Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
03/2003
03/05/2003EP1286964A1 Heterocyclic inhibitors of glycogen synthase kinase gsk-3
03/05/2003EP1286673A2 Ligands of integrin receptors
03/05/2003EP1202984B1 diphenyl-piperidine derivate
03/05/2003EP1194427B1 Thiophene-ethyl thiourea compounds and use in the treatment of hiv
03/05/2003EP1115719B1 Novel amidine derivatives, their preparation and application as medicines and pharmaceutical compositions containing same
03/05/2003EP1021411B1 Benzamide derivatives as thrombin inhibitors
03/05/2003EP0892791B1 N-[[4-(5-METHYL-3-PHENYLISOXAZOL-4-YL]PHENYL]SULFONYLPROPYLAMIDE and its SODIUMSALT AS PRODRUGS OF COX-2 INHIBITORS
03/05/2003EP0832069B1 BIPHENYL-2-CARBOXYLIC ACID-TETRAHYDRO-ISOQUINOLIN-6-YL AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND/OR APOLIPOPROTEIN B (Apo B) SECRETION
03/05/2003CN1400898A 回旋酶抑制剂及其用途 Gyrase inhibitors and their use
03/05/2003CN1102593C N-[4(heteroarylmethyl)phenyl]-heteroarylamines compound
03/05/2003CN1102583C Cationic polypeptide condensing agent of thiazole,its synthesizing process and its application
03/05/2003CN1102580C Arylethenesulfonamide derivatives and drug composition containing the same
03/05/2003CN1102573C Aryl or heteroaryl substd, 3,4-dihydroanthracene and benzo [1,2-g]-chrom-3-ene, benzo[1,2-g]-thiochrom-3-ene and benzo [1,2-g]-1,2-dihydroquinoline derivs having bioactivity of visual pigmentoid
03/04/2003US6528510 HIV protease inhibitors
03/04/2003US6528509 Pyrazole compositions useful as inhibitors of ERK
03/04/2003CA2218913C Substituted oximes, hydrazones and olefins as neurokinin antagonists
02/2003
02/27/2003WO2003016306A1 Hiv inhibiting pyrimidines derivatives
02/27/2003WO2003016303A1 Tetrazoyl oxime derivative and agricultural chemical containing the same as active ingredient
02/27/2003WO2003016302A1 Diamine derivatives
02/27/2003WO2003016286A1 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same
02/27/2003WO2003016284A1 Substituted anthranilamides for controlling invertebrate pests
02/27/2003WO2003016276A2 3-substituted oxindole beta-3 agonists
02/27/2003WO2003016275A1 Antiviral agent
02/27/2003WO2003016265A1 Cyclic compound and ppar agonist
02/27/2003WO2003015785A1 2h-phthalazin-1-ones and methods for use thereof
02/27/2003WO2003015778A1 Tyrosine kinase inhibitors
02/27/2003WO2003015776A1 2,4,5-trisubstituted thiazolyl derivatives and their antiinflammatory activity
02/27/2003WO2003015774A1 Compounds effecting glucokinase
02/27/2003WO2003015773A2 2-amino-4,5-trisubstituted thiazolyl derivatives and their use against autoimmune diseases
02/27/2003WO2003015772A1 Inhibitors of polyq-aggregation
02/27/2003WO2003015769A1 Aminoalkyl-substituted aromatic bicyclic compounds, method for the production thereof and their use as medicaments
02/27/2003WO2003015717A2 Tyrosine kinase inhibitors
02/27/2003WO2002100851A3 Thiophene derivatives as antiviral agents for flavivirus infection
02/27/2003WO2002092588A3 Aromatic sulfone hydroxamates and their use as protease inhibitors
02/27/2003WO2002089782A3 Dioxanes and uses thereof
02/27/2003WO2002089749A3 Arylsulfonamide ethers, and methods of use thereof
02/27/2003WO2002079149A3 Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases
02/27/2003WO2002074042A3 Combinations comprising an antidiarrheal agent and an epothilone or an epothilone derivative
02/27/2003WO2002067869A3 Acylated piperidine derivatives as melanocortin-4 receptor agonists
02/27/2003WO2002067675A3 Substituted 4,5-dihydro-1,2,4-triazin-6-ones, 1,2,4-triazin-6-ones, and their use as fungicides and insecticides
02/27/2003WO2002060904A3 A process for the preparation of epothilone analogs
02/27/2003WO2002060374A3 Benz-1,3-azole derivatives and their uses as heparanase inhibitors
02/27/2003US20030040631 As chemical intermediates used for the preparation of S-alpha-ethyl-2-oxo-1-pyrrolidine acetamide
02/27/2003US20030040608 Having good hue and capable of forming images having high lightfastness
02/27/2003US20030040536 For therapy of disease states in mammals that are alleviated by a protein kinase inhibitor, particularly diseases such as cancer, inflammatory disorders, restenosis, and cardiovascular disease
02/27/2003US20030040533 For use as hypoglycaemic and hypolipidaemic agents
02/27/2003US20030040524 Pyrimidine compounds and methods for making and using the same
02/27/2003US20030040518 For therapy of neurodegenerative diseases and for the regeneration or prevention of degeneration of lesioned and damaged neurons degeneration of lesioned and damaged neurons
02/27/2003US20030040513 P2x7 receptor antagonists for use in the treatment of inflammatory, immune or cardiovascular diseases
02/27/2003CA2457037A1 Aminoalkyl-substituted aromatic bicyclic compounds, method for the production thereof and their use as medicaments
02/27/2003CA2456985A1 2h-phthalazin-1-ones and methods for use thereof
02/27/2003CA2456868A1 Inhibitors of polyq-aggregation
02/27/2003CA2456841A1 Cyclohexyl and piperidine diamine derivatives useful as activated blood coagulation factor x inhibitors
02/26/2003EP1285918A1 C7 Ester substituted taxanes as antitumor agents
02/26/2003EP1285653A1 Use of alpha-1L agonists in the treatment of incontinence
02/26/2003EP1285651A1 Melanin concentrating hormone antagonists
02/26/2003EP1284970A2 Isothiazole derivatives and their use as microbicides
02/26/2003EP1284967A1 3-substituted isoquinolin-1-yl derivatives
02/26/2003EP1284737A1 Water soluble prodrugs of azole compounds
02/26/2003EP1100797B1 Heterocyclic compounds as inhibitors of rotamase enzymes
02/26/2003EP1021424B1 Thiadiazole amide mmp inhibitors
02/26/2003EP0971901B1 Phthalazinones
02/26/2003CN1399634A Hydroxyalkanoyl aminolactams and related structure as inhibitors of A beta protein production
02/26/2003CN1399631A Novel hydantoin, thiohydantoin, pyrimidinedione and thioxopyrimidinone derivatives, preparation method and use as medicines
02/26/2003CN1399515A Insecticidal and acaricidal agents
02/26/2003CN1102149C 4-haloalkyl-3-heterocycolyl pyridines and 4-haloalkyl-5-heterocyclylpyridines, method for producing same, composition containing same and use thereof
02/25/2003US6525220 Intermediates for the synthesis of benzimidazole derivatives and a process for the preparation thereof
02/25/2003US6525215 HIV protease inhibitors
02/25/2003US6525202 Cyclic amine phenyl beta-3 adrenergic receptor agonists
02/25/2003US6525193 Aminoaryl oxazolidinone N-oxides
02/25/2003US6525081 Antirheumatic
02/25/2003US6525076 Selective factor Xa inhibitors
02/25/2003US6525070 Bipiperidine derivatives as modulators of CCR3 activity and as H1 antagonists
02/25/2003US6525069 Such as N-(t-butyl)-N'-(2-((3-(4-fluorophenyl)methyl)piperi -dinyl)methyl)cyclohexyl)urea; prevention of asthma and other allergic diseases
02/25/2003US6525059 Substituted pyrazoles as p38 kinase inhibitors
02/25/2003US6525052 Compounds useful as reversible inhibitors of cysteine proteases
02/25/2003US6525036 Compounds and compositions as protease inhibitors
02/20/2003WO2003014095A1 Acylaminothiazole derivatives, their preparation and therapeutic use
02/20/2003WO2003014072A1 Disulfide and thiosulfonate ligands and libraries comprising these ligands
02/20/2003WO2003013571A1 Peptidomimetics of biologically active metallopeptides
02/20/2003WO2003013531A1 Phenyl derivatives as factor xa inhibitors
02/20/2003WO2003013518A1 Alpha-ketoamide derivatives as cathepsin k inhibitors
02/20/2003WO2003013517A1 Aminoisoxazole derivatives active as kinase inhibitors
02/20/2003WO2003013502A1 Compounds which mimic the chemical and biological properties of discodermolide
02/20/2003WO2003013484A2 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents
02/20/2003WO2002096516A8 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
02/20/2003WO2002085291A3 Nociceptin analogs
02/20/2003WO2002049993A3 High affinity small molecule c5a receptor modulators
02/20/2003WO2001079187A8 Substituted 1,4-thiazepine and analogs and their use as activators of caspases
02/20/2003US20030036655 2-(substituted-phenyl)amino-imidazoline derivatives
02/20/2003US20030036653 For prophylaxis and therapy of diseases associated with herpes viruses including human cytomegalovirus, herpes simplex viruses, Epstein-Barr virus, varicella-zoster virus, human herpesviruses- 6 and -7, and Kaposi herpesvirus
02/20/2003US20030036544 Pesticidal triazine-derivatives
02/20/2003US20030036543 Especially as inhibitors of Aurora-2 and GSK-3, for treating diseases such as cancer, diabetes and Alzheimer's disease.
02/20/2003CA2462200A1 Peptidomimetics of biologically active metallopeptides
02/20/2003CA2457814A1 Disulfide and thiosulfonate ligands and libraries comprising these ligands
02/20/2003CA2456553A1 Compounds which mimic the chemical and biological properties of discodermolide
02/20/2003CA2455631A1 Aminoisoxazole derivatives active as kinase inhibitors
02/19/2003EP1284268A1 Thiazolidinedione derivative and its use as antidiabetic
02/19/2003EP1284267A1 Triazole compounds having amide linkage
02/19/2003EP1284140A2 Use of ritonavir (ABT-538) for improving the pharmacokinetics of drugs metabolized by cytochrome P450 in a method of treating aids