Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
01/2000
01/20/2000WO2000002870A1 Antiviral macrocyclic compounds
01/20/2000WO2000002861A1 A3 adenosine receptor antagonists
01/20/2000WO1999058518A3 Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
01/20/2000CA2336884A1 Lk6-a derivatives
01/19/2000EP0972774A2 2-Benzylthio-8-amino(1,2,4)triazolo(1,5-pyridines
01/19/2000EP0972769A1 Novel amide derivatives and medicinal compositions thereof
01/19/2000EP0972525A1 Preventives and remedies for hyperphosphatemia
01/19/2000EP0972184A1 Luminescent transition metal-ligand complex and sensor, probe, system and method based thereon for detecting polar solvents
01/19/2000EP0971928A1 Quinoline-2(1h)-one and dihydroquinoline-2(1h)-one derivatives as ligands of 5-ht, 5-ht2 and 5-ht1-like receptors
01/19/2000EP0971922A1 Tetrahydropyrido compounds
01/19/2000EP0971921A1 2-aryl-naphthyridin-4-ones as antitumor agents
01/19/2000EP0971920A1 Compounds for inhibition of gastric acid secretion
01/19/2000EP0971744A2 COMBINATION THERAPY EMPLOYING ILEAL BILE ACID TRANSPORT INHIBITING BENZOTHIEPINES AND HMG Co-A REDUCTASE INHIBITORS
01/19/2000EP0971712A1 Compositions for the inhibition of bone resorption
01/19/2000EP0792257A4 Dichroic light polarizers
01/19/2000CN1242011A Tricyclic amine derivatives
01/19/2000CN1048492C Quinuclidine derivatives and its preparation
01/19/2000CN1048490C Cyclic derivatives, pharmacecctical compositions containg the same derivatives and their use
01/18/2000US6015912 Treating arthritis, cancer, cardiovascular disorders, skin disorders, ocular disorders, inflammation, gum disease
01/18/2000US6015901 S type 2-substituted hydroxy-2-indolidinylbutyric ester compounds and process for preparation thereof
01/18/2000US6015817 Inhibitors of farnesyl-protein transferase
01/18/2000US6015813 Heterocyclic compounds and their preparation and use
01/18/2000US6015807 Protein kinase C inhibitor
01/18/2000US6015458 Process for the preparation of highly chromatic perylene pigments
01/18/2000CA2172472C Pyrido[3,2-e]pyrazinones with anti-asthmatic action and processes for their manufacture
01/18/2000CA2168764C Novel quinolone carboxylic acid derivatives
01/18/2000CA2003837C Fused heterocyclic derivatives of 1,2,3,4-tetrahydroacridine, a process for their preparation and their use as medicaments
01/13/2000WO2000001716A2 Vasculoprotector
01/13/2000WO2000001704A2 Benzimidazoles, production thereof and use thereof as medicaments
01/13/2000WO2000001697A1 Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists
01/13/2000WO2000001696A1 3-ALKYLPYRROLO[3,2-c]QUINOLINE DERIVATIVES
01/13/2000WO2000001672A1 Naphthalimidobenzamide derivatives
01/13/2000WO2000001389A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
01/13/2000WO2000001376A2 Pharmaceutical compositions and their uses for treatment of demyelinating disorders
01/13/2000CA2336714A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
01/13/2000CA2335853A1 Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists
01/13/2000CA2301510A1 3-alkylpyrrolo[3,2-c]quinoline derivatives
01/12/2000EP0970957A1 Diaza-spiro[3,5] nonane derivatives
01/12/2000EP0970086A1 Spiro compounds and the use thereof
01/12/2000EP0970082A2 Biazacyclic crf antagonists
01/12/2000EP0970080A1 Imino-aza-anthracyclinone derivatives for the treatment of amyloidosis
01/12/2000EP0970079A1 Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with n- or c-linked imidazoles
01/12/2000EP0970070A1 Phthalazines with angiogenesis inhibiting activity
01/12/2000EP0862566B1 1-(1,2-disubstituted piperidinyl)-4-substituted piperazine derivatives
01/12/2000EP0781285B1 Fused indole and quinoxaline derivatives, their preparation and use as glutamate antagonists
01/12/2000EP0781284B1 Indole-2,3-dione-3-oxime derivatives, their preparation and use
01/12/2000CN1241192A Pro-drugs and counterparts of camptothecin, their application as medicines
01/12/2000CN1241191A Counterparts of camptothecin, their application as medicine and pharmaceutical compositions contg. them
01/12/2000CN1241187A Piperazino derivs as neurokinin antagonists
01/12/2000CN1241184A Indole derivs. for treatment of osteoporosis
01/12/2000CN1048296C Process for preparation of 9-amino camptothecin
01/12/2000CN1048249C Aminopyrrolizinetone compounds
01/11/2000US6013655 Hypotensive agents; respiratory system diisorders
01/11/2000US6013654 Imidazo[1,2-A]pyridines for the treatment of CNS and cardiac diseases
01/11/2000US6013653 Processes for producing pyridoindole derivatives
01/11/2000US6013652 Spiro-substituted azacycles as neurokinin antagonists
01/11/2000US6013648 Immunomodulators
01/11/2000US6013645 Hypocholesterolemic, antiatherosclerotic and hypotriglyceridemic mercaptoacetylamide disulfide derivatives
01/11/2000US6013127 Process for the preparation of quinacridone solid solutions
01/06/2000WO2000000487A1 5-ht1f agonists
01/06/2000WO2000000473A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000WO1999017759A3 Methods of modulating serine/threonine protein kinase function with 5-azaquinoxaline-based compounds
01/06/2000CA2336254A1 5-ht1f agonists
01/06/2000CA2335921A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000CA2330110A1 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones useful as hiv reverse transcriptase inhibitors
01/05/2000EP0968250A1 Soluble chromophores having improved solubilising groups
01/05/2000EP0968211A1 Novel tetrazoles
01/05/2000EP0968210A1 Method of making arylamino triazolopyridines
01/05/2000EP0968208A1 Quinoline and quinazoline compounds useful in therapy, particularly in the treatment of benign prostatic hyperplasia
01/05/2000EP0968179A1 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
01/05/2000EP0539420B1 substituted thiazolyl and substituted pyridinyl derivatives
01/05/2000DE19829964A1 New benzimidazolyl amidine or nitrile compounds, used as thrombin inhibitors, antithrombotic agents or intermediates
01/05/2000CN1240447A Spiro-substituted azacyclic-substituted piperazino derivatives as neurokinin
01/05/2000CN1240445A Preparation of [1S-[1a,2b,3b,4a(S*)]]-4-[7-[[1-(3-chloro-2-thienyl)methyl] propyl] amino]-3H-imidazo [4,5-b] pyridin-3-y1]-n-ethyl-2
01/05/2000CN1048015C Bicyclic tetrahydro pyrazolopyridines
01/05/2000CN1048014C Substituted pyrroles compound and preparational process, medicinal compositions and use
01/04/2000US6011052 Pyrazolone derivatives as MCP-1 antagonists
01/04/2000US6011045 Inhibitors of bone resorption; anticancer agents
01/04/2000US6011044 Antiulcer agents
01/04/2000US6011029 Benzodiazepine compounds
12/1999
12/29/1999WO1999067250A1 Syntheses of a variety of lamellarin compounds and analogues
12/29/1999WO1999067239A1 Pyrazolopyridine compounds and medicinal uses thereof
12/29/1999WO1999067238A2 Tetrahydroquinoline-indole derivatives antimicrobial agents, their uses and compositions containing them
12/29/1999WO1999067235A1 Five-membered ring compounds
12/29/1999WO1999067228A1 Fluorophenyl resin compounds
12/29/1999WO1999067220A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999WO1999067219A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999WO1999066944A1 Methods for identifying novel multimeric agents that modulate receptors
12/29/1999WO1999066934A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING β-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS
12/29/1999EP0966769A1 Novel electrode materials derived from polyquinoid ionic compounds and their uses in electrochemical generators
12/29/1999EP0966468A1 Crown ether-derivatised perylenes
12/29/1999EP0966467A1 Annulated azole derivatives useful as microbicidal agents
12/29/1999EP0966466A1 PYRROLO 3,2-c]QUINOLINE DERIVATIVES CONTAINING HALOALKOXY GROUP AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF
12/29/1999EP0966461A1 Pyrazole derivatives as herbicides
12/29/1999EP0966454A1 Disubstituted bicyclic heterocycles, their production and use as medicaments
12/29/1999EP0966443A1 Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of mip-1-alpha binding to its ccr1 receptor
12/29/1999EP0966442A1 Quinoline and quinazoline derivatives having corticotropin releasing factor (crf) antagonist activity
12/29/1999EP0966323A1 Catalysts and methods for catalytic oxidation
12/29/1999CN1239949A Novel heterocyclically substituted benzamides and their use in fighting diseases
12/29/1999CA2335760A1 Fluorophenyl resin compounds