Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
08/2000
08/22/2000US6107482 Nitrogenous macrocyclic compounds
08/22/2000US6107310 Heteroarylcarboxamide derivatives for treating CNS disorders
08/22/2000US6107304 Anemia
08/22/2000CA2143246C Imidazodiazepines
08/22/2000CA2020554C Process for the control of sea lice
08/17/2000WO2000047585A1 3-hydroxy-4-aryl-5-pyrazoline derivatives as herbicides
08/17/2000WO2000009109A3 Pipecolic acid derivatives for vision and memory disorders
08/16/2000EP1027341A1 High char yield benzoxazines
08/16/2000EP1026950A1 Treatment of schizophrenia with ampakines and neuroleptics
08/16/2000CN1263527A Cis-disubstituted aminocycloalykyl-pyrrolidine derivatives
08/16/2000CN1055472C Oxazolo quinolyl-one derivatives, their preparation method and application and use as medicine
08/15/2000US6103899 Bicyclic aminoimidazoles
08/15/2000US6103723 Inhibitors of farnesyl-protein transferase
08/15/2000US6103716 Bactericides; administering my mouth to mammals and humans; prophylaxis; cattle, sheep, swine, poultry
08/15/2000US6103712 Selective inhibitors of the beta isozyme of protein kinase c inhibits pulmonary vascular permeability, bronchial smooth muscle contractility, and airway hyperactivity, e.g. bisindolylmaleimides
08/10/2000WO2000046225A2 Pyridobenzodiazepine and pyridobenzoxazepine carboxyamide vasopressin agonists
08/10/2000WO2000046223A1 Tricyclic quinolonecarboxylic acid derivatives or salts thereof
08/10/2000DE19905278A1 Oxazolidinone und ihre Verwendung als antibakterielle Mittel Oxazolidinones and their use as antibacterial agents
08/10/2000CA2358895A1 Pyridobenzodiazepine and pyridobenzoxazepine carboxyamide vasopressin agonists
08/09/2000EP1025108A1 Photochromic spiro(indoline) fluoranthenoxazine compounds
08/09/2000EP1025107A1 Photochromic compounds
08/09/2000EP1025105A1 Condensed benzothiopyranic compounds
08/09/2000CN1262679A IL-5 inhibiting 6-azauracil derivatives
08/09/2000CN1055288C Cation-sensing composite structure and compounds for use therein
08/08/2000US6100397 Process for the preparation of N-[(1-n butyl-4-piperidyl)methyl]-3,4-dihydro-2H-[1,3]oxazino[3,2-a] indole-10-carboxamide and salts and intermediates in the process
08/08/2000US6100246 Spiro-piperidine derivatives as inhibitors of nitric oxide synthase
08/03/2000WO2000044749A1 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as tace inhibitors
08/03/2000WO2000044728A1 Substituted bicyclic derivatives useful as anticancer agents
08/03/2000WO1999064379A3 Biomimetic combinatorial synthesis
08/03/2000CA2355735A1 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as tace inhibitors
08/02/2000EP1023297A1 A process for the preparation of aminocarbonyl derivatives of geneseroline having selective brain anticholinesterase activity
08/02/2000EP1023270A1 Inhibitors of farnesyl-protein transferase
08/02/2000CN1055089C Intermediate of protein kinase C inhibitor and its preparation
08/01/2000US6096771 Isoxazole derivatives
08/01/2000US6096751 Substituted 1,2,3,4-tetrahydro-55-nitro-pyrimidines
08/01/2000US6096749 Pyrrolopyrimidine derivatives having pharmacological activity
08/01/2000US6096724 O(6)-alkylguanine-dna alkyltransferase (atase) enzyme inhibitors
07/2000
07/27/2000WO2000043398A2 Tricyclic benzodiazepines as vasopressin receptor antagonists
07/27/2000WO2000043375A2 Substituted aryl heterocyclic compounds
07/27/2000WO1999064033A9 Phosphodiesterase-v modulator drugs and their uses
07/27/2000WO1999063994A9 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE
07/26/2000EP1021415A1 Tricyclic aminoalkylcarboxamides; novel dopamine d 3? receptor subtype specific ligands
07/26/2000EP1021413A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
07/26/2000EP1021190A1 Novel amide derivatives
07/26/2000CN1261365A Crystalline macrolides and process for their preparation
07/26/2000CN1261284A Use of a CD40 : CD154 binding interruptor to prevent counter adaptive immune responses, particularly graft rejection
07/25/2000US6093726 Bicyclic amine derivatives
07/25/2000US6093713 A tyrosine kinase inhibitor for enhancing the function of a cholinergic neuron
07/25/2000US6093709 Administering a therapeutic beta isozyme of protein kinase c inhibitor for inducing smooth muscle relaxation and vasodilation
07/20/2000WO2000042030A1 Hypolipidemic and antioxidant morpholine derivatives
07/20/2000WO2000041474A2 Anti-cd3 immunotoxins and therapeutic uses therefor
07/20/2000WO1999064048A9 Inhibitors of hiv reverse transcriptase
07/20/2000DE19901846A1 New aryl-substituted aza-heterocyclic compounds, useful as pre- or post-emergence, total or selective herbicides, show defoliant, dessicant and especially weed-killing activity
07/20/2000DE19901306A1 New N-(imidazo-tetrahydrobenzazepinyl)-1,3-oxazolidin-2-ones, useful as broad-spectrum antibacterial agents having low toxicity
07/20/2000CA2359365A1 Anti-cd3 immunotoxins and therapeutic uses therefor
07/19/2000EP1020471A1 Process for producing UCN-01
07/19/2000EP1020467A1 N-acylamino acid amide compounds and intermediates for preparation thereof
07/19/2000EP1020459A1 Cis-disubstituted aminocycloalkyl-pyrrolidine derivatives
07/19/2000EP1020451A1 Novel anilide compounds and drugs containing the same
07/19/2000EP1019412A1 Biphenyl(thio)amide and biphenylethan(thi)one derivatives, their preparation and their use as 5-ht 1d? receptor antagonists
07/19/2000EP1019409A1 Poly(adp-ribose) polymerase ("parp") inhibitors, methods and pharmaceutical compositions for treating neural or cardiovascular tissue damage
07/19/2000EP1019408A1 1,2,3,4-TETRAHYDRO-BENZOFURO 3,2-c]PYRIDINE DERIVATIVES--
07/19/2000EP1019389A2 Epothilone derivatives
07/19/2000EP1019382A1 Compounds and compositions for treating diseases associated with serine protease, particularly tryptase, activity
07/19/2000EP1019380A2 Tricyclic 3-oxo-propanenitrile compounds
07/19/2000EP0760819B1 Tricyclic dicarbonyl derivatives
07/13/2000WO2000040569A1 2-amino-benzoxazinone derivatives for the treatment of obesity
07/13/2000WO2000040247A1 2-oxy-benzoxazinone derivatives for the treatment of obesity
07/13/2000WO2000040228A2 Formulations comprising imiquimod or other immune response modifiers for treating mucosal conditions
07/13/2000WO2000015208A3 New use of immunosupressants for mmp-mediated diseases
07/12/2000EP1018514A1 NF-$g(k)B INHIBITORS CONTAINING INDAN DERIVATIVES AS THE ACTIVE INGREDIENT
07/12/2000EP1017695A1 Resolution of optically-active compounds
07/12/2000EP0783910B1 Process for the vacuum distillation of crude petroleum, and a facility for carrying out the process
07/12/2000EP0561850B1 7-substituted-6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid compounds useful as antibacterial agents
07/12/2000CN1259942A Novel guanidine mimics as factor Xa inhibitors
07/12/2000CN1054380C Condensed cyclic compounds and their use
07/11/2000US6087358 Bactericides treating pathogenic infections of mycobacteria, clostridium, cryptosporidium or helicobacter and multidrug-resistant tuberculosis
07/06/2000WO2000039245A1 Photochromatic compounds, process for their preparation and their use in polymeric materials
07/06/2000WO2000039125A1 Piperidines as ccr5 modulators
07/06/2000WO2000039108A1 Thrombin or factor xa inhibitors
07/06/2000WO2000039102A1 THROMBIN OR FACTOR Xa INHIBITORS
07/06/2000WO2000038683A1 THROMBIN OR FACTOR Xa INHIBITORS
07/06/2000WO2000038680A1 Azabicycloalkanes as ccr5 modulators
07/06/2000CA2349557A1 Thrombin or factor xa inhibitors
07/06/2000CA2348740A1 Thrombin or factor xa inhibitors
07/06/2000CA2320730A1 Thrombin or factor xa inhibitors
07/05/2000EP1016664A1 Fused thiophene compounds and medicinal use thereof
07/05/2000EP1015459A1 Tetrazole-containing rapamycin analogs with shortened half-lives
07/05/2000EP1015448A1 Anti-cancer drug aldehyde conjugate drugs with enhanced cytotoxicity: compounds, compositions and methods
07/05/2000EP1015437A1 Benzoxazine and benzothiazine derivatives and their use in pharmaceuticals
07/05/2000EP1015427A1 Substituted 2-pyrrolidinone activators of pkc
07/05/2000EP0711296B1 IMIDAZOLYLALKYL DERIVATIVES OF IMIDAZOL[5,1-c][1,4]BENZOXAZIN-1-ONE AND THEIR USE AS THERAPEUTIC AGENTS
07/05/2000CN1259132A Compounds
07/04/2000US6084095 Including 6-amino-4-(3-bromoanilino)pyrido(3,2-d)pyrimidine; 4-(3-bromoanilino)-6-methylaminopyrido (3,2-d)pyrimidine; and 4-(3-bromoanilino)-6-methylaminopyrido(3,2-d)pyrimidine; useful in treating proliferative diseases such as cancer
07/04/2000US6083961 For prevention and/or treatment of bradykinin or its analogues mediated diseases such as allergy, inflammation, autoimmune disease, shock, pain
07/04/2000CA1341043C Piperazinyl derivatives of purines and isosteres thereof as hypoglycemic agents
06/2000
06/29/2000WO2000037470A1 Antihistaminic spiro compounds
06/29/2000WO2000037021A2 Products comprising trihydroxystilbenes and derivatives thereof and methods for their manufacture and use
06/29/2000CA2394949A1 Products comprising trihydroxystilbenes and derivatives thereof and methods for their manufacture and use
06/28/2000EP1013276A1 Aminoazacycloalkanes as CCR5 modulators