Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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08/31/2010 | US7786162 Agents useful for reducing amyloid precursor protein and treating dementia and methods of use thereof |
08/31/2010 | CA2603274C Tetracyclic compounds, their preparation process and the pharmaceutical compounds containing them |
08/26/2010 | WO2010095765A1 Ring compound |
08/26/2010 | WO2010095602A1 Heterocyclic compound |
08/26/2010 | WO2010011964A3 Imaging agents useful for identifying ad pathology |
08/26/2010 | WO2009098448A8 Compounds |
08/26/2010 | US20100217005 Epoxy compound and method for manufacturing the same |
08/26/2010 | US20100216821 Benzimidazoles With A Hetero Spiro-Decane Residue As NPY-Y5 Antagonists |
08/26/2010 | US20100216781 mTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY |
08/25/2010 | EP2221303A1 Benzoxazine-based monomer, polymer thereof, electrode for fuel cell including the polymer, electrolyte membrane for fuel cell including the polymer, and fuel cell using the electrode |
08/25/2010 | EP2221302A1 Pyrido-oxazine-based monomer, polymer thereof, electrode for fuel cell including the polymer, electrolyte membrane for fuel cell including the polymer, and fuel cell using the electrode |
08/25/2010 | EP2220068A1 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors |
08/25/2010 | EP2220048A2 Aryl- and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
08/25/2010 | EP2219453A1 Quinoxaline-containing compounds as hepatitis c virus inhibitors |
08/25/2010 | EP1366016B1 Process for the preparation of arylethanoldiamines useful as agonists of the beta-3-adrenoceptor |
08/25/2010 | EP0883403B1 Method for treating sexual dysfunctions |
08/25/2010 | CN101812078A Heterocyclic dihydropyridine compound and synthesis method thereof |
08/25/2010 | CN101812074A Method for preparing antofloxacin hydrochloride |
08/25/2010 | CN101812063A Alpha-naphthalenesulfonamide base quintuple heterocyclic compound and anti-tumor activity thereof |
08/24/2010 | US7781454 Substituted indazoles, benzotriazoles, and related bicyclic compounds; HIV (human immunodeficiency virus) reverse transcriptase inhibitors; delays onset of AIDS or AIDS related complex |
08/24/2010 | US7781447 O-methylated rapamycin derivatives for alleviation and inhibition of lymphoproliferative disorders |
08/24/2010 | US7781446 renal cancer; after standard chemotherapy; rapamycin 42-ester with 3-hydroxy-2-(hydroxymethyl)-2-methylpropionic acid (CCI-779) |
08/19/2010 | WO2010093341A1 C-7 isoxazolinyl quinolone/naphthyridine derivatives useful as antibacterial agents |
08/19/2010 | WO2010092181A1 Heterocyclic compounds, pharmaceutical compositions containing them, and their use as inhibitors of the glycine transporter 1 |
08/19/2010 | US20100210762 Heterocyclic compound, ultraviolet absorbent and composition containing the same |
08/19/2010 | US20100210636 Benzoxazinone derivative |
08/19/2010 | CA2750913A1 Heterocyclic compounds, pharmaceutical compositions containing them, and their use as inhibitors of the glycine transporter 1 |
08/18/2010 | EP2218722A2 Process for producing benzoxazine derivative and production intermediate thereof |
08/18/2010 | EP2217650A2 Curable benzoxazine-based compositions, their preparation and cured products thereof |
08/18/2010 | EP2217605A1 Compounds for inhibiting ksp kinesin activity |
08/18/2010 | EP2217604A1 Gamma secretase modulators |
08/18/2010 | EP2217600A2 Fungicidal bicyclic pyrazoles |
08/18/2010 | EP2217596A2 Bicyclic heterocycle derivatives and their use as modulators of the activity of gpr119 |
08/18/2010 | EP2217566A1 Bis-(sulfonylamino) derivatives in therapy 066 |
08/18/2010 | EP2217071A1 Antifungal agents |
08/18/2010 | EP2066677B1 Pyridooxazepine progesteron receptor modulators |
08/18/2010 | EP1940828B1 Heterocyclic aspartyl protease inhibitors |
08/18/2010 | CN101809019A Gamma secretase modulators |
08/18/2010 | CN101809016A Gamma secretase modulators |
08/18/2010 | CN101808988A Piperidine and piperazine derivatives |
08/18/2010 | CN101805748A 17-desmethylrapamycin and analogues thereof, methods for their production and their use as immunosupressants, anticancer agents, antifungal agents, etc |
08/18/2010 | CN101805358A Substituted (thiazol-2-yl) -amide or sulfonamide as glycokinase activators useful in treatment of type 2 diabetes |
08/18/2010 | CN101381372B Pazufloxacin mesylate and preparation method of powder for injection |
08/18/2010 | CN101024671B 丙型肝炎病毒抑制剂 Hepatitis C virus inhibitors |
08/17/2010 | US7777051 A compound with azo containing mono and a bicyclic rings attached with an aryl or heteroaryl ring; both therapeutic and diagnostic |
08/17/2010 | US7777032 N-4-[3-Chloro-4-(3-fluoro-benzyloxy)-phenyl]-N6-(3-ethyl-oxazolidin-2-ylidene)-quinazoline-4,6-diamine; use as type I receptor tyrosine kinase inhibitor; hyperproliferation diseases such as cancer; antiinflammatory agents |
08/17/2010 | US7776874 Cycloalkylcarbonyl-3H-spiro[2-benzofuran-1,3'-pyrrolidin]-3-ones: N-methyl-5-[4-(1-{[3-oxo-1'H,3H-spiro[2-benzofuran-1,3'-pyrrolidin]-1'-yl]carbonyl}cyclopropyl)phenyl]pyridine-2-carboxamide; 11- beta hydroxyl steroid dehydrogenase type 1 inhibitors; mineralcorticoid receptor antagonists; diabetes |
08/17/2010 | US7776853 Dietetics therapy; lipase inhibitor |
08/17/2010 | US7776791 N-heterocyclyl phenyl-substituted cyclic ketoenols |
08/12/2010 | WO2010090341A1 Method of manufacturing optically active trans-4-aminopiperidine-3-ol compound |
08/12/2010 | WO2010089127A1 Substituted spiro-amides as b1r modulators |
08/12/2010 | WO2010042489A3 Aminoquinoline derived heat shock protein 90 inhibitors, methods of preparing same, and methods for their use |
08/12/2010 | WO2009082437A9 Selective androgen receptor modulators (sarms) and uses thereof |
08/12/2010 | US20100204466 One pot synthesis of tetrazole derivatives of rapamycin |
08/12/2010 | US20100204216 PHARMACEUTICAL COMPOSITION FOR INHIBITING AMYLOID-beta PROTEIN ACCUMULATION |
08/12/2010 | US20100204201 Hiv integrase inhibitors |
08/12/2010 | US20100204197 Pyrrolopyrimidines |
08/12/2010 | US20100204119 4-amino-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5h)-yl phenyl derivatives |
08/12/2010 | US20100203007 Novel benzodiazepine derivatives |
08/12/2010 | CA2751535A1 Substituted spiro-amides as b1r modulators |
08/11/2010 | EP2215090A1 Purine derivatives useful as pi3 kinase inhibitors |
08/11/2010 | EP1797099B1 Piperidinylamino-thieno[2,3-d] pyrimidine compounds |
08/11/2010 | CN1649551B Drug-delivery endovascular stent and method for treating restenosis |
08/10/2010 | US7772252 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands |
08/10/2010 | US7772234 Bicyclic inhibitors of MEK and methods of use thereof |
08/10/2010 | US7772232 Quinazolinyl compounds as inhibitors of potassium channel function |
08/10/2010 | US7772229 Oxabispidine compounds useful in the treatment of cardiac arrhythmias |
08/10/2010 | US7772228 Administering a rifamycin microbiocides for treating infections caused by Mycobacterium tuberculosis, Mycobacterium avium complex, Chlamydia pneumoniae or Helicobacter pylori |
08/10/2010 | US7772227 such as (R)-3-Cyclohexyl-2,3-dihydro-6-(4-ethylpiperazin-1-ylcarbonyl)pyrrolo[1,2,3-de]-1,4-benzoxazine hydrochloride salt, used as analgesics for the treatment of post-operative pain, chronic pain neuropathic pain, cancer pain and spasticity associated with multiple sclerosis |
08/10/2010 | US7772226 such as 3-(2-Butynyl)-2-(piperazin-1-yl)-3,5-dihydroimidazo[4,5-d]pyridazin-4-one trifluoroacetate, used as dipeptidyl peptidase-IV (DPPIV) inhibitors for the treatment of obesity and diabetes |
08/10/2010 | CA2483159C Triazole derivatives as tachykinin receptor antagonists |
08/10/2010 | CA2477967C Purine derivatives as kinase inhibitors |
08/10/2010 | CA2451605C Diamine derivatives |
08/10/2010 | CA2366800C Carboxylic acid derivatives that inhibit the binding of integrins to their receptors |
08/05/2010 | WO2010086820A1 4-amino-5-oxo-7, 8-dihydropyrimido [5,4-f] [1,4] oxazepin-6 (5h) -yl) phenyl derivatives, pharmaceutical compositions and uses thereof |
08/05/2010 | WO2009100872A8 Urea derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
08/05/2010 | US20100197909 Mutilin derivative having heterocyclic aromatic ring carboxylic acid structure in subtituent at 14-position |
08/05/2010 | US20100197907 Phosphorus-containing compounds & uses thereof |
08/05/2010 | US20100197699 I-OXA-3-Azaspiro (4.5) Decan-2-One And 1-OXA-3, 8-Diazaspiro (4.5) Decan-2-One Derivatives For The Treatment of Eating Disorders |
08/05/2010 | US20100197679 Compounds |
08/05/2010 | US20100197678 Glucocorticoid Mimetics, Methods of Making Them, Pharmaceutical Compositions and Uses Thereof |
08/05/2010 | US20100197645 Thioamide Derivatives as Progesterone Receptor Modulators |
08/05/2010 | US20100196355 Immunophilin Ligands and Methods for Modulating Immunophilin and Calcium Channel Activity |
08/04/2010 | EP2213675A1 Pyridooxazepine derivative and use thereof |
08/04/2010 | EP1578705B1 Medical devices containing rapamycin analogs |
08/04/2010 | CN101792452A Preparation method of high-purity antofloxacin hydrochloride |
08/03/2010 | US7767823 washing, crystallizing |
08/03/2010 | US7767702 Combinations of oxazolidinones such as rivaroxaban with a platelet aggregation inhibitor such as a clopidogrel for the prophylaxis and/or treatment of thromboembolic disorders |
08/03/2010 | US7767663 Soluble 17-amino-analogs of geldanamycin in acid addition salt form; water solubility; anticancer agents; storage stability |
08/03/2010 | US7767662 17-amino analogs of geldanamycin, used for treating and modulating disorders associated with hyperproliferation, such as cancer; antiproliferative and anticarcinogenic agents |
08/03/2010 | CA2204748C Use of dioxomorpholines for combating endoparasites, new dioxomorpholines and processes for their preparation |
07/29/2010 | WO2010085684A1 Compositions and methods for inhibition of the jak pathway |
07/29/2010 | WO2010085570A1 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors |
07/29/2010 | WO2010084501A1 A method for determination of sirolimus stability and process for preparing its stable form |
07/29/2010 | WO2010042925A3 Compositions and methods for treating alcohol use disorders, pain and other diseases |
07/29/2010 | US20100190804 Macrocyclic compounds and their use as kinase inhibitors |
07/29/2010 | US20100190786 Indolin-2-ones and aza-indolin-2-ones |
07/29/2010 | US20100190768 Novel fused pyrole derivative |
07/29/2010 | US20100190763 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors |
07/29/2010 | US20100190745 Heterocyclic urea derivatives and methods of use thereof |