Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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10/27/2010 | EP1907399B1 5,6-di-substituted oxadiazolopyrazines and thiadiazolopyrazines as cxc-chemokine receptor ligands |
10/27/2010 | EP1838715B1 Method for the preparation of maytansinoid esters |
10/27/2010 | EP1432408B1 Pharmaceutical compositions comprising colloidal silicon dioxide |
10/27/2010 | CN1829722B Regioselective synthesis of CCI-779 |
10/27/2010 | CN101027309B Enantiomers of selected fused pyrimidones and uses in the treatment and prevention of cancer |
10/26/2010 | USRE41895 Epothilone derivatives |
10/26/2010 | USRE41893 Epothilone derivatives |
10/26/2010 | US7820838 Ecteinascidin 743; 5-(1,2-diaminoethyl-), 3,4-methylenedioxyphenol intermediate, of which the amine group cyclizes |
10/26/2010 | US7820823 Dual action antibiotics |
10/26/2010 | US7820812 Methods of manufacturing crystalline forms of rapamycin analogs |
10/26/2010 | US7820702 Sulfonylpyrrolidine modulators of androgen receptor function and method |
10/26/2010 | US7820664 N-(2-aylamino)aryl sulfonamides such as N-(7-(4-bromo-2-fluorophenylamino)imidazo[1,2-b]pyridazin-6-yl)-1-(2-hydroxyethyl)cyclopropane-1-sulfonamide; mitogen-activated ERK activating kinase (MEK) inhibitors; antiproliferative, anticarcinogenic, and antiinflammatory agents |
10/26/2010 | US7820655 Ethanol or 1,2-ethanediol cyclohexyl antibiotic derivatives |
10/26/2010 | CA2418921C Novel composition |
10/26/2010 | CA2133323C Self-assembling polynucleotide delivery system |
10/21/2010 | WO2010120998A1 Pyrimidine compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses |
10/21/2010 | WO2010084499A3 Bicyclic heterocyclic spiro compounds |
10/21/2010 | WO2009110007A8 Spiro derivatives of parthenin as novel anticancer agents |
10/21/2010 | WO2009020470A3 Cgrp receptor antagonists |
10/21/2010 | US20100268329 Drug/Drug Delivery Systems For The Prevention And Treatment Of Vascular Disease |
10/21/2010 | US20100267964 N-heterocyclylphenyl-substituted cyclic ketoenols |
10/21/2010 | US20100267945 Amine derivative having npy y5 receptor antagonistic activity |
10/21/2010 | US20100267685 Methods For The Prophylaxis And/or Treatment Of Thromboembolic Disorders By Combination Therapy With Substituted Oxazolidinones |
10/21/2010 | US20100266509 Heteroaryl amide analogues as p2x7 antagonists |
10/21/2010 | CA2755554A1 Pyrimidine compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses |
10/20/2010 | EP2240495A1 Nemorubicin metabolite and analog reagents, antibody-drug conjugates and methods |
10/20/2010 | EP2240485A1 Tricyclic compounds having corticotropin-releasing factor antagonistic activity and pharmaceutical compositions containing them |
10/20/2010 | EP2240467A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
10/20/2010 | EP2240454A1 Mesoionic pesticides |
10/20/2010 | EP2240016A1 Ampk modulators |
10/20/2010 | EP2049491B1 Heteroaryl compounds useful as inhibitors of e1 activating enzymes |
10/20/2010 | EP1789377B1 Alternative synthesis of renin inhibitors and intermediates thereof |
10/20/2010 | EP1732929B1 Tricyclic benzopyran compound as anti-arrhythmic agents |
10/20/2010 | CN101863909A Norcantharidin derivative and activity testing method and application thereof |
10/20/2010 | CN101863904A Preparation method of high-purity Levofloxacin semihydrate |
10/20/2010 | CN101863886A Heterocyclic aromatic compounds useful as growth hormone secretagogues |
10/20/2010 | CN101862233A Drug-delivery endovascular stent and method for treating restenosis |
10/19/2010 | US7816524 Methods of preparing quinolone analogs |
10/19/2010 | CA2400614C Synthetic process for an intermediate for ecteinascidin and phthalascidin compounds |
10/19/2010 | CA2393158C Substituted homopiperidinyl benzimidazole analogues as fundic relaxants |
10/19/2010 | CA2193130C New streptogramins and process for preparing streptogramins by mutasynthesis |
10/14/2010 | WO2010117077A1 Therapeutic agent for chorioretinal diseases comprising sirolimus derivative as active ingredient |
10/14/2010 | WO2010116270A1 Ep2/4 agonists |
10/14/2010 | US20100261719 Chemical compounds |
10/14/2010 | US20100261641 Spiro-piperidine compounds and medicinal use thereof |
10/14/2010 | CA2758072A1 Macrocyclic serine protease inhibitors |
10/13/2010 | EP2239565A1 Optical-isomer separating agent for chromatography and process for producing the same |
10/13/2010 | EP2239258A2 Tetrahydrobenzoxazine |
10/13/2010 | EP2238144A1 Compounds comprising a cyclobutoxy group |
10/13/2010 | EP2238138A1 Tricyclic nitrogen compounds and their use as antibacterial agents |
10/13/2010 | EP2004658B1 Condensed imidazole derivatives as aromatase inhibitors |
10/13/2010 | EP1783129B1 Spiropiperidyl rifamycins for the treatment of microbacterial infections |
10/13/2010 | EP1480644B1 Novel heterocyclic compounds which are active as inhibitors of beta+lactamases |
10/13/2010 | EP1204642B1 Fungicides |
10/13/2010 | CN101861309A SALARIN and TULEARIN, compositions and uses thereof |
10/13/2010 | CN101084217B Imidazo[4,5-b]pyridin-2-one and oxazolo[4,5-b]pyridin-2-one compounds and analogs thereof as therapeutic compounds |
10/12/2010 | US7812167 Substituted (thiazol-2-yl)-amides or sulfonamides as glucokinase activators useful in the treatment of type 2 diabetes |
10/12/2010 | US7812155 reacting rapamycin with an alkyl triflate, purifying the resulting reaction product with a normal phase chromatograph and further purifying with a reverse phase chromatography |
10/12/2010 | US7812038 such as vascular cell adhesion molecules and fibronectins, administered for the treatment of asthma, multiple sclerosis or inflammatory bowel diseases in mammals; (3S)-3-{[({1-[(2-chlorophenyl)methyl]-4-hydroxy-2-oxo-1,2-dihydro-3quinolinyl}amino)carbonyl]amino}-3-(4-methylphenyl)propanoic acid |
10/12/2010 | US7812032 crystalline forms of zotarolimus (ABT-578); bioavailability, solubility |
10/12/2010 | US7812024 such as (4R,11aR)-4-methyl-1,2,3,4,11,11a-hexahydropyrazino[1,2-b]isoquinolin-6-one, used for the treatment of obesity, diabetes, atherosclerosis, dyslipidemia, anxiety, depression, psychosis, schizophrenia, sleep, sexual, obsessive compulsive and gastrointestinal disorders |
10/12/2010 | US7812013 4-Imino-2-methyl-3,5,13-triazatetracyclo[15.3.1.1(2,5).1(7,11)]tricosa-1(21),7,9,11(22),17,19-hexaene-12,23-dione, used for treating cardiovascular diseases, cognitive and neurodegenerative diseases |
10/07/2010 | WO2010114971A1 Compounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof |
10/07/2010 | WO2010114958A1 Bridged bicyclic heterocycle derivatives and methods of use thereof |
10/07/2010 | WO2010112865A1 5-ht receptor modulating compounds |
10/07/2010 | US20100256388 3-3-Di-Substituted-Oxindoles As Inhibitors of Translation Initiation |
10/07/2010 | US20100256361 Thiazole derivatives |
10/07/2010 | US20100256170 Pyrazole compounds useful as protein kinase inhibitors |
10/07/2010 | US20100256129 Selective androgen receptor modulators (sarms) and uses thereof |
10/07/2010 | US20100256128 Gamma secretase modulators |
10/07/2010 | US20100256124 Substituted 1-Methyl-1H-Quinolin-2-Ones And 1-Methyl-1H-1,5-Naphthyridin-2-Ones As Antibacterials |
10/07/2010 | US20100256114 Amido Compounds And Their Use As Pharmaceuticals |
10/07/2010 | US20100255005 Gamma secretase modulators |
10/07/2010 | US20100251490 Reactive dyes, processes for their preparation and their use |
10/07/2010 | CA2757106A1 5-ht receptor modulating compounds |
10/07/2010 | CA2756989A1 Compounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof |
10/06/2010 | EP2235007A1 6h-dibenz0 [b, e] oxepine derived nonsteroidal mineralocorticoid receptor antagonists |
10/06/2010 | EP2234999A1 Heteroaryl derivatives as orexin receptor antagonists |
10/06/2010 | EP1781672B1 Solvent free amorphous rapamycin |
10/06/2010 | EP1515965B1 Phenylaminopyrimidines and their use as rho-kinase inhibitors |
10/06/2010 | CN1914212B Polymorphic forms of a GABAA agonist |
10/06/2010 | CN101855229A Spirocyclic aminoquinolones as GSK-3 inhibitors |
10/06/2010 | CN101855228A Cyanoaminoquinolones and tetrazoloaminoquinolones as GSK-3 inhibitors |
10/06/2010 | CN101855224A Equilibrative nucleoside transporter ENT1 inhibitors |
10/06/2010 | CN101851648A Method for preparing demethyl rapamycin by utilizing bacillus megaterium |
10/06/2010 | CN101851173A Inhibitors of histone deacetylase |
10/05/2010 | US7807833 Chemical intermediates for sulfiding under mild conditions forming ring compounds for use as marine alkaloids; connecting reaction of 4 components, transforming c22-tert-butyltriphenylsilyl to acety group, cyclization, hydroxy group to methanesulonyl group, reduction of amide, dehydration,Heck reaction |
10/05/2010 | US7807418 Method for producing hybrid polyketide synthases |
10/05/2010 | US7807191 Apparatus and methods for preventing or treating failure of hemodialysis vascular access and other vascular grafts |
10/05/2010 | US7807075 Photochromic compositions and light transmissible articles |
10/05/2010 | CA2322516C Sustained release macrolide compositions |
09/30/2010 | WO2010110380A1 Fused piperidine compound and pharmaceutical agent comprising same |
09/30/2010 | WO2010109299A2 Substituted 1, 4-dioxa-8-azaspiro [4,5] decanes useful as fungicides and a process for the preparation thereof |
09/30/2010 | WO2010108903A1 2,3-diaryl- or heteroaryl-substituted 1,1,1-trifluoro-2-hydroxypropyl compounds |
09/30/2010 | US20100249403 Use of oxazine compounds for making chromogenic materials |
09/30/2010 | US20100249201 3-3-Di-Substituted-Oxindoles As Inhibitors of Translation Initiation |
09/30/2010 | US20100249181 HIV Protease Inhibiting Compounds |
09/30/2010 | US20100249132 Imidazole derivatives |
09/30/2010 | US20100248264 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions |
09/30/2010 | US20100247519 Heterocyclic aspartyl protease inhibitors |