Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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11/22/2000 | CN1274353A Halogen substituted tetracyclic tetrahydrofuran derivatives |
11/22/2000 | CN1274283A Quinoline-containing & Alpha;-ketoamide cysteine and serine protease inhibitors |
11/22/2000 | CN1058723C D4T polymorphic form I process |
11/22/2000 | CN1058712C Microbicidal triazolyl derivatives |
11/22/2000 | CN1058710C Benzamide derivatives, process for prepn. thereof and pharmaceutical compsn. comprising same |
11/22/2000 | CN1058709C Amide compounds for medical treatment |
11/21/2000 | US6150557 Compounds |
11/21/2000 | US6150527 Synthetic multimerizing agents |
11/21/2000 | US6150526 Piperidine derivative having renin inhibiting activity |
11/21/2000 | US6150416 2-hydroxy-3-(substitued benzyl)-n,n'-bis(substituted carbonyl)-n-(substituted)-1,3-propanediamine based compounds; use in the detection, labelling and inhibition of cathepsin d |
11/21/2000 | US6150397 5-aroylnaphthalene derivatives as anti-inflammatory agents |
11/21/2000 | US6150394 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same |
11/21/2000 | US6150379 Compounds and compositions as anticoagulants |
11/21/2000 | US6150375 Inhibitors of both of the human 5ar isozymes; benign prostate hyperplasia, male pattern baldness, acne vulgaris, seborrhea, androgenic alopecia, hirsutism and prostate cancer; blocks the conversion of testosterone to 5-alpha-dihydrotestosterone |
11/21/2000 | US6150362 Administering 1,3,5-substituted triazine compounds to the patient suffering from angiogenic diseases |
11/21/2000 | US6150356 Potassium channel inhibitors and method |
11/21/2000 | US6150355 Phenylpiperidine derivative |
11/21/2000 | US6150352 Antagonists of gonadotropin releasing hormone |
11/16/2000 | WO2000068225A1 Substituted benzimidazole, the production thereof and the use thereof as means against parasitic protozoa |
11/16/2000 | WO2000068213A1 Substituted bicyclic compounds |
11/16/2000 | WO2000068208A1 Pyrimidinones derivatives for the treatment of atherosclerosis |
11/16/2000 | WO2000068206A1 Heterocyclically substituted benzimidazoles, the production and application thereof |
11/16/2000 | WO2000068203A1 Cyclic compounds and uses thereof |
11/16/2000 | WO2000068202A1 Substituted 4-oxo-quinoline-3-carboxamides: gaba brain receptor ligands |
11/16/2000 | WO2000068201A1 Quinoline derivatives as inhibitors of mek enzymes |
11/16/2000 | WO2000068198A2 Heterosubstituted pyridine derivatives as pde 4 inhibitors |
11/16/2000 | WO2000068197A1 3a,4,5,9b-TETRAHYDRO-1H-BENZ[e]INDOL-2-YL AMINE-DERIVED NEUROPEPTIDE Y RECEPTORS LIGANDS USEFUL IN THE TREATMENT OF OBESITY AND OTHER DISORDERS |
11/16/2000 | WO2000068188A1 Propanoic acid derivatives that inhibit the binding of integrins to their receptors |
11/16/2000 | WO2000067801A2 Prodrugs of chemotherapeutic agents with oxaalkanoic acids |
11/16/2000 | WO2000067746A1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors |
11/16/2000 | WO2000067735A2 USE OF SELECTIVE ANTAGONISTS OF THE α1b-ADRENERGIC RECEPTOR FOR IMPROVEMENT OF SEXUAL DYSFUNCTION |
11/16/2000 | WO2000067729A1 Regimen and kit for amelioration of premature ejaculation |
11/16/2000 | WO2000038665A3 Use of an integrin antagonist and one or more antineoplastic agents as a combination therapy in the treatment of neoplasia |
11/16/2000 | WO2000020358A3 NON-PEPTIDE GnRH AGENTS, METHODS AND INTERMEDIATES FOR THEIR PREPARATION |
11/16/2000 | WO2000015634A3 Hiv protease inhibitors |
11/16/2000 | DE19923001A1 New epothilone derivatives, used as mitosis regulators e.g. for treating malignant tumors, psoriasis or arthritis |
11/16/2000 | DE19922317A1 Preparation of N-(Benzofuranyl-alkoxycarbonyl)-tryptophan ester derivative, used as tachykinin antagonist intermediate, comprises reacting tryptophan ester with carbon dioxide and carbonate, then with benzofuran derivative |
11/16/2000 | DE19922316A1 N-(Benzofuranyl-alkoxycarbonyl)-tryptophan ester preparation, for use as tachykinin receptor antagonist intermediate, by reacting hydroxyalkyl-benzofuran with disuccinimidyl carbonate, then with tryptophan ester |
11/16/2000 | DE19922315A1 N-(Benzofuranyl-alkoxycarbonyl)-tryptophan ester preparation, for use as tachykinin receptor antagonist intermediate, by reacting tryptophan ester with N,N'-carbonyl diimidazole then benzofuran derivative |
11/16/2000 | CA2373073A1 Cyclic compounds and uses thereof |
11/16/2000 | CA2373035A1 3a,4,5,9b-tetrahydro-1h-benz¬e|indol-2-yl amine-derived neuropeptide y receptors ligands useful in the treatment of obesity and other disorders |
11/16/2000 | CA2372663A1 Quinoline derivatives as inhibitors of mek enzymes |
11/16/2000 | CA2371472A1 Substituted 4-oxo-quinoline-3-carboxamides: gaba brain receptor ligands |
11/16/2000 | CA2369323A1 Heterosubstituted pyridine derivatives as pde 4 inhibitors |
11/16/2000 | CA2368831A1 Permeable, water soluble, non-irritating prodrugs of chemotherapeutic agents with oxaalkanoic acids |
11/16/2000 | CA2366201A1 Use of selective antagonists of the .alpha.1b-adrenergic receptor for improvement of sexual dysfunction |
11/15/2000 | EP1052261A1 Pyran derivatives and use thereof |
11/15/2000 | EP1052255A1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics. |
11/15/2000 | EP1052254A1 Nitrogenous heterocyclic derivatives and medicine thereof |
11/15/2000 | EP1051413A1 Quinoline derivatives as antibacterials |
11/15/2000 | EP1051407A1 2,3,4,5-tetrahydro-1h-[1,4]-benzodiazepine-3-hydroxamic acids as matrix metalloproteinase inhibitors |
11/15/2000 | EP1051397A1 Method for preparing an n- (aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound |
11/15/2000 | EP1051176A1 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS |
11/15/2000 | CN1273584A Imidazolyl-cyclic acetals |
11/15/2000 | CN1058495C Polycyclic systems compound and derivatives thereof as neurotransmitter release enhancers useful in the treatment of cognitive disordes and medicine containing them and its use |
11/15/2000 | CN1058490C Tetrazolinone derivatives |
11/14/2000 | US6147232 Process of making 3-phenyl-1-methylenedioxyphenyl-indane-2-carboxylic acid derivatives |
11/14/2000 | US6147188 Irreversible cathepsin or calpain inhibitors |
11/14/2000 | US6147111 Kidney, brain, and cardiovascular disorders; vasodilation |
11/14/2000 | US6147110 Heterocyclic compounds |
11/14/2000 | US6147105 Use in the treatment of estrogen-related diseases |
11/14/2000 | US6147083 Novel substituted 1,2-ethanediamine derivatives which antagonize the pharmacological actions of the endogenous neuropeptide tachykinins known as neurokinins, useful for the treatment of asthma, etc. |
11/14/2000 | US6147080 Inhibitors of p38 |
11/14/2000 | US6147077 2R,4S-hydroxyitraconazole isomers |
11/14/2000 | CA2012432C N-(3-hydroxy-4piperidinyl)(dihydrobenzofuran, dihydro-2h-benzopyran or dihydrobenzodioxin) carboxamide derivatives |
11/09/2000 | WO2000066589A1 6-alkenyl-, 6-alkinyl- and 6-epoxy-epothilone derivatives, process for their production, and their use in pharmaceutical preparations |
11/09/2000 | WO2000066580A2 Antifungal ethers |
11/09/2000 | WO2000066568A1 Pesticidal triazine derivatives |
11/09/2000 | WO2000066563A1 Imidazoline derivatives as alpha-1a adrenoceptor ligands |
11/09/2000 | WO2000066562A1 Pyrazoles having antiinflammatory activity |
11/09/2000 | WO2000066559A1 Piperidine derivatives useful as ccr5 antagonists |
11/09/2000 | WO2000066558A1 Piperazine derivatives useful as ccr5 antagonists |
11/09/2000 | WO2000066556A1 Indoline derivatives as progesterone antagonists |
11/09/2000 | WO2000066551A1 Cyclic amide compounds, process for the preparation of the same and uses thereof |
11/09/2000 | WO2000066170A1 Prucalopride oral solution |
11/09/2000 | WO2000066120A1 Novel catechols as antimicrobial agents |
11/09/2000 | WO2000066119A1 Novel prolines as antimicrobial agents |
11/09/2000 | WO2000066112A1 Cxcr-4 receptor antagonists - thrombopoietin mimetics |
11/09/2000 | WO2000066104A2 Ace-2 inhibiting compounds and methods of use thereof |
11/09/2000 | WO2000066100A2 2r,4s-hydroxyitraconazole isomers |
11/09/2000 | WO2000038718A3 Use of matrix metalloproteinase inhibitor together with an antineoplastic agents, optionally also together with radiation, in the treatment of neoplasia |
11/09/2000 | WO2000035906A3 4- and 5-alkynyloxindoles and 4- and 5-alkenyloxindoles |
11/09/2000 | DE19920936A1 Heterozyklisch substituierte Benzimidazole, deren Herstellung und Anwendung Heterocyclic substituted benzimidazoles, their preparation and application |
11/09/2000 | DE19920551A1 Substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen Substituted benzimidazoles, their preparation and their use as agents against parasitic protozoa |
11/09/2000 | DE10021568A1 New pyrimidinyl aryl sulfoxide or sulfone derivatives useful as herbicides and plant growth inhibitors |
11/09/2000 | CA2372595A1 Contraceptive compositions containing indoline derivatives and progestational agents |
11/09/2000 | CA2372387A1 Ace-2 inhibiting compounds and methods of use thereof |
11/09/2000 | CA2372176A1 Novel prolines as antimicrobial agents |
11/09/2000 | CA2372079A1 Novel catechols as antimicrobial agents |
11/09/2000 | CA2371638A1 Indoline derivatives as progesterone antagonists |
11/09/2000 | CA2371629A1 3,3-substituted indoline derivatives |
11/09/2000 | CA2371618A1 Cyclic amide compounds, their production and use |
11/09/2000 | CA2369357A1 2r,4s-hydroxyitraconazole isomers |
11/08/2000 | EP1049700A1 Chemokine receptor antagonists and methods of use therefor |
11/08/2000 | EP1049691A1 Substituted 5-(2,2-difluoro-1,3-benzodioxol-5-yl) cyclopentenopyridine derivative |
11/08/2000 | EP1049680A1 Substituted aminoalkylidenamino triazines as herbicides |
11/08/2000 | EP1049676A1 4- aryl(piperidin-4-yl)] aminobenzamides which bind to the delta-opioid receptor |
11/08/2000 | EP1049675A1 Chemokine receptor antagonists and methods of use therefor |
11/08/2000 | EP1049674A1 Method for producing (-)cis-3-hydroxy-1-methyl-4-(2,4,6-trimethoxyphenyl)-piperidine |
11/08/2000 | EP1049673A1 Heterocyclic amidines as callicrein protease inhibitors |