Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
05/2002
05/16/2002WO2001079209A3 Diazafluorenone il-8 antagonists
05/16/2002WO2001079195A3 Pyridine and pyrazine derivatives as thrombin inhibitors
05/16/2002US20020058155 Cyclic tertiary amine compound and organic electroluminescent device containing the compound
05/15/2002EP1204675A1 Streptogramin derivatives, production thereof and compositions containing the same
05/15/2002EP1204642A1 Fungicides
05/15/2002EP1049694B1 Derivatives of benzoxadiazoles, benzothiadiazoles, benzotriazoles and quinoxalines
05/15/2002CN1349538A Cyclocarbamate and cyclic amide derivatives
05/15/2002CN1349537A Cyclic urea and cyclic amide derivatives
05/15/2002CN1349412A Contraceptive compositions containing cyclic urea and amide derivatives
05/14/2002US6387920 Isoxazole compounds; for treating estrogen receptor-mediated disorders such as osteoporosis, breast and endometrial cancers, atherosclerosis, alzheimer's disease
05/14/2002US6387919 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
05/14/2002US6387918 A tricyclic compound (with oxy and nitrogen atoms in the ring); perticularly useful for treating or preventing psoriasis and other skin diseases
05/10/2002WO2001097809A3 Method of treating cardiovascular disease using rapamycin
05/10/2002WO2001081342A3 Novel epothilone derivatives, method for the preparation thereof and their pharmaceutical use
05/10/2002WO2001041780A3 Use of an immunosuppressant for increasing an antifugal activity of a lipopeptide
05/10/2002WO2001029036A3 Allosteric sites on muscarinic receptors
05/09/2002US20020055518 Polyoxyethylated hydroxyesters of rapamycin useful in inducing immunosuppression and in the treatment of transplantation rejection, autoimmune diseases, solid tumors, fungal infections, and vascular disease.
05/09/2002US20020055508 Benzofurazan compounds which enhance AMPA receptor activity
05/09/2002US20020055502 New compounds, their preparation and use
05/08/2002EP1203766A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors
05/08/2002EP1202985A2 Chemokine receptor antagonists
05/08/2002EP0737197B1 Amino alkanoic esters of rapamycin
05/08/2002CN1348454A Tetracyclic azepinoindole compounds as 5-HT receptor ligands
05/07/2002US6384218 Prepared by reacting amino acid, oligo- or polypeptide or polyamino acid with trialdehyde; molecular recognition agent for use in neurotransmission studies
05/07/2002US6384073 Use of macrolide compounds for treating glaucoma
05/07/2002US6384050 Tricyclic amine derivatives
05/07/2002US6384046 Treating neointimal proliferation and thickening
05/07/2002CA2216535C Protein kinase c inhibitors
05/07/2002CA2098612C Arthropodicidal carboxanilides
05/02/2002WO2002034718A1 Amide derivatives as nmda receptor antagonists
05/02/2002WO2002002562A3 Heteropolycyclic inhibitors
05/02/2002US20020052364 Condensed 2,3-benzodiazepine derivatives and their use as AMPA-receptor inhibitors
05/02/2002EP1201718A2 Mixed crystals of benzimidazoloneoxazine derivatives
05/02/2002EP1201670A2 Process for preparing 2-oxaisocephem derivatives
05/02/2002EP1201668A1 Staurosporin derivatives
05/02/2002EP1200447A1 Oxazinocarbazoles for the treatment of cns diseases
05/02/2002EP0888359B1 Pyrimidin-4-one derivatives as pesticide
05/02/2002EP0812838B1 Pyridonecarboxylic acid derivative substituted by bicyclic amino group, ester thereof, salt thereof, and bicyclic amine as intermediate therefor
05/02/2002DE10052221A1 Verfahren zur Herstellung neuer Kristallmodifikationen eines methylsubstituierten Benzimidazolon-Dioxazin-Pigmentes Process for the preparation of new crystal forms of a methyl-substituted benzimidazolone-dioxazine pigment
04/2002
04/30/2002USRE37686 Biosynthesis of polypeptides
04/30/2002US6380228 E.g., n-(2-phenylsulfonyl-1-ethyl)-3-(4-cyanophenyl)-2,3-dihydro-imidazo(2,1 -b)thiazole-5-carboxamide hydrochloride; treating cancer, neurofibromin benign proliferative disorder, retinal vascularization, and hepatitis delta
04/30/2002US6380211 For treating diabetes
04/30/2002US6380178 Cyclic regimens using cyclocarbamate and cyclic amide derivatives
04/30/2002US6380134 N-pyridyl herbicide compounds
04/30/2002US6379823 Electroluminescence device, cyclic azine compound and production process of cyclic azine dye
04/25/2002WO2002032904A1 New cephalotaxanes, their method of preparation and their use in treatment of cancers, leukemias, parasites including thus resistant to usual chemotherapeutic agents and as reversal agents
04/25/2002WO2002032893A2 Piperidine compounds as anti-allergic
04/25/2002WO2001087283A3 New use of citreamicins
04/25/2002WO2001081341A3 9-oxa-epothilon derivatives, method for the production and use thereof in pharmaceutical preparations
04/25/2002US20020049327 Such as 7-(3-chlorophenyl)-9-((4-chlorophenyl)-1H-imidazol-1-ylmethyl)-2,3-dihydro -1H,5H-benzo(ij)quinolizin-5-one; for forming oncogenes for signalling transformation of tumor cells
04/25/2002US20020049242 Condensed 4,5,6,7-tetrahydrobenzo[C]thiopenes as enhancer for cell differentiation induction factor action
04/25/2002US20020049203 CRF receptor antagonists and methods relating thereto
04/25/2002US20020049197 Aminoquinazolines and their use as medicaments
04/25/2002DE10052858A1 Mixed crystals of different benzimidazolone-dioxazine compounds give fast red shades e.g. for pigmenting plastics or use in toners or developers, are obtained by co-synthesis, acidic cyclization, precipitation or sublimation
04/25/2002CA2426103A1 New cephalotaxanes, their method of preparation and their use in treatment of cancers, leukemias, parasites including thus resistant to usual chemotherapeutic agents and as reversal agents
04/24/2002EP1199309A1 Process for producing new crystalline modifications of a methyl-substituted benzimidazolonedioxazine pigment
04/24/2002EP1199306A1 Biarylurea derivatives
04/24/2002EP0714299B1 Benzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonists
04/24/2002CN1346074A Silver halide picture photosensitive material, compound forming azoheterocyclic dye, and process for preparing dye
04/24/2002CN1083453C Fused imidazole derivatives as emultidrug resistance modulators
04/23/2002US6376656 Disazo dyes, triazine dyes
04/23/2002US6376517 For treating vision loss, preventing vision degeneration, and promoting vision regeneration (?neopsis?)
04/23/2002US6376487 Oxadiazine derivatives
04/18/2002WO2002030938A1 Benzhydryl derivatives
04/18/2002WO2002030925A1 Benzopyranyl heterocycle derivatives, process for preparation thereof, and pharmaceutical compositions containing them
04/18/2002WO2002002541A3 Inhibitors of copper-containing amine oxidases
04/18/2002WO2001087830A3 Substituted thioacetamides
04/18/2002WO2001077112A3 Photochromic spiro(indoline)naphthoxazines
04/18/2002US20020045759 E.g., N-(2-Phenylsulfonyl-1-ethyl)-3-(4-Cyanophenyl)-2,3-dihydro-imidazo(2,1 -b)thiazole-5-carboxamide hydrochloride; treating cancer, neurofibromin benign proliferative disorder, retinal vascularization, and hepatitis delta
04/18/2002US20020045629 Sleep, eating and brain disorders, wakefulness promoters; Parkinson's disease, antiischemic agents, stroke, chronic fatigue syndrome; antidepressants; schizophrenia, nervous system disorders; multiple sclerosis, cognition activators
04/18/2002US20020044967 Sustained release preparations
04/17/2002EP1196384A1 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
04/17/2002EP1196170A2 New use of a macrolide compound for treating neurodegenerative disorders
04/17/2002EP0804186B1 Indole diterpene alkaloid compounds
04/17/2002CN1082963C Isoxazolidine derivatives
04/16/2002US6372775 Reversal of multidrug resistance in human colon carcinoma cells
04/11/2002WO2002028867A2 Ethers of 7-desmethylrapamycin for use in immunosuppression
04/11/2002WO2002028866A2 Hydroxyesters of 7-desmethylrapamycin
04/11/2002WO2002028865A2 Condensed pyridoindole derivatives
04/11/2002WO2002028864A1 New process for the production of oxabispidines
04/11/2002WO2002028863A1 New oxabispidine compound useful in the treatment of cardiac arrhythmias
04/11/2002WO2002028834A1 Process for the preparation of aryl-piperidine carbinols and intermediates thereof
04/11/2002WO2001087342A3 Delivery devices for treatment of vascular disease
04/11/2002US20020042415 Dipeptide derivatives
04/11/2002US20020042411 Condensed thiophene compounds and pharmaceutical use thereof
04/11/2002CA2423898A1 Ethers of 7-desmethylrapamycin for use in immunosuppression
04/11/2002CA2423888A1 Hydroxyesters of 7-desmethylrapamycin
04/11/2002CA2423312A1 Condensed pyridoindole derivatives
04/11/2002CA2422810A1 New oxabispidine compound useful in the treatment of cardiac arrhythmias
04/11/2002CA2421776A1 New process for the production of oxabispidines
04/10/2002EP1194135A2 Methods of treating fungal infections with inhibitors of nad synthetase enzyme
04/10/2002EP0918774B9 Androgen receptor modulator compounds and methods
04/10/2002EP0813535B1 Hexacyclic camptothecin analogues, and process for preparing them
04/10/2002EP0712402B1 Hydroisoquinoline derivatives
04/09/2002US6369227 Thrombin or factor Xa inhibitors
04/09/2002US6369086 Substituted oxidole derivatives as protein tyrosine and as protein serine/threonine kinase inhibitors
04/09/2002US6369070 Methods for inhibiting mrp1
04/09/2002US6369056 Agonists and antagonists of the progesterone receptor; contraceptives; 6-(3-chlorophenyl)-4,4-dimethyl-1,4-dihydro -3-oxa-1,8-diaza-naphthalene-2-one and 6-chloro-4,4-dimethyl-1,4-dihydro-3-oxa-1,5-diaza-naphthalen-2-one
04/09/2002US6369002 Hetero is pyrimidine or pyridazine; 1-(3-fluoro-5-chloro pyridin-2-yl)-3-methyl-4-trifluoromethylpyrimidin-2,6-dione
04/09/2002US6368520 Synergistic stabilizer mixture