Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
08/2001
08/02/2001WO2001005385A3 New use of a macrolide compound for treating neurodegenerative disorders
08/02/2001US20010010920 Complex of rapamycin-42 ester with dicarboxylic acid and fluorescein; antibody detection/generation; immunoglobulins; hybridomas; ring opening; precipitation
08/02/2001DE10004157A1 New pyridyl- or pyrimidinyl-substituted bicyclic pyrrole derivatives, are cyclokine release inhibitors useful for treating immune system-related disorders, e.g. cancer, multiple sclerosis or arthritis
08/02/2001DE10003287A1 Neue Isoxazolopyrimidinone und ihre Verwendung New Isoxazolopyrimidinone and their use
08/01/2001EP1120421A2 New triphendioxazine compounds
08/01/2001EP1120420A2 New triphendioxazine compounds
08/01/2001EP1120414A1 Disubstituted maleimide compounds and medicinal utilization thereof
08/01/2001EP1119568A1 4,5-dihydro-isoxazole derivatives and their pharmaceutical use
08/01/2001EP0719268B1 K-252a DERIVATIVES WHICH ENHANCE NEUROTROPHIN-INDUCED ACTIVITY
08/01/2001EP0625984B1 Cephalosporin compounds
08/01/2001CN1306526A Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
08/01/2001CN1306427A Acylbenzoxazines for enhancing synaptic response(s)
07/2001
07/31/2001US6268383 Containing a phenanthrene ring; e.g., desbutylhalofantrine.
07/31/2001CA2040774C Compounds formed from o-hydroxyphenyl-1,3,5-triazines and sterically hindered amines
07/26/2001WO2001053302A1 5H-QUINOXALINO[2,3-b]NAPHTHO[2,1][1,4]OXAZIN-5-ONE AND INTERMEDIATE FOR THE PREPARATION THEREOF
07/26/2001WO2001053273A1 3-aminoquinazolin-2,4-dione antibacterial agents
07/26/2001WO2001053262A1 Alpha v integrin receptor antagonists
07/26/2001WO2001018007A3 Method for separating lactone-containing high-molecular weight compounds
07/26/2001CA2397665A1 Alpha v integrin receptor antagonists
07/25/2001EP1117801A2 Polyketide synthase enzymes and recombinant dna constructs therefor
07/25/2001EP0794955B1 Hindered n-oxide esters of rapamycin and their use as medicaments
07/24/2001US6265418 N-acylamino acid amide compounds and intermediates for preparation thereof
07/24/2001US6265410 Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
07/24/2001CA2066191C Tricyclic ¬6,5,5|/¬6,6,5|-fused oxazolidinone antibacterial agents
07/19/2001WO2001051494A1 Inhibitors of prenyl-protein transferase
07/19/2001WO2001051128A1 Inhibitors of prenyl-protein transferase
07/19/2001WO2001051125A1 Inhibitors of prenyl-protein transferase
07/19/2001WO2001051049A1 O-methylated rapamycin derivatives for alleviation and inhibition of lymphoproliferative disorders
07/19/2001WO2000041474A3 Anti-cd3 immunotoxins and therapeutic uses therefor
07/18/2001CN1304311A Bridged indenopyrrolocarbazoles
07/18/2001CN1304306A Method for inhibiting MRP1
07/17/2001US6262257 Selective ion- and neutral molecule-binding agents forming supramolecular ensembles, and ion- and neutral molecule-separation agents
07/17/2001US6262098 Estrogen receptor modulators
07/17/2001US6262058 Pyrimidin-4-one derivatives as pesticide
07/12/2001WO2001049682A1 Condensed azepines as vasopressin agonists
07/12/2001WO2001049508A1 Benzbisazole compound and optical recording medium containing the compound
07/12/2001US20010007867 Substituted 6,5-hetero-bicyclic derivatives
07/12/2001US20010007761 Novel process for the isolation of clavulanic acid and of pharmaceutically acceptable salts thereof
07/11/2001EP0876371B1 Reverse-turn mimetics and methods relating thereto
07/11/2001EP0683783B1 Rapamycin derivative process for its preparation and its use
07/10/2001US6258948 An n-acylamino compound; antiinflammatory agents, autoimmune diseases
07/10/2001US6258823 Materials and method for treating or preventing pathogenic fungal infection
07/10/2001CA2175502C Cyclic amide derivatives
07/05/2001WO2001047934A1 Isoxazolo pyrimidinones and the use thereof
07/05/2001WO2001047921A1 Pyrimidine and triazine kinase inhibitors
07/05/2001WO2001047919A1 Substituted oxazolidinones and their use in the field of blood coagulation
07/05/2001WO2001047897A1 Cytokine, especially tnf-alpha, inhibitors
07/05/2001WO2001047836A1 Novel selective deacetylating agents
07/05/2001WO2001047507A2 Combinations of receptor tyrosine kinase inhibitor with an a1-acidic glycoprotein binding compound
07/05/2001WO2000040247A8 2-oxy-benzoxazinone derivatives for the treatment of obesity
07/05/2001DE19962924A1 Substituierte Oxazolidinone und ihre Verwendung Substituted oxazolidinones and their use
07/05/2001CA2396693A1 Cytokine, especially tnf-alpha, inhibitors
07/05/2001CA2395418A1 Isoxazolo pyrimidinones and the use thereof
07/05/2001CA2394944A1 Combinations of a receptor tyrosine kinase inhibitor with an organic compound capable of binding to .alpha.1-acidic glycoprotein
07/05/2001CA2394727A1 Pyrimidine and triazine kinase inhibitors
07/03/2001US6255482 Triphendioxazine compounds
06/2001
06/28/2001WO2001046199A1 Methods and compounds for inhibiting mrp1
06/28/2001WO2001046190A1 Tricyclic compounds and addition salts thereof
06/28/2001WO2001046189A1 Substituted homopiperidinyl benzimidazole analogues as fundic relaxants
06/28/2001WO2001045707A1 Inhibitors of prenyl-protein transferase
06/28/2001WO2000077010A3 Substituted heterocycle fused gamma-carbolines
06/28/2001WO2000040569A8 2-amino-benzoxazinone derivatives for the treatment of obesity
06/28/2001WO1999063937A9 Multivalent macrolide antibiotics
06/28/2001DE19962925A1 New aminosulfonyl-substituted isoxazolo (4,5-d) pyrimidin-7(6H)-one derivatives, are phosphodiesterase inhibitors useful for treating cardiovascular, cerebrovascular or urogenital disorders
06/28/2001CA2395513A1 Methods and compounds for inhibiting mrp1
06/27/2001EP1109804A1 Chemokine receptor antagonists and methods of use therefor
06/27/2001EP1109554A2 Pipecolic acid derivatives for vision and memory disorders
06/27/2001EP0572454B1 Process for the preparation of 29-desmethylrapamycin and its use as antifungal or immunosuppressant agent
06/27/2001CN1301265A Novel substituted arylhydroxamic acids as metalloproteinase inhibitors
06/27/2001CN1301262A Novel herbicides
06/27/2001CN1301157A Sustained release preparations
06/27/2001CN1067686C Fused polycyclic heterocycle derivatives
06/26/2001US6251902 Dipeptide derivatives as growth hormone secretagogues
06/26/2001US6251894 1-(1,2-disubstituted piperidinyl)-4 (fused imidazole)-piperidine derivatives
06/20/2001EP0796260B1 Rapamycin 42-oximes and hydroxylamines
06/20/2001CN1067419C Reactive dyestuffs their preparation and their use
06/14/2001WO2001042242A1 Antibacterial heterobicyclic substituted phenyl oxazolidinones
06/14/2001WO2001041780A2 Use of an immunosuppressant for increasing an antifugal activity of a lipopeptide
06/14/2001CA2393587A1 Use of an immunosuppressant for increasing an antifungal activity of a lipopeptide
06/13/2001EP1105395A1 Photocyclized rapamycins
06/13/2001EP1105394A1 ISOXAZOLO 4,5-d]PYRIMIDINES AS CRF ANTAGONISTS
06/13/2001EP0805812B1 Bicyclic substituted hexahydrobenz(e)isoindole alpha-1- adrenergic antagonists
06/12/2001US6245796 Tricyclic pyrrole or pyrazole derivative
06/12/2001US6245776 Drug mixture of immune response modifier, fatty acid, preservative and carbomer
06/12/2001US6245449 Material for organoelectroluminescence device and use thereof
06/07/2001WO1999063940A3 INHIBITORS OF H+K+-ATPase
06/06/2001EP1104755A1 Process for the preparation of (S)-N-tertbutyl-1,2,3,4- tetrahydroisoquinoline-3-carboxamide
06/06/2001EP0737188B1 Arthropodicidal oxadiazine carboxanilides
06/06/2001EP0681584B1 Condensed heterocyclic glutamic acid derivatives as antiproliferative agents
06/06/2001EP0676961B1 Use of macrolides for the treatment of cerebral ischemia
06/06/2001CN1066734C Novel intermediates and their use to prepare N,N'-bridged bisindolylmaleimides
06/06/2001CN1066733C 1-(1,2-disubstituted piperidinyl)-4-(fused imidazole)-piperidine derivatives
06/05/2001US6242471 Bone disorders, osteoporosis, rheumatoid arthritis, arteriosclerosis, cancer metastasis, nervous system and brain disorders
06/05/2001CA2047848C Azabicyclo derivatives
05/2001
05/31/2001WO2000066593A3 Novel spirocyclic compounds, method for the production thereof and their use for treating hyperproliferative diseases
05/30/2001EP1103553A2 Substituted heterocyclic derivatives
05/30/2001EP1103551A1 Pyrazole derivatives and salts thereof
05/30/2001EP1102755A1 Substituted isoxazole derivatives as estrogen receptor modulators
05/30/2001EP1102753A2 Pyrazoles as estrogen receptor modulators
05/30/2001EP0672043B1 Novel 4-(3-benzofuranyl)piperidinyl and 4-(3-benzothienyl)piperidinyl derivatives and pharmaceutical compositions containing them