Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
12/2000
12/26/2000US6166017 Method of using ketoconazole and related substances in medicaments for treatment of type II diabetes and methods of treating same
12/26/2000US6166015 Pyrrolidine derivatives-CCR-3 receptor antagonists
12/26/2000US6166008 Treatment of schizophrenia with ampakines and neuroleptics
12/26/2000US6166006 Having antagonistic activity on mcp-1 (monocyte chemoattractant protein-1) receptor; antiinflammatory agents
12/26/2000US6166005 Heterocyclic metalloprotease inhibitors
12/26/2000US6165996 Compounds with chelation affinity selectivity for first transition series elements: use in medical therapy and diagnosis
12/26/2000US6165944 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
12/26/2000US6165941 Substituted 2-phenylpyridines
12/26/2000US6165729 Electrochemiluminescent reaction utilizing amine-derived reductant
12/26/2000US6164282 Methods for restoring and/or enhancing accommodation in pseudo phakia
12/26/2000CA2203494C Energy transfer dyes with enhanced fluorescence
12/21/2000WO2000077027A2 Serine protease inhibitors
12/21/2000WO2000076993A1 Benzazepine derivatives, process for the preparation of the same and uses thereof
12/21/2000WO2000076984A2 Novel compounds, their use and preparation
12/21/2000WO2000076983A1 1-(4-arylsulfonyl)-3-substituted-5-aryl-2-pyrazolines as inhibitors of cyclooxygenase-2
12/21/2000WO2000076980A1 Novel nitrogen-contaiing heterocyclic derivatives or salts thereof
12/21/2000WO2000076979A1 Pyridine carboxamides and their use as plant protection agents
12/21/2000WO2000076972A1 N-cyclopentyl modulators of chemokine receptor activity
12/21/2000WO2000076971A2 Serine protease inhibitors
12/21/2000WO2000076970A2 Serine protease inhibitors
12/21/2000WO2000076966A2 Indolinylamide derivatives and the use thereof as antiviral drugs
12/21/2000WO2000076521A1 Antiviral indoleoxoacetyl piperazine derivatives
12/21/2000WO2000053597A3 Benzofuran-2-ones as colorants for organic materials
12/21/2000WO2000053579A3 Solid phase synthesis of 4-aminoproline derivatives and/or combinatorial libraries thereof
12/21/2000DE19927415A1 Indolinylharnstoffderivate Indolinylharnstoffderivate
12/21/2000DE10006210A1 New 5-fluoro-6-phenoxypyrimidine derivatives useful as fungicides and bactericides in agriculture and industry, and as herbicides and pesticides
12/21/2000DE10005039A1 New halopyrimidinyloxyphenyl substituted methoxyimino-acetic acid methyl esters useful as pesticides, especially as fungicides in the protection of plants and materials
12/21/2000CA2383008A1 Compounds
12/21/2000CA2380860A1 Benzazepine derivative, production and use thereof
12/21/2000CA2375920A1 Compounds
12/21/2000CA2340663A1 Antiviral indoleoxoacetyl piperazine derivatives
12/20/2000EP1061080A1 Optically active epoxy compound
12/20/2000EP1061073A1 (R-(R*R*))-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl-3-phenyl-4((phenylamino)-carbonyl)-1H-pyrrole-1-heptanoic acid, its lactone form and salts thereof
12/20/2000EP1061072A1 Pyrrolic compounds with a high herbicidal activity and their agronomic use
12/20/2000EP1060178A1 Heterocyclic compounds as inhibitors of rotamase enzymes
12/20/2000EP1060177A1 Method for producing doxazodin mesylate in a crystal modification designated as form a and intermediate product for producing the same
12/20/2000EP1060176A1 Oxyranyle-triazoline thiones and their use as microbicides
12/20/2000EP1060170A1 Optically active substituted 2,4-diamino-1,3,5-triazines as herbicides
12/20/2000EP1060167A1 Novel unsymmetrically substituted carboxylic acid derivatives, method for producing them, and their use as mixed et a?/et b?-receptor antagonists
12/20/2000EP1060166A1 Five-membered, benzo-condensed heterocycles used as antithrombotic agents
12/20/2000EP1060163A1 New piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides
12/20/2000CN1277609A Oxyranyle-triazoline thiones and their use as microbicides
12/20/2000CN1277605A Arylpyridazinones as prostaglandin endoperoxide H synthase biosynthesis inhibitors
12/20/2000CN1277604A Heteraryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
12/19/2000US6162927 (2s,3r,4s)-2-(2,2-dimethylpentyl)-4-(7-methoxy-1,3-benzodioxol-5-yl)-1-(n,n-di(n-butyl)aminocarbonylmethyl)-pyrrolidine-3-carboxylic acid, or salt or ester thereof, in pure form; adminstering to treat hypertension, other diseases
12/19/2000US6162920 Taxane derivatives having a pyridyl substituted C13 side chain, their preparation and their use as anti-tumor agents
12/19/2000US6162918 Tetramethylacridinedione derivatives are inhibitors of herpes simplex virus thymidine kinase in the treatment and prophylaxis of infections caused by herpes simplex virus.
12/19/2000US6162819 Pyrazole derivatives, their preparation and their use in pharmaceuticals
12/19/2000US6162809 Pyridylthio compounds for controlling helicobacter bacteria
12/19/2000US6162808 Compounds
12/19/2000US6162800 N-(pyrimidinyl)-aspartic acid analogs as interleukin-1β converting enzyme inhibitors
12/19/2000US6162798 Cerebrovascular contraction after subarachnoid hemorrhage with quinoline compounds
12/19/2000US6162765 Herbicides and antigrowth agents
12/19/2000CA2184822C Intranasal antimigraine composition
12/19/2000CA2159787C Dibenzofuran aromatic derivatives; pharmaceutical and cosmetic compositions containing the same
12/14/2000WO2000075238A1 Chromene compounds
12/14/2000WO2000075137A1 Pyrrolidinyl, piperidinyl or homopiperidinyl substituted (benzodioxan, benzofuran or benzopyran) derivatives
12/14/2000WO2000075136A1 Aminoalkyl substituted (benzodioxan, benzofuran or benzopyran) derivatives
12/14/2000WO2000075133A1 Novel isoquinoline derivatives or salts thereof
12/14/2000WO2000075131A1 Substituted pyrazole compounds
12/14/2000WO2000075130A1 Indolylpiperidine derivatives as antihistaminic and antiallergic agents
12/14/2000WO2000075127A1 Tricyclic fused heterocycle compounds, process for preparing the same and use thereof
12/14/2000WO2000075123A1 Substituted 5-oxo-5,6,7,8-tetrahydro-4h-1-benzopyrans and benzothiopyrans and the use thereof as potentiators of ampa
12/14/2000WO2000075122A1 Novel processes for the preparation of substituted propenone derivatives
12/14/2000WO2000075119A2 Substituted 2-aryl-1,2,4-triazine-3,5-di(thi)ones used as herbicides
12/14/2000WO2000075114A1 Beta2-adrenoceptor agonists
12/14/2000WO2000075111A1 Formazan metal complex
12/14/2000WO2000074681A1 Metalloprotease inhibitors
12/14/2000WO2000074679A1 Substituted piperidines as melanocortin-4 receptor agonists
12/14/2000WO2000043032A3 Baff, inhibitors thereof and their use in the modulation of b-cell response
12/14/2000DE19958166A1 Pyridincarbamide Pyridincarbamide
12/14/2000CA2377369A1 Substituted piperidines as melanocortin-4 receptor agonists
12/14/2000CA2376043A1 Novel processes for the preparation of substituted propenone derivatives
12/14/2000CA2375985A1 Indolylpiperidine derivatives as antihistaminic and antiallergic agents
12/14/2000CA2375942A1 Substituted 2-aryl-1,2,4-triazine-3,5-di(thi)ones
12/14/2000CA2375882A1 Metalloprotease inhibitors
12/14/2000CA2370013A1 Tricyclic fused heterocycle compounds, process for preparing the same and use thereof
12/13/2000EP1058686A1 2'-fluoronucleosides
12/13/2000EP1058684A1 Glycine transport inhibitors
12/13/2000EP1058680A1 2-arylethyl-(piperidin-4-ylmethyl)amine derivatives as muscarinic receptor antagonists
12/13/2000CN1276370A Process for preparing anticancer compound, and intermediate
12/13/2000CN1276211A Use of non-peptides NK3-antagonist
12/12/2000US6159982 Treating psychological disorders, schizophrenia
12/12/2000US6159980 Anxiolytic agents, antidepressants; psychological and eating disorders
12/12/2000US6159979 Bicyclic aryl or a bicyclic heterocyclic ring containing compounds having a combined 5HT1A, 5HT1B and 5HT1D receptor antagonistic activity
12/12/2000US6159978 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
12/12/2000US6159974 LDL receptor gene expression promoters
12/12/2000US6159964 Vitronectin receptor antagonists
12/12/2000CA2167397C Indoles
12/12/2000CA2011087C Use of trifluoromethylphenylazolylmethyloxiranes as crop protection agents
12/07/2000WO2000073298A1 Mutual prodrugs of amlodipine and atorvastatin
12/07/2000WO2000073284A2 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
12/07/2000WO2000073269A2 Nicotine receptor ligands
12/07/2000WO2000072832A2 Novel use of 1-[4-(cyanoindol-3yl)butyl]-4-(carbamoyl-benzofuran-5yl)-piperazine and its physiologically acceptable salts
12/07/2000WO2000072815A1 Indole derivatives
12/07/2000DE19925593A1 Substituierte 2-Aryl-1,2,4-triazin-3,5-di(thi)one Substituted 2-aryl-1,2,4-triazine-3,5-di (thi) ones
12/07/2000CA2694866A1 Novel use of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts
12/07/2000CA2370141A1 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
12/06/2000EP1057826A1 Substituted dimeric carboxamide derivatives, method for preparing them, and pharmaceutical compositions containing them
12/06/2000EP1057814A1 Tetrahydrobenzindole derivatives