Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
02/1999
02/23/1999US5874432 Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof
02/23/1999US5874427 Substituted heteroaromatic 5-HT1F agonists
02/23/1999US5874382 Cyclic sulfonamide herbicides
02/18/1999WO1999007704A1 1-aryl-1,8-naphthylidin-4-one derivative as type iv phosphodiesterase inhibitor
02/18/1999WO1999007703A1 4-AMINOPYRROLE(3,2-d) PYRIMIDINES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS
02/18/1999WO1999007696A1 Quinolizine carboxylic acid derivatives
02/18/1999WO1999007687A1 Pesticidal 4-benzyl-1,2,4-triazolin-5-one derivatives
02/18/1999WO1999007380A1 5,11-DIHYDRO-6H-DIPYRIDO[3,2-b:2',3'-e] AZEPIN-6-ONES AND THEIR USE IN THE PREVENTION OR TREATMENT OF HIV INFECTION
02/18/1999WO1999007379A1 5,6-HETEROARYL-DIPYRIDO[2,3-b:3',2'-f]AZEPINES AND THEIR USE IN THE PREVENTION OR TREATMENT OF HIV INFECTION
02/18/1999WO1999007378A1 Nicotine antagonists for nicotine-responsive neuropsychiatric disorders
02/18/1999WO1999007366A1 Swainsonine derivatives and methods for preparing the same
02/18/1999DE19735198A1 Optical resolution of cis- or trans-pyrrolo:piperidine derivatives
02/18/1999CA2295620A1 5,6-heteroaryl-dipyrido¬2,3-b:3',2'-f|azepines and their use in the prevention or treatment of hiv infection
02/18/1999CA2268190A1 1-aryl-1,8-naphthylidin-4-one derivative as type iv phosphodiesterase inhibitor
02/17/1999EP0896964A2 Perylenehydrazideimides as carbonyl derivatizing agents
02/17/1999CN1208415A Angiogenesis inhibiting pyridazinamines
02/17/1999CN1208413A Antagonists of gonadotropin releasing hormone
02/17/1999CN1208412A Antagonists of gonadotropin releasing hormone
02/17/1999CN1208347A Substituted N-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides
02/17/1999CN1042133C N-substituted azabicycloheptane derivatives, the preparation and use thereof
02/16/1999US5872256 Cyclobutenedione derivative, process for preparing the same, and nonlinear optical element
02/16/1999US5872251 Process for preparing intermediates of inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof
02/11/1999WO1999007028A1 Electroluminescent device
02/11/1999WO1999006405A1 Pyrazolo-acridine derivatives having antitumour activity
02/11/1999WO1999006404A1 1,2,4-triazolo[4,3-b]pyrido[3,2-d]pyridazine derivatives and pharmaceutical compositions containing them
02/11/1999WO1999006403A1 Tricyclic vasopressin agonists
02/11/1999WO1999006402A1 N-acylamino acid amide compounds and intermediates for preparation thereof
02/11/1999WO1999006401A1 2-ARYL-2,5-DIHYDRO-PYRAZOLO[4,3-c]QUINOLIN-3-ONES AS GABA ALPHA 5 RECEPTOR INVERSE AGONISTS
02/11/1999WO1999006400A1 Pyrazoloquinolinone derivatives as gaba alpha 5 receptor inverse agonists
02/11/1999WO1999006399A1 Aryl-substituted pyrazoloquinolinone derivatives as gaba alpha 5 receptor inverse agonists
02/11/1999WO1999006396A1 Irreversible bicyclic inhibitors of tyrosine kinases
02/11/1999WO1999006378A1 Irreversible inhibitors of tyrosine kinases
02/11/1999WO1999006372A1 Bis-acridinecarboxamides having antitumor activity
02/11/1999WO1999006368A1 Special 3-azabicyclo[3.1.0]hexanes, method for producing and modifying the same, and their use
02/11/1999WO1999006351A1 Process for converting propargylic amine-n-oxides to enaminones
02/11/1999WO1999006041A1 SUBSTITUTED ALKANOHYDROXAMIC ACIDS AND METHOD OF REDUCING TNFα LEVELS
02/11/1999WO1999006032A2 Oral pharmaceutical preparation comprising an antiulcer activity compound, and process for its production
02/11/1999CA2298935A1 1,2,4-triazolo[4,3-b]pyrido[3,2-d]pyridazine derivatives and pharmaceutical compositions containing them
02/11/1999CA2298595A1 Process for converting propargylic amine-n-oxides to enaminones
02/11/1999CA2298509A1 Special 3-azabicyclo[3.1.0]hexanes, method for producing and modifying the same, and their use
02/11/1999CA2297815A1 N-acylamino acid amide compounds and intermediates for preparation thereof
02/11/1999CA2297407A1 Tricyclic vasopressin agonists
02/11/1999CA2295295A1 Substituted alkanohydroxamic acids and method of reducing tnf.alpha. levels
02/10/1999EP0895988A1 Arylsulfonylamino hydroxamic acid derivatives
02/10/1999EP0710239B1 Novel 9-n-bicyclic nucleoside agents useful as selective inhibitors of proinflammatory cytokines
02/10/1999CN1207402A Process for preparation of quinacridone solid solutions
02/09/1999US5869691 Aminoalkyl-indoles
02/09/1999US5869686 Substituted pyrazole derivatives, processes for their preparation and their use as herbicides
02/09/1999US5869670 7-(4-aminomethyl-3-methyloxyiminopyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof
02/09/1999US5869659 Microbiocides
02/09/1999US5869655 Diamine compounds, methods of making same, method of use of same and intermediates
02/09/1999US5869500 Pyridone compounds useful in treating Alzheimer's disease
02/09/1999US5869489 Trypthophan ureas as neurokinnin antagonists
02/09/1999US5869487 Pyrido 3,4-B!pyrazines for use as thrombin inhibitors
02/09/1999US5869483 Tricyclic benzazepine vasopressin antagonists
02/09/1999US5869482 Dipyridio 2,3-b:3',2'-! azepines and their use in the prevention or treatment of HIV infection
02/09/1999CA2163274C Intermediates for producing neuroleptic perhydro-1h-pyrido¬1,2-a| pyrazines
02/04/1999WO1999005521A2 Conjugate for differentiating between healthy and unhealthy tissue
02/04/1999WO1999005116A1 Nitrophenyl-sulfonyl-imidazoles and use thereof for controlling vegetable and animal pests
02/04/1999WO1999005107A1 Vitronectin receptor antagonist
02/04/1999WO1999004795A1 Delta opioid receptor agonist for reducing ischemic damage
02/04/1999WO1999004794A1 Cyclic amine modulators of chemokine receptor activity
02/04/1999DE19733439A1 Neue 6-endo-Amino-3-azabicyclo(3.1.0)hexande, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung von Chinolon- und Naphthyridincarbonsäure-Derviaten mit verbesserten Eigenschaften New 6-endo-amino-3-azabicyclo (3.1.0) hexande, processes for their preparation and their use for the preparation of quinolone and naphthyridine-Derviaten with improved properties
02/04/1999CA2297910A1 Vitronectin receptor antagonist
02/04/1999CA2297251A1 Delta opioid receptor agonist for reducing ischemic damage
02/04/1999CA2296314A1 Cyclic amine modulators of chemokine receptor activity
02/03/1999EP0894832A2 Process for the preparation of quinacridone solid solutions
02/03/1999EP0894797A1 Novel amide derivatives and intermediates for the synthesis thereof
02/03/1999EP0894795A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them
02/03/1999EP0894003A1 N-formyl hydroxylamine containing compounds useful as ace inhibitors and/or nep inhibitors
02/03/1999EP0786996A4 Cysteine protease and serine protease inhibitors
02/03/1999CN1207101A Novel tricyclic compounds for the inhibition of the ice/ced-3 protease family of enzymes
02/03/1999CN1207100A Novel indole-2,3-done-3-oxime derivatives
02/03/1999CN1207098A Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase
02/03/1999CN1041932C Tricyclic quinoxalinedione derivatives
02/02/1999US5866598 4h-carbazol-4-ones
02/02/1999US5866588 Dual histamine (h1) and platelet activating factor (paf) receptor antagonists.
02/02/1999US5866587 Hydroxamide derivatives of fused piperidine derivatives
02/02/1999US5866586 CNS-active pyridinylurea derivatives
02/02/1999US5866580 Treating an illness caused by p. carinii and t. gondii
02/02/1999US5866579 Imidazole and imidazoline derivatives and uses thereof
01/1999
01/30/1999CA2244438A1 New benzimidazole, benzoxazole and benzothiazole derivatives, their preparation process and the pharmaceutical compositions containing them
01/28/1999WO1999003857A1 5-substituted-3-oxadiazolyl-1,6-naphthyridin-2(1h)-one derivatives
01/28/1999WO1999003832A1 Piperidine oligomers and combinatorial libraries thereof
01/28/1999WO1999003498A1 USE OF FVIIa OR FVIIai FOR THE TREATMENT OF ADVERSE CONDITIONS RELATED TO THE FVIIa MEDIATED INTRACELLULAR SIGNALLING PATHWAY
01/28/1999DE19731741A1 Konjugat zur Unterscheidung von krankhaftem und gesundem Gewebe Conjugate to distinguish between diseased and healthy tissue
01/28/1999CA2296428A1 Piperidine oligomers and combinatorial libraries thereof
01/27/1999EP0892804A1 Isoxazolidine derivatives
01/27/1999EP0892802A1 Spiro(cyclopent(b)indole-piperidines) and n-phenyl-hydrazon intermediates for their preparation, both being acetylcholinesterase and mao inhibitors
01/27/1999EP0892801A1 Acridone-derived compounds useful as antineoplastic and antiretroviral agents
01/27/1999EP0892797A1 Inhibitors of farnesyl protein transferase
01/27/1999EP0892789A1 Irreversible inhibitors of tyrosine kinases
01/27/1999EP0892787A1 NOVEL $g(a)-HYDROXYLIC ACID DERIVATIVES, THEIR PRODUCTION AND USE
01/27/1999EP0892780A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS
01/27/1999CN1206422A Growth-hormone secretagogues
01/27/1999CN1206417A 1-(1,2-disubstituted piperidinyl)-4-(fused imidazole)-piperidine derivatives
01/27/1999CN1206416A N-([1,2,4] triazoloazinyl- benzenesulfonamide and pyridinesulfonamide composes and their use as herbicides
01/27/1999CN1206414A N-acyl-2-substituted-4-(benzimidazolyl-or imidazopyridinyl-substituted pesidues)-piperidines as tachykinin antagonists
01/27/1999CN1206406A 1-(1,2-disubstituted piperidinyl)-4-substituted piperidine derivatives as tachykinin receptor antagonists
01/27/1999CN1206347A Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters