Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
07/2003
07/23/2003CN1431904A Protease inhitors
07/22/2003US6596876 Prostaglandin I2 inhibitors
07/22/2003US6596875 Method for synthesizing epothilones and epothilone analogs
07/22/2003US6596873 2-and 2,5-substituted phenylketoenols
07/22/2003US6596747 For therapy of diseases associdated with Factor VIIa and or inosine monophosphate dehydrogenase (IMPDH)
07/22/2003US6596746 Cyclic protein tyrosine kinase inhibitors
07/22/2003US6596745 Method for treating fibrotic diseases with azolium chroman compounds
07/22/2003US6596744 Method for treating fibrotic diseases or other indications IIC
07/22/2003US6596738 Inhibiting activity to adenosine deaminase (hereinafter described as ADA) An adenosine deaminase inhibiting agent comprising a compound of the formula (I):
07/22/2003US6596728 A pharmaceutical composition, comprising at least one compound or salt thereof as claimed in claim 1 and a polypeptides with excipients
07/22/2003US6596724 Oxadiazole and thiadiazole derivatives of dihydropyridine NPY antagonists
07/22/2003US6596723 Fungal efflux pump inhibitors
07/22/2003US6596718 7-Morpholin-4yl-benzothiazole amide derivatives
07/22/2003CA2228572C Nk-1 receptor antagonists for prevention of neurogenic inflammation in gene therapy
07/17/2003WO2003057693A1 5-membered cyclic compounds
07/17/2003WO2003057692A1 Novel crystalline forms of meloxicam and the preparation and interconversion methods thereof
07/17/2003WO2003057676A1 3,4-di-substituted pyridazinediones as cxc chemokine receptor antagonists
07/17/2003WO2003057674A1 4-sulfide / sulfoxide / sulfonyl-1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
07/17/2003WO2003057672A2 Tetrahydroquinoline analogues as muscarinic agonists
07/17/2003WO2003057669A1 Androgen receptor antagonists
07/17/2003WO2003057668A1 Nitrogenous cyclic ketone derivative, process for producing the same, and use
07/17/2003WO2003057666A2 Inhibitors of dipeptidyl peptidase iv
07/17/2003WO2003057144A2 Change inhibitors of dipeptidyl peptidase iv
07/17/2003WO2002055496A8 Aryl piperidine and piperazine derivatives as inducers of ldl-receptor expression
07/17/2003WO2002006280A3 INHIBITORS OF FACTOR Xa
07/17/2003US20030135057 5-amino- and 5-thio- substituted; prepared from a methylenedithietane intermediate
07/17/2003US20030134888 Substituted diaminopyrazoles; treating diseases, such as cancer, inflammatory disorders, restenosis, and cardiovascular disease. coatings for implantable medical devices, such as prostheses, artificial valves, etc.
07/17/2003US20030134885 Biaromatic ligand activators of PPARgamma receptors
07/17/2003US20030134883 Use in the treatment of cancer and other diseases characterized by undesired cellular hyperproliferation.
07/17/2003US20030134876 Inhibiting TNF alpha
07/17/2003US20030134859 Substituted 2-chloro-5-nitrobenzamides; treating retrograde osteoporosis and diabetes mellitus
07/17/2003US20030134855 P-acylaminomethyl-N-(4-methoxy-7-morpholin-4-yl-benzothiazol-2 -yl)-benzamides; treatment of diseases related to the adenosine receptor, such as Alzheimer's disease, depression, drug addiction, Parkinson's and ADHD
07/17/2003US20030134854 Treatment of diseases related to the adenosine receptor, such as Alzheimer's disease, depression, drug addiction, neuroprotection, Parkinson's disease, and attention deficit hyperactivity disorder.
07/17/2003US20030134849 Thiazepinyl hydroxamic acid derivatives as matrix metalloproteinase inhibitors
07/17/2003US20030134848 Substituted 1-aza-2-imino-heterocycles and their use as nicotinic acetylcholin receptors activators
07/17/2003US20030134840 Novel compounds
07/17/2003US20030134836 Substituted arylamine derivatives and methods of use
07/17/2003US20030134827 Lactams or pharmaceutically acceptable salt forms thereof, wherein rings ring B is a 4-8 membered cyclic amide containing from 0-3 additional heteroatoms selected from N, O, and S, which are useful as metalloprotease inhibitors.
07/17/2003US20030134802 Novel effectors of dipepetidyl peptidase IV
07/17/2003US20030134801 Pharmaceutical compositions containing them are of the class of thrombin inhibitors which are useful as anticoagulants.
07/17/2003US20030134237 Methine dyes, manufacturing methods thereof, and silver halide photoraphic materials contaning same dyes
07/17/2003US20030134148 Red fluorescent dyes having high fluorescent strength and high color purity; high luminance; high efficacy by low voltage-driving; stability; durability; color conversion filter, pulp dyeing; photographic dye; sensitizers
07/17/2003CA2472165A1 3,4-di-substituted pyridazinediones as cxc chemokine receptor antagonists
07/17/2003CA2471885A1 4-sulfide / sulfoxide / sulfonyl-1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
07/17/2003CA2471754A1 Androgen receptor antagonist
07/17/2003CA2471204A1 Inhibitors of dipeptidyl peptidase iv
07/17/2003CA2470164A1 New crystalline forms of meloxicam and processes for their preparation and interconversion.
07/16/2003EP1326864A2 Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
07/16/2003EP1326861A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
07/16/2003EP1326860A1 Quinazoline derivatives
07/16/2003EP1326858A2 Piperidine compounds as anti-allergic
07/16/2003EP1326853A1 New thiadiazoles and oxadiazoles and their use as phosphodiesterase-7 inhibitors
07/16/2003EP1326852A1 Aromatic and heterocyclic thiazolyl thiourea compounds and use
07/16/2003EP1326850A1 A process for the preparation of bis-benzazolyl compounds
07/16/2003EP1326829A2 17-beta-hydroxysteroid dehydrogenase-ii inhibitors
07/16/2003EP1326606A2 Ep4 receptor inhibitors to treat rheumatoid arthritis
07/16/2003EP1175416B1 Heteroaryl diazacycloalkanes, their preparation and use
07/16/2003EP1028955B1 Pyrimidinone compounds and pharmaceutical compositions containing them
07/16/2003EP0832076B1 Novel isoxazoline and isoxazole fibrinogen receptor antagonists
07/16/2003CN1430615A Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
07/16/2003CN1430614A Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
07/16/2003CN1430612A Hete rocyclic derivatives
07/16/2003CN1430610A Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
07/16/2003CN1430609A Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
07/16/2003CN1430608A Substituted iminoazines
07/16/2003CN1114604C Bicyclic aryl carboxamides and their therapeutic use
07/16/2003CN1114603C Hydrazono-1,3-dithiocyclopentane derivative and synthesizing method thereof
07/16/2003CN1114598C Aromatic compounds and pharmaceutical compositions containing them
07/16/2003CN1114403C Vitronectin receptor antagonists
07/16/2003CN1114402C Isothiazolones compound, preparation containing them and its use
07/15/2003USRE38188 Ethylene derivatives and pesticides containing said derivatives
07/15/2003US6593472 NK-1 receptor active amine oxide prodrugs
07/15/2003US6593357 Treating disease states in mammals that are alleviated by a protein kinase inhibitor, particularly diseases such as cancer, inflammatory disorders, restenosis, and cardiovascular disease.
07/15/2003US6593346 Substituted 3-(piperidin-1-ylmethyl)cyclopentylamines, useful as modulators of the chemokine receptors CCR-5 and/or CC R-3.
07/15/2003US6593344 These substances have especially high cytostatic activities and pronounced immunosuppressive properties which make them suitable for therapeutic treatment in broad tumor spectrum and autoimmune diseases
07/15/2003US6593327 Compounds and compositions as protease inhibitors
07/15/2003US6593326 Useful as anti-cancer agents; and processes for their manufacture and pharmaceutical compositions containing them are described. Apoptotic effect in a warm-blooded animal such as man.
07/15/2003US6593322 Compounds and methods for modulation of estrogen receptors
07/15/2003US6593013 Electroluminescence device, cyclic azine compound and production process of cyclic azine dye
07/15/2003US6592633 Less selective colorations and which are particularly resistant to the various attacking factors to which the hair may be subjected
07/10/2003WO2003055868A1 Benzothiazole- and benzoxazole-4,7-dione derivatives and their use as cdc25 phosphatase inhibitors
07/10/2003WO2003055867A1 Biphenylmethyl-thiazolidinediones and analogues and their use as ppar-gamma activators
07/10/2003WO2003055866A1 Quinazoline and quinoline derivative compounds as inhibitors of prolylpeptidase, inducers of apoptosis and cancer treatment agents
07/10/2003WO2003055860A1 3,4-diarylpyrazoles and their use in the therapy of cancer
07/10/2003WO2003055482A1 Amide derivatives as gk activators
07/10/2003WO2003055478A1 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders
07/10/2003WO2003055447A2 Heterocyclic acridone inhibitors of impdh enzyme
07/10/2003WO2003010140A3 Hepatitis c virus polymerase inhibitors with heterobicyclic structure
07/10/2003WO2003006440A8 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
07/10/2003WO2001098269A3 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
07/10/2003WO2001096297A3 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
07/10/2003US20030130520 Producing substituted 2-nitro-guanidine derivatives.
07/10/2003US20030130515 Aryl or heteroaryl substituted 3,4-dihydroanthracene and aryl or heteroaryl substituted benzo[1,2-g]-chrom-3-ene, benzo[1,2-g]-thiochrom-3-ene and benzo [1,2-g]-1,2-dihydroquinoline derivatives having retinoid antagonist or retinoid inverse agonist type biological activity
07/10/2003US20030130506 4-phenoxy or 4-(pyrid-4-yloxy)- benzensulfonic acid derivatives; antitumor and antiarthritic agents
07/10/2003US20030130505 Nonsteroidal agonists and antagonists
07/10/2003US20030130340 Novel benzothiophene derivatives
07/10/2003US20030130318 2-sulfonamido-thiazole derivatives
07/10/2003US20030130289 Inhibitors of glycogen synthase kinase 3
07/10/2003US20030130287 Psychological disorders; central nervous system disorders; antidepressants; Parkinson's disease; Alzheimer's disease;cardiovascular disorders
07/10/2003US20030130282 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto