Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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08/22/2000 | US6107482 Nitrogenous macrocyclic compounds |
08/22/2000 | US6107310 Heteroarylcarboxamide derivatives for treating CNS disorders |
08/22/2000 | US6107304 Anemia |
08/22/2000 | CA2143246C Imidazodiazepines |
08/22/2000 | CA2020554C Process for the control of sea lice |
08/17/2000 | WO2000047585A1 3-hydroxy-4-aryl-5-pyrazoline derivatives as herbicides |
08/17/2000 | WO2000009109A3 Pipecolic acid derivatives for vision and memory disorders |
08/16/2000 | EP1027341A1 High char yield benzoxazines |
08/16/2000 | EP1026950A1 Treatment of schizophrenia with ampakines and neuroleptics |
08/16/2000 | CN1263527A Cis-disubstituted aminocycloalykyl-pyrrolidine derivatives |
08/16/2000 | CN1055472C Oxazolo quinolyl-one derivatives, their preparation method and application and use as medicine |
08/15/2000 | US6103899 Bicyclic aminoimidazoles |
08/15/2000 | US6103723 Inhibitors of farnesyl-protein transferase |
08/15/2000 | US6103716 Bactericides; administering my mouth to mammals and humans; prophylaxis; cattle, sheep, swine, poultry |
08/15/2000 | US6103712 Selective inhibitors of the beta isozyme of protein kinase c inhibits pulmonary vascular permeability, bronchial smooth muscle contractility, and airway hyperactivity, e.g. bisindolylmaleimides |
08/10/2000 | WO2000046225A2 Pyridobenzodiazepine and pyridobenzoxazepine carboxyamide vasopressin agonists |
08/10/2000 | WO2000046223A1 Tricyclic quinolonecarboxylic acid derivatives or salts thereof |
08/10/2000 | DE19905278A1 Oxazolidinone und ihre Verwendung als antibakterielle Mittel Oxazolidinones and their use as antibacterial agents |
08/10/2000 | CA2358895A1 Pyridobenzodiazepine and pyridobenzoxazepine carboxyamide vasopressin agonists |
08/09/2000 | EP1025108A1 Photochromic spiro(indoline) fluoranthenoxazine compounds |
08/09/2000 | EP1025107A1 Photochromic compounds |
08/09/2000 | EP1025105A1 Condensed benzothiopyranic compounds |
08/09/2000 | CN1262679A IL-5 inhibiting 6-azauracil derivatives |
08/09/2000 | CN1055288C Cation-sensing composite structure and compounds for use therein |
08/08/2000 | US6100397 Process for the preparation of N-[(1-n butyl-4-piperidyl)methyl]-3,4-dihydro-2H-[1,3]oxazino[3,2-a] indole-10-carboxamide and salts and intermediates in the process |
08/08/2000 | US6100246 Spiro-piperidine derivatives as inhibitors of nitric oxide synthase |
08/03/2000 | WO2000044749A1 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as tace inhibitors |
08/03/2000 | WO2000044728A1 Substituted bicyclic derivatives useful as anticancer agents |
08/03/2000 | WO1999064379A3 Biomimetic combinatorial synthesis |
08/03/2000 | CA2355735A1 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as tace inhibitors |
08/02/2000 | EP1023297A1 A process for the preparation of aminocarbonyl derivatives of geneseroline having selective brain anticholinesterase activity |
08/02/2000 | EP1023270A1 Inhibitors of farnesyl-protein transferase |
08/02/2000 | CN1055089C Intermediate of protein kinase C inhibitor and its preparation |
08/01/2000 | US6096771 Isoxazole derivatives |
08/01/2000 | US6096751 Substituted 1,2,3,4-tetrahydro-55-nitro-pyrimidines |
08/01/2000 | US6096749 Pyrrolopyrimidine derivatives having pharmacological activity |
08/01/2000 | US6096724 O(6)-alkylguanine-dna alkyltransferase (atase) enzyme inhibitors |
07/27/2000 | WO2000043398A2 Tricyclic benzodiazepines as vasopressin receptor antagonists |
07/27/2000 | WO2000043375A2 Substituted aryl heterocyclic compounds |
07/27/2000 | WO1999064033A9 Phosphodiesterase-v modulator drugs and their uses |
07/27/2000 | WO1999063994A9 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE |
07/26/2000 | EP1021415A1 Tricyclic aminoalkylcarboxamides; novel dopamine d 3? receptor subtype specific ligands |
07/26/2000 | EP1021413A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors |
07/26/2000 | EP1021190A1 Novel amide derivatives |
07/26/2000 | CN1261365A Crystalline macrolides and process for their preparation |
07/26/2000 | CN1261284A Use of a CD40 : CD154 binding interruptor to prevent counter adaptive immune responses, particularly graft rejection |
07/25/2000 | US6093726 Bicyclic amine derivatives |
07/25/2000 | US6093713 A tyrosine kinase inhibitor for enhancing the function of a cholinergic neuron |
07/25/2000 | US6093709 Administering a therapeutic beta isozyme of protein kinase c inhibitor for inducing smooth muscle relaxation and vasodilation |
07/20/2000 | WO2000042030A1 Hypolipidemic and antioxidant morpholine derivatives |
07/20/2000 | WO2000041474A2 Anti-cd3 immunotoxins and therapeutic uses therefor |
07/20/2000 | WO1999064048A9 Inhibitors of hiv reverse transcriptase |
07/20/2000 | DE19901846A1 New aryl-substituted aza-heterocyclic compounds, useful as pre- or post-emergence, total or selective herbicides, show defoliant, dessicant and especially weed-killing activity |
07/20/2000 | DE19901306A1 New N-(imidazo-tetrahydrobenzazepinyl)-1,3-oxazolidin-2-ones, useful as broad-spectrum antibacterial agents having low toxicity |
07/20/2000 | CA2359365A1 Anti-cd3 immunotoxins and therapeutic uses therefor |
07/19/2000 | EP1020471A1 Process for producing UCN-01 |
07/19/2000 | EP1020467A1 N-acylamino acid amide compounds and intermediates for preparation thereof |
07/19/2000 | EP1020459A1 Cis-disubstituted aminocycloalkyl-pyrrolidine derivatives |
07/19/2000 | EP1020451A1 Novel anilide compounds and drugs containing the same |
07/19/2000 | EP1019412A1 Biphenyl(thio)amide and biphenylethan(thi)one derivatives, their preparation and their use as 5-ht 1d? receptor antagonists |
07/19/2000 | EP1019409A1 Poly(adp-ribose) polymerase ("parp") inhibitors, methods and pharmaceutical compositions for treating neural or cardiovascular tissue damage |
07/19/2000 | EP1019408A1 1,2,3,4-TETRAHYDRO-BENZOFURO 3,2-c]PYRIDINE DERIVATIVES-- |
07/19/2000 | EP1019389A2 Epothilone derivatives |
07/19/2000 | EP1019382A1 Compounds and compositions for treating diseases associated with serine protease, particularly tryptase, activity |
07/19/2000 | EP1019380A2 Tricyclic 3-oxo-propanenitrile compounds |
07/19/2000 | EP0760819B1 Tricyclic dicarbonyl derivatives |
07/13/2000 | WO2000040569A1 2-amino-benzoxazinone derivatives for the treatment of obesity |
07/13/2000 | WO2000040247A1 2-oxy-benzoxazinone derivatives for the treatment of obesity |
07/13/2000 | WO2000040228A2 Formulations comprising imiquimod or other immune response modifiers for treating mucosal conditions |
07/13/2000 | WO2000015208A3 New use of immunosupressants for mmp-mediated diseases |
07/12/2000 | EP1018514A1 NF-$g(k)B INHIBITORS CONTAINING INDAN DERIVATIVES AS THE ACTIVE INGREDIENT |
07/12/2000 | EP1017695A1 Resolution of optically-active compounds |
07/12/2000 | EP0783910B1 Process for the vacuum distillation of crude petroleum, and a facility for carrying out the process |
07/12/2000 | EP0561850B1 7-substituted-6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid compounds useful as antibacterial agents |
07/12/2000 | CN1259942A Novel guanidine mimics as factor Xa inhibitors |
07/12/2000 | CN1054380C Condensed cyclic compounds and their use |
07/11/2000 | US6087358 Bactericides treating pathogenic infections of mycobacteria, clostridium, cryptosporidium or helicobacter and multidrug-resistant tuberculosis |
07/06/2000 | WO2000039245A1 Photochromatic compounds, process for their preparation and their use in polymeric materials |
07/06/2000 | WO2000039125A1 Piperidines as ccr5 modulators |
07/06/2000 | WO2000039108A1 Thrombin or factor xa inhibitors |
07/06/2000 | WO2000039102A1 THROMBIN OR FACTOR Xa INHIBITORS |
07/06/2000 | WO2000038683A1 THROMBIN OR FACTOR Xa INHIBITORS |
07/06/2000 | WO2000038680A1 Azabicycloalkanes as ccr5 modulators |
07/06/2000 | CA2349557A1 Thrombin or factor xa inhibitors |
07/06/2000 | CA2348740A1 Thrombin or factor xa inhibitors |
07/06/2000 | CA2320730A1 Thrombin or factor xa inhibitors |
07/05/2000 | EP1016664A1 Fused thiophene compounds and medicinal use thereof |
07/05/2000 | EP1015459A1 Tetrazole-containing rapamycin analogs with shortened half-lives |
07/05/2000 | EP1015448A1 Anti-cancer drug aldehyde conjugate drugs with enhanced cytotoxicity: compounds, compositions and methods |
07/05/2000 | EP1015437A1 Benzoxazine and benzothiazine derivatives and their use in pharmaceuticals |
07/05/2000 | EP1015427A1 Substituted 2-pyrrolidinone activators of pkc |
07/05/2000 | EP0711296B1 IMIDAZOLYLALKYL DERIVATIVES OF IMIDAZOL[5,1-c][1,4]BENZOXAZIN-1-ONE AND THEIR USE AS THERAPEUTIC AGENTS |
07/05/2000 | CN1259132A Compounds |
07/04/2000 | US6084095 Including 6-amino-4-(3-bromoanilino)pyrido(3,2-d)pyrimidine; 4-(3-bromoanilino)-6-methylaminopyrido (3,2-d)pyrimidine; and 4-(3-bromoanilino)-6-methylaminopyrido(3,2-d)pyrimidine; useful in treating proliferative diseases such as cancer |
07/04/2000 | US6083961 For prevention and/or treatment of bradykinin or its analogues mediated diseases such as allergy, inflammation, autoimmune disease, shock, pain |
07/04/2000 | CA1341043C Piperazinyl derivatives of purines and isosteres thereof as hypoglycemic agents |
06/29/2000 | WO2000037470A1 Antihistaminic spiro compounds |
06/29/2000 | WO2000037021A2 Products comprising trihydroxystilbenes and derivatives thereof and methods for their manufacture and use |
06/29/2000 | CA2394949A1 Products comprising trihydroxystilbenes and derivatives thereof and methods for their manufacture and use |
06/28/2000 | EP1013276A1 Aminoazacycloalkanes as CCR5 modulators |