Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
04/2003
04/22/2003US6552018 As antitumor agents
04/22/2003CA2253951C .delta.1,2bicyclo[4,4,0] functional dyes for contrast enhancement in optical imaging
04/22/2003CA2239187C Inhibitors of farnesyl protein transferase
04/22/2003CA2079646C Succinimide derivatives of 2,5-dimercapto-1,3,4-thiadiazole
04/19/2003CA2361863A1 Composition and method for use of pyridinium derivatives in cosmetic and therapeutic applications
04/17/2003WO2003031440A1 3,4-di-substituted maleimide compounds as cxc-chemokine receptor antagonists
04/17/2003WO2003031437A1 Propylcarbamate derivatives as inhibitors of serine and cysteine proteases
04/17/2003WO2003031436A1 Heterocyclic compounds for use in the treatment of disorders of the urinary tract
04/17/2003WO2003031435A1 Pyrazole derivatives as glycine transporter inhibitors
04/17/2003WO2003031428A1 Stereospecific process for the synthesis of 2-yl chroman derivatives
04/17/2003WO2003031422A1 Novel benzothiazine derivatives, their preparation and use
04/17/2003WO2003031420A1 Isothiazole derivatives
04/17/2003WO2003031419A1 Substituted diphenyloxazoles, the synthesis thereof, and the use thereof as fluorescence probes
04/17/2003WO2003031414A1 Novel heterocyclic compound and anti-inflammatory agent
04/17/2003WO2003031407A2 β-LACTAMYL VASOPRESSIN VlaANTAGONISTS
04/17/2003WO2003031397A1 Acylsulfonamides as inhibitors of steroid sulfatase
04/17/2003WO2003031376A1 Solid phase synthesis of substituted 1,5-benzodiazepine-2-one and 1,5-benzothiazepine-2-one
04/17/2003WO2003030909A1 2- and 4-aminopyrimidines n-substtituded by a bicyclic ring for use as kinase inhibitors in the treatment of cancer
04/17/2003WO2003030898A1 Modulators of ccr5 chemokine receptor activity
04/17/2003WO2003013484A3 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents
04/17/2003WO2003006454A3 Heterocyclic carboxamides and their use as fungicides
04/17/2003WO2002069968A8 New use
04/17/2003WO2001094341A9 Quinazoline derivatives for the treatment of tumours
04/17/2003WO2001017965A3 Cyanopiperidines as pesticides
04/17/2003US20030073852 Anticancer agents
04/17/2003US20030073850 Incontinence; nasal congestion
04/17/2003US20030073842 Psychological disorders; hypotensive agents
04/17/2003US20030073836 Heteroarylcarboxylic acid amides, the preparation thereof and their use as pharmaceutical compositions
04/17/2003US20030073834 Purine compounds having PDE IV inhibitory activity and methods of synthesis
04/17/2003US20030073732 Antiinflammatory agents
04/17/2003US20030073726 Heterocyclic inhibitors of glycine transporter 2
04/17/2003US20030073718 Enzyme inhibitors; cardiovascular disorders; antiinflammatory agents; autoimmune disease
04/17/2003US20030073706 Fused thiophone derivatives and drugs containing the same as the active ingredient
04/17/2003US20030073687 Alzheimer's disease; anticancer agents; antidiabetic agents
04/17/2003US20030073684 Respiratory system disorders; cardiovascular disorders; hemorrhage therapy
04/17/2003US20030073682 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors
04/17/2003US20030073677 Synergistic mixtures; anticancer agents; 2-(2 -methyl-4-thiazolyl)ethenyl)-4,17-dioxabicyclo(14.1.0)heptadecane-5,9 -dione or 4-aza-17-oxabicyclo(14.1.0) heptadecane-5,9-dione or 1-aza-13-cyclohexadecene-2,6-dione or 1-oxa-13-cyclohexadecene-2,6-dione derivatives
04/17/2003US20030073669 N-heterocyclic derivatives as NOS inhibitors
04/17/2003US20030073205 Production of polyketides
04/17/2003US20030073047 Forms an azomethine dye upon a coupling reaction with an oxidized product of a developing agent
04/17/2003CA2462862A1 3,4-di-substituted maleimide compounds as cxc-chemokine receptor antagonists
04/17/2003CA2462860A1 Stereospecific process for the synthesis of 2-yl chroman derivatives
04/17/2003CA2462000A1 Substituted diphenyloxazoles, the synthesis thereof, and the use thereof as fluorescence probes
04/17/2003CA2458456A1 Heterocyclic compounds for use in the treatment of disorders of the urinary tract
04/17/2003CA2458453A1 Acylsulfonamides as inhibitors of steroid sulfatase
04/17/2003CA2458388A1 Novel benzothiazine derivatives, their preparation and use
04/16/2003EP1302468A1 Processes and intermediates for manufacturing retroviral protease inhibiting compounds
04/16/2003EP1302467A2 Process for the preparation of substituted thiazoline derivatives and their intermediate
04/16/2003EP1302466A1 Benzoxazole compound, process for producing the same, and herbicide
04/16/2003EP1302463A1 Medicine comprising dicyanopyridine derivative
04/16/2003EP1302462A1 Sulfone derivatives, process for their production and use thereof
04/16/2003EP1302461A1 Tnf-alpha production inhibitors
04/16/2003EP1301487A2 Viral polymerase inhibitors
04/16/2003EP1301484A2 Capsaicin receptor ligands
04/16/2003EP1301483A1 1-aryl-4-alkyl halide-2(1h)-pyridones and their use as herbicides
04/16/2003EP1301482A1 Cyclic amine phenyl beta-3 adrenergic receptor agonists
04/16/2003EP1301481A1 Pyrrole derivatives for treating aids
04/16/2003EP1301480A1 1,3-disubstituted and 1,3,3-trisubstituted pyrrolidines as histamine-3 receptor ligands and their therapeutic applications
04/16/2003EP1181017B1 Metalloprotease inhibitors
04/16/2003EP0880508B1 Quinazoline derivatives as vegf inhibitors
04/16/2003CN1411460A Substituted homopiperidinyl benzimidazole analogues as fundic relaxants
04/16/2003CN1411457A Substituted pyrroles
04/16/2003CN1411456A Chemokine receptor binding heterocyclic compounds
04/16/2003CN1411445A Method for preparing 3-hydroxypicolinic acid derivatives
04/16/2003CN1411379A Preventives or remedies for arrhythmia
04/16/2003CN1105718C Improved method for producing thiazolidinediones, and new thiazolidinediones
04/16/2003CN1105707C Pyrazole derivative
04/16/2003CN1105706C Cyclic amidino agents useful as nitric oxide synthase inhibitors
04/15/2003US6548667 For prevention and treatment of diseases caused by overexpression and overactivation of matrix metalloproteinase
04/15/2003US6548666 Tricyclic compounds and their use in medicine process for their preparation and pharmaceutical compositions containing them
04/15/2003US6548638 Peptoid and nonpeptoid containing α-keto oxadiazoles as serine protease inhibitors
04/15/2003US6548526 Isothiazole derivatives useful as anticancer agents
04/15/2003US6548516 (NMDA=N-methyl-D-aspartate); where the heteroaryl is 3H-benzoxazol-2-one, 3H-benzothiazol-2-one, 3H-benzimidazol-2-one or indolin-2-one; excitatory amino acid antagonists for combating neurodegenerative disorders
04/15/2003US6548512 Nitrogen containing heteroaromatics as factor Xa inhibitors
04/15/2003US6548499 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
04/15/2003US6548495 Dihydro-benzo [B] [1,4] diazepin-2-one derivatives
04/15/2003US6548481 A salt form of a dipeptide compound formed from an amino acid and a thiazolidine or pyrrolidine group, and the salts are selected from acetates, tartrates, fumarates, succinates, phosphates and sulfates
04/15/2003US6548451 Use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
04/15/2003CA2274338C Ziprasidone formulations
04/15/2003CA2169737C Endothelin antagonistic heteroaromatic ring-fused cyclopentene derivatives
04/15/2003CA2099588C Prevention of synovial adhesions
04/15/2003CA2037975C 5-hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors
04/10/2003WO2003029251A1 Novel process for the synthesis of thiazolidinedione derivatives
04/10/2003WO2003029250A1 Benzisothiazolyl-substituted aminomethyl chromanes for treating diseases of the central nervous system
04/10/2003WO2003029249A1 Thiazolyl substituted aminopyrimidines as plant protection agents
04/10/2003WO2003029248A1 N-(4-(4-methylthiazol-5-yl) pyrimidin-2-yl) -n-phenylamines as antiproliferative compounds
04/10/2003WO2003029238A1 Chroman derivatives as 5-hydroxytryptamine-6 ligands
04/10/2003WO2003029215A1 4[piperidin-4-yliden-(3-carbamoylphenyl)methyl] benzamide derivatives and their use for the treatment of pain, spinal injuries or gastrointestinal disorders
04/10/2003WO2003029210A2 Heteroaryl substituted tetrazole modulators of metabotropic glutamate receptor-5
04/10/2003WO2003029195A1 Intermediates for epothilone derivative and process for producing these
04/10/2003WO2003028729A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
04/10/2003WO2003028720A1 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
04/10/2003WO2003028719A1 Substituted 2,5-diamidoindoles as ece inhibitors for the treatment of cardiovascular diseases
04/10/2003WO2003028650A2 Benzimidazolidinone derivatives as muscarinic agents
04/10/2003WO2003028641A2 Mch receptor antagonists
04/10/2003WO2003028458A1 N-thio-nicotinamide derivatives and related compounds for use as pesticides
04/10/2003WO2003004493A8 Novel compounds, their preparation and use
04/10/2003WO2002094203A3 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
04/10/2003WO2002078596A3 Novel dyeing composition for dyeing keratinous fibres comprising a particular dicationic diazo dye
04/10/2003WO2002070540A3 Peptide deformylase inhibitors