Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
07/2003
07/10/2003US20030130281 DPP IV inhibitors
07/10/2003US20030130279 Hyperglycemic agents; dietetics; cardiovascular disorders; immunology modulation; osteoporosis; cognition activators
07/10/2003US20030130273 Hydantoins and related heterocycles as inhibitors of matrix metalloproteinases and/or TNF-alpha converting enzyme (TACE)
07/10/2003US20030130258 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
07/10/2003US20030130254 Respiratory system disorders; antihistamines; antiarthritic agents
07/10/2003US20030130251 Blocking amyloid deposits; Alzheimer's disease, Down syndrome
07/10/2003US20030130203 Sleep disorders
07/10/2003US20030130125 Pesticides; herbicides
07/10/2003CA2471713A1 Benzothiazole- and benzoxazole-4,7-dione derivatives and their use as cdc25 phosphatase inhibitors
07/10/2003CA2471049A1 Amide derivatives as gk activators
07/09/2003EP1325920A1 N-substituted benzothiophenesulfonamide derivatives
07/09/2003EP1325918A1 Heart muscular cell apoptosis inhibitors and remedies/preventives for heart diseases
07/09/2003EP1325910A1 Aliphatic nitrogenous five-membered ring compounds
07/09/2003EP1325000A1 A thiazolidinedione derivative and its use as antidiabetic
07/09/2003EP1324999A1 Novel aminophenyl piperazine or aminophenyl piperidine derivatives inhibiting prenyl transferase proteins and methods for preparing same
07/09/2003EP1324998A1 Novel aminotriazolone compounds, method for preparing same and pharmaceutical compositions containing same
07/09/2003EP1324993A2 Substituted 1,4-thiazepine and analogs as activators of caspases and inducers of apoptosis and the use thereof
07/09/2003EP1324991A1 Compounds useful in the treatment of inflammatory diseases
07/09/2003EP1324990A1 Morpholin-acetamide derivatives for the treatment of inflammatory diseases
07/09/2003EP1324974A2 Drugs for diabetes
07/09/2003EP1165496B1 Substituted aniline compounds
07/09/2003EP0966465B1 Inhibitors of impdh enzyme
07/09/2003CN1429224A Novel benzothiophene derivatives
07/09/2003CN1429222A 激酶抑制剂 Kinase inhibitors
07/09/2003CN1429215A 三唑衍生物 Triazole derivatives
07/09/2003CN1429210A Substituted thioacetamides
07/09/2003CN1428145A Quinoline derivative as tachykinin NK3 receptor agonist
07/09/2003CN1113875C Substituted aromatic thiocarboxylic acid amides and their use as herbicides
07/08/2003US6589984 Blood cholesterol and triglycerides (TG) themselves are generally insoluble in blood, and they exist as lipoproteins by binding with apolipoproteins. In the body, triglycerides are biosynthesized primarily in the liver from acetyl CoA as
07/08/2003US6589969 Carboxylic acid derivatives and drugs containing the same as the active ingredient
07/08/2003US6589968 Epothilone compounds and methods for making and using the same
07/08/2003US6589962 Certain alpha -hydroxy- gamma -(((carbocyclic- or heterocyclic- substituted)amino)carbonyl)alkanamide derivatives are described as inhibitors of HIV protease and inhibitors of HIV replication. These compounds are useful in
07/08/2003US6589956 Its enantiomers, diastereoisomers, and addition salts thereof with a pharmaceutically acceptable acid or base, and medicinal products containing the same which are useful as a TXA2 receptor antagonist and 5-HT2 receptor antagonist.
07/08/2003US6589953 Indole derivatives as 5-HT1B and 5-HT1D agonists
07/08/2003CA2285208C Improved method for producing thiazolidinediones, and new thiazolidinediones
07/03/2003WO2003053979A1 Novel benzothiazine and benzothiadiazine derivatives, method for preparing same and pharmaceutical compositions containing same
07/03/2003WO2003053965A1 Salicylate salt of a thiazolidinedione derivative
07/03/2003WO2003053964A1 5- (4- (2- (n-methyl-n- (2-pyridil) amino) ethoxy) benzyl) thiazolidine-2, 4-dione nephtalenesulfonate salt and use against diabetes mellitus
07/03/2003WO2003053963A1 Novel pharmaceutical
07/03/2003WO2003053962A1 5- (4- (2- (n-methyl-n- (2-pyridyl) amino) ethoxy) benzyl) thiazolidine-2, 4-dione malic acid salt and use against diabetes mellitus
07/03/2003WO2003053961A1 Benzothiazoles
07/03/2003WO2003053959A1 Heterocyclylamino carbonyluracils
07/03/2003WO2003053955A1 Thiochromenones used to combat painful conditions and neurodegenerative diseases
07/03/2003WO2003053948A1 Isochroman compounds for treatment of cns disorders
07/03/2003WO2003053946A1 7-amino-benzothiazole derivatives as adenosine receptor ligands
07/03/2003WO2003053941A2 Barbituric acid derivatives as inhibitors of tnf-alpha converting enzyme (tace) and/or matrix metalloproteinases
07/03/2003WO2003053939A1 Benzimidazole derivatives and their use as gnrh antagonists
07/03/2003WO2003053928A1 Serotonine reuptake inhibitor
07/03/2003WO2003053925A1 Pyrrolidine-2-ones as factor xa inhibitors
07/03/2003WO2003053915A2 Compounds for the treatment of inflammatory disorders
07/03/2003WO2003053443A1 Substituted diketopiperazines as oxytocin antagonists
07/03/2003WO2003053441A1 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and the use of the same
07/03/2003WO2003053435A1 Broadspectrum heterocyclic substituted phenyl containing sulfonamide hiv protease inhibitors
07/03/2003WO2003053367A2 Hydrogenation of precursors to thiazolidinedione antihyperglycemics
07/03/2003WO2003053366A2 Pyrimidine a2b selective antagonist compounds, their synthesis and use
07/03/2003WO2002101073A3 Aryl-benzimidazole compounds having antiinfective activity
07/03/2003WO2002062295A3 Pyridine-substituted benzanilides as potassium ion channel openers
07/03/2003US20030125369 New indenoindolone compounds
07/03/2003US20030125364 Antirheumatic agent
07/03/2003US20030125362 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
07/03/2003US20030125358 Pharmaceutical compositions containing thiazolidinedione derivatives and process for their preparation
07/03/2003US20030125356 Reacting a methylketophenolic compound with a benzaldehyde compound to produce an intermediate, cyclizing the intermediate in presence of a base; anticarcinogenic agent, and treats diseases induced by cell proliferation
07/03/2003US20030125346 Amino-substituted pyrimidinyl derivatives and methods of use
07/03/2003US20030125340 3-(Amino-or aminoalkyl) pyridinone derivatives and their use for the treatment of HIV related diseases
07/03/2003US20030125339 Substituted alkylamine derivatives and methods of use
07/03/2003US20030125334 5-HT receptor ligands and uses thereof
07/03/2003US20030125324 Alpha 4 beta 1 integrin and CD49d/ CD29 (vla-4); antiinflammatory agents
07/03/2003US20030125318 Benzothiazole derivatives with activity as adenosine receptor ligands
07/03/2003US20030125317 Vitronectin receptor antagonists
07/03/2003US20030124082 Method of repairing or restoring damaged or imperfect hair
07/03/2003CA2471461A1 Pyrrolidine-2-ones as factor xa inhibitors
07/03/2003CA2471355A1 Substituted diketopiperazines as oxytocin antagonists
07/03/2003CA2471263A1 Novel benzothiazine and benzothiadiazine derivatives, method for preparing same and pharmaceutical compositions containing same
07/03/2003CA2470964A1 Broadspectrum heterocyclic substituted phenyl containing sulfonamide hiv protease inhibitors
07/03/2003CA2470075A1 Hydrogenation of precursors to thiazolidinedione antihyperglycemics
07/03/2003CA2469884A1 7-amino-benzothiazole derivatives as adenosine receptor ligands
07/03/2003CA2469278A1 Isochroman compounds for treatment of cns disorders
07/03/2003CA2448811A1 Thiochromenones used to combat painful conditions and neurodegenerative diseases
07/02/2003EP1323710A1 Nitrogenous five-membered ring compounds
07/02/2003EP1322710A1 Modified carbocyanine dyes and their conjugates
07/02/2003EP1322650A2 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives
07/02/2003EP1322648A1 3-(heteroaryl acetamido)-2-oxo-azetidine-1-sulfonic acids derivatives as antibacterial agents
07/02/2003EP1322647A1 Novel polymorphic forms of 5-[4-[2-[n-methyl-n-(2-pyridyl)amino]ethoxy]benzyl]thiazolidine-2,4-dione maleic acid salt and process for their preparation
07/02/2003EP1322646A1 2-(1h-indol-3-yl)-2-oxo-acetic acid amides with antitumor activity
07/02/2003EP1322644A1 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinolinone derivatives
07/02/2003EP1322639A1 Substituted aryl ketones and their use as herbicides
07/02/2003EP1322636A1 Farnesyl transferase inhibiting 6- (substituted phenyl)methyl]-quinoline and quinazoline derivatives
07/02/2003EP1322635A1 Farnesyl transferase inhibiting quinoline and quinazoline derivatives as farnesyl transferase inhibitors
07/02/2003EP1322628A2 Substituted urea neuropeptide y y5 receptor antagonists
07/02/2003EP1322627A1 Cyclic sulfonyl compounds as inhibitors of metalloproteases
07/02/2003EP1322617A1 Compounds and methods for modulation of estrogen receptors
07/02/2003EP1322613A1 Spiroheterocyclic nitriles useful as reversible inhibitors of cysteine proteases
07/02/2003EP1322611A1 Chemical compounds
07/02/2003EP1322608A1 Delta1-pyrrolines used as pesticides
07/02/2003EP1322598A1 Nitroso diphenylamine derivatives
07/02/2003EP1322309A2 High affinity small molecule c5a receptor modulators
07/02/2003EP1218372B1 Novel heterocyclic compounds useful as reversible inhibitors of cysteine proteases
07/02/2003EP0991627B1 Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
07/02/2003EP0913392B1 Ethylene derivatives and pest controlling agents
07/02/2003EP0900211B1 Thiadiazolyl(thio)ureas useful as matrix metalloprotease inhibitors