Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
09/2002
09/12/2002WO2001012600A9 INHIBITORS OF FACTOR Xa
09/12/2002US20020128510 Antiarthritic agents; rheumatic diseases; osteoarthritis; inhibition of the inducible nitric oxide synthase - induced after activation of vascular smooth muscle, macrophages, endothelial cells by enotoxin and cytokines
09/12/2002US20020128290 Derivatives of benzofuran or benzodioxole
09/12/2002US20020128272 4,5,6, and 7-indole and indoline derivatives, their preparation and use
09/12/2002US20020128270 Treating stroke, arhtritis, cancer, tissue ulceration, decubitis ulcer, restenosis, periodontal disease, epidermolysis bullosa, scleritis, psoriasis, AIDS, sepsis, and septic shock.
09/12/2002US20020128266 ABCA-1 elevating compounds
09/12/2002US20020128263 Treatment or prevention of mGluR5 receptor mediated disorders.
09/12/2002US20020128262 Styrylbenzodiazepines
09/12/2002US20020128247 Phenyl sulfamide derivatives as dietetics, antidiabetics, and hypotensive agents
09/12/2002US20020128185 Cryptophycin compounds useful for disrupting the microtubulin system; antineoplastic, antifungal, and anticancer agents
09/12/2002CA2439827A1 Peptide deformylase inhibitors
09/12/2002CA2439666A1 Nitrogen-containing heteroaryl compounds having hiv integrase inhibitory activity
09/12/2002CA2439644A1 Phenyl derivatives and their use in the treatment of thromboembolic disorders or tumours
09/12/2002CA2437840A1 Heterocyclic diamide invertebrate pest control agents
09/12/2002CA2437594A1 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
09/12/2002CA2433467A1 Substituted quinolinecarboxamides as antiviral agents
09/12/2002CA2431549A1 Substituted 8-arylquinoline phosphodiesterase-4 inhibitors
09/11/2002EP1238975A1 Difluoromethyltriazolone compounds, use of the same and intermediates for the production thereof
09/11/2002EP1238974A1 Heterocycle derivatives and drugs
09/11/2002EP1238970A1 Cycloamine ccr5 receptor antagonists
09/11/2002EP1237953A2 Polymerization of olefins
09/11/2002EP1237895A2 Phosphorylation of terminal primary alcohol groups
09/11/2002EP1237889A1 Antibiotic sultam and sultone derived oxazolidinones
09/11/2002EP1237888A2 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
09/11/2002EP1237887A1 9-(piperazinylalkyl)carbazoles as bax-modulators
09/11/2002EP1237875A1 Substituted imidazole neuropeptide y y5 receptor antagonists
09/11/2002EP1237874A2 Selective neurokinin antagonists
09/11/2002EP1237869A1 Compounds, compositions, and methods for stimulating neuronal growth and elongation
09/11/2002EP1237868A1 Hydroxamic acid derivatives as matrix metalloproteinase (mmp) inhibitors
09/11/2002EP1237867A1 Hydroxamic acid derivatives as matrix metalloproteinase (mmp) inhibitors
09/11/2002EP1237862A1 Succinate compounds, compositions and methods of use and preparation
09/11/2002EP1237551A1 Pharmaceutical formulations containing zolmitriptan
09/11/2002EP0934309B1 New pyridyl alkane acid amides as cytostatics and immunosuppressives
09/11/2002EP0799206B1 Aryl- and hetaryl-sulfonamide derivatives, their preparation and their use as endothelin antagonists
09/11/2002EP0668860B1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hiv and other retroviruses
09/11/2002CN1368972A Nonsteroid IL-5 inhibitor, its preparation method and medical composition containing the inhibitor
09/11/2002CN1368961A Compounds for modulation of PPAP gamma activity
09/11/2002CN1090631C Heterocyclic compounds, preparation process thereof and medicinal composition containing same
09/11/2002CN1090629C Novel Heterocyclic compounds
09/11/2002CN1090627C 2-amino-1,2-indene compounds, process for their preparation and pharmaceutical compositions containing them
09/11/2002CN1090625C Method for selective protection of baccation derivatives and its application to taxane synthesis
09/11/2002CN1090623C 3-aryl-1,2,4-triazole derivatives with herbicidal properties
09/10/2002US6448405 Coupling a 2-halo-5-nitrobenzoic acid and a 2-methoxyphenyl boronic acid; cyclizing to a nitrobenzocoumarin; reducing to the amine; converting to a coumarino(3,4-f)quinoline; reduction to a 5h-chromeno(3,4-f)quinoline
09/10/2002US6448396 Compounds useful as neuro-protective agents
09/10/2002US6448281 Inhibitors of hepatitis c virus replication; treatment of hepatitis c
09/10/2002US6448277 VEGF receptor tyrosine kinase inhibitors
09/10/2002US6448276 Such as 1-pyridin-3-yl-4-pyrrolidin-1-yl-but-1-ene; increasing hydration and lubrication of vaginal and cervical tissues; nicotine, epibatidine alkaloids and analogs
09/10/2002US6448270 4-substituted piperidine analogs and their use as subtype selective NMDA receptor antagonists
09/10/2002US6448250 Sulfamato hydroxamic acid metalloprotease inhibitor
09/10/2002US6448247 Tachykinin receptor antagonist; especially to the receptors for substance p (which receptors are generally referred to as ?neurokinin 1 receptors?)
09/10/2002US6448244 Broad-spectrum antifungals, against which there is no existing resistance and which can be administered intravenously or transungually
09/10/2002US6448203 Substituted aryluracils
09/10/2002US6448201 Benzoylcyclohexanediones and benzoylpyrazoles, their preparation, and their use as herbicides and plant growth regulators
09/10/2002CA2240946C Isoxazoline, isothiazoline and pyrazoline factor xa inhibitors
09/10/2002CA2195129C Substituted piperidine intermediates for producing heterocyclic-cyclic amine derivatives capable of inhibiting cholinesterase
09/06/2002WO2002068417A2 Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
09/06/2002WO2002068415A1 Pyrazole compounds useful as protein kinase inhibitors
09/06/2002WO2002068409A1 N-substituted nonaryl-heterocyclic nmda/nr2b antagonists
09/06/2002WO2002068406A2 Substituted amine derivatives and their use for the treatment of angiogenesis
09/06/2002WO2002068393A1 Phenylalanine enamide derivatives possessing a cyclobutene group, for use as integrin inhibitors
09/06/2002WO2002068388A2 Acylated piperidine derivatives as melanocortin-4 receptor agonists
09/06/2002WO2002068387A2 Acylated piperidine derivatives as melanocortin-4 receptor agonists
09/06/2002WO2002067939A1 Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
09/06/2002WO2002067869A2 Acylated piperidine derivatives as melanocortin-4 receptor agonists
09/06/2002WO2002067865A2 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof
09/06/2002WO2002067684A1 Pyridyl pyrimidines for use as pesticides
09/06/2002WO2002022577A3 Hydroxamate derivatives useful as deacetylase inhibitors
09/06/2002WO2002012534A3 Bio-intermediates for use in the chemical synthesis of polyketides
09/06/2002WO2002008475A3 Method for recovery of copper from sulfidic ore materials using super-fine grinding and medium temperature pressure leaching
09/06/2002CA2439265A1 Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
09/06/2002CA2439119A1 Acylated piperidine derivatives as melanocortin-4 receptor agonists
09/06/2002CA2438895A1 N-substituted nonaryl-heterocyclic nmda/nr2b antagonists
09/06/2002CA2434666A1 Phenylalanine enamide derivatives possessing a cyclobutene group, for use as integrin inhibitors
09/05/2002US20020123629 Benzothiadiazoles and derivatives
09/05/2002US20020123513 Administering indole-2-carboxylic amide derivatives of given formula
09/05/2002US20020123502 5-(4-(2-(2,4-dimethyl-6-oxo-1,6-dihydro-1-pyrimidinyl) -ethoxy)phenyl methyl)thiazolidine-2,4-dione for example; also oxazolidine-2,4-dione, and 1,2,4-oxadiazolidine-3,5-dione derivatives; reducing blood glucose levels
09/05/2002US20020123491 Selective neurokinin antagonists
09/05/2002DE10110325A1 Phenylderivate 2 Phenyl derivatives 2
09/05/2002DE10109867A1 Verwendung von Triazolverbindungen zur Prophylaxe und Therapie neurodegenerativer Erkrankungen, Hirntrauma und zerebraler Ischämie Use of triazole compounds for the prophylaxis and treatment of neurodegenerative diseases, brain trauma and cerebral ischemia
09/04/2002EP1236723A1 Sulfamide derivatives useful as beta3 agonists and pharmaceutical uses thereof
09/04/2002EP1236719A1 Novel heterocyclic compounds and salts thereof and medicinal use of the same
09/04/2002EP1235825A1 Novel benzoimidazole derivatives useful as antiproliferative agents
09/04/2002EP1235816A1 Benzoylcyclohexandione and benzoylpyrazols, method for the production and use thereof as herbicides and plant growth regulators
09/04/2002EP1235803A1 Urea compounds having muscarinic receptor antagonist activity
09/04/2002EP1235802A1 Carbamate derivatives having muscarinic receptor antagonist activity
09/04/2002EP1054886B1 Heteroaryl amidines, methylamidines and guanidines as protease inhibitors, in particular as urokinase inhibitors
09/04/2002EP0944672B1 Helium-neon excitable reticulocyte dyes derivable from halolepidines
09/04/2002EP0882043B1 Halogen pyrimidines and its use thereof as parasite abatement means
09/04/2002EP0809636B1 Substituted isoxazoles for the treatment of inflammation
09/04/2002EP0642506B1 Heterocyclically bisubstituted sulphonyl amino(thio)carbonyl compounds
09/04/2002CN1367780A Oxazolidinones and their preparing method and use thereof
09/04/2002CN1090020C 4,4-(disubstituted) cyclohexan-1-ols and related compounds
09/04/2002CN1090019C 组合物 The composition
09/03/2002US6444827 From beta-methyl l-aspartate via chemical intermediate; efficiency; antidiabetic agents
09/03/2002US6444823 Pyridyl alkane acid amides as cytostatics and immunosuppressives
09/03/2002US6444811 Central nervous system disorders; cardiovascular disorders
09/03/2002US6444809 Antihistamines
09/03/2002US6444687 Eating disorders and diabetes
09/03/2002US6444686 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
09/03/2002US6444679 Neurological and gastrointestinal disorders; delta opioid ligands or opioid receptors