Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
12/1999
12/16/1999CA2319495A1 Multibinding inhibitors of microsomal triglyceride transferase protein
12/16/1999CA2319477A1 Inhibitors of h+k+-atpase
12/16/1999CA2319474A1 Inhibitors of nitric oxide synthase
12/16/1999CA2319175A1 Multibinding agents that modulate nmda receptors
12/16/1999CA2319159A1 Novel therapeutic agents that modulate neurokinin receptors
12/16/1999CA2319120A1 Phosphodiesterase-v modulator drugs and their uses
12/16/1999CA2319068A1 Novel angiotensin receptor modulators and their uses
12/16/1999CA2318894A1 .beta.2-adrenergic receptor agonists
12/16/1999CA2318547A1 Combinatorial synthesis of multibinding libraries
12/16/1999CA2318286A1 Multibinding agents that modulate ppar.gamma. and rxr receptors
12/16/1999CA2318055A1 .beta.2-adrenergic receptor agonists
12/16/1999CA2316999A1 Inhibitors of hiv reverse transcriptase
12/15/1999EP0963988A2 Method of making camptothecin and camptothecin analogs
12/15/1999EP0963987A2 Spiro(piperidine-4,1'-pyrrolo(3,4-c)pyrrole)
12/15/1999EP0963986A2 5,10-Dihydrodipyrido(2,3-b:2,3-e)pyrazine and 5,10-dihydro(2,3-b:3,2-e)pyrazine, process for their preparation and pharmaceutical compositions containing them
12/15/1999EP0963985A2 Di-or triaza-spiro(4,5)decane derivatives
12/15/1999EP0963984A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
12/15/1999EP0963977A1 Process for the preparation of quinolone- and naphthyridonecarboxylic acids and their esters
12/15/1999EP0750612B1 Acridone-derived bisintercalators as chemotherapeutic agents
12/15/1999EP0638079B1 Deazaaminopterins for treatment of inflammation
12/15/1999CN1238773A Novel substituted pyrazole derivatives for the treatment of cardiocirculatory diseases
12/15/1999CN1238772A Novel phenanethridinium derivatives
12/15/1999CN1238770A Tricyclic antitumor compounds being farnesyl protein transferase inhibitors
12/15/1999CN1047386C Novel spiro [indole-pyrrolidine] derivatives as melatoninergic agonists, method for preparing same and use thereof as drug
12/14/1999US6002000 Chemiluminescent compounds and methods of use
12/14/1999US6001905 Polyalkylene glycol group-containing hindered amines
12/14/1999US6001849 Furopyridine, thienopyridine pyrrolopyridine useful in controlling chemical synaptic transmission
12/14/1999US6001847 Chemical compounds
12/14/1999US6001834 [(4-heteroaryl-1-piperazinyl)alkoxy]-3,4-dihydro-1(2h)-naphthalenones and related compounds and their therapeutic utility
12/14/1999CA2136007C Novel compound with platelet aggregation inhibitor activity
12/14/1999CA2081805C Process for the manufacture of substituted maleimides
12/14/1999CA2010636C Substituted pyrroles
12/12/1999CA2274733A1 New derivatives of 5,10-dihydrodipyrido[2,3-b:2,3-e]pyrazine and of 5,10- dihydrodipyrido[2,3-b:3,2-e]pyrazine, their preparation process and pharmaceutical compositions made thereof
12/12/1999CA2274202A1 Diaza-spiro[3,5]nonane derivatives
12/12/1999CA2273802A1 Process for preparing quinolone- and naphthyridonecarboxylic acids and esters thereof
12/09/1999WO1999062908A2 Cell adhesion-inhibiting antinflammatory compounds
12/09/1999WO1999062904A1 Sulfonic acid or sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
12/09/1999WO1999062883A1 2-aminopyridines containing fused ring substituents as nitric oxide synthase inhibitors
12/09/1999WO1999062882A1 Substituted indolinones, the production thereof and their use as medicaments
12/09/1999WO1999062553A1 Remedies for male sterility
12/09/1999DE19824922A1 Neue substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel New substituted indolinones, their preparation and their use as medicaments
12/09/1999CA2333994A1 Sulfonic acid or sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
12/09/1999CA2333770A1 Cell adhesion-inhibiting antinflammatory compounds
12/09/1999CA2328291A1 Substituted indolinones, the preparation thereof and their use as pharmaceutical compositions
12/08/1999EP0962458A1 New naphthalenetetracarboxylic acid diimides as electron transporting agents in photosensitive material for electrophotography
12/08/1999CN1237963A Qinoline derivatives inhibiting effect of growth factors such as VEGF
12/08/1999CN1047172C Improved purification method for quinolone compounds
12/07/1999US5998622 Analgesics; antiinflammatory agents; side effect reduction
12/07/1999US5998619 Process for preparing imidazoquinolinamines
12/07/1999US5998594 Self-assembling, chromogenic receptors for the recognition of medically important substrates and their method of use
12/07/1999US5998436 Pyridonecarboxylic acid derivatives or their salts and antibacterial agent comprising the same as the active ingredient
12/07/1999US5998434 Composition for treating pain
12/07/1999US5998429 Azabicyclic esters of carbamic acids useful in therapy
12/07/1999US5998417 N-[(4-heteroaryl-1-piperazinyl) alkyl]phthalimides and related compounds and their therapeutic utility
12/07/1999US5998405 Psychological disorders
12/07/1999US5998404 Nervous system disorders
12/07/1999US5998333 Pyrimidinone derivatives and herbicides containing them
12/07/1999CA2198231C Dihydropyridine derivatives as bradykinin antagonists
12/02/1999WO1999061444A2 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation
12/02/1999WO1999061442A1 Imidazopyridine thrombin inhibitors
12/02/1999WO1999061441A1 Polymorphs of crystalline (7s,9as)-7-[ 3-cyanophenoxy] methyl-2-(5- fluoropyrimidin-2- yl)-2,3,4,6,7,8,9a -octahydro-1h-pyrido[1,2-a] pyrazine- monohydrochloride and their pharmaceutical compositions
12/02/1999WO1999061436A1 Heterocyclic indole derivatives and mono- or diazaindole derivatives
12/02/1999WO1999061023A1 Cocaine receptor binding ligands
12/02/1999CA2333040A1 Imidazopyridine thrombin inhibitors
12/01/1999EP0960102A1 AMIDINOINDOLES, AMIDINOAZOLES, AND ANALOGS THEREOF AS INHIBITORS OF FACTOR Xa AND OF THROMBIN
12/01/1999EP0800504B1 Tricyclic retinoids, methods for their production and use
12/01/1999EP0655056B1 Azacyclyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
12/01/1999CN1237177A Fused bicyclic pyrimidine derivatives
12/01/1999CN1237164A Compounds useful for inhibition of farnesyl protein transferase
12/01/1999CN1046942C Imidazopyridines
11/1999
11/30/1999US5994544 Producing a 5h-chromeno(3,4-f)quinoline
11/30/1999US5994389 Insecticide
11/30/1999US5994379 Analgesics; antiinflammatory agent; antipyretics
11/30/1999US5994368 Antiallergens, antiinflammatory agents, analgesics
11/30/1999US5994367 Method for treating tumors using 2-aryl-naphthyridin-4-ones
11/30/1999US5994366 Psychological disorders
11/30/1999US5994365 Bactericides; fungicides; antitumor agent
11/30/1999US5994364 Antitumor, anticarcinogenic agents
11/25/1999WO1999059997A1 Novel 1,3,8-triazaspiro[4.5]decanones with high affinity for opioid receptor subtypes
11/25/1999WO1999059996A1 Antitumour 1,5-diazaanthraquinones
11/25/1999WO1999059975A1 Fused tricyclic compounds which inhibit parp activity
11/25/1999WO1999059587A1 Anti-viral compounds
11/25/1999WO1999059409A1 Compounds and uses thereof
11/25/1999WO1999050249A3 Pyrimidines and triazines as integrin antagonists
11/25/1999CA2345917A1 Antitumour 1,5-diazaanthraquinones
11/25/1999CA2332403A1 Anti-viral compounds
11/25/1999CA2332239A1 Fused tricyclic compounds which inhibit parp activity
11/24/1999EP0959076A1 Heteroarylperidines and piperazines and their use as antipsychotics and analgetics
11/24/1999EP0959075A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
11/24/1999EP0958297A1 1-aryl-1,8-naphthylidin-4-one derivative as type iv phosphodiesterase inhibitor
11/24/1999EP0958296A1 Novel heterocyclic compounds process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
11/24/1999CN1236367A Benzonaphthyrindines as bronchial therapeutics
11/24/1999CN1236358A Substituted N-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides
11/24/1999CN1235968A Substituted tricyclics
11/24/1999CN1046726C Imidazopyridine-pyrrolidone, its preparation and medical use
11/24/1999CN1046725C Condensed imidazole compounds, their preparation and use
11/24/1999CN1046724C Pyrazolopyridine compounds, pharmaceutical containing them, and its preparing method and use
11/24/1999CN1046722C Heterocyclic compounds and their preparation and use
11/23/1999US5990145 Antiinflammatory,-carcinogenic,-tumor,-metastasis agents; cardiovascular disorders, e.g., arteriosclerosis, restenosis; retinopaathies and nephropathies; osteoporosis
11/23/1999US5990132 Polycyclic systems, and derivatives thereof, as neurotransmitter release enhancers useful in the treatment of cognitive disorders