Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/2003
01/08/2003EP1272477A1 Pyrimidine compounds
01/08/2003EP1272474A1 Substituted 5-methyldihydropyridazinones and their use in the prophylaxis and/or treatment of anemias
01/08/2003EP1272178A2 Bilirubin or biliverdin degradation fragments
01/08/2003EP1272168A2 Small organic molecule regulators of cell proliferation
01/08/2003EP1123284B1 Method for the preparation of citalopram
01/08/2003EP1077945B1 Isoquinolines as urokinase inhibitors
01/08/2003EP0946175B1 USE OF A COMBINATION OF H+, K+ -ATPase INHIBITORS AND GLUCOCORTICOIDS IN THE TREATMENT OF NASAL POLYPS
01/08/2003EP0934286B1 3-alkoxyisoxazol-4-yl-substituted 2-amino carboxylic acid compounds
01/08/2003EP0892795B1 Piperidinylpyramidine derivatives
01/08/2003EP0889033B1 Alpha-substituted benzyl heterocyclic derivatives, intermediates for producing the same, and pesticides containing the same as active ingredient
01/08/2003CN1390214A New phenylpiperazines
01/08/2003CN1390210A Process for preparing oxazolines from tetrahydrofurans
01/08/2003CN1390204A Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/08/2003CN1390201A Cyclic amine compounds as CCR5-antagonists
01/08/2003CN1098263C Pyridin-2-yl-methylaminederivatives, method of preparing and application as medicine
01/08/2003CN1098259C Novel carboxy substituted cyclic carboxamide derivatives
01/08/2003CN1098104C New oral pharmaceutical dosage form
01/07/2003US6503935 Imidazoles and related compounds as α1A agonists
01/07/2003US6503926 Nitrogen heterocycle compounds
01/07/2003US6503925 Treating anxiety, anesthesia, and epilepsy
01/07/2003US6503913 2-heterocyclically substituted dihydropyrimidines
01/07/2003US6503907 Indole and dihydroindole derivatives
01/07/2003US6503905 3,3-biarylpiperidine and 2,2-biarylmorpholine derivatives
01/07/2003US6503901 Amino lactam sulfonamides as inhibitors of Aβ protein production
01/07/2003US6503898 Administering 4,7-dibenzyl-5,6-dihydroxy-N,N*-di(m-aminobenzyl)--1,3-diazepin-2-one or salt to treat human immunodeficiency virus infection
01/07/2003CA2143208C Sulfonamide inhibitors of hiv-aspartyl protease
01/07/2003CA2047531C 1-(substituted pyridinylamino)-1h-indol-5-yl substituted carbamates, a process and intermediates for their preparation and their use as medicaments
01/06/2003CA2392187A1 Combination preparation for the therapy of immunological diseases
01/03/2003WO2003000692A2 Oxytocin agonists
01/03/2003WO2003000686A1 Isoxazoline derivatives and herbicides
01/03/2003WO2003000685A1 5-membered heterocycle derivatives
01/03/2003WO2003000677A1 Spiropiperidine compounds as ligands for orl-1 receptor
01/03/2003WO2003000676A1 1,2,4-trioxolane antimalarials
01/03/2003WO2003000669A1 2-(2,6-disubstituted phenyl)-4-aryl-5-alkyl-1,3-oxazoline compounds useful as insecticides and acaricides
01/03/2003WO2003000668A1 Oxa(thia)zolidine compounds, process for preparation thereof and anti-inflammatory agents
01/03/2003WO2003000660A1 Quinoline derivative and quinazoline derivative inhibiting self-phosphorylation of hepatocytus proliferator receptor, and medicinal composition containing the same
01/03/2003WO2003000267A1 Amino nicotinate derivatives as glucokinase (glk) modulators
01/03/2003WO2003000262A1 Vinyl phenyl derivatives as glk activators
01/03/2003WO2003000256A1 Substituted oxazolidinones for combinational therapy
01/03/2003WO2003000180A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003WO2002046170A8 Anilinopyrimidine derivatives as jnk pathway inhibitors and compositions and methods related thereto
01/03/2003WO2002020531A3 Method for producing anellated tetrahydro-[1h]-triazoles
01/03/2003WO2001083800A8 Heterologous production of polyketides
01/03/2003CA2454538A1 Quinoline derivatives and quinazoline derivatives capable of inhibiting autophosphorylation of hepatocyte growth factor receptors, and pharmaceutical composition comprising the same
01/03/2003CA2451249A1 Amino nicotinate derivatives as glucokinase (glk) modulators
01/03/2003CA2450579A1 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003CA2450550A1 Spiropiperidine compounds as ligands for orl-1 receptor
01/03/2003CA2450480A1 Oxytocin agonists
01/02/2003WO2002002529A1 Bicyclic lactams and sulfonamides with 5-ht1a-affinity and use thereof for preventing and treating cerebral ischaemia
01/02/2003US20030004354 Thienylsulphonylamino(thio)carbonyl compounds
01/02/2003US20030004351 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
01/02/2003US20030004344 Thrombin or factor Xa inhibitors
01/02/2003US20030004340 Skin disorders; gastrointestinal disorders
01/02/2003US20030004212 Cyclohexylamine derivatives as subtype selective N-Methyl-D-Aspartate antagonists
01/02/2003US20030004210 Coupling to cell binding agent; killing cells
01/02/2003US20030004196 Antiinflamamtory agents; autoimmune disease
01/02/2003US20030004195 Reducing pressure in eye
01/02/2003US20030004194 Method for treating fibrotic diseases or other indications VI
01/02/2003US20030004187 Method for preventing dyskinesias
01/02/2003US20030004185 Viricides, organ transplants, antiarthritic agents
01/02/2003US20030004174 Antiinflammatory agents, anticancer agents, antihistamines, central nervous system disorders
01/02/2003US20030004164 Anticancer agents; autoimmune diseases
01/02/2003US20030004162 Antidiabetic agents; dietetics
01/02/2003US20030004161 Anticancer agents; autoimmune diseases
01/02/2003US20030004137 Muscle relaxants, controlling immunology, strokes, antidiabetic agents
01/02/2003US20030003396 Reflection, protective or covering layers which can be written on or read by blue, red or infrared light
01/02/2003EP1270571A1 Heterocyclic compounds, their production and use
01/02/2003EP1270569A1 Substituted tryptophan derivatives
01/02/2003EP1268473A1 Oxazole derivatives and their uses as tyrosine kinase inhibitors
01/02/2003EP1268472A1 3-aminopyrazole inhibitors of cyclin dependent kinases
01/02/2003EP1268466A1 Decahydro-isoquinolines
01/02/2003EP1268465A1 Triarylimidazole derivatives as cytokine inhibitors
01/02/2003EP1268449A1 Substituted piperidines as melanocortin receptor agonists
01/02/2003EP1268446A1 Method for producing asymmetrical 4,6-bis(aryloxy)pyrimidine derivatives
01/02/2003EP1268431A1 3-cyanoquinolines,3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors
01/02/2003EP1268422A1 Indoles for treating diseases that can be treated using thyroid hormones
01/02/2003EP1268412A1 Sulphonamido-substituted bridged bicycloalkyl derivatives
01/02/2003EP1268407A1 Propenecarboxylic acid amidoxime derivatives, a process for the preparation thereof, and pharmaceutical compositions containing the same
01/02/2003EP0934265B1 Amidinophenyl-pyrrolidines, -pyrrolines, and -isoxazolidines and derivatives thereof
01/02/2003EP0925286B1 Substituted pyrimidine derivatives and their pharmaceutical use
01/02/2003EP0891341B1 1,3,4-oxadiazine derivatives and their use as pesticides
01/02/2003EP0821719B1 Liquid crystal compounds having a chiral fluorinated terminal portion
01/02/2003CA2414726A1 Bicyclic lactams and sulfonamides with 5-ht1a-affinity and use thereof for preventing and treating cerebral ischaemia
01/01/2003CN1388804A Amino acid-N-carboxy anhydrides having substitent at nitrogen
01/01/2003CN1387849A Use of thiazolidinedione for preventing or retaining non-insulin-dependent diabets mellitus (NIDDM) attack
01/01/2003CN1387848A Use of thiazolidinedione for preventing or retaining non-insulin-dependent diabets mellitus (NIDDM) attack
12/2002
12/31/2002US6500966 Process for the preparation of taxanes from 10-deacetylbaccatin III
12/31/2002US6500950 Benzylidenepyrazolones, their preparation and use
12/31/2002US6500855 Nitrogen containing aromatic heterocycles with ortho-substituted p1 groups; anticoagulants
12/31/2002US6500848 Pesticides
12/31/2002US6500846 2-(4-chlorophenyl)-7-methoxychromen-4-one, as cyclin-dependent kinase inhibitors, used as anticarcinogenic agents or for prophylaxis of neurodegenerative disease
12/31/2002US6500844 Cyclopentyl modulators of chemokine receptor activity
12/31/2002US6500842 N-((4-chlorophenyl)methyl)-8-hydroxy-7-quinolinecarboxamide administered as viricides against herpes virus
12/31/2002US6500822 Benzocycloalkylenylamine derivatives as muscarinic receptor antagonists
12/27/2002WO2002102800A1 5-(2-aminopyrimidin-4-yl) benzisoxazoles as protein kinase inhibitors
12/27/2002WO2002102799A2 Pyrrolidine oxadiazole- and thiadiazole oxime derivatives being oxytocin receptor antagonists
12/27/2002WO2002102795A1 Fluorescent probes for zinc
12/27/2002WO2002102793A2 Quinazolinediones as antibacterial agents
12/27/2002WO2002102791A1 Pyrrolidine bicyclic compounds
12/27/2002WO2002102785A1 Novel bicyclic isoxazolinones as antibacterial agents