Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
09/1999
09/15/1999CN1045084C Novel compound with platelet aggregation inhibitor activity and its use, and drug composition containing the same
09/14/1999US5952504 Reacting a sulfonated, halogenated or phosphonated 1,7-naphthyridine compounds with an aromatic amine derivative; antiulcer agent
09/14/1999US5952498 Synthesizing the chemical intermediates for antiatherosclerotically active drug
09/14/1999US5952359 Thiazoles and their agricultural compositions
09/14/1999US5952343 HIV protease inhibitors
09/14/1999US5952342 1,6-naphthyridines effective in treating atherosclerosis, restenosis and psoriasis; anticarcinogenic and -proliferative agents; bactericides
09/14/1999US5952341 Integrin antagonists
09/14/1999US5952340 Use of granisetron for the treatment of postoperative nausea and vomiting
09/14/1999US5952335 Antitumor agents
09/14/1999US5952306 Integrin receptor antagonists
09/14/1999US5952140 Bipolar charge transport materials useful in electrophotography
09/14/1999CA1340734C Substituted bridged-diazabicycloalkyl quinolone carboxylic acids
09/13/1999CA2232074A1 Granulatimide compounds as g2 checkpoint inhibitors
09/10/1999WO1999045011A1 Glycine transport inhibitors
09/10/1999WO1999045009A1 Heterocyclo-substituted imidazopyrazine protein tyrosine kinase inhibitors
09/10/1999WO1999045007A1 Crf antagonistic pyrazolo[4,3-b]pyridines
09/10/1999WO1999044991A1 Process for preparing a protected 4-aminomethyl-pyrrolidin-3-one
09/10/1999WO1999044596A2 Glycine transport inhibitors
09/10/1999CA2322164A1 Glycine transport inhibitors
09/10/1999CA2322136A1 Glycine transport inhibitors
09/09/1999CA2264460A1 1-alkoxy-polyalkyl-piperidine derivatives and their use as polymerization regulators
09/08/1999EP0939757A1 Novel integrin receptor antagonists
09/08/1999EP0730594B1 9-HYDROXY-PYRIDO [1,2-a]PYRIMIDIN-4-ONE ETHER DERIVATIVES
09/08/1999CN1228091A Substituted 6,6-hetero-bicyclic derivatives
09/08/1999CN1228090A Naphthyridines with affect IL-4 and G-CSF
09/08/1999CN1227743A Trovafloxacin mesylate tablet
09/07/1999US5948933 Tropane analogs and methods for inhibition of monoamine transport
09/07/1999US5948789 Process for synthesis of substituted sulphoxides
09/07/1999US5948782 Antiinflammatory agent; rheumatic diseases
09/07/1999CA2134445C Methods for regenerating a sulfur scavenging compound from a product of a sulfur scavenging reaction
09/07/1999CA2014884C 5,11-dihydro-6h-pyrido[2,3-b][1,4]benzodiazepin-6-ones and -thiones and their use in the prevention or treatment of aids
09/07/1999CA1340721C 1,4-dihydro-quinoline-and naphthyridine-3-carboxylic acid antibacterial agents
09/02/1999WO1999043682A1 2-(het-)aryl-4-(cyclic amino substituted) heteroaryl fused pyridine derivatives, their preparation and their use as (ant-)agonists for gaba (a) brain receptors
09/02/1999WO1999043681A1 4-(4-piperidylmethylamino) substituted heteroaryl fused pyridines: gaba brain receptor ligands
09/02/1999WO1999043674A1 Remedies for erectile dysfunction
09/02/1999WO1999043673A1 1-azaindolizine derivatives
09/02/1999WO1999043671A1 Substituted aminomethyl isoxazoline derivatives useful as antimicrobials
09/02/1999WO1999043659A1 Pyridone derivatives and process for producing the same
09/02/1999WO1999043649A1 Arylphenyl-substituted cyclic keto-enols
09/02/1999WO1999043648A1 Cyclic amino compounds
09/02/1999DE19807993A1 Treating tumor necrosis factor mediated inflammatory disease, e.g. arteriosclerosis, using new or known beta-carboline derivatives
09/02/1999CA2321237A1 Pyridone derivatives and process for producing the same
09/02/1999CA2318762A1 Substituted aminomethyl isoxazoline derivatives useful as antimicrobials
09/01/1999EP0938315A1 Immune response modifier compounds for treatment of th2 mediated and related diseases
09/01/1999EP0687267B1 Pyrrolo-pyridine derivatives as ligands of dopamine receptor
09/01/1999CN1227555A Cytokine production inhibitors triazepine compounds, and intermediates thereof
09/01/1999CN1227554A Substituted 6,5-hetero-bicyclic derivatives
09/01/1999CN1227552A Substituted pyrido- or pyrimido-containing 6,6- or 6,7-bicyclic derivatives
08/1999
08/31/1999US5945431 Cytomegalovirus inhibiting compounds
08/31/1999US5945429 Benzo(5,6)cycloheptapyridine or dibenzo(a,d)cycloheptene compounds that inhibit ras function, use for treating tumor cells expressing an activated ras oncogene in mammals
08/31/1999US5945428 Substituted oximes for treatment of asthma, cough, bronchospasm, inflammatory diseases, and gastrointestinal disorders
08/31/1999US5945422 N-oxides of amino containing pyrido 2,3-D! pyrimidines
08/31/1999US5945418 Administering to the mammal to inhibit a mammalian protein kinase p38 which causes cell proliferation, cell death and response to extracellular stimuli
08/31/1999US5945417 Nervous system disorders
08/31/1999CA2173328C Hiv protease inhibitors
08/26/1999WO1999042465A2 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
08/26/1999WO1999042464A1 SUBSTITUTED IMIDAZO[1,2-a;3,4-a']DIQUINOLINYLIUM INTERLEUKIN-8 RECEPTOR ANTAGONISTS
08/26/1999WO1999042452A1 Phthalazine derivatives and remedies for erectile dysfunction
08/26/1999WO1999042443A1 Sulfonylamino derivatives which inhibit matrix-degrading metalloproteinases
08/26/1999WO1999042100A1 Cell death inhibitors
08/26/1999WO1999031098A8 Novel pyridine and pyrimidine derivatives
08/26/1999WO1999031060A3 Piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides as cytostatics and immunesuppressants
08/26/1999WO1999030697A3 Combination effective for the treatment of impotence
08/26/1999DE19808088A1 New tris(hydroxynaphthylazo) bridged triphenylamine pigments for electrophotographic charge generating layer
08/26/1999CA2321278A1 Novel compounds
08/25/1999EP0937724A1 Perylene compounds and their use as pigment dispersants
08/25/1999EP0937077A1 Pyridone-fused azabicyclic- or cytisine derivatives, their preparation and their use in addiction therapy
08/25/1999EP0937076A1 Substituted oximes, hydrazones and olefins as neurokinin antagonists
08/25/1999EP0937075A1 New imidazopyridines and oxazolopyridines
08/25/1999EP0937074A1 Benzonaphthyridines as bronchial therapeutics
08/25/1999EP0937069A1 Piperazino derivatives as neurokinin antagonists
08/25/1999EP0937044A1 Cftr channel activator compounds and pharmaceutical compositions containing same
08/25/1999EP0612321B1 Pyrido pyridazinone and pyridazinthione compounds with pde iv inhibiting activity
08/24/1999US5942616 A metal ion coordination complex crystal comprises protonated derivative of a compound containing atleast one basic nitrogen and aromatic heterocyclic ring, an anion of triiodine, a positive metal ion and an optional acid
08/24/1999US5942535 a!-Annelated pyrrole derivatives and pharmaceutical use thereof
08/24/1999US5942493 LH-RH antagonists having improved action
08/24/1999CA2064853C Indole derivatives
08/19/1999WO1999041276A1 β-SHEET MIMETICS AND METHODS RELATING TO THE USE THEREOF
08/19/1999WO1999041252A1 Antagonists of gonadotropin releasing hormone
08/19/1999WO1999041251A1 Antagonists of gonadotropin releasing hormone
08/19/1999WO1999041250A1 1,4-dihydropyridine derivatives
08/19/1999WO1999041230A1 Processes and intermediates useful to make antifolates
08/19/1999WO1999041224A1 Biaryl-acetic acid derivatives and their use as cox-2 inhibitors
08/19/1999WO1999040931A1 Cyclic dipeptides and azetidinone compounds and their use in treating cns injury and neurodegenerative disorders
08/19/1999WO1999040910A1 Anti-inflammatory agents
08/19/1999WO1999025354A3 Aqueous suspensions of submicron 9-hydroxyrisperidone fatty acid esters
08/19/1999WO1999015894A3 Method of identification of leads or active compounds
08/19/1999CA2320378A1 Cyclic dipeptides and azetidinone compounds and their use in treating cns injury and neurodegenerative disorders
08/19/1999CA2320319A1 1,4-dihydropyridine derivatives
08/19/1999CA2320285A1 Anti-inflammatory agents
08/19/1999CA2319766A1 .beta.-sheet mimetics and methods relating to the use thereof
08/19/1999CA2319424A1 Processes and intermediates useful to make antifolates
08/19/1999CA2318966A1 Biaryl-acetic acid derivatives and their use as cox-2 inhibitors
08/19/1999CA2318957A1 Antagonists of gonadotropin releasing hormone
08/19/1999CA2317451A1 Antagonists of gonadotropin releasing hormone
08/18/1999EP0935601A2 Arylamino fused pyridines and pyrimidines
08/18/1999EP0935600A1 Method or producing naphthyridine compounds and novel intermediate products
08/18/1999EP0935599A1 2-methoxyphenylpiperazine derivatives
08/18/1999EP0935598A1 5-HETEROATOM-CONTAINING ALKYL SUBSTITUTED-3-OXO-PYRIDO(1,2-a) BENZIMIDAZOLE-4-CARBOXAMIDE DERIVATIVES USEFUL IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS
08/18/1999CN1226246A Noval tricyclic N-cyanoimines useful as inhibitors of farnesyl-protein transferase