Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
11/2002
11/07/2002WO2002087587A2 4-aminosulfonylquinazolines and -quinolines as tyrosine kinase inhibitors
11/07/2002WO2002087580A1 Abc expression promoters
11/07/2002WO2001042243A3 Protein kinase inhibitors
11/07/2002US20020165412 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof
11/07/2002US20020165400 Antagonists of the platelet glycoprotein IIb/IIIa fibrinogen receptor complex; thrombolytic agents
11/07/2002US20020165398 Amino-thiophene-amido derivatives
11/07/2002US20020165393 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids
11/07/2002US20020165253 Such as N-(4-chlorobenzyl)-8-(4-hydroxybut-1-ynyl)-1-methyl-6-(morpholin-4-ylmethyl)-4-oxo-1,4-dihydroquinoline-3-carboxamide for treatment against herpes viruse; enzyme inhibitors
11/07/2002US20020165241 Such as 4-((methyl-pyrimidin-2-ylamino)-methyl)-piperidine-1-carboxylic acid benzyl ester; useful for pain relief; treating migraine, depression, anxiety, schizophrenia, Parkinson's disease, and stroke; N-methyl-D-aspartate (NMDA)
11/07/2002US20020165240 Method of treating proliferative diseases using Eg5 inhibitors
11/07/2002US20020165234 Selective B3 adrenergic agonists
11/07/2002US20020165230 Gamma-ketoacid dipeptides as inhibitors of caspase-3
11/07/2002US20020165228 Antiproliferative agents; antidiabetic agents
11/07/2002US20020165219 Novel heterocycles useful in the treatment of benign prostatic hyperplasia
11/07/2002US20020165203 Enzyme inhibitors; antiinflammatory agents; rheumatic diseases; antidiabetic agents
11/07/2002CA2445348A1 Novel benzylpiperidine compound
11/07/2002CA2444500A1 Triazole compounds useful in treating diseases associated with unwanted cytokine activity
11/07/2002CA2444499A1 Triazole compounds useful in treating diseases associated with unwanted cytokine activity
11/06/2002EP1254906A1 Tetrahydrothiopyran phenyloxazolidinone S,S-dioxides
11/06/2002EP1254904A1 Novel piperidine compounds and drugs containing the same
11/06/2002EP1254901A1 Nitrogen-containing 5-membered cyclic compounds and drugs containing these compounds as the active ingredient
11/06/2002EP1254899A2 Piperazine derivatives and their use as anti-inflammatory agents
11/06/2002EP1254897A1 Tricyclic compounds
11/06/2002EP1254895A1 Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
11/06/2002EP1254667A1 Drug comprising combination
11/06/2002EP1254661A1 Method for preventing dyskinesias with selective NMDA-Antagonists
11/06/2002EP1254136A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF
11/06/2002EP1254134A2 1,3-dihydro-2h-indol-2-one derivatives,and their use as ligands for v1b or v1b and v1a arginine-vasopressin-receptors
11/06/2002EP1254129A1 Method for the preparation of 5-cyanophthalide
11/06/2002EP1254119A1 Pyrimidine derivatives as selective inhibitors of cox-2
11/06/2002EP1254115A2 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators for treating respiratory and non-respiratory diseases
11/06/2002EP1253925A1 Tetrahydropyrimidone inhibitors of fatty acid binding protein and method
11/06/2002EP1253916A1 Method of treating vaginal dryness with nicotinic acetylcholine receptor agonists
11/06/2002EP1135387B1 3-(heterocyclyl)-benzoylpyrazole-derivatives
11/06/2002EP0993459B1 Compounds useful for inhibition of farnesyl protein transferase
11/06/2002EP0927168B1 1,3-diheterocyclic metalloprotease inhibitors
11/06/2002EP0920421B1 Isoxazoline derivatives useful as antimicrobials
11/06/2002EP0912559B1 Fused heterocyclic compounds as protein tyrosine kinase inhibitors
11/06/2002EP0898566B1 Substituted benzylamines and their use for the treatment of depression
11/06/2002EP0879229B1 Arylpyrazole insecticides
11/06/2002CN1378546A Antibiotic sultam and sultone drived oxazolidiones
11/06/2002CN1378544A Substituted azoles compounds
11/06/2002CN1378541A Inhibitors of c-JUN N-terminal kinase (JNK) and other protein kinases
11/06/2002CN1378540A New piperazine and piperidine compounds
11/06/2002CN1378539A Thiocarbamic acid derivatives
11/06/2002CN1378537A 嘧啶衍生物 Pyrimidine derivatives
11/06/2002CN1378533A Phenoxypropylamine compounds
11/06/2002CN1378446A Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
11/06/2002CN1093858C Quinoline and quinozoline compounds useful in therapy, particularly in the treatment of begnin prostatic hyperplasia
11/06/2002CN1093857C New piperazine and piperidine compounds
11/06/2002CN1093856C Substituted sulfonic acid N-[(aminoiminomethyl)phenylalkyl]-azaheterocyclamide compounds
11/05/2002US6476235 Process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1H-pyrrole-3-carboxylic acid phenylamide
11/05/2002US6476232 4-(2-amino-1-hydroxyethyl)oxazoline derivative and method for producing same
11/05/2002US6476226 Isoxazoline fibrinogen receptor antagonists
11/05/2002US6476040 Processes and intermediates for preparing anti-cancer compounds
11/05/2002US6476024 Pyridazine derivatives and related composition
11/05/2002US6476016 Inhibiting loss of blood platelets, inhibiting formation of blood platelet aggregates, inhibiting formation of fibrin, inhibiting thrombus formation, and inhibiting embolus formation
11/04/2002WO2004001058A2 Transcription factor modulating compounds and methods of use thereof
10/2002
10/31/2002WO2002085906A2 Phthalazinones derivatives useful as pde4/7 inhibitors
10/31/2002WO2002085898A1 Clathrate of azithromycin hydrate with 1,2-propyleneglycol, method for the manufacture thereof and pharmaceutical composition comprising same
10/31/2002WO2002085897A1 Heterocyclic compounds for aging-related and diabetic vascular complications
10/31/2002WO2002085891A1 2,6-substituted chroman derivatives useful as beta-3 adrenoreceptor agonists
10/31/2002WO2002085886A2 Chiral, broad-spectrum antibacterial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation and compositions
10/31/2002WO2002085885A1 Piperazino-derivatives and their use as pde4 inhibitor
10/31/2002WO2002085869A1 Arylsulfonamides as antiviral agents
10/31/2002WO2002085866A1 Novel compounds
10/31/2002WO2002085860A1 Pyrazole derivatives for treating hiv
10/31/2002WO2002085855A1 2-iminopyrrolidine derivatives
10/31/2002WO2002085854A1 5-aryl-1.3.3.-trimethyl-2-methylene-indoline derivatives and salts thereof, methods for the production and use of said compounds for the temporary coloration of fibres
10/31/2002WO2002085850A1 Cyclic amidine derivative
10/31/2002WO2002085849A2 Process to prepare oxazolidinones
10/31/2002WO2002085412A1 Tissue fibrosis inhibitors
10/31/2002WO2002085357A1 Nociceptin analogs
10/31/2002WO2002064574A3 Pyridoarylphenyl oxazolidinone antibacterials, and related compositions and methods
10/31/2002WO2002022611A3 Caspase inhibitors and uses thereof
10/31/2002US20020161238 Novel methods for the preparation of taxanes using oxazolidine intermediates
10/31/2002US20020161236 2-methyl-3-(protected hydroxy) benzyl chloride; use making nelfinavir mesylate
10/31/2002US20020161038 Inosine 5'-monophosphate dehydrogenase (IMPDH); prodrug having functional group -CO-N(-R)-COO-, a carrier, and an immunosuppressant, anticancer agent, antiviral agent, or anti-vascular hyperproliferation agent
10/31/2002US20020161029 Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods
10/31/2002US20020161005 Nitrogen heterocycle compounds
10/31/2002US20020161004 Antiinflammation agents
10/31/2002US20020160984 For example, 2,3-dihydro-1H-benz(de)isoquinolin-1-one; treating diabetes, cancer, radiosensitizing tumor cells, cardiovascular disorders, septic shock, inflammatory bowel disease, senescent cells
10/31/2002US20020160983 Substituted benzopyranones as telomerase inhibitors
10/31/2002CA2445888A1 Chiral, broad-spectrum antibacterial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation and compositions
10/31/2002CA2445236A1 Piperazino-derivatives and their use as pde4 inhibitor
10/31/2002CA2445233A1 Phthalazinones derivatives useful as pde4/7 inhibitors
10/31/2002CA2445114A1 Clathrate of azithromycin hydrate with 1,2-propyleneglycol, method for the manufacture thereof and pharmaceutical composition comprising same
10/31/2002CA2444563A1 Tissue fibrosis inhibitors
10/31/2002CA2444381A1 Novel compounds
10/31/2002CA2440600A1 Process to prepare oxazolidinones
10/30/2002EP1252158A1 Nicotinamide benzofused-heterocyclyl derivatives useful as selective inhibitors of pde4 isozymes
10/30/2002EP1252156A1 Blockade of voltage dependent sodium channels
10/30/2002EP1252154A1 Heterocyclic amide derivatives
10/30/2002EP1252145A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
10/30/2002EP1252140A1 Pyrrolecarboxamides and pyrrolethioamides as fungicides
10/30/2002EP1252139A1 Trifluoromethylpyrrole carboxamides and trifluoromethylpyrrolethioamides as fungicides
10/30/2002EP1251848A1 Gyrase inhibitors and uses thereof
10/30/2002EP1000172A4 Detection of targets with green fluorescent protein and fluorescent variants thereof
10/30/2002EP0852225B1 Fibrinogen receptor antagonists and medicinal preparations containing the same as the active ingredient
10/30/2002CN1377348A 4,5-diaryloxazole compounds with prostaglandin 12 (PG12) agonistic activity