Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
02/2003
02/06/2003WO2002096420A3 Method for treating nerve injury caused by surgery
02/06/2003WO2002079146A3 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
02/06/2003WO2002070516A3 Cyclopropaheterocycles as non-nucleoside reverse transcriptase inhibitors
02/06/2003WO2002059112A3 Pyrazole compounds useful as protein kinase inhibitors
02/06/2003WO2002048134A3 Di-substituted aminomethyl chroman derivative beta-3 adrenoreceptor agonists
02/06/2003WO2002041843A3 Antiinflammation agents
02/06/2003WO2002010137A9 Indazole derivatives as jnk inhibitors
02/06/2003US20030028022 Preferably tertiary amines comprising tetrahydroquinoline and benzimidazole; use treating human immunodeficiency virus (HIV) and Feline Immunodeficiency Virus (FIV)
02/06/2003US20030028018 Treating diseases characterized by activity of vascular endothelial growth factor receptor tyrosine kinases such as cancer
02/06/2003US20030027845 Ether derivatives useful as inhibitors of PDE4 isozymes
02/06/2003US20030027842 Halogenobenzimidazoles
02/06/2003US20030027829 Potassium channel inhibitors
02/06/2003US20030027798 For therapy
02/06/2003US20030027797 For therapy of metabolic disorders related to insulin resistance or hyperglycemia
02/06/2003US20030027795 N-(4-sulfonylaryl)cyclylamine-2-hydroxyethylamines as beta-3 adrenergic receptor agonists
02/06/2003US20030027794 N-heterocyclic derivatives as NOS inhibitors
02/06/2003CA2454903A1 Substituted piperazines as modulators of the melanocortin receptor
02/06/2003CA2452328A1 Substituted piperidines as modulators of the melanocortin receptor
02/05/2003EP1280802A1 Indazoles substituted with 1,1-dioxoisothiazolidine useful as inhibitors of cell proliferation
02/05/2003EP1280801A2 Hydantoin-containing glucokinase activators
02/05/2003EP1280797A1 Inhibitors of dipeptidyl peptidase iv
02/05/2003EP1280795A2 N-substituted carbamoyloxyalkyl-azolium derivatives
02/05/2003EP1280793A2 Cyclic amidine compounds and their use as alpha4beta2 nicotinic acetylcholine receptor ligands
02/05/2003EP1280789A1 Cdk inhibitors having 3-hydroxychromen-4-one structure
02/05/2003EP1280777A1 Tetrahydroisoquinoline analogs useful as growth hormone secretagogues
02/05/2003CN1395575A Novel piperidine compounds and drugs containing the same
02/05/2003CN1395566A Corticotropin releasing factor antagonists
02/05/2003CN1395563A Isatine derivatives with neurotrophic activity
02/05/2003CN1395562A Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
02/05/2003CN1395485A Water soluble prodrugs of azole compounds
02/05/2003CN1394855A Substituted heterocyclic compound
02/05/2003CN1100884C Homogenous method for assay of double-stranded nucleic acids using flourescent dyes and kit useful therein
02/05/2003CN1100777C N-heterocyclic derivatives as NOS inhibitor
02/04/2003US6515135 Aminoaryl oxazolidinone N-oxides
02/04/2003US6515133 Certain diaryl imidazoles act as partial agonists or antagonists for NPY receptors, in particular NPY 5 receptors. They are of use, for example in treating loss of appetite. Such compounds bear aryl groups in the 2 position.
02/04/2003US6515124 Dehydroamino acids
02/04/2003US6515013 For diseases or conditions caused by or exacerbated by histamine-3 receptor activity
02/04/2003US6515005 Substituted azole derivatives as inhibitors of corticotropin releasing factor
02/04/2003US6515004 Useful in the treatment of Alzheimer's disease, chemotherapy-induced alopecia, and cardiovascular disease
02/04/2003US6515003 Useful in the treatment of diseases related to lipid and carbohydrate metabolism
02/04/2003US6515002 Compounds and compositions for treating C1s-mediated diseases and conditions
02/04/2003US6514977 For treating p38 kinase mediated disorders
02/04/2003US6514971 Cinnoline derivatives and use as medicine
02/04/2003US6514968 Treating a disease or condition in a mammal wherein the 5-HT receptor is implicated and modulation of 5-HT function is desired comprising
02/04/2003US6514964 Treating diseases, conditions or disorders mediated by integrin receptors, such as vitronectin and fibronectin receptors
02/04/2003US6514633 Light emitting device material, light emitting device using thereof, and amine compound
01/2003
01/31/2003CA2354486A1 C7 ester substituted taxanes
01/30/2003WO2003008411A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors
01/30/2003WO2003008409A1 Quinoline derivatives and their use as tyrosine kinase inhibitors
01/30/2003WO2003008407A2 Phenylsulfonyl-1,3-dihydro-2h-indole-2-one derivatives, their preparation and their therapeutic use
01/30/2003WO2003008398A1 Aryl substituted thiazolidinones and the use thereof
01/30/2003WO2003008395A1 Substituted isoxazoles and the use thereof as antibiotics
01/30/2003WO2003008384A1 Substituted 2-thio-3, 5-dicyano-4-phenyl-6-aminopyridines and their use as adenosine receptor-selective ligands
01/30/2003WO2003008365A2 Phenylacetamido-thiazole derivatives, process for their preparation and their use as antitumor agents
01/30/2003WO2003007948A1 Antimalarial agent containing rhodacyanine dye compound
01/30/2003WO2003007946A1 Secondary 1,3-thiazole-5-yl sulfonamide derivatives and their use as antiviral agents
01/30/2003WO2003007945A1 Viral polymerase inhibitors
01/30/2003WO2002088079A3 Dual inhibitors of pde 7 and pde 4
01/30/2003WO2002012247A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof
01/30/2003US20030023086 For therapy of thrombosis in humans and other mammals
01/30/2003US20030023082 Epothilone derivatives and methods for making and using the same
01/30/2003US20030022905 Prevention and/or therapy of ischaemia and reperfusion damage; poly(ADP-ribose)-synthetase inhibitors
01/30/2003US20030022895 2-Amino-benzoxazinones for the treatment of viral infections
01/30/2003US20030022885 Pyrazole compounds useful as protein kinase inhibitors
01/30/2003US20030020603 Vehicular sound-processing system incorporating an interior mirror user-interaction site for a restricted-range wireless communication system
01/30/2003CA2454059A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors
01/30/2003CA2453846A1 Substituted isoxazoles and the use thereof as antibiotics
01/30/2003CA2453633A1 Aryl substituted thiazolidinones and the use thereof
01/30/2003CA2453294A1 Phenylacetamido-thiazole derivatives, process for their preparation and their use as antitumor agents
01/30/2003CA2450437A1 1-phenylsulphonyl-1,3-dihydro-2h-indol-2-one derivatives, their preparation and their therapeutic application
01/30/2003CA2417804A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof
01/29/2003EP1278744A1 Heterobicyclic sulfonamides and their use as platelet adp receptor inhibitors
01/29/2003EP1278743A1 Novel anti-infectives
01/29/2003EP1278741A1 Muscarinic agonists
01/29/2003EP1278739A1 Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by the np y5 receptor
01/29/2003EP1278520A1 Diaryl piperidyl pyrrole derivatives as antiprotozoal agents
01/29/2003EP1278502A2 Protease inhibitors
01/29/2003EP1105387B1 Prodrugs of proton pump inhibitors
01/29/2003EP0906294B1 Benzoxazinone dopamine d4 receptor antagonists
01/29/2003EP0835243B1 Dialkyl phenyl halide-substituted keto-enols for use as herbicides and pesticides
01/29/2003EP0708769B1 Substituted 2-fused phenylpyridines with herbicidal activity
01/29/2003CN1394203A Piperidine and piperazine derivatives which function as 5-HT2A receptor antagonists
01/29/2003CN1394202A Picolinic acid derivatives and their use as fungicides
01/29/2003CN1100048C 1,2,3-thiadiazole derivatives, plant disease controlling agent, and method for use thereof
01/28/2003WO2002010155A1 Substituted aryl ketones and their use as herbicides
01/28/2003US6512112 Useful as prodrugs, easily convert to parent amine in vivo; antibiotic activity versus gram negative aerobic and anaerobic bacteria
01/28/2003US6512001 D-proline derivatives
01/28/2003US6511998 Pyrazole carboxamides useful for the treatment of obesity and other disorders
01/28/2003US6511994 Modulators of CCR5 chemokine receptor activity
01/28/2003US6511993 Metalloprotease inhibitors
01/28/2003US6511977 For preventing or treating cardiac arrhythmia or atrial arrhythmia
01/28/2003US6511942 Animal husbandry, veterinary medicine
01/28/2003CA2417385A1 Substituted aryl ketones and their use as herbicides
01/28/2003CA2254905C Tricyclic functional dyes for contrast enhancement in optical imaging
01/23/2003WO2003006506A2 Protease inhibitor conjugates and antibodies useful in immunoassay
01/23/2003WO2003006495A2 Human papillomavirus e2 transactivation domain/inhibitor co-crystal and x-ray coordinates defining the inhibitor-binding pocket
01/23/2003WO2003006463A1 Acaricide
01/23/2003WO2003006461A1 Substituted benzo-nitro-heterocycles
01/23/2003WO2003006454A2 Heterocyclic carboxamides and their use as fungicides
01/23/2003WO2003006447A2 Interaction inhibitors of tcf-4 with beta-catenin