Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
10/2002
10/30/2002CN1377347A 药学活性磺酰胺衍生物 Pharmaceutically active sulfonamide derivatives
10/30/2002CN1377346A Z-pyrazoline-5-ones
10/30/2002CN1377344A Inhibitor of cysteinyl aspartic acid proteinase
10/30/2002CN1377343A Substituted aryl ketones
10/30/2002CN1377269A Vitronectin receptor antagonists
10/30/2002CN1377259A ACE-2 inhibiting compounds and methods of use thereof
10/29/2002US6472534 Treating tetrahydrofuran derivativ with an oxophilic electrophilic reagent in a manner that is effective to provide the oxazoline compound
10/29/2002US6472529 Viricides
10/29/2002US6472526 Shows an inhibitory activity against farnesyl transferase or pharmaceutically acceptable salts or isomers thereof, in pharmaceutical composition and intermediates
10/29/2002US6472418 Non-peptide NK1 receptors antagonists
10/29/2002US6472412 Compounds as PDE IV and TNF inhibitors
10/29/2002US6472404 HIV protease inhibitors
10/29/2002US6472394 MCH antagonists and their use in the treatment of obesity
10/29/2002US6472392 Triazole compounds and the use thereof as dopamine-D3 -ligands
10/29/2002US6472388 Psychotherapeutic agents.
10/29/2002US6472387 Methods of using compounds as neuro-protective agents
10/29/2002US6472386 Cyclic diamine compound with 5-membered ring groups
10/29/2002US6472349 Pyridine-2,3-dicarboxylic acid diamides
10/29/2002CA2342471C Heterocyclecarbonylmethyl amine intermediates
10/24/2002WO2002083863A2 Thiazole and other heterocyclic ligands and use thereof
10/24/2002WO2002083668A1 Isoxaxole derivatives as inhibitors of src and other protein kinases
10/24/2002WO2002083665A1 DIHYDRO-BENZO[b][1,4]DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS I
10/24/2002WO2002083655A1 Prodrugs of cox-2 inhibitors
10/24/2002WO2002083652A1 DIHYDRO-BENZO [b] [1, 4] DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II
10/24/2002WO2002083649A1 Novel imidazolidinedione derivatives and use thereof as drugs
10/24/2002WO2002083645A1 Novel compounds
10/24/2002WO2002083642A1 Compounds useful as anti-inflammatory agents
10/24/2002WO2002083628A1 1,4-disubstituted benzo-fused compounds
10/24/2002WO2002083624A1 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands
10/24/2002WO2002083143A1 Cxcr3 antagonists
10/24/2002WO2002083130A1 Enantiomers of n-[[2'-[[(4,5-dimethyl-3-isoxazolyl) amino]sulfonyl]-4-(2-oxazolyl)[1,1'-biphenyl]-2-yl]methyl]-n,3,3-trimethylbutanamide
10/24/2002WO2002083111A2 Imidazole, thiazole and oxazole derivatives and their use for the manufacture of a medicament for the treatment and/or prevention of pollakiuria or urinary incontinence
10/24/2002WO2002074763A9 Benzimidazol derivatives modulate chemokine receptors
10/24/2002WO2002050065A3 Pyrazole compounds useful as protein kinase inhibitors
10/24/2002WO2001040221A3 Cyclopropyl-anellated 3-(4,5-dihydroisoxazol-3-yl)-substituted benzoylpyrazoles as herbicides
10/24/2002WO2000040247A9 2-oxy-benzoxazinone derivatives for the treatment of obesity
10/24/2002US20020156111 Substituted bicyclic compounds
10/24/2002US20020156110 Anticancer, antiproliferative and antiarthritic agents
10/24/2002US20020156102 Piperidine amides as modulators of chemo kine receptor activity
10/24/2002US20020156087 Pyrimidine or pyridine derivatives
10/24/2002US20020156076 Imidazole derivatives used to reduce ocular pressure or treat glaucoma and other diseases
10/24/2002US20020156063 Heterocyclic amide compounds useful for treating diseases associated with activity of cathepsin K
10/24/2002US20020156018 Treating parasitic diseases, which are mediated by such proteases. In particular, treating malaria by inhibiting the cysteine protease falcipain.
10/24/2002DE10148598A1 New N-(acylaminophenyl)-heteroaryl-benzenesulfonamide derivatives, useful as antiviral agents, especially effective against human cytomegalovirus infections
10/24/2002DE10119204A1 Production of new or known 5-aryl-1,3,3-trimethyl-2-methylene-indoline derivatives useful in compositions for dyeing keratin and other fibers, especially human hair
10/24/2002DE10108481A1 Pyridylpyrimidine Pyridylpyrimidines
10/24/2002CA2490819A1 Compounds useful as anti-inflammatory agents
10/24/2002CA2444596A1 Large conductance calcium-activated k channel opener
10/24/2002CA2444267A1 Prodrugs of cox-2 inhibitors
10/24/2002CA2443697A1 1,4-disubstituted benzo-fused compounds
10/24/2002CA2443234A1 Isoxaxole derivatives as inhibitors of src and other protein kinases
10/24/2002CA2431553A1 Cxcr3 antagonists
10/23/2002EP1251129A1 Pyrimidine derivatives having antitumor effect
10/23/2002EP1251128A1 Cyclohexylamine derivatives as subtype selective N-methyl-D-aspartate antagonists
10/23/2002EP1251127A1 Novel sidechain-bearing taxanes and intermediates thereof
10/23/2002EP1251125A2 New camptothecin analogues, preparation methods thereof, use thereof as drugs, and pharmaceutical compositions containing them
10/23/2002EP1250337A1 Substituted homopiperidinyl benzimidazole analogues as fundic relaxants
10/23/2002EP1250332A1 Inhibitors of interleukin 5 gene expression
10/23/2002EP1250328A1 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses
10/23/2002EP1196384A4 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
10/23/2002EP0979229B1 2-oxo-1-azetidine sulfonic acid derivatives as potent beta-lactamase inhibitors
10/23/2002EP0923561B1 Heterocyclic metalloprotease inhibitors
10/23/2002EP0783499B1 Benzofuran derivatives as tachykinin antagonists
10/23/2002EP0674630B1 7-HALO- AND 7$g(b),8$g(b)-METHANO-TAXOLS, ANTINEOPLASTIC USE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
10/23/2002CN1376149A 2,4-diamino-1,3,5-triazine, method for the production and use of the same as herbicides and plant growth regulators
10/23/2002CN1376147A 吡唑类衍生物 Pyrazole derivatives
10/23/2002CN1093124C Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to PPAR-gamma
10/23/2002CN1093123C Aralkyl and aralkylidene heterocyclic lactams and imides
10/23/2002CA2381630A1 Method for preventing dyskinesias
10/22/2002US6469176 Method and novel intermediate products for producing isoxazolin-3-yl-acylbenzenenes
10/22/2002US6469037 Prophylactic or therapeutic drug for renal diseases
10/22/2002US6469032 3-(4′-bromobenzylindenyl)-2-indolinone and analogues thereof for the treatment of disease
10/22/2002US6469025 For the prophylaxis or treatment of a disease or disorder in a mammal in which the extravasation of leukocytes plays a role; inhibiting the binding of alpha 4 integrins to their ligands
10/22/2002US6469011 Benzenesulfonamide compounds useful as TXA2 and 5-HT2 receptor antagonists
10/22/2002US6469006 Particularly for treating hiv infections
10/22/2002US6469001 IL-5 inhibiting 6-azauracil derivatives
10/22/2002US6469000 1,3-diheterocyclic metalloprotease inhibitors
10/17/2002WO2002081483A2 Inhibitors of acyl glucosaminyl inositol amidase and methods of use
10/17/2002WO2002081478A2 Broadspectrum 2-(substituted-amino)-benzoxazole sulfonamide hiv protease inhibitors
10/17/2002WO2002081470A1 Oxazolidinones containing a sulfonimid group as antibiotics
10/17/2002WO2002081469A1 Oxazolidinone-sulfoximines and -sulfilimines as antibiotics
10/17/2002WO2002081468A1 Oxazolidinones and their use as antibacterial agents
10/17/2002WO2002081467A1 Quinazoline and quinazoline-like compounds for the treatment of integrin-mediated disorders
10/17/2002WO2002081453A1 Thiohydantoins and use thereof for treating diabetes
10/17/2002WO2002081448A1 Benzamidine derivative
10/17/2002WO2002080928A1 N-substituted nonaryl-heterocyclo amidyl nmda/nr2b antagonists
10/17/2002WO2002080920A1 Arylacetamido-ketobenzoxazole as cysteine protease inhibitors
10/17/2002WO2002080853A2 Fused heterocyclic inhibitors of factor xa
10/17/2002WO2002080846A2 Epothilone derivatives and methods for making and using the same
10/17/2002WO2002080841A2 Antibacterial oxazolidinones with a cyclic sulphilimine or sulphoximine
10/17/2002WO2002066468A3 Heterocyclic urea derivatives and their use as dopamine d3 receptor ligands
10/17/2002WO2002044156A3 Benzimidazole derivatives useful as tie-2 and/or vegfr-2 inhibitors
10/17/2002WO2002034726A3 Pyrimidine-2,4,6-trione metalloproteinase inhibitors
10/17/2002WO2002032884A3 Methods for the preparation of biphenyl isoxazole sulfonamides
10/17/2002WO2001083463A1 Oxadiazole derivatives having anticancer effects
10/17/2002US20020151720 Naphthol derivatives
10/17/2002US20020151555 Pyrimidine matrix metalloproteinase inhibitors
10/17/2002US20020151547 Substituted phenyl-piperidine methanone compounds
10/17/2002US20020151535 Heterocyclic 1,2,4-oxadiazole or oxazole ring containing propanohydroxamic acids useful as antiscarring agent
10/17/2002CA2444024A1 Thiohydantoins and use thereof for treating diabetes