Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
10/1999
10/12/1999CA1340782C Naphthyridone antibacterial compounds
10/07/1999WO1999050249A2 Pyrimidines and triazines as integrin antagonists
10/07/1999WO1999049864A1 Indole-2,3-dione-3-oxime derivatives for therapeutic use
10/07/1999DE3153481C2 New herbicides and intermediates
10/07/1999DE19815020A1 Neue substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel New substituted indolinones, their preparation and their use as medicaments
10/07/1999CA2333927A1 Pyrimidines and triazines as integrin antagonists
10/07/1999CA2326576A1 Indole-2,3-dione-3-oxime derivatives for therapeutic use
10/06/1999EP0947515A1 Novel naphthyridine derivatives
10/06/1999EP0947514A1 Novel phenanethridinium derivatives
10/06/1999EP0947513A1 Tricyclic amine derivatives
10/06/1999EP0946567A1 Novel counterparts of camptothecin, their application as medicine and pharmaceutical compositions containing them
10/06/1999EP0946566A1 Pro-drugs and counterparts of camptothecin, their application as medicines
10/06/1999EP0946555A1 Pyrrole derivatives, their preparation and pharmaceutical compositions containing them
10/06/1999EP0946554A1 Fused bicyclic pyrimidine derivatives
10/06/1999EP0946550A1 PREPARATION OF 1S- 1a,2b,3b,4a(S*)]]-4- 7- 1-(3-CHLORO-2-THIENYL) METHYL]PROPYL]AMINO]-3H-IMIDAZO 4,5-b]PYRIDIN-3-yl]-N-ETHYL-2,3-DIHYDROXYCYCLOPENTANECARBOXAMIDE
10/06/1999EP0946549A1 Combinatorial process for preparing fused pyrimidine libraries
10/06/1999EP0946523A1 Fused polycyclic 2-aminopyrimidine derivatives, their preparation and their use as protein tyrosine kinase inhibitors
10/06/1999EP0946519A1 Benzamide derivatives having a vasopressin antagonistic activity
10/06/1999EP0946518A1 Modulators of proteins with phosphotyrosine recognition units
10/06/1999EP0946509A1 Novel heterocyclically substituted benzamides and their use in fighting diseases
10/06/1999EP0946175A1 USE OF AN H+, K+ -ATPase INHIBITOR IN THE TREATMENT OF NASAL POLYPS
10/06/1999EP0946165A1 Integrin antagonists
10/06/1999EP0946164A1 Integrin antagonists
10/06/1999CN1230958A Oxazolone derivatives and their use as anti-helicobacter pylori agents
10/06/1999CN1045442C Levo- and dextro- chloroscouriline (tetrahydroprotoberberines) and preparation and application thereof
10/05/1999US5962683 Oxazoline compounds as stabilizers
10/05/1999US5962502 Polyamidic acid derivatives with antigastrin activity, a method for their preparation, and their pharmaceutical use
10/05/1999US5962479 Psychological and nervous sytem disorders
10/05/1999US5962470 Heterocyclic compounds having anti-diabetic activity and their use
10/05/1999US5962468 Antibacterial activity
10/05/1999US5962467 Derivatives of swainsonine and their use as therapeutic agents
10/05/1999US5962462 Spiro-substituted azacycles as modulators of chemokine receptor activity
10/05/1999US5962457 2,3 Disubstituted- (5,6)-heteroarylfused-pyrimidine-4-ones
10/05/1999CA2175204C Certain fused pyrrolecarboxanilides; a new class of gaba brain receptor ligands
09/1999
09/30/1999WO1999048892A1 Pyrazolo-pyridine derivatives as ligands for gaba receptors
09/30/1999WO1999042465A3 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
09/30/1999CA2324266A1 Pyrazolo-pyridine derivatives as ligands for gaba receptors
09/29/1999EP0945435A1 Novel pyridonecarboxylic acid derivatives or salts thereof and drugs containing the same as the active ingredient
09/29/1999EP0944631A1 Novel substituted pyrazole derivatives for the treatment of cardiocirculatory diseases
09/29/1999EP0944629A1 Biaryl-pyridoquinazolinone derivatives as anti-cancer agents
09/29/1999EP0944628A1 Hetero-biaryl-pyridoquinazolinone derivatives as anti-cancer agents
09/29/1999EP0944627A1 8-azabicyclo 3.2.1]octane-, 8-azabicyclo 3.2.1]oct-6-ene-, 9-azabicyclo 3.3.1]nonane-, 9-aza-3-oxabicyclo 3.3.1]nonane- and 9-aza-3-thiabicyclo 3.3.1]nonane derivatives, their preparation and their use as insecticides
09/29/1999EP0944619A1 Novel integrin receptor antagonists
09/29/1999EP0944386A1 Sulfonic acid or sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
09/29/1999CN1230196A Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn.
09/29/1999CN1230187A Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
09/29/1999CN1230186A Pyrazolopyridine compound and pharmaceutical use thereof
09/29/1999CN1230185A Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
09/29/1999CN1230184A Arylamino fused pyridines and pyrimidines
09/29/1999CN1230110A Cell adhesion inhibitors
09/29/1999CN1045295C Process for prepn. of 14,15-dihydro-14-hydroxy-(3,16)-eburnamenine-14-carboxylic acid
09/28/1999US5959116 Pyridine-2, 3-dicarboximides their preparation and their use for controlling undesired plant growth
09/28/1999US5959111 Treating an octahydro-1,6,7,8-indolizinetetrol with bis/tributyltin/oxide in an organic solvent and then treating the reaction mixture with alkyl or phenyl acid halide
09/28/1999US5959109 Compounds and methods for increasing endogenous levels of corticotropin-releasing factor
09/28/1999US5958947 DNA-affinic hypoxia selective cytotoxins
09/28/1999US5958944 Treatment of circulatory diseases in coronary, cerebral, renal and peripheral arteries, as a therapeutic agent for hypertension, angina pectoris, and renal and peripheral circulation disorder, antiasthmatic agent
09/28/1999US5958943 A!-anellated pyrrole derivatives and their use in pharmacology
09/28/1999US5958942 Tricyclic nitrogen ring compounds, their production and use
09/28/1999US5958936 For inducing antiandrogenic activity in warm-blooded animals, including humans
09/28/1999US5958930 Treating cancer, and secondary infections caused by pneumocystis carinii and toxoplasmosis gondii in immunocompromised patients.
09/28/1999US5958926 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
09/28/1999US5958920 Aralkyl diazabicycloalkane derivatives for CNS disorders
09/28/1999US5958683 Screening method using the RZR receptor family
09/28/1999CA2181351C Process and intermediates for preparing naphthyridonecarboxylic acid salts
09/23/1999WO1999047549A1 PIPERAZINES AS INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE (FBPase)
09/23/1999WO1999047522A1 Granulatimide derivatives for use in cancer treatment
09/23/1999WO1999047521A1 HYPNOTIC β-CARBOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINAL PRODUCTS
09/23/1999WO1999047490A1 Bicyclo[2.2.1]heptanes and related compounds
09/23/1999CA2324270A1 Hypnotic .beta.-carboline derivatives, process for their preparation and their use as medicinal products
09/23/1999CA2289621A1 Piperazines as inhibitors of fructose-1,6-bisphosphatase (fbpase)
09/22/1999EP0943615A1 1,4-dihydropyridine derivatives
09/22/1999EP0942906A2 Compounds useful for inhibition of farnesyl protein transferase
09/22/1999EP0942722A1 Tetrahydro-beta-carboline compounds
09/22/1999CN1229412A Inhibitors of interleukin-1'beta' converting emzyme
09/22/1999CN1229082A Amine compound and its acid addition salt
09/22/1999CN1229080A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229079A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229078A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1045206C Method for preparing cyclic amide derivative
09/21/1999US5955615 Couplers
09/21/1999US5955613 Agonists or antagonists at human corticotropin-releasing factor 1 (crf1) receptors and are useful in the diagnosis and treatment of treating stress related disorders such as post trumatic stress disorder (ptsd) as well as depression,
09/21/1999CA2135751C 4-mercaptoacetylamino-¬2| benzazepinone(3) derivatives, and use as enkephalinase inhibitors
09/16/1999WO1999046268A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
09/16/1999WO1999046260A1 New compounds
09/16/1999WO1999045927A1 Vitronectin receptor antagonists
09/16/1999DE19909767A1 New 1-alkoxy-polyalkyl-piperidine derivatives used as initiators in free radical polymerization processes
09/16/1999CA2323208A1 Vitronectin receptor antagonists
09/15/1999EP0941086A1 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
09/15/1999EP0741697B1 Amino acid derivatives and their use as phospholipase a2 inhibitors
09/15/1999EP0656001B1 Novel 2-substituted indane-2-mercaptoacetylamide tricyclic derivatives useful as inhibitors of enkephalinase
09/15/1999EP0641339B1 Azaspiro quinolone antibacterial agents
09/15/1999CN1228779A Spirocyclic metalloprotease inhibitors
09/15/1999CN1228778A Pyridazino [4,5-b]-quinoline 5-oxide derivatives, their preparation and their use as glycine antagonists
09/15/1999CN1228776A Cis-substituted aminocyclopropane derivatives
09/15/1999CN1228770A Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties
09/15/1999CN1228701A Heterocyclic compounds with thrombolytic activity and their use for treating thrombosis
09/15/1999CN1228431A Derivative of 2-aryl imidazo [2,1-a] isoquinoline and its use
09/15/1999CN1228424A 1-alkoxy-polyalkyl-piperidine derivatives and their use as polymerization regulators
09/15/1999CN1228422A Process for preparing naphthyridones and intermediates
09/15/1999CN1045087C Preparation of imidazopyridine derivative