Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
04/2000
04/26/2000EP0554247B1 Neuroprotective indolone and related derivatives
04/26/2000CN1251588A Novel 3,5 and/or 6 substituted analogues of swainsonine, process for their preparation and their use as therapeutic agents
04/26/2000CN1251579A Compound and compositions for treating diseases associated with serine protease, particularly tryptase, activity
04/25/2000US6054466 Inhibitors of farnesyl-protein transferase
04/25/2000US6054464 Azabicyclic esters of carbamic acids useful in therapy
04/25/2000CA2196538C Process for making antimicrobial compounds
04/25/2000CA2105575C Esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions
04/21/2000CA2287122A1 Treatment of bph with cgmp elevators
04/20/2000WO2000021962A1 Method of stabilizing aqueous pyrazoloacridone derivative solution
04/20/2000WO2000021961A1 Imidazo-isoquinoline compounds, their compositions and uses
04/20/2000WO2000021952A1 Quinoline derivatives and their use as antibacterial agents
04/20/2000WO2000021951A1 Tetrahydrobenzazepine derivatives useful as modulators of dopamine d3 receptors (antipsychotic agents)
04/20/2000WO2000021950A1 2,3-dihydro-1h-isoindole derivatives useful as modulators of dopamine d3 receptors (antipsychotic agents)
04/20/2000WO2000021948A1 Naphthrydine compounds and their azaisosteric analogues as antibacterials
04/20/2000WO2000021927A2 Pyrrole-2,5-diones as gsk-3 inhibitors
04/20/2000WO2000021926A2 6-SUBSTITUTED PYRAZOLO[3,4-d]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS
04/20/2000WO2000021563A1 Remedies or preventives for ischemic reflow failure
04/20/2000WO2000021533A1 A dried or frozen pharmaceutical preparation containing a class iii antiarrhythmic compound
04/20/2000WO2000021530A1 Peripherally acting anti-pruritic opiates
04/20/2000WO2000006525A9 Synthesis of combinatorial libraries of compounds reminiscent of natural products
04/20/2000WO1999064000A9 Novel therapeutic agents that modulate neurokinin receptors
04/20/2000CA2346834A1 Method of stabilizing aqueous pyrazoloacridone derivative solution
04/20/2000CA2346689A1 Tetrahydrobenzazepine derivatives useful as modulators of dopamine d3 receptors (antipsychotic agents)
04/20/2000CA2346464A1 Peripherally acting anti-pruritic opiates
04/20/2000CA2346414A1 Imidazo-isoquinoline compounds, their compositions and uses
04/20/2000CA2346334A1 Composition for treating or preventing ischemia reperfusion injury
04/20/2000CA2315375A1 A dried or frozen pharmaceutical preparation containing a class iii antiarrhythmic compound
04/19/2000EP0994113A2 7-Aminopyrido(2,3-d)-pyrimidine derivatives for treatment of bronchial asthma
04/19/2000EP0994102A1 Cyclic derivatives with a cycloalkylenic chain, process for their preparation and pharmaceutical compositions containing them
04/19/2000EP0713487B1 Novel quinolone carboxylic acid derivatives
04/19/2000CN1251102A Tetrahydropyrido compounds
04/19/2000CN1251101A Salt of naphthyridine carobxylic acide derivative
04/19/2000CN1251100A Method for making arylamino triazolopyridines
04/19/2000CN1251097A Phthalazines with angiogenesis inhibiting activity
04/19/2000CN1250777A 5,10-dihydrodi pyridino [2,3-b: 2,3-e] pyrazine and 5,10 dihydrodipyridino [2,3-b:3,2-3] pyrazine compound, and prepn.therefor
04/19/2000CN1250776A Heterodicyclic compound derivatives
04/19/2000CN1250771A Novel cyclocompound having cycloalkylene chain, prepn. method and pharmaceutical compositions contg. same
04/19/2000CN1051549C 2-aminoalkyl-5-aminoalkylamino substituted isoquinoindazole-6-(2h)-ones, pharmaceutical composition and prepn. thereof
04/19/2000CN1051548C Heterobicyclic derivatives, pharmaceutical compositions contg. same, mfg. method and use thereof
04/19/2000CN1051547C Beta-lactams derivative and its prepn.and use
04/18/2000US6051712 Piperidine derivatives having renin inhibiting activity
04/18/2000US6051711 Acid hydrolysis in the presence of a c1-c4 alkanol to obtain a crystalline salt of swainsonine
04/18/2000US6051586 Sulfonamide substituted chroman derivatives useful as beta 3 adrenoreceptor agonists
04/18/2000CA2166700C Heterocyclic amines having central nervous system activity
04/13/2000WO2000020416A1 Imidazo[4,5-c-]-pyridine-4-one derivatives with factor xa inhibiting effect
04/13/2000WO2000020401A1 New bis-benzimidazoles
04/13/2000WO2000020400A1 Novel compounds and compositions for treating hepatitis c infections
04/13/2000WO2000020393A1 Substituted 1,3-diaryl-2-pyridine-2-yl-3-(pyridine-2-ylamino)-propanol derivatives, methods for their production, pharmaceutical compositions containing the same and their use
04/13/2000WO2000020358A2 NON-PEPTIDE GnRH AGENTS, METHODS AND INTERMEDIATES FOR THEIR PREPARATION
04/13/2000DE19845406A1 Substituierte 1,3-Diaryl-2-pyridin-2-yl-3-(pyridin-2-ylamino)- propanolderivate, Verfahren zu deren Herstellung, diese Verbindungen enthaltende Arzneimittel und deren Verwendung Substituted 1,3-diaryl-2-pyridin-2-yl-3- (pyridin-2-ylamino) - propanol derivatives, process for their preparation, pharmaceutical compositions containing them and their use
04/13/2000CA2346040A1 New bis-benzimidazoles
04/13/2000CA2346033A1 Imidazo[4,5-c-]-pyridin-4-one(sic) derivatives having factor xa-inhibiting action
04/13/2000CA2341346A1 Non-peptide gnrh agents, methods and intermediates for their preparation
04/12/2000EP0992501A2 Pyridonecarboxylic acid derivatives as antibacterial agents
04/12/2000EP0992496A1 Annulated 4-carboxyamino-2-methyl-1,2,3,4-tetrahydroquinolines as CETP inhibitors
04/12/2000EP0991650A1 Novel n-benzenesulphonyl-l-proline compounds, preparation method and use in therapy
04/12/2000EP0991638A1 NOVEL GUANIDINE MIMICS AS FACTOR Xa INHIBITORS
04/12/2000EP0991623A2 Quinoline-indole antimicrobial agents, uses and compositions related thereto
04/12/2000CN1250446A Pyrazole derivatives as herbicides
04/12/2000CN1051313C 5-arylindole derivatives and its use, pharmaceutical composition containing the same and intermediate for preparing them
04/11/2000US6049428 Coating a substrate with a solution of an organic dye occurring in the lyotropic liquid-crystal state in a solvent while simultaneously orienting the dye and removing the solvent
04/11/2000US6048884 Antidiabetic agents; hypoglycemic agents
04/11/2000US6048870 Mannosidase inhibitor; immunostimulant
04/11/2000US6048868 Melatonin-antagonist β-carboline derivatives and analogues thereof containing naphthalenic structure, process for their preparation and their use as medicinal products
04/11/2000US6048864 Benign prostatic hyperplasia
04/11/2000US6048861 Osteoporosis; bone disorders; cardiovascular disorders; antiinflammatroy agents; wound healing agents
04/06/2000WO2000018769A2 INDOLO[2,1-b]QUINAZOLE-6,12-DIONE ANTIMALARIAL COMPOUNDS AND METHODS OF TREATING MALARIA THEREWITH
04/06/2000WO2000018768A1 Novel salts of pyridopyrazine compound and crystals thereof
04/06/2000WO2000018735A1 2-substituted heterocyclic sulfonamides
04/06/2000WO2000018733A1 Heterocyclic 2-substituted ketoamides useful for treating hair loss in mammals
04/06/2000WO2000018391A1 Drugs for improving vesical excretory strength
04/06/2000WO2000018388A2 Antibiotic compositions for treatment of the eye, ear and nose
04/06/2000WO2000018386A2 Antibiotic compositions for treatment of the eye, ear and nose
04/06/2000WO2000018233A1 Synthetic analogs of ecteinascidin-743
04/06/2000WO2000006173A8 5-ht1f agonists
04/06/2000WO2000001704A3 Benzimidazoles, production thereof and use thereof as medicaments
04/06/2000WO1999064421A8 Acetylcholine enhancers
04/06/2000DE19845153A1 Imidazo[4,5]-pyridin-4-on-derivate Imidazo [4,5] pyridin-4-one derivatives
04/06/2000CA2774207A1 Antibiotic compositions for treatment of the eye
04/06/2000CA2659064A1 Antibiotic compositions for treatment of the ear and nose
04/06/2000CA2345362A1 Novel salts of pyridopyrazine compound and crystals thereof
04/06/2000CA2344894A1 Agents for improving excretory potency of urinary bladder
04/06/2000CA2342603A1 Antibiotic compositions for treatment of the eye, ear and nose
04/06/2000CA2317711A1 Indolo[2,1-b]quinazole-6,12-dione antimalarial compounds and methods of treating malaria therewith
04/05/2000EP0989993A1 Tartrate salt of a substituted dipeptide as growth hormone secretagogue
04/05/2000EP0989986A1 5,7-disubstituted 4-aminopyrido 2,3-d]pyrimidine compounds and their use as adenosine kinase inhibitors
04/05/2000EP0989984A1 Bispyrido-cycloheptane compounds useful for inhibition of farnesyl protein transferase
04/05/2000EP0989857A1 Novel therapeutic agents that modulate enzymatic processes
04/05/2000EP0716661B1 Pseudo- and non-peptide bradykinin receptor antagonists
04/05/2000CN1249753A Farnesyl transferase inhibiting 1,8-annelated quinolinone derivs. substd. with N- or C-linked imidazoles
04/05/2000CN1249752A Annulated azole derivs. useful as microbicidal agents
04/05/2000CN1051086C Heterocycle-condensed morphinoid derivs. and use thereof
04/04/2000US6046335 Heterocyclic compounds
04/04/2000US6046333 Convergent process for the preparation of a growth hormone secretagogue
04/04/2000US6046211 Amidino derivatives useful as nitric oxide synthase inhibitors
04/04/2000US6046136 Herbicidal heterocyclic N-oxides compounds
04/04/2000US6045398 Battery accepting unit and battery pack
04/04/2000CA2107432C Quaternary basic amides, method of preparing them and pharmaceutical compositions in which they are present
03/2000
03/30/2000WO2000017200A1 Tetrahydropyridoethers
03/30/2000WO2000017199A1 Process for the production of a naphthyridine carboxylic acid derivative (methanesulfonate sesquihydrate)