| 09/15/2009 | CA2429220C Gaba enhancers in the treatment of diseases relating to reduced neurosteroid activity |
| 09/15/2009 | CA2274204C Spiro[piperidine-4,1'-pyrrolo[3,4-c]pyrrole] |
| 09/15/2009 | CA2148871C Method of preventing hyperproliferative vascular disease |
| 09/11/2009 | WO2009110901A1 Substituted dihydro, trihydro and tetrahydro cycloalkyloxazolopyrimidinones, preparation and use thereof as allosteric modulators of mglur |
| 09/11/2009 | WO2009110510A1 Alkylaminopyridine derivative |
| 09/11/2009 | WO2009110007A1 Spiro derivatives of parthenin as novel anticancer agents |
| 09/11/2009 | WO2009075746A3 Curable benzoxazine macromonomers, their preparation and cured products thereof |
| 09/11/2009 | CA2728855A1 Spiro derivatives of parthenin as novel anticancer agents |
| 09/11/2009 | CA2716664A1 Oxadiazoanthracene compounds for the treatment of diabetes |
| 09/11/2009 | CA2714617A1 Alkylaminopyridine derivative |
| 09/10/2009 | US20090227789 Ethylenediamine derivatives |
| 09/10/2009 | US20090226948 Enzyme-based time temperature indicator |
| 09/09/2009 | EP2097400A2 Fused substituted aminopyrrolidine derivative |
| 09/09/2009 | EP1902050B1 Oxazolidinone derivatives and use thereof as antibiotics |
| 09/09/2009 | EP1664061A4 Process for the synthesis of morphinane compounds and intermediates thereof |