Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
02/2003
02/27/2003US20030040483 Compounds with growth hormone releasing properties
02/27/2003CA2457405A1 Compositions and methods relating to benzodiazepine compounds
02/27/2003CA2457037A1 Aminoalkyl-substituted aromatic bicyclic compounds, method for the production thereof and their use as medicaments
02/27/2003CA2456985A1 2h-phthalazin-1-ones and methods for use thereof
02/27/2003CA2456868A1 Inhibitors of polyq-aggregation
02/27/2003CA2454298A1 Substituted 1h-dihydropyrazoles, their preparation and use
02/26/2003EP1284967A1 3-substituted isoquinolin-1-yl derivatives
02/26/2003EP1284961A1 Glycinamides
02/26/2003EP1284741A2 3'-or 2'-hydroxymethyl substituted nucleoside derivatives for treatment of hepatitis virus infections
02/26/2003EP1284731A1 Use of compounds having combined dopamine d2, 5-ht1a and alpha adrenoreceptor agonistic action for treating cns disorders
02/26/2003EP1100797B1 Heterocyclic compounds as inhibitors of rotamase enzymes
02/26/2003EP0938483B1 Muscarinic antagonists
02/26/2003EP0832068B1 Stable reagents for the preparation of radiopharmaceuticals
02/26/2003EP0708763B1 Process for making hiv protease inhibitors
02/26/2003CN1399635A Piperazing derivatives as 5-HT1B antagonists
02/26/2003CN1399632A Pyrimidine derivatives, process for preparing the derivatives and drugs containing the same as active ingredient
02/26/2003CN1102149C 4-haloalkyl-3-heterocycolyl pyridines and 4-haloalkyl-5-heterocyclylpyridines, method for producing same, composition containing same and use thereof
02/25/2003US6525204 Oximination reaction of nitro-o-methylphenyl compound with organic nitrite; cyclization with alkene in basic catalyst presence; reduction, bromination, oxidation, carboxylation
02/25/2003US6525202 Cyclic amine phenyl beta-3 adrenergic receptor agonists
02/25/2003US6525193 Aminoaryl oxazolidinone N-oxides
02/25/2003US6525079 Antiparasitic compounds such as 4-(2,2-dibromocyclopropyl)-1-(2,6-dichloro-4-trifluoromethylphenyl)-1,2,3 -triazole
02/25/2003US6525076 Selective factor Xa inhibitors
02/25/2003US6525074 Peptidomimetic macrocyclic compounds which inhibit prenyl-protein transferase and the prenylation of the oncogene protein Ras
02/25/2003US6525070 Bipiperidine derivatives as modulators of CCR3 activity and as H1 antagonists
02/25/2003US6525069 Such as N-(t-butyl)-N'-(2-((3-(4-fluorophenyl)methyl)piperi -dinyl)methyl)cyclohexyl)urea; prevention of asthma and other allergic diseases
02/25/2003US6525059 Substituted pyrazoles as p38 kinase inhibitors
02/25/2003US6525052 Compounds useful as reversible inhibitors of cysteine proteases
02/25/2003US6525025 Controlling apoptosis; cardiovascular disorders; central nervous system disorders
02/20/2003WO2003014133A1 Isoxazoline derivatives as p, n ligands
02/20/2003WO2003014094A2 Heterocyclic aryl sulphonamides
02/20/2003WO2003014075A2 Novel gamma secretase inhibitors
02/20/2003WO2003013545A1 Novel benzo-fused heterocycles as endothelin antagonisits
02/20/2003WO2003013531A1 Phenyl derivatives as factor xa inhibitors
02/20/2003WO2003013528A1 Substituted pyridin-4-ones and their use as gonadotropin-releasing hormone receptor antagonists.
02/20/2003WO2003013527A1 Sulfonamide derivatives as gamma secretase inhibitors
02/20/2003WO2003013518A1 Alpha-ketoamide derivatives as cathepsin k inhibitors
02/20/2003WO2003013517A1 Aminoisoxazole derivatives active as kinase inhibitors
02/20/2003WO2003013502A1 Compounds which mimic the chemical and biological properties of discodermolide
02/20/2003WO2003013484A2 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents
02/20/2003WO2002068387A3 Acylated piperidine derivatives as melanocortin-4 receptor agonists
02/20/2003WO2002015940A3 Solution of an oxazolidinone antibiotic drug
02/20/2003US20030036557 Heterocyclo-substituted imidazoles for the treatment of inflammation
02/20/2003US20030036543 Especially as inhibitors of Aurora-2 and GSK-3, for treating diseases such as cancer, diabetes and Alzheimer's disease.
02/20/2003CA2456553A1 Compounds which mimic the chemical and biological properties of discodermolide
02/20/2003CA2456175A1 Benzoquinone ansamycins
02/20/2003CA2455871A1 Substituted pyridin-4-ones and their use as gonadotropin-releasing hormone receptor antagonists.
02/20/2003CA2455861A1 Sulfonamide derivatives as gamma secretase inhibitors
02/20/2003CA2455631A1 Aminoisoxazole derivatives active as kinase inhibitors
02/20/2003CA2454417A1 Novel benzo-fused heterocycles as endothelin antagonists
02/19/2003EP1284267A1 Triazole compounds having amide linkage
02/19/2003EP1283838A1 Piperazine and piperidine compounds
02/19/2003EP1283837A1 New thiochromane derivatives and their use as thrombin inhibitors
02/19/2003EP1020466B1 5,11-DIHYDRODIBENZ[b,e][1,4]OXAZEPINE DERIVATIVES AND MEDICINAL COMPOSITION CONTAINING THE SAME
02/19/2003EP0917530B1 Tetrahydroisoquinoline derivatives as modulators of dopamine d3 receptors
02/19/2003EP0750618B1 Oxazolidinone derivatives and pharmaceutical compositions containing them
02/19/2003EP0690867B1 Taxanes having furyl or thienyl substituted side-chain
02/19/2003CN1398265A 杂环酰胺衍生物 Heterocyclic amide derivatives
02/19/2003CN1398258A 4-hydroxycinnoline-3-carboxyamides as antiviral agents
02/19/2003CN1398189A Combination therapy of radiation and COX-2 inhibitor for treatment of neoplasia
02/19/2003CN1397550A Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them
02/19/2003CN1397547A Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them
02/18/2003US6521653 Microbicidal benzotriazoles
02/18/2003US6521650 Amines as pharmaceutical agents
02/18/2003US6521643 Pyridine compounds and their pharmaceutical use
02/18/2003US6521629 2-amine substituted quinoline or quinozoline derivatives useful for treating benign prostatic hyperplasia
02/18/2003US6521622 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
02/18/2003US6521621 1-(1,2-disubstituted piperidinyl)-4-substituted piperazine derivatives
02/18/2003US6521614 N-(amidinophenyl)cyclourea analogs as factor Xa inhibitors
02/18/2003US6521611 2-(azetidin-2-on-1-yl) acetic acid derivatives; treatment of obsessive-compulsive disorder
02/18/2003US6521610 4-Haloalkyl-3-heterocyclylpyridines and 4-haloalkyl-5-heterocyclyl-pyrimidines, processes for their preparation, compositions comprising them, and their use as pesticides
02/18/2003US6521592 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
02/13/2003WO2003011861A1 Azole derivatives useful as insecticide
02/13/2003WO2003011859A2 Oxazolidinone derivatives as antibacterial agents
02/13/2003WO2003011853A1 6-aryl-4-aminopicolinates and their use as herbicides
02/13/2003WO2003011842A1 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation
02/13/2003WO2003011836A1 Tyrosine kinase inhibitors
02/13/2003WO2003011833A1 Indazole or indole derivatives, their use in human medicine and more particularly in cancerology
02/13/2003WO2003011830A1 Heteroarylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase
02/13/2003WO2003011396A1 Tetrahydroindolone and purine derivatives linked to arylpiperazines
02/13/2003WO2003011297A1 N3-substituted 6-anilinopyrimidines and methods to treat gram-positive bacterial and mycoplasmal infections
02/13/2003WO2001077107A8 Oxazole derivatives and their uses as tyrosine kinase inhibitors
02/13/2003US20030032811 Sulfonyltriazol derivatives and their use for combating micro-organisms
02/13/2003US20030032654 Useful for the treatment or prevention of asthma and other allergic diseases.
02/13/2003US20030032647 Aromatic nitrogen-containing 6-membered cyclic compounds
02/13/2003CA2753329A1 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation
02/13/2003CA2452751A1 Azole derivatives useful as insecticide
02/12/2003EP1283205A1 Naphthol derivatives
02/12/2003EP1283199A1 Melanin-concentrating hormone antagonist
02/12/2003EP1283055A1 Soluble beta amyloid precursor protein secretion promoters
02/12/2003EP1282621A1 Novel vitronectin receptor antagonists
02/12/2003EP1282619A1 Processes for the preparation of thiazolidinedione derivatives and intermediates
02/12/2003EP1282618A2 9-oxa-epothilon derivatives, method for the production and use thereof in pharmaceutical preparations
02/12/2003EP1282606A2 Hiv replication inhibiting pyrimidines and triazines
02/12/2003EP1282601A1 Process and intermediates for the preparation of 1-(9h-carbazol-4-yloxy)-3-[2-(2-methoxy-phenoxy)-ethylamino]-propan-2-ol, carvedilol or acid addition salt thereof
02/12/2003EP1282600A1 Inhibitors of dipeptidyl peptidase iv
02/12/2003EP1282420A2 Halogenated 2-amino-3, 4 heptenoic acid derivatives useful as nitric oxide synthase inhibitors
02/12/2003EP1282413A1 Halogenated 2-amino-5,6 heptenoic acid derivatives useful as nitric oxide synthase inhibitors
02/12/2003EP0988292B1 Piperazine derivatives and their use as anti-inflammatory agents
02/12/2003EP0868424B1 4-pyrimidinyl- or 4-pyrazinyl-piperazinyl-phenyl-oxazolidinone derivatives, their preparation and their use as anti-bacterial agents
02/12/2003EP0861239B1 Biphenyl ether oxazolines and their use as pest-control agents