Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/2003
01/30/2003US20030022907 Anxiolytic agents and analgesics
01/30/2003US20030022905 Prevention and/or therapy of ischaemia and reperfusion damage; poly(ADP-ribose)-synthetase inhibitors
01/30/2003US20030022895 2-Amino-benzoxazinones for the treatment of viral infections
01/30/2003US20030022885 Pyrazole compounds useful as protein kinase inhibitors
01/30/2003US20030022884 Heterocycle derivatives and drugs
01/30/2003CA2454059A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors
01/30/2003CA2454007A1 Tetrahydroquinoxalines acting as bradykinin antagonists
01/30/2003CA2453846A1 Substituted isoxazoles and the use thereof as antibiotics
01/30/2003CA2453650A1 Substituted isoindoles and the use thereof
01/30/2003CA2417955A1 Quinazolines, pharmaceutical compositions containing these compounds, their use and processes for preparing them
01/30/2003CA2417907A1 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for preparing them
01/30/2003CA2417804A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof
01/29/2003EP1278744A1 Heterobicyclic sulfonamides and their use as platelet adp receptor inhibitors
01/29/2003EP1278741A1 Muscarinic agonists
01/29/2003EP1278739A1 Amino substituted dibenzothiophene derivatives for the treatment of disorders mediated by the np y5 receptor
01/29/2003EP1278735A1 2,4-di(hetero-)arylamino(-oxy)-5-substituted pyrimidines as antineoplastic agents
01/29/2003EP1278728A1 Pyrrolidine and piperidine derivatives and their use for the treatment of neurodegenerative disorders
01/29/2003EP1278520A1 Diaryl piperidyl pyrrole derivatives as antiprotozoal agents
01/29/2003EP1192145A4 Process for preparing chiral cyclopropane carboxylic acids and acyl guanidines
01/29/2003EP1036074B1 S-oxide tetrahydrothiopyran phenyloxazolidinones
01/29/2003EP0906294B1 Benzoxazinone dopamine d4 receptor antagonists
01/29/2003EP0708769B1 Substituted 2-fused phenylpyridines with herbicidal activity
01/29/2003CN1394207A Linezolid-crystal form II
01/29/2003CN1394202A Picolinic acid derivatives and their use as fungicides
01/29/2003CN1100055C Piperazine and piperidine compounds
01/29/2003CN1100046C 喹唑啉衍生物 Quinazoline derivatives
01/28/2003WO2002018372A1 Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
01/28/2003US6512135 2-methyl-3-(protected hydroxy) benzyl chloride; use making nelfinavir mesylate
01/28/2003US6512112 Useful as prodrugs, easily convert to parent amine in vivo; antibiotic activity versus gram negative aerobic and anaerobic bacteria
01/28/2003US6512001 D-proline derivatives
01/28/2003US6511994 Modulators of CCR5 chemokine receptor activity
01/28/2003US6511977 For preventing or treating cardiac arrhythmia or atrial arrhythmia
01/28/2003US6511975 Spiropiperidine derivatives
01/28/2003US6511973 Enzyme inhibitors of blood coaggulation factor X for use as anticoaggulants in the treatment of cardiovascular diseases associated with thromboses
01/24/2003WO2002010145A1 Urethane derivatives
01/24/2003CA2417268A1 Urethane derivatives
01/23/2003WO2003006462A1 Processes for the manufacture of thrombin inhibitors and n-pyridin-4-yl-oxazolidin-2-ones as intermediate therefor
01/23/2003WO2003006461A1 Substituted benzo-nitro-heterocycles
01/23/2003WO2003006459A1 Piperazine oxime derivatives having nk-1 receptor antagonistic activity
01/23/2003WO2003006447A2 Interaction inhibitors of tcf-4 with beta-catenin
01/23/2003WO2003006440A2 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
01/23/2003WO2003006437A1 Imidazole derivatives as adenosine deaminase inhibitors
01/23/2003WO2003006423A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003WO2003006016A2 Use of nk-1 receptor antagonists with pyridinic structure, for the treatment of brain, spinal or nerve injury
01/23/2003WO2003006012A1 Compounds and methods for the inhibition of trypanosoma cruz i
01/23/2003WO2003005999A2 Methods of treating cytokine mediated diseases
01/23/2003WO2003005824A2 Substituted 3-heteroaryl (amino-or-oxy)-pyrrolidin-2-ones, method for the production thereof and use thereof as herbicides or as plant growth regulators
01/23/2003WO2002050066A3 Pyrazole compounds useful as protein kinase inhibitors
01/23/2003WO2002046171A3 Anilinopyrimidine derivatives as ikk inhibitors and compositions and methods related thereto
01/23/2003WO2002036562A3 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
01/23/2003WO2002034760A3 Compounds and methods
01/23/2003WO2002022559A3 2-amino-2-alkyl-4 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors
01/23/2003WO2002008177A2 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
01/23/2003US20030018200 Preparation of isoxazolin-3-ylacylbenzenes
01/23/2003US20030018199 Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors
01/23/2003US20030018197 Administering a therapeutically effective amount of a pyrrazole sulfide or ether compound to treat the human immunodeficiency virus infection
01/23/2003US20030018193 Beta-alanine derivatives and their use as receptor anatgonists
01/23/2003US20030018059 Antiinflammatory agents; antihistamines; antiallergens
01/23/2003US20030018058 3-aminopyrazole inhibitors of cyclin dependent kinases
01/23/2003US20030018046 Chemokine receptor binding heterocyclic compounds
01/23/2003US20030018029 Tyrosine kinase inhbitor; antiproliferative agents
01/23/2003US20030018021 Piperidine derivatives as subtype selective N-methyl-D-aspartate antagonists
01/23/2003US20030018016 Cell adhesion inhibitors
01/23/2003US20030017166 Combination preparation for the therapy of immunological diseases
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003CA2453421A1 Substituted benzo-nitro-heterocycles
01/23/2003CA2453396A1 Compounds and methods for the inhibition of trypanosoma cruzi
01/23/2003CA2453175A1 Interaction inhibitors of tcf-4 with beta-catenin
01/23/2003CA2453147A1 Methods of treating cytokine mediated diseases
01/23/2003CA2452513A1 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
01/23/2003CA2451566A1 Use of nk-1 receptor antagonists for the treatment of brain, spinal or nerve injury
01/23/2003CA2446726A1 Piperazine oxime derivatives having nk-1 receptor antagonistic activity
01/23/2003CA2418173A1 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
01/23/2003CA2417156A1 3,4-dihydroisoquinoline derivative compound and a pharmaceutical agent comprising it as active ingredient
01/22/2003EP1277744A1 Oxadiazole derivatives having anticancer effects
01/22/2003EP1277743A1 Oxa(thia)zolidine derivative and anti-inflammatory drug
01/22/2003EP1277741A1 Cyclic compounds
01/22/2003EP1277738A1 Condensed heteroaryl derivatives
01/22/2003EP1276740A2 Novel epothilone derivatives, method for the preparation thereof and their pharmaceutical use
01/22/2003EP1276739A2 Heterocycles that are inhibitors of impdh enzyme
01/22/2003EP1276730A2 Thiazolidinedione analogues and their use for the treatment of diabetes
01/22/2003EP1276729A1 New neurokinin antagonists for use as medicaments
01/22/2003EP1276726A2 Substituted phenyl farnesyltransferase inhibitors
01/22/2003EP1276725A2 5-substituted tetralones as inhibitors of ras farnesyl transferase
01/22/2003EP1276723A2 Pyrazole compounds having anti proliferative activity
01/22/2003EP1157018B1 A process for the preparation of taxanes from 10-deacetylbaccatin iii
01/22/2003EP1030835B1 Urea derivatives and their use as integrin inhibitors
01/22/2003EP1006114B1 Pyrazole derivatives and cox inhibitors containing them
01/22/2003EP0782575B1 Substituted pyrazolyl-pyrazole derivatives, processes for their preparation and their use as agents with herbicidal action
01/22/2003EP0729465B1 Pyrone derivatives as protease inhibitors and antiviral agents
01/22/2003EP0646115B1 Heterocyclic-cyclic amine derivatives
01/22/2003CN1392875A Condensed azepines as vasopressino agonists
01/22/2003CN1392874A Cyclic amidine compounds
01/22/2003CN1099413C Certain fused N-pyrrolylaniline: new class of GABA brain receptor ligand
01/21/2003US6509464 1-Heteroaryl-pyrrolidine, piperidine, or homopiperidine derivates; nervous system disorder treatment; amidation
01/21/2003US6509335 This invention discloses benzoxazinone and benzothiazinone compounds which display inhibitory effects on serine proteases such as factor Xa, thrombin, and/or factor VIIa. The invention also discloses pharmaceutically acceptable salts of
01/21/2003US6509334 Cyclocarbamate derivatives as progesterone receptor modulators
01/21/2003US6509328 Glutamate receptor antagonists
01/17/2003WO2002006269A1 Cyclic amino acid derivatives
01/17/2003CA2415964A1 Cyclic amino acid derivatives