| Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
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| 09/21/2000 | DE19912690A1 New benzimidazolyl amidine or nitrile compounds, useful as thrombin inhibitors or antithrombotic agents, for treating deep leg vein thrombosis |
| 09/21/2000 | DE19912638A1 Naphthylcarbonsäureamid-substituierte Sulfonamide Naphthylcarbonsäureamid-substituted sulfonamides |
| 09/21/2000 | DE19911510A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation |
| 09/21/2000 | CA2366838A1 A method of treating bulimia nervosa and related eating disorders by administration of atypical antipsychotic medications |
| 09/21/2000 | CA2361939A1 Modified amino acid amides, pharmaceutical compositions containing these compounds and processes for preparing them |
| 09/21/2000 | CA2361810A1 Pharmaceutical composition based on polyaromatic compounds |
| 09/21/2000 | CA2361770A1 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for preparing them |
| 09/20/2000 | EP1036072A1 Thrombin receptor antagonists |
| 09/20/2000 | EP1035850A1 Inhibitors of farnesyl-protein transferase |
| 09/20/2000 | EP1035849A1 Inhibitors of farnesyl-protein transferase |
| 09/20/2000 | EP1035848A1 Substituted alkanohydroxamic acids and method of reducing tnf-alpha levels |
| 09/20/2000 | CN1267334A Method for racemic biochemical resolusion of cis- and trans-pyrrolopiperidine |
| 09/20/2000 | CN1266852A Process for aqueous preparation of small size linear quinacridone |
| 09/20/2000 | CN1056611C Pyrazolo and pyrrolopyridines, their use and intermidiates for preparing same |
| 09/19/2000 | US6121456 2-(2'Hydroxyphenyl) benzotriazoles and process for their preparation |
| 09/19/2000 | US6121451 Anticancer drugs |
| 09/19/2000 | US6121450 Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors |
| 09/19/2000 | US6121325 Naphthyl compounds promote release of growth hormone |
| 09/19/2000 | US6121308 Indole and benzimidazole antithrombotic compounds, such as 1-methyl-2-(n-(4-amidinophenyl)-aminomethyl)-5-(n-(hydroxycarbonylmethyl) -quinoline-8-sulphonylamino)-indole |
| 09/19/2000 | US6121285 Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives |
| 09/19/2000 | US6121284 Specified 1-(alkyl or cycloalkyl)-2-methyl-3-(alkoxycarbonyl)-4-(substituted pyridyl or aryl)-5-oxo-1,4,5,6,7,8-hexahydroquinoline compounds; treating sickle cell anemia, psychoses, depression |
| 09/19/2000 | US6121281 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use |
| 09/19/2000 | US6121278 Di-n-heterocyclic compounds, methods, and compositions for inhibiting parp activity |
| 09/19/2000 | US6121277 Antitumor agents |
| 09/19/2000 | US6121262 Neurokin (tachykinin) antagonists |
| 09/19/2000 | US6120793 Transdermal administering |
| 09/14/2000 | WO2000053582A1 HETEROCYCLIC COMPOUNDS HAVING EFFECT OF ACTIVATING NICOTINIC ACETYLCHOLINE α4β2 RECEPTOR |
| 09/14/2000 | WO2000053185A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone |
| 09/14/2000 | WO2000053181A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone |
| 09/14/2000 | WO2000053179A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone |
| 09/14/2000 | WO2000053178A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone |
| 09/14/2000 | WO2000037469A3 Process for preparing n6-substituted deaza-adenosine derivatives |
| 09/14/2000 | WO2000024717A3 Isoquinoline derivatives |
| 09/14/2000 | WO1999063999A8 H1-histamine receptor antagonists |
| 09/14/2000 | DE19911039A1 Abgewandelte Aminosäureamide, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung Modified amino acid amides, pharmaceutical compositions containing them and methods for their preparation |
| 09/14/2000 | CA2367130A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone |
| 09/14/2000 | CA2367126A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone |
| 09/14/2000 | CA2367116A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone |
| 09/14/2000 | CA2367113A1 6-azaindole compounds as antagonists of gonadotropin releasing hormone |
| 09/14/2000 | CA2366260A1 Heterocyclic compounds having effect of activating .alpha.4.beta.2 nicotinic acetylcholine receptors |
| 09/13/2000 | EP1034793A1 Preventives/remedies for glaucoma |
| 09/13/2000 | EP1034173A2 Method for producing 8-methoxy-quinoline carboxylic acids |
| 09/13/2000 | EP1033987A2 Aqueous suspensions of submicron 9-hydroxyrisperidone fatty acid esters |
| 09/13/2000 | EP0817787A4 Nitrogenous macrocyclic compounds |
| 09/13/2000 | EP0764166B1 Corticotropin releasing factor antagonists |
| 09/13/2000 | CN1266434A 1,2,4-triazolo [4,3-B] pyrido [3,2-D] pyridazine derivatives and pharmaceutical compositions containing them |
| 09/13/2000 | CN1266432A Bispyrido-cyclohepatne compounds useful for inhibition of farnesyl protein transferase |
| 09/13/2000 | CN1056373C Process for preparation of fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles |
| 09/12/2000 | US6117940 Solid phase synthesis of compounds such as the imidazoles, benzodiazepines, pyrazines, and steroid mimics. |
| 09/12/2000 | US6117893 Heterocyclic compounds having anti-diabetic activity and their use |
| 09/12/2000 | US6117885 Biphenyl-substituted quinoline derivatives |
| 09/12/2000 | US6117883 Useful for modulating a muscarinic receptor. |
| 09/12/2000 | US6117881 N-cinnamoyl derivatives of (β) carbolines |
| 09/12/2000 | US6117875 Prophylactic or therapeutic treatment of phosphodiesterase iv (pde-iv) and tumor necrosis factor (tnf) mediated diseases |
| 09/12/2000 | US6117861 Protein kinase C inhibitor |
| 09/12/2000 | CA2047773C Derivatives of benzofuran, benzothiophene, indole and indolizine, process for their preparation as well as the compositions containing them |
| 09/08/2000 | WO2000052010A1 Crystal modification d of 8-cyano-1-cyclopropyl-7- (1s, 6s- 2,8- diazabicyclo- [4.3.0] nonan-8-yl) -6-fluoro -1,4-dihydro -4-oxo -3-quinoline carboxylic acid |
| 09/08/2000 | WO2000052009A1 Crystal modification c of 8-cyano-1-cyclopropyl-7- (1s, 6s-2,8- diazabicyclo -[4.3.0] nonan-8-yl) -6-fluoro-1,4-dihydro-4-oxo-3-quinoline carboxylic |
| 09/08/2000 | WO2000052008A1 Pyrazolopyridines |
| 09/08/2000 | WO2000051608A1 3-thienyl and 3-furanyl pyrrolidine modulators of chemokine receptor activity |
| 09/08/2000 | WO2000037465A3 Novel derivatives of swainsonine, processes for their preparation, and their use as therapeutic agents |
| 09/08/2000 | WO2000037021A3 Products comprising trihydroxystilbenes and derivatives thereof and methods for their manufacture and use |
| 09/08/2000 | WO2000018769A3 INDOLO[2,1-b]QUINAZOLE-6,12-DIONE ANTIMALARIAL COMPOUNDS AND METHODS OF TREATING MALARIA THEREWITH |
| 09/08/2000 | WO2000012497B1 Quinazoline derivatives as medicaments |
| 09/08/2000 | CA2362804A1 Crystal modification d of 8-cyano-1-cyclopropyl-7- (1s, 6s- 2,8- diazabicyclo- [4.3.0] nonan-8-yl) -6-fluoro -1,4-dihydro -4-oxo -3-quinoline carboxylic acid |
| 09/08/2000 | CA2362801A1 Crystal modification c of 8-cyano-1-cyclopropyl-7-(1s, 6s-2,8- diazabicyclo-[4.3.0]nonan-8-yl)-6-fluoro-1,4-dihydro-4-oxo-3-quinoline carboxylic |
| 09/06/2000 | EP1032574A2 INDOLO 2,1-b]QUINAZOLE-6,12-DIONE ANTIMALARIAL COMPOUNDS AND METHODS OF TREATING MALARIA THEREWITH |
| 09/06/2000 | EP0697864B1 Use of ferrioxamine b in the treatment os septic shock |
| 09/06/2000 | EP0593766B1 Pyridonecarboxylic acid derivative |
| 09/06/2000 | CN1265661A N-acylamino acid amide compounds and intermediates for preparation thereof |
| 09/06/2000 | CN1265650A Special 3-azabicyclo [3,1,0] hexanes, method for producing and modifying the same, and their use |
| 09/06/2000 | CN1265590A Substituted alkanohydroxamic acid and method of reducing TNF 'alpha' levels |
| 09/06/2000 | CN1056140C Biphenyl derivatives, their preparation and theirt use for treatment of hypertension and cardiac disease |
| 09/05/2000 | US6114531 Reacting 7-chloro-1-(2,4-difluorophenyl)-6-fluoro-1,4-dihydro-4-oxo-1,8 -naphthyridine-3-carboxylic acid with a fused aminoaromatic salt to from trovafloxacin |
| 09/05/2000 | US6114529 Useful for preparing camptothecin derivatives having antitumor activities |
| 09/05/2000 | US6114526 Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases |
| 09/05/2000 | US6114351 N-oxides as antibacterial agents |
| 09/05/2000 | US6114339 Derivatives of pyrido [2,3-D] and [3,2-D] pyrimidine method of using these derivatives |
| 09/05/2000 | US6113527 3,3-bis-hydroxymethyl-7-(cis-4-isopropyl-cyclohexyl)-1-phenyl -1,7-diaza-spiro-(3.5)nonane-2-one, for example; agonists of the orphanin fq (ofq) receptor; useful in the treatment of psychiatric, neurological and physiological disorders |
| 09/05/2000 | CA2020340C Enantioselective synthesis of antifolates |
| 08/31/2000 | WO2000050424A1 [1,8] naphthyridine derivatives having antiviral activity |
| 08/31/2000 | WO2000050406A1 Isoquinoline derivatives and isoquinoline combinatorial libraries |
| 08/31/2000 | WO2000012074A3 Use of piperidines and/or piperazines as inhibitors of p38-alpha kinase |
| 08/31/2000 | WO2000007996A3 Pyrazoles as estrogen receptor modulators |
| 08/31/2000 | DE19908449A1 Kristallmodifikation C von Crystal modification of C 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicylo-[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chino/incarbonsäure |
| 08/31/2000 | DE19908448A1 Kristallmodifikation D von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicylo[4.3.0)nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chino incarbonsäure Crystal modification D of 8-cyano-1-cyclopropyl-7- (1S, 6S-2,8-diazabicyclo [4.3.0) nonane-8-yl) -6-fluoro-1,4-dihydro-4-oxo-3 -chino incarbonsäure |
| 08/31/2000 | CA2364652A1 ¬1,8| naphthyridine derivatives having antiviral activity |
| 08/30/2000 | EP1031615A2 Aqueous process for the preparation of linear quinacridones having a reduced particle size |
| 08/30/2000 | EP1031575A1 Process for preparing growth hormone secretagogues |
| 08/30/2000 | EP1031571A1 Sulfamoyl compounds and agricultural or horticultural bactericide |
| 08/30/2000 | EP1030843A1 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them |
| 08/30/2000 | EP0765328B1 Pirydyl imidazole derivatives and processes for the preparation thereof |
| 08/29/2000 | US6110939 As a substance p antagonists treating tachykinin-mediated disease, asthma, central nervous system disorder |
| 08/29/2000 | US6110938 1-(arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-4-(heteroaryl)piperidines and related compounds useful as antipsychotics and analgesics |
| 08/29/2000 | US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor |
| 08/29/2000 | US6110932 Increase the level of endogenous growth hormone for the treatment and prevention of osteoporosis, congestive heart failure, frailty associated with aging, obesity; accelerating bone fracture repair, accelerating wound healing |
| 08/29/2000 | US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
| 08/29/2000 | US6110919 Diazabicyclic neurokinin antagonists |
| 08/29/2000 | US6110910 Antiinflammatory agents, antiarthritic agents, antirheumatic agents, anticarcinogenic agents |
| 08/26/2000 | CA2299494A1 Aqueous process for the preparation of linear quinacridones having a reduced particle size |