Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
01/2003
01/23/2003WO2003006443A2 2- 4-(naphtalin-2-yl)-thiazol-2-ylaminocarbonyl benzoic acid and 2- 4-(naphtalin-2-yl)-pyrimidin-2-ylaminocarbonyl benzoic acid and additional compounds serving as telomerase inhibitors for use in tumor therapy
01/23/2003WO2003006440A2 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
01/23/2003WO2003006437A1 Imidazole derivatives as adenosine deaminase inhibitors
01/23/2003WO2003006423A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003WO2003006015A1 Substituted thiazoles and oxazoles as corticotropin releasing hormone ligands
01/23/2003WO2003006012A1 Compounds and methods for the inhibition of trypanosoma cruz i
01/23/2003WO2003005824A2 Substituted 3-heteroaryl (amino-or-oxy)-pyrrolidin-2-ones, method for the production thereof and use thereof as herbicides or as plant growth regulators
01/23/2003WO2002050066A3 Pyrazole compounds useful as protein kinase inhibitors
01/23/2003WO2002046171A3 Anilinopyrimidine derivatives as ikk inhibitors and compositions and methods related thereto
01/23/2003WO2002044174A3 3-(2,4-dimethylthiazol-5-yl) indeno[1,2-c]pyrazol-4-one derivatives as cdk inhibitors
01/23/2003WO2002036562A3 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
01/23/2003US20030018199 Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors
01/23/2003US20030018193 Beta-alanine derivatives and their use as receptor anatgonists
01/23/2003US20030018059 Antiinflammatory agents; antihistamines; antiallergens
01/23/2003US20030018053 Substituted indolealkanoic acids
01/23/2003US20030018046 Chemokine receptor binding heterocyclic compounds
01/23/2003US20030018045 Heterocyclic beta-3 adrenergic receptor agonists
01/23/2003US20030018034 Piperazine compounds and medicinal use thereof
01/23/2003US20030018022 Antiinflammatory agents; antiallergens
01/23/2003US20030018021 Piperidine derivatives as subtype selective N-methyl-D-aspartate antagonists
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003CA2453421A1 Substituted benzo-nitro-heterocycles
01/23/2003CA2453396A1 Compounds and methods for the inhibition of trypanosoma cruzi
01/23/2003CA2453175A1 Interaction inhibitors of tcf-4 with beta-catenin
01/23/2003CA2452513A1 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
01/23/2003CA2449243A1 Protease inhibitor conjugates and antibodies useful in immunoassay
01/23/2003CA2417156A1 3,4-dihydroisoquinoline derivative compound and a pharmaceutical agent comprising it as active ingredient
01/22/2003EP1277753A1 Thiazolidinedione derivative and its use as antidiabetic
01/22/2003EP1277752A1 Process for producing optically active sulfoxide derivative
01/22/2003EP1277751A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277749A1 2- and 2,5-substituted phenylketo enols
01/22/2003EP1277743A1 Oxa(thia)zolidine derivative and anti-inflammatory drug
01/22/2003EP1277741A1 Cyclic compounds
01/22/2003EP1277738A1 Condensed heteroaryl derivatives
01/22/2003EP1277735A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277734A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277733A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277729A1 Ppar (gamma) modulators
01/22/2003EP1276740A2 Novel epothilone derivatives, method for the preparation thereof and their pharmaceutical use
01/22/2003EP1276739A2 Heterocycles that are inhibitors of impdh enzyme
01/22/2003EP1276730A2 Thiazolidinedione analogues and their use for the treatment of diabetes
01/22/2003EP1276726A2 Substituted phenyl farnesyltransferase inhibitors
01/22/2003EP1276725A2 5-substituted tetralones as inhibitors of ras farnesyl transferase
01/22/2003EP1276723A2 Pyrazole compounds having anti proliferative activity
01/22/2003EP1030835B1 Urea derivatives and their use as integrin inhibitors
01/22/2003EP1006114B1 Pyrazole derivatives and cox inhibitors containing them
01/22/2003EP0898562B1 Hydroxamic acid derivatives for use with the treatment of diseases related to connective tissue degradation
01/22/2003EP0646115B1 Heterocyclic-cyclic amine derivatives
01/22/2003CN1392874A Cyclic amidine compounds
01/22/2003CN1392144A 3-amino-2-mercapto phenyl formic acid erivative and its preparation
01/21/2003US6509358 For therapy of metabolic disorders related to insulin resistance or hyperglycemia, typically associated with obesity or glucose intolerance), atherosclerosis, gastrointestinal disorders, neurogenic inflammation, glaucoma
01/21/2003US6509339 Gastrointestinal disorders; cardiovascular disorders
01/21/2003US6509335 This invention discloses benzoxazinone and benzothiazinone compounds which display inhibitory effects on serine proteases such as factor Xa, thrombin, and/or factor VIIa. The invention also discloses pharmaceutically acceptable salts of
01/21/2003US6509334 Cyclocarbamate derivatives as progesterone receptor modulators
01/21/2003US6509331 Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds
01/21/2003US6509328 Glutamate receptor antagonists
01/16/2003WO2003004493A1 Novel compounds, their preparation and use
01/16/2003WO2003004489A1 Compositions and methods for inhibiting prenyltransferases
01/16/2003WO2003004467A2 Thiazole benzamide derivatives and pharmaceutical compositions for inhibiting cell proliferation, and methods for their use
01/16/2003WO2003004028A1 Tetrahydroquinoline derivatives
01/16/2003WO2003004027A1 Substituted anilinic piperidines as mch selective antagonists
01/16/2003WO2003004020A1 Heteroaryl carboxylic acid amides, the production thereof and the use of the same as inhibitors of the microsomal triglyceride transfer protein (mtp)
01/16/2003WO2002051837A3 Heterocyclindazole and azaindazole compounds as 5-hydroxytryptamine-6 ligands
01/16/2003WO2002050062A3 Benzimidazole and pyridylimidazole derivatives as ligands for gaba receptors
01/16/2003WO2002046129A3 Inhibitors of histone deacetylase
01/16/2003WO2002012196A3 Lactam compounds and their use as inhibitors of serine proteases and method
01/16/2003WO2001074898A3 Charged compounds comprising a nucleic acid binding moiety and uses therefor
01/16/2003US20030013886 Such as (E)-1-(2-Pyridyl)-2-styryl-1H-benzimidazole; antiinflammatory and analgesic agents; prostaglandin inhibitors
01/16/2003US20030013875 3-azabicyclo[3.1.0]hexane derivatives useful in therapy
01/16/2003US20030013874 Non-opioid analgesics for chronic and acute pain; 1-[1-(p-phenylbenzyl)-4-piperidinyl]-2,1,3-benzothiadiazol-2,2-dione; modulation of the opioid and ORL I receptors; agonist or antagonist activity at the CNS mu, delta and kappa receptors greater than morphine
01/16/2003US20030013751 Viricides; enzyme inhibitors
01/16/2003US20030013750 Bactericides; fungicides; miticides; nematocides; for agriculture
01/16/2003US20030013742 Antiinflammatory agents; skin disorders
01/16/2003US20030013741 Antihistamines; antiallergens
01/16/2003US20030013725 Amino acid derivatives
01/16/2003US20030013724 Novel prolines as antimicrobial agents
01/16/2003US20030013712 Antiinflammatory agents
01/16/2003US20030013708 Therapeutic heterocyclic compounds
01/16/2003US20030013706 Autoimmune disease; antiinflammatory agents
01/16/2003US20030013041 Write-once optical data carrier
01/16/2003CA2454613A1 Substituted anilinic piperidines as mch selective antagonists
01/16/2003CA2452609A1 Thiazole benzamide derivatives and pharmaceutical compositions for inhibiting cell proliferation, and methods for their use
01/16/2003CA2448913A1 Sulfone containing bicyclic aromatic ring compounds, their preparation and use as nicotinic acetyl-chloine receptors
01/15/2003WO2002006233A1 1-aryl-4-alkyl halide-2(1h)-pyridones and their use as herbicides
01/15/2003EP1275648A1 Epothilone minor constituents
01/15/2003EP1275644A1 Benzenesulfonamide derivatives, process for their preparation and pharmaceutical compositions containing them
01/15/2003EP1275641A2 Benzenesulfonamide derivatives, process for their preparation and pharmaceutical compositions containing them
01/15/2003EP1275301A1 Trisubstituted heterocyclic compounds and their use as fungicides
01/15/2003EP1274708A1 Herbicidal 3-heterocyclic substituted benzisothiazole and benzisoxazole compounds
01/15/2003EP1274707A1 Therapeutically useful new salts of cck inhibitors, process for the preparation thereof and pharmaceutical preparations containing them
01/15/2003EP1274705A1 2-substituted 4-heteroaryl-pyrimidines and their use in the treatment of proliferative disorders
01/15/2003EP1274701A1 Chemical compounds
01/15/2003EP1274696A1 Oxime derivatives for controlling undesired microorganisms and animal pests
01/15/2003EP1274692A1 Quinazoline compounds
01/15/2003EP1274683A2 Heterocyclic acylsulfimides, a method for their production, agents containing the same and their use as pesticides
01/15/2003EP1274407A2 Uses of ppar-gamma agonists in neutrophil-induced diseases
01/15/2003EP1023265B1 Azetidinone derivatives for the treatment of hcmv infections
01/15/2003EP0934938B1 Substituted benzoylaminothiazole derivatives and drugs containing the same
01/15/2003EP0925287B1 Heterocyclic metalloprotease inhibitors
01/15/2003EP0787723B1 Cyclopropachromenecarboxylate derivatives