Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
10/1999
10/14/1999CA2327617A1 Methods for inhibiting mrp1
10/14/1999CA2327452A1 Methods for inhibiting mrp1
10/13/1999CN1231608A Use of PKC inhibitors for the manufacture of a medicament for the treatment of HTLV-1 infections
10/13/1999CN1231607A Use of inhibitors of PKG for the manufacture of a medicament for the treatment of central nervous system diseases associated with HIV infection
10/12/1999US5965591 Monoamine oxidase inhibitor; for prophylaxis and treating parkinson's disease, depression and alzheimer's disease
10/07/1999WO1999050244A1 Nitroxide free radical dual indicator agents
10/07/1999WO1999049863A1 Sustained release preparations
10/06/1999EP0947513A1 Tricyclic amine derivatives
10/06/1999EP0946689A1 Antioxidants and antioxidant boosters capable of producing hydroperoxyl radicals
10/06/1999EP0946567A1 Novel counterparts of camptothecin, their application as medicine and pharmaceutical compositions containing them
10/06/1999EP0946566A1 Pro-drugs and counterparts of camptothecin, their application as medicines
10/06/1999EP0946553A1 8-azabicyclo 3.2.1]octane derivatives, their preparation and their use as insecticides
10/06/1999EP0946176A1 The use of 7-(2-oxa-5,8-diazabicyclo 4.3.0]non-8-yl)-quinolone carboxylic acid and naphthyridon carboxylic acid derivatives for the treatment of helicobacter pylori infections and associated gastroduodenal diseases
10/05/1999US5962504 Activator of protein kinase; anticancer agent
10/05/1999US5962447 Psychological disorders, cognition activators, schizophrenia
10/05/1999US5962446 Administering protein kinase inhibitors
09/1999
09/30/1999WO1999048461A2 Substituted aromatic compounds for treatment of antibiotic resistant infections
09/30/1999CA2325689A1 Substituted aromatic compounds for treatment of antibiotic resistant infections
09/29/1999EP0945455A1 Thriphendioxazine pigments
09/29/1999EP0944627A1 8-azabicyclo 3.2.1]octane-, 8-azabicyclo 3.2.1]oct-6-ene-, 9-azabicyclo 3.3.1]nonane-, 9-aza-3-oxabicyclo 3.3.1]nonane- and 9-aza-3-thiabicyclo 3.3.1]nonane derivatives, their preparation and their use as insecticides
09/29/1999EP0944625A1 8-azabicyclo 3.2.1]octane-, 8-azabicyclo 3.2.1]oct-6-ene-, 9-azabicyclo 3.3.1]nonane-, 9-aza-3-oxabicyclo 3.3.1]nonane-, 9-aza-3-thiabicyclo 3.3.1]nonane derivatives, their preparation and their use as insecticides
09/29/1999EP0944311A1 Heregulin antagonists and methods for their use
09/29/1999EP0573573B1 Mesogenic glycidyl amines
09/29/1999CN1230211A Antioxidants and antioxidant boosters capable of producing hydroperoxyl radicals
09/29/1999CN1230179A Prepn. of 1-butyl-4-piperidinylmethylamine
09/28/1999US5958959 Administering 5-methylisoxazole-4-carboxylic acid-(4-trifluoromethyl)anilide or 2-cyano-3-hydroxy-n-(4-(trifluoromethyl)phenyl)-2-butenamide
09/28/1999US5958943 A!-anellated pyrrole derivatives and their use in pharmacology
09/28/1999US5958782 Cation-sensing composite structure and compounds for use therein
09/23/1999WO1999047525A1 Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
09/23/1999WO1999047524A1 Novel heterocyclic compounds
09/23/1999WO1999047522A1 Granulatimide derivatives for use in cancer treatment
09/23/1999WO1999047490A1 Bicyclo[2.2.1]heptanes and related compounds
09/22/1999EP0943661A2 Chromophoric compounds and their preparation process
09/22/1999EP0942912A1 Antibacterial agents
09/22/1999CN1229438A Erythromycins and process for their preparation
09/22/1999CN1229412A Inhibitors of interleukin-1'beta' converting emzyme
09/22/1999CN1045206C Method for preparing cyclic amide derivative
09/21/1999US5955460 Oxazolidinone antibacterial agent with tricyclic substituents
09/21/1999US5955457 Water soluble rapamycin esters
09/21/1999CA2135751C 4-mercaptoacetylamino-¬2| benzazepinone(3) derivatives, and use as enkephalinase inhibitors
09/15/1999EP0656001B1 Novel 2-substituted indane-2-mercaptoacetylamide tricyclic derivatives useful as inhibitors of enkephalinase
09/15/1999EP0641339B1 Azaspiro quinolone antibacterial agents
09/14/1999US5952494 Method for the preparation of pyrido benzoxazine derivatives
09/14/1999US5952491 Method of determining an alkali ion
09/14/1999US5952335 Antitumor agents
09/14/1999US5952334 Carbocyclic compounds
09/14/1999CA2086924C Method for the preparation of sulphinyl pristinamycin iib
09/14/1999CA1340734C Substituted bridged-diazabicycloalkyl quinolone carboxylic acids
09/10/1999WO1999044612A1 Substituted quinazolines and analogs and the use thereof
09/10/1999WO1999044606A1 Use of pkc-inhibitors for the manufacture of a medicament for the treatment of asthma
09/10/1999WO1999044599A1 Therapeutic treatment for renal dysfunction
09/10/1999WO1999044597A2 Use of macrolide compounds for the treatment of ards
09/10/1999CA2323173A1 Use of pkc-inhibitors for the manufacture of a medicament for the treatment of asthma
09/10/1999CA2323172A1 Therapeutic treatment for renal dysfunction
09/08/1999EP0940143A2 Use of PKC-inhibitors for the manufacture of a medicament for the treatment of asthma
09/08/1999CN1228091A Substituted 6,6-hetero-bicyclic derivatives
09/08/1999CN1228082A Synthesis of bisindolylmalimides
09/08/1999CN1228024A Use of K-252A derivative for treatment of peripheral or central nerve disorders, and cytokine overproduction
09/07/1999US5948907 Synthesis of bisindolylmaleimides
09/07/1999US5948816 Non-tolerance-inducing antiviral agents
09/07/1999US5948811 Psychological disorders; parkinson's disease
09/07/1999CA1340721C 1,4-dihydro-quinoline-and naphthyridine-3-carboxylic acid antibacterial agents
09/01/1999CN1227553A Bicyclic pyrimidine derivatives and their use as anti-coagulants
09/01/1999CN1227552A Substituted pyrido- or pyrimido-containing 6,6- or 6,7-bicyclic derivatives
09/01/1999CN1227488A Improved method for preparing potassim clavulanate
08/1999
08/31/1999US5944854 Process for the preparation of triphendioxazine dyestuffs amidated on both sides, and novel triphendioxazine dyestuffs
08/26/1999WO1999042452A1 Phthalazine derivatives and remedies for erectile dysfunction
08/26/1999WO1999042104A1 Use of macrolide compounds for treating glaucoma
08/26/1999WO1999031060A3 Piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides as cytostatics and immunesuppressants
08/25/1999EP0937458A2 Pyrrolidine and piperidine derivatives
08/25/1999EP0937082A2 Materials and method for treating or preventing pathogenic fungal infection
08/25/1999EP0937075A1 New imidazopyridines and oxazolopyridines
08/25/1999EP0937042A1 Heteroaryl succinamides and their use as metalloproteinase inhibitors
08/25/1999CN1226893A Selected derivatives of K-252a
08/25/1999CN1226891A Processes for preparing indeno [1,2-E] (1,3,4) oxadiazine-dicarboxylates
08/24/1999US5942547 2-Deoxystreptamine derivatives, pharmaceutical compositions thereof and therapeutic methods using same
08/19/1999WO1999041276A1 β-SHEET MIMETICS AND METHODS RELATING TO THE USE THEREOF
08/19/1999WO1999041275A1 Prodrugs
08/19/1999WO1999041258A1 Novel dimerizing agents, their production and use
08/19/1999WO1999041252A1 Antagonists of gonadotropin releasing hormone
08/19/1999WO1999041245A1 Insecticidal dihydro-oxadiazines, -thiadiazines and -triazines
08/19/1999CA2319766A1 .beta.-sheet mimetics and methods relating to the use thereof
08/19/1999CA2319492A1 Novel dimerizing agents, their production and use
08/19/1999CA2318978A1 Prodrugs
08/19/1999CA2318957A1 Antagonists of gonadotropin releasing hormone
08/18/1999EP0935602A1 Pyrido (3,2,1-ij)-1,3,4-benzoxadiazine
08/17/1999US5939427 Lotion with 17-allyl-1,4-dihydroxy-12-(2-(4-hydroxy-3-methoxy cyclohexyl)-1-methylvinyl)-23,25-dimethoxy-13,19,21,27-tetrame thyl-11,28-dioxa-4-azatricyclo(22.3.1.0(4,9))octacos-18-ene-1, 3,10,16-tetraone or salt as antiinflammatory agent
08/17/1999US5939418 Isoxazoline, isothiazoline and pyrazoline factor Xa inhibitors
08/17/1999US5939415 A!-annellated pyrrole derivatives and their use in pharmacology
08/17/1999CA2142920C Sulfonamidodioxepanes, methods of preparation, intermediates, salts and use thereof
08/12/1999WO1999040094A1 Agent for sealing metallic ground coats, especially ground coats consisting of zinc or zinc alloys
08/12/1999WO1999040093A2 Synthesis of quinobenzoxazine analogues with topoisomerase ii and quadruplex interactions for use as antineoplastic agents
08/12/1999WO1999040089A1 Benzothiadiazoles and derivatives
08/12/1999WO1999026940A3 Method for producing 8-methoxy-quinoline carboxylic acids
08/12/1999WO1999002130A3 Storage-stable ophthalmic compositions comprising diclofenac and ofloxacin
08/12/1999DE19805117A1 Neue Oxazolidinone mit azolhaltigen Tricyclen Novel oxazolidinones with azole tricycles
08/12/1999CA2318977A1 Derivatives of benzoxadiazoles, benzothiadiazoles, benzotriazoles and quinoxalines
08/11/1999EP0934937A1 Azole derivatives as superoxide radical inhibitor
08/11/1999EP0934318A1 Novel 3, 5, and/or 6 substituted analogues of swainsonine, processes for their preparation and their use as therapeutic agents
08/11/1999EP0669127B1 Prolonged-action pharmaceutical preparation