| Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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| 02/25/2010 | US20100048890 Conjugated small molecules |
| 02/25/2010 | US20100048667 Thiolactones |
| 02/25/2010 | US20100048528 Heterocyclic compounds as inhibitors of beta-lactamases |
| 02/24/2010 | EP2157077A1 Method for producing triarylamine compound |
| 02/24/2010 | EP2155737A1 Gamma secretase modulators |
| 02/23/2010 | US7666880 Hydroxamate compounds which are inhibitors of histone deacetylase; may be useful as medicaments for treatment of proliferative disorders as well as other diseases involving, relating to, or associated with enzymes having histone deacetylase activities such as neurodegenerative, cardiovascular disorders |
| 02/23/2010 | US7666879 enzyme inhibitor; 2-{2-Fluoro-4-[7-(2-methyl-pyridin-4-yl)-imidazo[1,2-a]pyridin-3-yl]-phenyl}-N-(3-trifluoromethyl-phenyl)-acetamide; angiogenesis inhibitor; antitumor agent; treating hyperglycemia, psoriasis, rheumatoid arthritis, Kaposi's sarcoma, autoimmune diseases, inflammation, and eye disorders |
| 02/23/2010 | US7666876 Buprenorphine formulations for intranasal delivery |
| 02/23/2010 | US7666864 Bicyclic nitroimidazole-substituted phenyl oxazolidinones |
| 02/18/2010 | WO2010018686A1 Nitrogenated heterocyclic derivative, and agricultural or horticultural bactericidal agent |
| 02/18/2010 | WO2009155017A3 Novel substituted azabenzoxazoles |
| 02/18/2010 | WO2009117728A3 Compounds and compositions for the detection and treatment of alzheimer's disease and related disorders |
| 02/18/2010 | US20100041676 Kinase inhibitors |
| 02/18/2010 | US20100041647 3-Substituted-[1,2,3]-Benzotriazinone compounds for enhancing glutamatergic synaptic responses |
| 02/18/2010 | US20100040548 High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds |
| 02/17/2010 | EP2152719A1 Bicyclic heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
| 02/17/2010 | EP2152695A2 Gamma secretase modulators |
| 02/17/2010 | EP2152664A1 Dipeptide analogs as coagulation factor inhibitors |
| 02/17/2010 | EP2152082A1 Tetracyclic inhibitors of fatty acid amide hydrolase |
| 02/17/2010 | CN101652373A Oxazinyl isoflavonoid compounds, medicaments and use |
| 02/17/2010 | CN101648960A Method for preparing ofloxacin |
| 02/16/2010 | US7662971 enzyme inhibitor for treating sleep disorders |
| 02/16/2010 | US7662958 e.g. N-[3-{1-[(cyclobutyl)amino]-4-hydroxy-2-oxo-1,2-dihydro-quinolin -3-yl}-1,1-dioxo-1,4-dihydro-1 lambda 6-thieno[2,3-e][1,2,4]thiadiazin-7-yl)methyl]methane-sulfonamide; viricides for infections caused by an RNA-containing virus; hepatitis C virus (HCV) polymerase inhibitor; liver cirrhosis |
| 02/16/2010 | US7662846 Selective spirocyclic glucocorticoid receptor modulators |
| 02/16/2010 | US7662833 metalloproteinases inhibitor, particular Peptide Deformylase (Pdf) inhibitor; antibiotic; e.g. 2-(6-fluoro-imidazo[1,2-a]pyridin-3-ylamino)-N-hydroxy-acetamide |
| 02/16/2010 | US7662828 Substituted 5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine-2-yl compounds and 5,6,7,8-tetrahydroquinazoline-2-yl compounds |
| 02/16/2010 | CA2562532C Crystalline clopidogrel naphthalenesulfonate or hydrate thereof, method for preparing same and pharmaceutical composition containing same |
| 02/16/2010 | CA2533548C Method of purifying macrolides |
| 02/16/2010 | CA2225822C Nitroimidazole antibacterial compounds and methods of use thereof |
| 02/11/2010 | WO2010017093A2 Dopamine receptor ligands with enhanced duration of action |
| 02/11/2010 | WO2010016851A1 Process for selectively producing a pyridobenzoxazine carboxylic acid hemihydrate |
| 02/11/2010 | WO2010016552A1 Therapeutic agent for irritable bowel syndrome |
| 02/11/2010 | WO2010015628A1 Pyrazolo [5,1-b] oxazole derivatives as crf1 antagonists |
| 02/11/2010 | WO2010015626A1 Crystalline forms of a pyridine derivative |
| 02/11/2010 | US20100035947 Method for manufacturing neuraminic acid derivatives |
| 02/11/2010 | US20100035946 Indoline anti-cancer agents |
| 02/11/2010 | US20100035874 Organic compounds |
| 02/11/2010 | CA2733235A1 Crystalline forms of a pyridine derivative |
| 02/11/2010 | CA2733176A1 Pyrazolo [5,1-b] oxazole derivatives as crf1 antagonists |
| 02/10/2010 | EP2150551A1 2-oxo-3-benzyl-benzoxazol-2-one derivatives and related compounds as met kinase inhibitors for the treatment of tumors |
| 02/10/2010 | EP2150115A1 Cyclopropyl pyrrolidine orexin receptor antagonists |
| 02/10/2010 | EP2066678B1 Spiro antibiotic derivatives |
| 02/10/2010 | EP1701951B1 Modulators of peripheral 5-ht receptors |
| 02/10/2010 | EP1411932B1 Substituted oxazolidinones for combinational therapy |
| 02/10/2010 | CN101646679A Heterocyclic antiviral compounds |
| 02/09/2010 | US7659296 2-{1-[4-(3,3-dimethyl-2-oxo-butoxy)-3-methyl-phenyl]-1-ethyl-propyl}-benzooxazole-6-carboxylic acid; 1-[4-(3,3-Dimethyl-2-oxo-butoxy)-3-methyl-phenyl]-1-ethyl-propyl}-benzooxazole-6-carboxylic acid amide; stimulate bone formation, restore bone quality, acne, alopecia, Alzheimer's disease etc. |
| 02/09/2010 | US7659265 5-(4,4-dimethyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbothioamide; menopause therapy; contraceptive; anticancer agents |
| 02/09/2010 | US7659263 (E)-3-[4-({1-[(11-cyclohexyl-8-methoxy-4,5-dihydro-6-oxa-1-thia-3b-azabenzo[e]cyclopenta[a]azulene-2-carbonyl)amino]cyclobutanecarbonyl}amino)phenyl]acrylic acid; RNA-dependent RNA polymerase inhibitory activity; hepatitis C |
| 02/09/2010 | US7659244 Rapamycin peptides conjugates: synthesis and uses thereof |
| 02/09/2010 | CA2437505C Isoxazoline derivatives as anti-depressants |
| 02/09/2010 | CA2274201C Di-or triaza-spiro[4,5]decane derivatives |
| 02/09/2010 | CA2201863C Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitors |
| 02/04/2010 | US20100029937 Novel and practical process for exclusively producing (s)-9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7h-pyrido-[1,2,3,de][1,4]benzoxazine-6-carboxylic acid hemihydrate |
| 02/04/2010 | US20100029933 Pure form of rapamycin and a process for recovery and purification thereof |
| 02/04/2010 | US20100029731 Method for preparing largazole analogs and uses thereof |
| 02/04/2010 | US20100029669 3-(substituted ethyl)-rifamycin derivatives useful as antimicrobial agents |
| 02/04/2010 | US20100029666 Macrocyclic Quinoxaline Compounds as HCV NS3 Protease Inhibitors |
| 02/04/2010 | US20100029633 Imidazo[1,2-a]pyridine compounds as receptor tyrosine kinase inhibitors |
| 02/04/2010 | US20100029632 improved pharmacokinetics |
| 02/04/2010 | US20100029623 4-(1-amino-ethyl)-cyclohexylamine derivatives |
| 02/04/2010 | CA2729045A1 Pyrimidine compounds, compositions and methods of use |
| 02/03/2010 | EP2149571A1 Mutilin derivative having heterocyclic aromatic ring carboxylic acid structure in substituent at 14-position |
| 02/03/2010 | EP1778677B1 Heterocyclic condensed compounds useful as antidiuretic agents |
| 02/03/2010 | CN101637624A Medical devices containing rapamycin analogs |
| 02/03/2010 | CN100586952C Derivative of oxazolocamptothecin ester, preparation method and application |
| 02/03/2010 | CN100586945C Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivatives and their use as neurokinin antagonists |
| 02/02/2010 | US7655673 39-desmethoxyrapamycin, compositions and methods of use thereof |
| 02/02/2010 | US7655658 Thieno [2,3-D]pyrimidine-2,4-dione melanocortin-specific compounds |
| 02/02/2010 | US7655650 Oxadiazine derivatives |
| 02/02/2010 | US7655649 Inhibitors of Akt activity |
| 02/02/2010 | US7655648 Antibacterial agents |
| 02/02/2010 | US7655642 3-cyano-quinoline derivatives with antiproliferative activity |
| 01/28/2010 | WO2010011964A2 Imaging agents useful for identifying ad pathology |
| 01/28/2010 | WO2010011959A1 Antiviral compounds |
| 01/28/2010 | WO2010010435A2 Fused oxazole and thiazole derivatives as trpms modulators |
| 01/28/2010 | WO2009122176A3 Rapamycin carbonate esters |
| 01/28/2010 | WO2009107850A3 Fused heterocyclic derivative and use thereof |
| 01/28/2010 | US20100022766 Biosynthetic gene cluster for the production of a complex polyketide |
| 01/28/2010 | US20100022607 Diazonamide analogs |
| 01/28/2010 | US20100022593 Process for Producing Anticancer Agent LL-D45042 |
| 01/28/2010 | US20100022524 Tricyclic tetrahydroquinoline antibacterial agents |
| 01/28/2010 | US20100022516 4,5-Disubstituted-2-aryl pyrimidines |
| 01/28/2010 | US20100022508 Antiviral compounds |
| 01/28/2010 | US20100022500 Macrocyclic Lactams and Pharmaceutical Use Thereof |
| 01/28/2010 | CA2731738A1 Imaging agents useful for identifying ad pathology |
| 01/27/2010 | EP2147000A1 Method of purification of rapamycin and its analogs by use of cascade chromatography |
| 01/27/2010 | EP2146983A1 Pyrazoles useful in the treatment of inflammation |
| 01/27/2010 | EP2146972A2 Heterocyclic compounds containing the morpholine nucleus their preparation and use |
| 01/27/2010 | EP1554286B1 Fused heterocyclic isoxazoline derivatives and their use as anti-depressants |
| 01/26/2010 | US7652032 5-Thioxylopyranose compounds |
| 01/26/2010 | US7652020 novel hydantoin derivatives to inhibit matrix metalloproteinases (MMPs), a disintegrin and metalloproteases (ADAMs) and/or tumor necrosis factor alpha converting enzyme (TACE) and in so doing prevent the release of tumor necrosis factor alpha (TNF- alpha ); autoimmune diseases; side effect reduction |
| 01/26/2010 | US7652010 Azabicyclic aryl derivatives and their medical use |
| 01/26/2010 | US7652008 Tricyclic benzopyran compound as anti-arrhythmic agents |
| 01/26/2010 | US7652006 Substituted 1(2H)-phthalazinones and pharmaceutical compositions thereof |
| 01/26/2010 | CA2303934C Tetrazole-containing rapamycin analogs with shortened half-lives |
| 01/26/2010 | CA2275345C Pro-drugs and counterparts of camptothecin, their application as medicines |
| 01/21/2010 | WO2010006704A1 Oxazolopyrimidines as edg-1 receptor agonists |
| 01/21/2010 | WO2010006521A1 2-methyl-5h-pyrazolo[1,5-a][3,1]benzoxazin-5-imine compound, the preparation and the use thereof |
| 01/21/2010 | WO2010006485A1 Benzoxazinopyrazoles and their ring-opening compound |
| 01/21/2010 | WO2009145456A3 Heterocyclic derivatives |