Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
---|
04/14/2010 | CN1360592B Streptogramin derivs., production thereof and composition containing same |
04/13/2010 | US7696195 Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions |
04/13/2010 | US7695930 Method for the detection, identification and/or quantification of microoganisms with peptidase activity using phenoxazinone derivatives as enzyme substrates |
04/13/2010 | CA2432303C Pyrazole compounds useful as protein kinase inhibitors |
04/13/2010 | CA2422377C Pyrazole compounds useful as protein kinase inhibitors |
04/08/2010 | WO2010040020A1 Methods of treating hepatic encephalopathy |
04/08/2010 | WO2010037225A1 Heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
04/08/2010 | US20100087429 Spiro-tricyclic ring compounds as beta-secretase modulators and methods of use |
04/08/2010 | US20100087424 Tricyclic nitrogen containing heterocycles as antibacterial agents |
04/08/2010 | US20100087326 Heterocylic compounds containing the morpholine nucleus their preparation and use |
04/08/2010 | DE19820157B4 Neue Verbindungen auf Basis von Polyalkyl-1-oxa-diazaspirodecan-Verbindungen New connections based on polyalkyl-1-oxa-diazaspirodecan connections |
04/08/2010 | CA2739436A1 Methods of treating hepatic encephalopathy |
04/08/2010 | CA2738348A1 Heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
04/07/2010 | EP2170904A1 Process for preparing amorphous rifaximin and the amorphous rifaximin thus obtained |
04/07/2010 | EP2170807A1 Spiro compounds useful as antagonists of the h1 receptor |
04/07/2010 | EP2007771B1 Imidazo compounds |
04/07/2010 | EP1590340B1 Inhibitors of histone deacetylase |
04/06/2010 | US7691857 3-Benzyl-3a-cyclobutyl-7-methoxymethyl-2-oxo-octahydro-oxazolo[4,5-c]pyridin-5-ium; useful as agents for stimulating the cognitive functions of the brain |
04/06/2010 | US7691853 Pyrazole compounds useful as protein kinase inhibitors |
04/06/2010 | US7691851 increased potency and selectivity in relation to currently known MMP-13 inhibitors; treating rheumatoid arthritis, osteoarthritis or inflammation; modified benzoxazine moiety |
04/06/2010 | US7691840 Analogs of benzoquinone-containing ansamycins and methods of use thereof |
04/06/2010 | CA2566108C Proline derivatives and their use as dipeptidyl peptidase iv inhibitors |
04/01/2010 | WO2010036921A2 Slow release of organoboronic acids in cross-coupling reactions |
04/01/2010 | WO2010036871A1 Macrocyclic compounds as hepatitis c virus inhibitors |
04/01/2010 | WO2010036551A1 Hepatitis c virus inhibitors |
04/01/2010 | WO2010034740A1 (r)-3-(n,n-dimethylamino)pyrrolidine derivatives |
04/01/2010 | WO2010034656A1 Isoxazolo[4,5]pyridin-3-yl-piperazin derivatives useful as modulatorsof dopamine d3 receptors |
04/01/2010 | WO2010034243A1 Novel gene cluster |
04/01/2010 | US20100081682 39-Desmethoxy Derivatives of Rapamycin |
04/01/2010 | US20100081654 Oncogenic-RAS-signal dependent lethal compounds |
04/01/2010 | US20100081650 Antimicrobial Compounds |
04/01/2010 | US20100080771 Hepatitis C Virus Inhibitors |
04/01/2010 | US20100080770 Hepatitis C Virus Inhibitors |
04/01/2010 | CA2737252A1 Isoxazolo[4,5]pyridin-3-yl-piperazin derivatives useful as modulators of dopamine d3 receptors |
03/31/2010 | EP2168972A2 Preparation and use of carbohydrate-based ring structures with antimicrobial and cytostatic activity |
03/31/2010 | EP2167508A1 Compounds for treating duchenne muscular dystrophy |
03/31/2010 | EP2167494A1 3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives |
03/31/2010 | EP2167484A2 Condensed anthranilamide insecticides |
03/31/2010 | EP2166846A1 Inhibitors of janus kinases |
03/31/2010 | CN101687884A macrolactone derivatives |
03/31/2010 | CN101687871A Spiro condensed barbituric acid derivatives for use as antibacterial |
03/31/2010 | CN101687861A Pyrazoles useful in the treatment of inflammation |
03/30/2010 | US7687627 Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy |
03/25/2010 | WO2010031251A1 Rapamycin carbonic ester analogues, pharmaceutical compositions, preparations and uses thereof |
03/25/2010 | WO2010008777A3 Fused azabicyclic pyridines |
03/25/2010 | US20100075994 Substituted dihydro and tetrahydro oxazolopyrimidinones, preparation and use thereof |
03/25/2010 | CA2737355A1 Rapalogs, pharmaceutical compositions, preparation methods and uses thereof |
03/24/2010 | EP1615699B1 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |
03/24/2010 | CN101679455A New progesterone receptor modulators |
03/24/2010 | CN101679454A Antimicrobial heterocyclic compounds for treatment of bacterial infections |
03/24/2010 | CN101679453A New process for preparing 3-methyl-4-phenylisoxazolo[3,4-d]pyridazin-7(6H)-one |
03/24/2010 | CN101679405A 2-aminopyridine analogs as glucokinase activators |
03/24/2010 | CN101679401A 2-oxo-3-benzyl-benzoxazol-2-one derivatives and related compounds as MET kinase inhibitors for the treatment of tumors |
03/24/2010 | CN101679348A 5-pyridinone substituted indazoles |
03/24/2010 | CN101679339A Method for manufacturing neuraminic acid derivatives |
03/24/2010 | CN101679257A Process and intermediates for the synthesis of 8-[{1-(3,5-bis-(trifluoromethyl)phenyl)-ethoxy}-methyl]-8-phenyl-1,7-diaza-spiro[4.5]decan-2-one compounds |
03/24/2010 | CN101676291A Rapamycin carbonate analog, pharmaceutical composition thereof, and preparation method and uses thereof |
03/24/2010 | CN101676290A Levofloxacin salt, and preparation method thereof and medicament composition |
03/23/2010 | US7683164 Nucleic acid derivatives |
03/23/2010 | US7683056 Pyridine derivatives and their use in the treatment of psychotic disorders |
03/23/2010 | US7682387 Drug-delivery endovascular stent and method for treating restenosis |
03/23/2010 | CA2460177C 3-substituted-4-pyrimidone derivatives |
03/18/2010 | WO2010030954A1 Spiro-tetracyclic ring compounds as betasecretase modulators and methods of use |
03/18/2010 | WO2010029379A1 Compounds for inhibiting semicarbazide-sensitive amine oxidase (ssao) / vascular adhesion protein-1 (vap-1) and uses thereof for treatment and prevention of diseases |
03/18/2010 | WO2010003133A3 Cdk modulators |
03/18/2010 | WO2009126806A3 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene a4 hydrolase |
03/18/2010 | US20100069424 3-cyano-quinoline derivatives with antiproliferative activity |
03/18/2010 | US20100069376 5-hydroxymethyl-oxazolidin-2-one antibacterials |
03/18/2010 | US20100069374 Tricyclic benzopyrane compound |
03/18/2010 | US20100069360 Organic compounds |
03/18/2010 | CA2736130A1 Spiro-tetracyclic ring compounds as beta-secretase modulators and methods of use |
03/17/2010 | EP1948666B1 Hiv integrase inhibitors |
03/17/2010 | CN101675060A Substituted dihydro and tetrahydro oxazolopyrimidinones, preparation and use thereof |
03/17/2010 | CN101675044A Epoxy compound and method for manufacturing the same |
03/16/2010 | US7678903 Preparation of levofloxacin hemihydrate free of levofloxacin monohydrate by reacting (S)-(-) 9,10-difluoro-3-methyl-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4] benzoxazine-6-carboxylic acid with N-methyl piperazine to yield crude levofloxacin which is suspended in isopropanol, adding water, precipitating |
03/16/2010 | US7678901 Rapamycin analogs containing an antioxidant moiety |
03/16/2010 | US7678802 Voltage gated sodium and calcium channel inhibitors |
03/16/2010 | US7678791 4-Deoxy-3,4-[2-spiro-[1-[2-(2-methyl-5-nitro-imidazol-1-yl)ethyl]-piperidin-4-yl]]-(1H)-imidazo-(2,5-dihydro)rifamycin; antibiotic resistance; synergistic effects of covalently linking antibacterial pharmacophores together; pharmacokinetics; aerobic, anaerobic gram-positive and gram-negative bacteria |
03/16/2010 | CA2512683C Tricyclic compounds protein kinase inhibitors for enhancing the efficacy of anti-neoplastic agents and radiation therapy |
03/11/2010 | WO2010028232A1 Process and intermediates for the synthesis of 8-[{1-(3,5-bis-(trifluoromethyl)phenyl)-ethoxy}-methyl]-8-phenyl-1,7-diaza-spiro[4.5]decan-2-one compounds |
03/11/2010 | WO2010028116A1 Macrocyclics pyrimidines as aurora kinase inhibitors |
03/11/2010 | WO2010027567A2 Tricyclic spirocycle derivatives and methods of use thereof |
03/11/2010 | WO2010027002A1 Ring-fused morpholine derivative having pi3k-inhibiting activity |
03/11/2010 | US20100063041 Novel phenylpropionic acid derivatives as peroxisome proliferator-activated gamma receptor modulators, method of the same, and pharmaceutical composition comprising the same |
03/11/2010 | US20100061982 3-substituted-1h-indole, 3-substituted-1h-pyrrolo[2,3-b]pyridine and 3-substituted-1h-pyrrolo[3,2-b]pyridine compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses |
03/11/2010 | CA2736195A1 Process and intermediates for the synthesis of 8-[{1-(3,5-bis-(trifluoromethyl)phenyl)-ethoxy}-methyl]-8-phenyl-1,7-diaza-spiro[4.5]decan-2-one compounds |
03/11/2010 | CA2735775A1 6-substituted benzoxazines |
03/11/2010 | CA2735420A1 Macrocyclic pyrimidines as protein kinase inhibitors |
03/10/2010 | EP2161275A1 Prodrugs of 2,4-pyrimidinediamine compounds and their uses |
03/10/2010 | EP2161239A1 Semiconductor nanocrystals |
03/10/2010 | CN101665498A Organic compounds |
03/04/2010 | US20100056605 Oxidative degradation products of atorvastatin calcium |
03/04/2010 | US20100056509 Heteroaryl sulfonamides and ccr2 |
03/04/2010 | US20100056502 Compounds |
03/03/2010 | EP2159216A1 Ih - Modulators |
03/03/2010 | CN101659669A Method for preparing levofloxacin |
03/02/2010 | US7671079 Sulfonyltetrahydro-3H-benzo(e)indole-8-amine compounds as 5-hydroxytryptamine-6 ligands |
03/02/2010 | US7671068 N-(alkoxyalkyl) carbamoyl-substituted 6-phenyl-benzonaphthyridine derivatives and their use as PDE ¾ inhibitors |
02/25/2010 | WO2010020548A1 Glyt1 receptor antagonists |
02/25/2010 | WO2004092124A8 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |